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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-fluoro-3-{4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1-(2,2,2-trifluoroethyl)-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one 1231190-23-0 C23H18F4N6O2
6-fluoro-3-{4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1-(2,2,2-trifluoroethyl)-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one
—— 6-{4-[(2-chlorobenzyl)amino]phenyl}-N-[3-(4-methylpiperazin-1-yl)propyl]-5,6-dihydrobenzo[h]quinazolin-2-amine 1234356-41-2 C33H37ClN6
6-{4-[(2-chlorobenzyl)amino]phenyl}-N-[3-(4-methylpiperazin-1-yl)propyl]-5,6-dihydrobenzo[h]quinazolin-2-amine
—— 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(tetrahydropyran-4-yloxy)pyrimidin-2-yl]benzyl}-2H-pyridazin-3-one 1103506-52-0 C24H24N6O3
6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(tetrahydropyran-4-yloxy)pyrimidin-2-yl]benzyl}-2H-pyridazin-3-one
—— —— 130971-38-9 C24H20B*C52H96ClOsP4
—— —— 1415242-38-4 C26H25Cl2F3N4O4
—— ethyl 2-(3-(4-chlorobenzo[d]thiazole-2-yl)thioureido)acetate 1233692-59-5 C12H12ClN3O2S2
ethyl 2-(3-(4-chlorobenzo[d]thiazole-2-yl)thioureido)acetate
—— (S)-1-(4-chloro-phenyl)-pyrrolidine-2-carboxylic acid (5,5-dimethyl-3-oxo-cyclohex-1-enyl)-amide 1234314-40-9 C19H23ClN2O2
(S)-1-(4-chloro-phenyl)-pyrrolidine-2-carboxylic acid (5,5-dimethyl-3-oxo-cyclohex-1-enyl)-amide
—— 4-{4-[(4'-chloro-1,1'-biphenyl-2-yl)methyl]piperazin-1-yl}-N-{[5-(1,3-dimethyl-1H-pyrazol-5-yl)isoxazol-4-yl]sulfonyl}benzamide 1235865-36-7 C32H31ClN6O4S
4-{4-[(4'-chloro-1,1'-biphenyl-2-yl)methyl]piperazin-1-yl}-N-{[5-(1,3-dimethyl-1H-pyrazol-5-yl)isoxazol-4-yl]sulfonyl}benzamide
—— 3-benzyl-6-methyl-2H-1,3-benzoxazine-2,4(3H)-dithione 1233944-40-5 C16H13NOS2
3-benzyl-6-methyl-2H-1,3-benzoxazine-2,4(3H)-dithione
—— —— 1415571-81-1 C25H29ClN4O3
—— lithium 2-[(1R,5S,6s)-6-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-azabicyclo[3.1.0]hex-3-yl]-4-(2-ethoxybenzyl)-1,3-thiazole-5-carboxylate 1206909-73-0 C24H23Cl2N4O4S*Li
lithium 2-[(1R,5S,6s)-6-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-azabicyclo[3.1.0]hex-3-yl]-4-(2-ethoxybenzyl)-1,3-thiazole-5-carboxylate
—— —— 1414776-52-5 C29H30F2N2O3S
—— —— 1444175-02-3 C26H21Cl2F3N2O2S
—— —— 1342806-98-7 C36H55N5O3Si
—— —— 1414777-64-2 C24H20F4N2O3S
—— —— 1363285-83-9 C28H32N4O2
—— —— 1413284-72-6 C24H17Cl3F3N3O2S
—— —— 1404536-45-3 C31H38N6O3*ClH
—— —— 1192426-77-9 C19H26FN3O2S
—— 8,8-dimethyl-3-(4-(pyridin-2-yl)thiazol-2-yl)-8,9-dihydro-6H-pyrido[2,1-b]quinazolin-11(7H)-one 1416011-76-1 C22H20N4OS
8,8-dimethyl-3-(4-(pyridin-2-yl)thiazol-2-yl)-8,9-dihydro-6H-pyrido[2,1-b]quinazolin-11(7H)-one
—— 6-fluoro-1H-indazole-3-carboxylic acid ((S)-2-fluoro-4-morpholin-2-yl-phenyl)amide 1415756-04-5 C18H16F2N4O2
6-fluoro-1H-indazole-3-carboxylic acid ((S)-2-fluoro-4-morpholin-2-yl-phenyl)amide
—— N-[6-amino-5-(2,3,5-trichlorophenyl)pyridin-2-yl]-1-methyl-1,2,3-triazole-5-carboxamide 1079400-87-5 C15H11Cl3N6O
N-[6-amino-5-(2,3,5-trichlorophenyl)pyridin-2-yl]-1-methyl-1,2,3-triazole-5-carboxamide
—— 8-methyl-12-oxo-N'-picolinoyl-6,7,8,9,10,12-hexahydroazepino[2,1-b]quinazoline-3-carbohydrazide 1416011-63-6 C21H21N5O3
8-methyl-12-oxo-N'-picolinoyl-6,7,8,9,10,12-hexahydroazepino[2,1-b]quinazoline-3-carbohydrazide
—— tert-butyl 4'-((2,3-dimethyl-5-((2-phenylpropan-2-yl)carbamoyl)-1H-indol-1-yl)methyl)-[1,1'-biphenyl]-2-carboxylate 1415256-55-1 C38H40N2O3
tert-butyl 4'-((2,3-dimethyl-5-((2-phenylpropan-2-yl)carbamoyl)-1H-indol-1-yl)methyl)-[1,1'-biphenyl]-2-carboxylate
—— (2S)-1-[(11cR)-10-(trifluoromethyl)-1,2,3,5,6,11c-hexahydroindolizino[7,8-b]indol-7-yl]-2-(4-pyridyl)propan-2-ol 1570094-54-0 C23H24F3N3O
(2S)-1-[(11cR)-10-(trifluoromethyl)-1,2,3,5,6,11c-hexahydroindolizino[7,8-b]indol-7-yl]-2-(4-pyridyl)propan-2-ol
—— 6-(((3R,4R)-4-((5-(3-amino-5-methylphenyl)pentyl)oxy)pyrrolidin-3-yl)methyl)-4-methylpyridin-2-amine 1402971-59-8 C23H34N4O
6-(((3R,4R)-4-((5-(3-amino-5-methylphenyl)pentyl)oxy)pyrrolidin-3-yl)methyl)-4-methylpyridin-2-amine
—— [3-(3-ethyl-ureido)-isoquinolin-8-ylmethyl]-carbamic acid benzyl ester 1401310-26-6 C21H22N4O3
[3-(3-ethyl-ureido)-isoquinolin-8-ylmethyl]-carbamic acid benzyl ester
—— tert-butyl methyl((2S,3S)-3-methyl-1-oxo-1-((3aS,4R,6aR)-2-(3-(trifluoromethyl)phenylsulfonyl)octahydrocyclopenta[c]pyrrol-4-ylamino)pentan-2-yl)carbamate 1228027-19-7 C26H38F3N3O5S
tert-butyl methyl((2S,3S)-3-methyl-1-oxo-1-((3aS,4R,6aR)-2-(3-(trifluoromethyl)phenylsulfonyl)octahydrocyclopenta[c]pyrrol-4-ylamino)pentan-2-yl)carbamate
—— 3-(morpholin-4-ylcarbonyl)-1-[1-(tetrahydro-2H-pyran-4-yl)azepan-4-yl]-1,4-dihydrochromeno[4,3-c]pyrazole 5,5-dioxide 1305271-96-8 C26H34N4O5S
3-(morpholin-4-ylcarbonyl)-1-[1-(tetrahydro-2H-pyran-4-yl)azepan-4-yl]-1,4-dihydrochromeno[4,3-c]pyrazole 5,5-dioxide
—— N1-[(3aS,4R,6aR)-2-benzyloctahydrocyclopenta[c]pyrrol-4-yl]-N2-neopentyl-L-norvalinamide 1228026-31-0 C24H39N3O
N1-[(3aS,4R,6aR)-2-benzyloctahydrocyclopenta[c]pyrrol-4-yl]-N2-neopentyl-L-norvalinamide
—— 4-benzyloxymethyl-1-{4-[5-(2-chlorobiphenyl-4-yl)-1,2,4-oxadiazol-3-yl]benzyl}piperidine-4-carboxylic acid tert-butylamine 1403232-47-2 C4H11N*C35H32ClN3O4
4-benzyloxymethyl-1-{4-[5-(2-chlorobiphenyl-4-yl)-1,2,4-oxadiazol-3-yl]benzyl}piperidine-4-carboxylic acid tert-butylamine
—— 2-(4-fluorobenzyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-6-carboxylic acid 1354633-92-3 C14H9FN2O3S
2-(4-fluorobenzyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-6-carboxylic acid
—— 4-[2-(cyclobutylmethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine 1403988-17-9 C22H23FN4O3S
4-[2-(cyclobutylmethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine
—— 1-[1-(3,3-dimethylbutyl)piperidin-3-yl]-3-(morpholin-4-ylcarbonyl)-1,4-dihydrothiochromeno[4,3-c]pyrazole 5,5-dioxide 1305268-68-1 C26H36N4O4S
1-[1-(3,3-dimethylbutyl)piperidin-3-yl]-3-(morpholin-4-ylcarbonyl)-1,4-dihydrothiochromeno[4,3-c]pyrazole 5,5-dioxide
—— N,N-dimethyl-2-{3-[3-(morpholin-4-ylcarbonyl)-5,5-dioxidothiochromeno[4,3-c]pyrazol-1(4H)-yl]piperidin-1-yl}ethanamide 1305268-74-9 C24H33N5O4S
N,N-dimethyl-2-{3-[3-(morpholin-4-ylcarbonyl)-5,5-dioxidothiochromeno[4,3-c]pyrazol-1(4H)-yl]piperidin-1-yl}ethanamide
—— 4-[4-fluoro-2-(pentyloxy)phenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine 1403988-06-6 C22H25FN4O3S
4-[4-fluoro-2-(pentyloxy)phenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine
—— 5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]-2-(tetrahydro-2H-pyran-4-yloxy)benzonitrile 1403247-17-5 C21H19N5O2
5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]-2-(tetrahydro-2H-pyran-4-yloxy)benzonitrile
—— 1-{4-[4-(4-methylphenyl)-6-morpholin-4-yl-1,3,5-triazin-2-yl]phenyl}-3-[4-(piperidin-1-ylcarbonyl)phenyl]urea 1197166-32-7 C33H35N7O3
1-{4-[4-(4-methylphenyl)-6-morpholin-4-yl-1,3,5-triazin-2-yl]phenyl}-3-[4-(piperidin-1-ylcarbonyl)phenyl]urea
—— 3-[3-isopropyl-8-(trifluoromethyl)quinolin-4-yl]phenyl 2-methyl-5-(methylsulfonyl)benzoate 1354628-49-1 C28H24F3NO4S
3-[3-isopropyl-8-(trifluoromethyl)quinolin-4-yl]phenyl 2-methyl-5-(methylsulfonyl)benzoate
—— 2-methylthio-3-phenyl-naphtho[2,3-b]furan-4,9-dione 1361227-30-6 C19H12O3S
2-methylthio-3-phenyl-naphtho[2,3-b]furan-4,9-dione
—— N-[(S)-1-((3aS,6S,6aS)-6-fluoro-3-oxo-hexahydro-furo[3,2-b]pyrrole-4-carbonyl)-3-methyl-butyl]-4-[2-(4-methyl-piperazin-1-yl)-thiazol-4-yl]-benzamide L-ascorbate 1015251-95-2 C6H8O6*C27H34FN5O4S
N-[(S)-1-((3aS,6S,6aS)-6-fluoro-3-oxo-hexahydro-furo[3,2-b]pyrrole-4-carbonyl)-3-methyl-butyl]-4-[2-(4-methyl-piperazin-1-yl)-thiazol-4-yl]-benzamide L-ascorbate
—— —— 1055901-31-9 C21H20ClFN2O
—— 1-methyl-1H-imidazole-4-carboxylic acid [4-(3-fluoro-azetidin-1-yl)-cyclohexyl]-(4-fluoro-3-isopropoxy-benzyl)-amide 1031310-84-5 C24H32F2N4O2
1-methyl-1H-imidazole-4-carboxylic acid [4-(3-fluoro-azetidin-1-yl)-cyclohexyl]-(4-fluoro-3-isopropoxy-benzyl)-amide
—— 1-methyl-1H-imidazole-4-carboxylic acid (4-fluoro-3-trifluoromethyl-benzyl)-[4-(3-methanesulfonylamino-azetidin-1-yl)-cyclohexyl]-amide 1031310-46-9 C23H29F4N5O3S
1-methyl-1H-imidazole-4-carboxylic acid (4-fluoro-3-trifluoromethyl-benzyl)-[4-(3-methanesulfonylamino-azetidin-1-yl)-cyclohexyl]-amide
—— 1,2,3-trimethoxy-5-[2-nitro-3-(3,4,5-trimethoxyphenyl)prop-2-enyl]benzene 1393750-77-0 C21H25NO8
1,2,3-trimethoxy-5-[2-nitro-3-(3,4,5-trimethoxyphenyl)prop-2-enyl]benzene
—— 4-(6-(4-(3-(5-(1,3-difluoro-2-methylpropan-2-yl)isoxazol-3-yl)ureido)phenylcarbamoyl)pyridin-3-yloxy)-1,2,2,6,6-pentamethylpiperidinium methanesulfonate 1351521-98-6 CH4O3S*C30H38F2N6O4
4-(6-(4-(3-(5-(1,3-difluoro-2-methylpropan-2-yl)isoxazol-3-yl)ureido)phenylcarbamoyl)pyridin-3-yloxy)-1,2,2,6,6-pentamethylpiperidinium methanesulfonate
—— 6-cyclopropyl-3-(pyrimidin-5-ylamino)pyrazine-2-carboxylic acid [5-(2-hydroxy-2-methyl-propylcarbamoyl)-1-(3,3,3-trifluoro-propyl)-1H-pyrazol-4-yl]amide 1352197-62-6 C23H26F3N9O3
6-cyclopropyl-3-(pyrimidin-5-ylamino)pyrazine-2-carboxylic acid [5-(2-hydroxy-2-methyl-propylcarbamoyl)-1-(3,3,3-trifluoro-propyl)-1H-pyrazol-4-yl]amide
—— (2S,3R,4R,5S,6R)-2-(4-hydroxy-3-((5-phenylthiazol-2-yl)methyl)naphthalen-1-yl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol 1352714-21-6 C26H25NO6S
(2S,3R,4R,5S,6R)-2-(4-hydroxy-3-((5-phenylthiazol-2-yl)methyl)naphthalen-1-yl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
—— N-[[5-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-4H-1,2-oxazol-3-yl]-3-methylthiophen-2-yl]methyl]-3-methylsulfanylpropanamide 1352712-29-8 C20H19Cl2F3N2O2S2
N-[[5-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-4H-1,2-oxazol-3-yl]-3-methylthiophen-2-yl]methyl]-3-methylsulfanylpropanamide
—— 5-[1-(cyclopropylmethyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2-fluorobenzonitrile 1352420-93-9 C18H15FN4O
5-[1-(cyclopropylmethyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2-fluorobenzonitrile