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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-methyl-1-(3-methylthiophen-2-yl)-7-(3-phenylpiperidine-1-carbonyl)-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one 1243156-64-0 C27H25N5O2S
8-methyl-1-(3-methylthiophen-2-yl)-7-(3-phenylpiperidine-1-carbonyl)-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one
—— ethyl 3-[2-[(1R)-1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]propyl]-4-fluorophenyl]propanoate 1232405-80-9 C30H42FNO4
ethyl 3-[2-[(1R)-1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]propyl]-4-fluorophenyl]propanoate
—— (2,5-dioxopyrrolidin-1-yl) 2-(2,5-dioxopyrrolidin-1-yl)oxycarbonyloxyethyl carbonate 122375-06-8 C12H12N2O10
(2,5-dioxopyrrolidin-1-yl) 2-(2,5-dioxopyrrolidin-1-yl)oxycarbonyloxyethyl carbonate
—— 1-[(4-Fluorophenyl)methyl]-6-(3-methylsulfanylanilino)-3-propan-2-yl-1,3,5-triazine-2,4-dione 1239686-71-5 C20H21FN4O2S
1-[(4-Fluorophenyl)methyl]-6-(3-methylsulfanylanilino)-3-propan-2-yl-1,3,5-triazine-2,4-dione
—— tert-butyl (2S)-2-[(4-chloro-3-fluorophenyl)methyl]pyrrolidine-1-carboxylate 1232829-71-8 C16H21ClFNO2
tert-butyl (2S)-2-[(4-chloro-3-fluorophenyl)methyl]pyrrolidine-1-carboxylate
—— 3-((S)-2-((3S,5R,6S)-3-allyl-5-(3-chlorophenyl)-6-(4-chlorophenyl)-3-methyl-2-oxopiperidin-1-yl)butyl)-5,5-dimethyloxazolidin-2-one 1352075-31-0 C30H36Cl2N2O3
3-((S)-2-((3S,5R,6S)-3-allyl-5-(3-chlorophenyl)-6-(4-chlorophenyl)-3-methyl-2-oxopiperidin-1-yl)butyl)-5,5-dimethyloxazolidin-2-one
—— 5-Phenoxypyrazine-2-carboxylic acid 1342960-29-5 C11H8N2O3
5-Phenoxypyrazine-2-carboxylic acid
—— 3-[4-(3,4-Dimethoxyphenyl)piperazin-1-yl]-1-[4-(3-ethoxy-4-nitrophenoxy)piperidin-1-yl]propan-1-one 1247034-80-5 C28H38N4O7
3-[4-(3,4-Dimethoxyphenyl)piperazin-1-yl]-1-[4-(3-ethoxy-4-nitrophenoxy)piperidin-1-yl]propan-1-one
—— 1-[4-(3-Methoxy-4-nitroanilino)piperidin-1-yl]-3-[4-(4-methylphenyl)piperidin-1-yl]propan-1-one 1247033-25-5 C27H36N4O4
1-[4-(3-Methoxy-4-nitroanilino)piperidin-1-yl]-3-[4-(4-methylphenyl)piperidin-1-yl]propan-1-one
—— (2S)-2-(3-(5-(2'-methyl-2-(trifluoromethyl)biphenyl-4-yl)-1,2,4-oxadiazol-3-yl)phenethylamino)propanoic acid 1355158-36-9 C27H24F3N3O3
(2S)-2-(3-(5-(2'-methyl-2-(trifluoromethyl)biphenyl-4-yl)-1,2,4-oxadiazol-3-yl)phenethylamino)propanoic acid
—— 2-(5-chloro-2-fluoro-phenyl)-4-([2,6]naphthyridin-1-yl)-[1,8]naphthyridine 1353967-71-1 C22H12ClFN4
2-(5-chloro-2-fluoro-phenyl)-4-([2,6]naphthyridin-1-yl)-[1,8]naphthyridine
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(cyclopropylcarbamoyl)-6-methylphenyl]-5-[[5-(trifluoromethyl)tetrazol-1-yl]methyl]pyrazole-3-carboxamide 1229656-19-2 C24H18ClF3N10O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(cyclopropylcarbamoyl)-6-methylphenyl]-5-[[5-(trifluoromethyl)tetrazol-1-yl]methyl]pyrazole-3-carboxamide
—— N-(2-methyl-3,4-dihydro-1H-isoquinolin-7-yl)-3-[[[4-(1,2,4-triazol-1-ylmethyl)benzoyl]amino]methyl]benzamide 1354553-99-3 C28H28N6O2
N-(2-methyl-3,4-dihydro-1H-isoquinolin-7-yl)-3-[[[4-(1,2,4-triazol-1-ylmethyl)benzoyl]amino]methyl]benzamide
—— 1-biphenyl-3-yl-3-(4-tert-butyl-benzoyl)-thiourea 1352481-19-6 C24H24N2OS
1-biphenyl-3-yl-3-(4-tert-butyl-benzoyl)-thiourea
—— 2-(2-(4-chlorophenoxy)ethyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one 1354198-80-3 C21H15ClF3N3O3
2-(2-(4-chlorophenoxy)ethyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— 5-(4-methylphenyl)-3-(2-morpholinoethyl)imino-2-(3-pyridyl)amino-3,5-dihydrophenazine 1353732-47-4 C30H30N6O
5-(4-methylphenyl)-3-(2-morpholinoethyl)imino-2-(3-pyridyl)amino-3,5-dihydrophenazine
—— <i>N</i>,<i>N</i>'-bis-(1,3-dimethyl-2,4,6-trioxo-tetrahydro-pyrimidin-5-ylidenemethyl)-<i>o</i>-phenylenediamine 110553-74-7 C20H20N6O6
<i>N</i>,<i>N</i>'-bis-(1,3-dimethyl-2,4,6-trioxo-tetrahydro-pyrimidin-5-ylidenemethyl)-<i>o</i>-phenylenediamine
—— N-benzyl-N-(2-methoxyethyl)-4-oxo-1-propyl-5H-[1,2,4]triazolo[4,3-a]quinoxaline-7-carboxamide 1243157-11-0 C23H25N5O3
N-benzyl-N-(2-methoxyethyl)-4-oxo-1-propyl-5H-[1,2,4]triazolo[4,3-a]quinoxaline-7-carboxamide
—— 3-methoxybenzo[b]naphtho[1,2-d]furan-5-carbonitrile 1079791-90-4 C18H11NO2
3-methoxybenzo[b]naphtho[1,2-d]furan-5-carbonitrile
—— (5R,8S)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-vinylcyclopropyl}-7-[(2S)-2-{[(2S)-2-{[(3,5-dimethylisoxazol-4-yl)sulfonyl]amino}-3,3-dimethylbutanoyl]amino}-3,3-dimethylbutanoyl]-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide 1247708-63-9 C38H58N6O9S2
(5R,8S)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-vinylcyclopropyl}-7-[(2S)-2-{[(2S)-2-{[(3,5-dimethylisoxazol-4-yl)sulfonyl]amino}-3,3-dimethylbutanoyl]amino}-3,3-dimethylbutanoyl]-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide
—— (S)-4-fluoro-N<sup>1</sup>-{4-[2-(methoxymethyl)pyrrolidin-1-yl]-6-propylpyrimidin-2-yl}benzene-1,3-diamine 1394318-65-0 C19H26FN5O
(S)-4-fluoro-N<sup>1</sup>-{4-[2-(methoxymethyl)pyrrolidin-1-yl]-6-propylpyrimidin-2-yl}benzene-1,3-diamine
—— 3-[4-(1,5-dimethylpyrazol-4-yl)triazol-1-yl]-4-methyl-N-[3-[(propan-2-ylamino)methyl]-5-(trifluoromethyl)phenyl]benzamide 1096691-78-9 C26H28F3N7O
3-[4-(1,5-dimethylpyrazol-4-yl)triazol-1-yl]-4-methyl-N-[3-[(propan-2-ylamino)methyl]-5-(trifluoromethyl)phenyl]benzamide
—— adamantan-2-yl-(4-hydroxy-2-methyl-1,1-dioxo-1,2-dihydro-2H-benzo[e][1,2]thiazin-3-yl)-methanone 1242133-68-1 C20H23NO4S
adamantan-2-yl-(4-hydroxy-2-methyl-1,1-dioxo-1,2-dihydro-2H-benzo[e][1,2]thiazin-3-yl)-methanone
—— 2,2-dimethyl-3-(5-(2-methyl-4-(2-propylphenylcarbamoyl)quinolin-7-yl)pyridin-2-yloxy)propanoic acid 1246211-81-3 C30H31N3O4
2,2-dimethyl-3-(5-(2-methyl-4-(2-propylphenylcarbamoyl)quinolin-7-yl)pyridin-2-yloxy)propanoic acid
—— 6-[4-[3-amino-2-(3-oxo-4H-quinoxalin-2-yl)-1H-indole-6-carbonyl]piperazin-1-yl]pyridine-3-carbonitrile 1055897-48-7 C27H22N8O2
6-[4-[3-amino-2-(3-oxo-4H-quinoxalin-2-yl)-1H-indole-6-carbonyl]piperazin-1-yl]pyridine-3-carbonitrile
—— 3-[4-(3,4-dihydropyrimido[1,2-a]benzimidazol-1(2H)-yl)phenyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1353678-83-7 C22H18N6O
3-[4-(3,4-dihydropyrimido[1,2-a]benzimidazol-1(2H)-yl)phenyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— ethyl (4E)-5-{2-[(1R)-1-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}ethyl]phenyl}pent-4-enoate 1356494-01-3 C31H43NO4
ethyl (4E)-5-{2-[(1R)-1-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}ethyl]phenyl}pent-4-enoate
—— 2,6-difluoro-N-[3-[5-[2-[2-methoxy-5-methyl-4-[4-(2-methylsulfonylethyl)piperazin-1-yl]anilino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide 1244644-59-4 C38H42F2N8O6S3
2,6-difluoro-N-[3-[5-[2-[2-methoxy-5-methyl-4-[4-(2-methylsulfonylethyl)piperazin-1-yl]anilino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide
—— 6-{2-[2-(4-cyclopropanesulfonyl-phenyl)-2-(2,4-difluoro-phenoxy)-acetylamino]-thiazol-5-yloxy}-nicotinic acid methyl ester 1328992-73-9 C27H21F2N3O7S2
6-{2-[2-(4-cyclopropanesulfonyl-phenyl)-2-(2,4-difluoro-phenoxy)-acetylamino]-thiazol-5-yloxy}-nicotinic acid methyl ester
—— 1-(4-chloro-benzyl)-3-(4-methyl-benzoyl)-thiourea 1352480-93-3 C16H15ClN2OS
1-(4-chloro-benzyl)-3-(4-methyl-benzoyl)-thiourea
—— (S,E)-N-(3-cyano-4-(3-ethynylphenylamino)-7-(tetrahydrofuran-3-yl-oxy)quinolin-6-yl)-4-(morpholin-4-yl)-but-2-enamide 1351941-76-8 C30H29N5O4
(S,E)-N-(3-cyano-4-(3-ethynylphenylamino)-7-(tetrahydrofuran-3-yl-oxy)quinolin-6-yl)-4-(morpholin-4-yl)-but-2-enamide
—— N-[(2-fluorophenyl)methyl]-N-methyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.5]octane-8-sulfonamide 1384874-40-1 C20H23FN6O2S
N-[(2-fluorophenyl)methyl]-N-methyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.5]octane-8-sulfonamide
—— 5-(1-acetylindolin-5-yl)-4-methyl-3-(4-sulfamoylphenyl)thiophene-2-carboxylic acid 1394374-77-6 C22H20N2O5S2
5-(1-acetylindolin-5-yl)-4-methyl-3-(4-sulfamoylphenyl)thiophene-2-carboxylic acid
—— 5-chloro-3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-1-[(3-methoxyphenyl)methyl]-N-methylsulfonylindole-2-carboxamide 1154598-75-0 C24H19ClN4O6S2
5-chloro-3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-1-[(3-methoxyphenyl)methyl]-N-methylsulfonylindole-2-carboxamide
—— 4-(2-methylpiperidin-4-yl)benzonitrile 1399182-01-4 C13H16N2
4-(2-methylpiperidin-4-yl)benzonitrile
—— (3-Methyl-butyl)-[1-pyridin-3-yl-meth-(Z)-ylidene]-amine 111603-77-1 C11H16N2
(3-Methyl-butyl)-[1-pyridin-3-yl-meth-(Z)-ylidene]-amine
—— 2-Bromo-propionic acid 5-oxo-pentyl ester 107289-60-1 C8H13BrO3
2-Bromo-propionic acid 5-oxo-pentyl ester
—— 3-(4-aminophenyl) [1,3]oxazolo[4,5-b]pyridin-2(3H)-one 1353677-05-0 C12H9N3O2
3-(4-aminophenyl) [1,3]oxazolo[4,5-b]pyridin-2(3H)-one
—— (1R,2S,3R,5R)-5-(hydroxymethyl)-2-methoxy-3-[[6-methyl-2-[[(1R)-1-(4-methylphenyl)ethyl]amino]-5-([1,3]thiazolo[4,5-c]pyridin-2-yl)pyrimidin-4-yl]amino]cyclopentan-1-ol 1208996-70-6 C27H32N6O3S
(1R,2S,3R,5R)-5-(hydroxymethyl)-2-methoxy-3-[[6-methyl-2-[[(1R)-1-(4-methylphenyl)ethyl]amino]-5-([1,3]thiazolo[4,5-c]pyridin-2-yl)pyrimidin-4-yl]amino]cyclopentan-1-ol
—— [4-[(2S)-3-[[(3S,6S,10aS)-3-[[(2S)-1-(benzylamino)-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-5-oxo-2,3,6,7,8,9,10,10a-octahydro-1H-pyrrolo[1,2-a]azocin-6-yl]amino]-2-(dimethylamino)-3-oxopropyl]phenyl]methylphosphonic acid 1233085-37-4 C36H48N7O7P
[4-[(2S)-3-[[(3S,6S,10aS)-3-[[(2S)-1-(benzylamino)-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-5-oxo-2,3,6,7,8,9,10,10a-octahydro-1H-pyrrolo[1,2-a]azocin-6-yl]amino]-2-(dimethylamino)-3-oxopropyl]phenyl]methylphosphonic acid
—— (S)-3-{6,6-dimethyl-5-[4-(1-methylpiperidin-4-yl)phenyl]-4,4-dioxo-5,6-dihydro-4H-4lambda6-[1,4,3]-oxathiazin-2-ylamino}-3-(2-fluorophenyl)propan-1-ol 1397713-33-5 C26H34FN3O4S
(S)-3-{6,6-dimethyl-5-[4-(1-methylpiperidin-4-yl)phenyl]-4,4-dioxo-5,6-dihydro-4H-4lambda6-[1,4,3]-oxathiazin-2-ylamino}-3-(2-fluorophenyl)propan-1-ol
—— ethyl 1-amino-4-chloro-1H-pyrrole-2-carboxylate 1400688-80-3 C7H9ClN2O2
ethyl 1-amino-4-chloro-1H-pyrrole-2-carboxylate
—— 2,2,2-trichloroethyl 2-benzoylindoline-1-carboxylate 1394031-53-8 C18H14Cl3NO3
2,2,2-trichloroethyl 2-benzoylindoline-1-carboxylate
—— [(1,1-dimethylethyl)oxy][4-(8-fluoro-5-methyl-3,4-dihydro-2H-chromen-6-yl)-2-methyl-1-oxo-1,2-dihydro-3-isoquinolinyl]acetic acid 1392200-12-2 C26H28FNO5
[(1,1-dimethylethyl)oxy][4-(8-fluoro-5-methyl-3,4-dihydro-2H-chromen-6-yl)-2-methyl-1-oxo-1,2-dihydro-3-isoquinolinyl]acetic acid
—— methyl 6-(2,6-difluoro-4-(tetrahydro-2H-pyran-4-yloxy)phenyl)picolinate 1395997-17-7 C18H17F2NO4
methyl 6-(2,6-difluoro-4-(tetrahydro-2H-pyran-4-yloxy)phenyl)picolinate
—— rac-(1-methyl-1H-indol-3-yl)-[7-(3-pyrazol-1-ylbenzyl)-4,7-dihydro-5H-thieno[2,3-c]pyridin-6-yl]methanone 1394177-34-4 C27H24N4OS
rac-(1-methyl-1H-indol-3-yl)-[7-(3-pyrazol-1-ylbenzyl)-4,7-dihydro-5H-thieno[2,3-c]pyridin-6-yl]methanone
—— 4-[3-(4-carbamoylphenoxy)propyl]-N-pyridin-3-ylpiperidine-1-carboxamide 1008765-93-2 C21H26N4O3
4-[3-(4-carbamoylphenoxy)propyl]-N-pyridin-3-ylpiperidine-1-carboxamide
—— (R)-tert-butyl 4-((3-carbamoyl-6-(hydrazinecarbonyl)pyrrolo[1,2-b]pyridazin-4-yl)amino)-3,3-dimethylpiperidine-1-carboxylate 1400580-78-0 C21H31N7O4
(R)-tert-butyl 4-((3-carbamoyl-6-(hydrazinecarbonyl)pyrrolo[1,2-b]pyridazin-4-yl)amino)-3,3-dimethylpiperidine-1-carboxylate
—— 3-({[1-(4-fluorophenyl)ethyl][(2-methyl-1H-benzimidazol-5-yl)carbonyl]amino}methyl)benzoic acid 1398583-61-3 C25H22FN3O3
3-({[1-(4-fluorophenyl)ethyl][(2-methyl-1H-benzimidazol-5-yl)carbonyl]amino}methyl)benzoic acid
—— (R)-2-benzyl-1,6-bis((S)-benzyl-2-oxooxazolidin-3-yl)hexane-1,6-dione 1400676-02-9 C33H34N2O6
(R)-2-benzyl-1,6-bis((S)-benzyl-2-oxooxazolidin-3-yl)hexane-1,6-dione