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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(3-{3-[(2-morpholin-4-yl-2-oxoethyl)sulfanyl]-4-(trifluoromethyl)phenyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl)-3-[4-(pyrrolidin-1-ylcarbonyl)piperidin-1-yl]propan-2-ol 1049099-01-5 C32H43F3N6O4S
1-(3-{3-[(2-morpholin-4-yl-2-oxoethyl)sulfanyl]-4-(trifluoromethyl)phenyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl)-3-[4-(pyrrolidin-1-ylcarbonyl)piperidin-1-yl]propan-2-ol
—— 2-(5-(4-bromopyridin-2-yl)-1-(2-fluorobenzyl)-1H-1,2,4-triazol-3-yl)thiazole 1375182-39-0 C17H11BrFN5S
2-(5-(4-bromopyridin-2-yl)-1-(2-fluorobenzyl)-1H-1,2,4-triazol-3-yl)thiazole
—— 5-chloro-N2-(5-cyclopropyl-2-methyl-2H-pyrazol-3-yl)-N4-methylpyrimidine-2,4-diamine 1374825-27-0 C12H15ClN6
5-chloro-N2-(5-cyclopropyl-2-methyl-2H-pyrazol-3-yl)-N4-methylpyrimidine-2,4-diamine
—— 4-(5-isopropyl-2,4-dimethoxyphenyl)-1-(4-n-butyl-phenyl)-1H-1,2,3-triazole 1155371-54-2 C23H29N3O2
4-(5-isopropyl-2,4-dimethoxyphenyl)-1-(4-n-butyl-phenyl)-1H-1,2,3-triazole
—— (2S)-1-[4-(dimethylamino)piperidin-1-yl]-3-{3-[3-{[2-(4-fluoropiperidin-1-yl)ethyl]sulfanyl}-4-(trifluoromethyl)phenyl]-5-(methylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl}propan-2-ol 1049100-11-9 C31H46F4N6O3S2
(2S)-1-[4-(dimethylamino)piperidin-1-yl]-3-{3-[3-{[2-(4-fluoropiperidin-1-yl)ethyl]sulfanyl}-4-(trifluoromethyl)phenyl]-5-(methylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl}propan-2-ol
—— 2-(2-Chloroethyl)-1,4-dioxaspiro[4.4]nonane 1823377-09-8 C9H15ClO2
2-(2-Chloroethyl)-1,4-dioxaspiro[4.4]nonane
—— 3-(Cyclopropylmethyl)pyrrolidine hydrochloride 1707604-64-5 C8H16ClN
3-(Cyclopropylmethyl)pyrrolidine hydrochloride
—— 1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N'-(4-phenoxyphenyl)-1H-pyrrole-2-carbohydrazide 1188476-33-6 C23H16ClF3N4O2
1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N'-(4-phenoxyphenyl)-1H-pyrrole-2-carbohydrazide
—— (2S)-1-(4-fluoropiperidin-1-yl)-3-{3-[3-{[2-(4-fluoropiperidin-1-yl)ethyl]sulfanyl}-4-(trifluoromethyl)phenyl]-5-(methylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl}propan-2-ol 1049099-09-3 C29H40F5N5O3S2
(2S)-1-(4-fluoropiperidin-1-yl)-3-{3-[3-{[2-(4-fluoropiperidin-1-yl)ethyl]sulfanyl}-4-(trifluoromethyl)phenyl]-5-(methylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl}propan-2-ol
—— methyl 1-(2-chloro-4-nitrophenyl)-1H-pyrrole-2-carboxylate 1188446-27-6 C12H9ClN2O4
methyl 1-(2-chloro-4-nitrophenyl)-1H-pyrrole-2-carboxylate
—— methyl 6-[(2-butan-2-yl-6-methoxy-1H-indol-3-yl)methyl]pyridine-2-carboxylate 1262877-40-6 C21H24N2O3
methyl 6-[(2-butan-2-yl-6-methoxy-1H-indol-3-yl)methyl]pyridine-2-carboxylate
—— 6-[(6-fluoro-2-phenyl-1H-indol-3-yl)methyl]pyridine-2-carboxylic acid 1262876-67-4 C21H15FN2O2
6-[(6-fluoro-2-phenyl-1H-indol-3-yl)methyl]pyridine-2-carboxylic acid
—— 6-ethoxy-5-fluoro-2-pyridin-3-yl-1H-indole 1262882-02-9 C15H13FN2O
6-ethoxy-5-fluoro-2-pyridin-3-yl-1H-indole
—— 4-(3,5-difluoro-4-methoxyphenyl)-5-methyl-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine 1375457-13-8 C16H15F2N5O
4-(3,5-difluoro-4-methoxyphenyl)-5-methyl-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
—— 1-(dibenzo[b,d]furan-2-ylmethyl)-6-(3,5-dimethoxypyridin-4-yl)piperidin-2-one 1375093-59-6 C25H24N2O4
1-(dibenzo[b,d]furan-2-ylmethyl)-6-(3,5-dimethoxypyridin-4-yl)piperidin-2-one
—— (4-methoxy-5-trifluoromethylpyrimidin-2-yl)-(3-methyl-1-phenyl-1H-pyrazol-4-yl)amine 1374825-60-1 C16H14F3N5O
(4-methoxy-5-trifluoromethylpyrimidin-2-yl)-(3-methyl-1-phenyl-1H-pyrazol-4-yl)amine
—— 4-(4-chlorobenzylsulfinyl)-1-(ethoxycarbonylmethyloxy)-8-methylimidazo[1,5-d][1,2,4]triazine 179316-91-7 C17H17ClN4O4S
4-(4-chlorobenzylsulfinyl)-1-(ethoxycarbonylmethyloxy)-8-methylimidazo[1,5-d][1,2,4]triazine
—— tert-butyl (1-(4-(3-phenyl-9H-benzo[f]imidazo[1,2-d]pyrido[2,3-b][1,4]diazepin-2-yl)phenyl)cyclobutyl)carbamate 1374263-11-2 C35H33N5O2
tert-butyl (1-(4-(3-phenyl-9H-benzo[f]imidazo[1,2-d]pyrido[2,3-b][1,4]diazepin-2-yl)phenyl)cyclobutyl)carbamate
—— (3aR,5R,6S,7R,7aR)-5-((S)-1-hydroxyethyl)-2-(methyl(propyl)amino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol 1374660-91-9 C12H22N2O4S
(3aR,5R,6S,7R,7aR)-5-((S)-1-hydroxyethyl)-2-(methyl(propyl)amino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol
—— 2-methyl-2'-(2-(pyrrolidin-1-yl)ethyl)-3,3',4,4'-tetrahydro-6,6'-biisoquinoline-1,1'(2H,2'H)-dione hydrochloride 1131218-14-8 C25H29N3O2*ClH
2-methyl-2'-(2-(pyrrolidin-1-yl)ethyl)-3,3',4,4'-tetrahydro-6,6'-biisoquinoline-1,1'(2H,2'H)-dione hydrochloride
—— 1-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(2-fluorobenzyl)-1H-pyrrole-2-carboxamide 1188434-17-4 C18H12ClF4N3O
1-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(2-fluorobenzyl)-1H-pyrrole-2-carboxamide
—— 2-(3-methyl-1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)-1H-pyrazol-4-ylamino)-4-(methylamino)pyrimidine-5-carbonitrile 1374828-30-4 C17H21F3N8
2-(3-methyl-1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)-1H-pyrazol-4-ylamino)-4-(methylamino)pyrimidine-5-carbonitrile
—— 5-chloro-N-(1-isopropyl-3-methyl-1H-pyrazol-4-yl)-4-methoxypyrimidin-2-amine 1374825-09-8 C12H16ClN5O
5-chloro-N-(1-isopropyl-3-methyl-1H-pyrazol-4-yl)-4-methoxypyrimidin-2-amine
—— 3-(2-(1H-indazol-5-ylamino)-5-(trifluoromethyl)pyridin-4-ylamino)-N-methylpicolinamide hydrochloride 1061357-12-7 C20H16F3N7O*ClH
3-(2-(1H-indazol-5-ylamino)-5-(trifluoromethyl)pyridin-4-ylamino)-N-methylpicolinamide hydrochloride
—— 1-(3,5-dichloropyridin-2-yl)-N-{[4-(4-fluorophenoxy)phenyl]methyl}-1H-pyrrole-2-carboxamide 1188477-06-6 C23H16Cl2FN3O2
1-(3,5-dichloropyridin-2-yl)-N-{[4-(4-fluorophenoxy)phenyl]methyl}-1H-pyrrole-2-carboxamide
—— 6-(2-methoxy-6-methylphenyl)-1-(4-(trifluoromethoxy)benzyl)piperidin-2-one 1375095-35-4 C21H22F3NO3
6-(2-methoxy-6-methylphenyl)-1-(4-(trifluoromethoxy)benzyl)piperidin-2-one
—— N-methyl-4-oxo-3,4-dihydrospiro[chromene-2,4-piperidine]-6-carboxylamide 1031416-78-0 C15H18N2O3
N-methyl-4-oxo-3,4-dihydrospiro[chromene-2,4-piperidine]-6-carboxylamide
—— N-(1-{[1-(difluoromethyl)-1H-indol-3-yl]methyl}-4-piperidinyl)-4-methyl-3,5-bis(methyloxy)benzamide 1206885-31-5 C25H29F2N3O3
N-(1-{[1-(difluoromethyl)-1H-indol-3-yl]methyl}-4-piperidinyl)-4-methyl-3,5-bis(methyloxy)benzamide
—— N-[2-oxo-6-(pyridin-3-yl)-2H-pyran-3-yl]-4-methylbenzamide 1294393-92-2 C18H14N2O3
N-[2-oxo-6-(pyridin-3-yl)-2H-pyran-3-yl]-4-methylbenzamide
—— 4-methyl-N-{1-[(1-methyl-1-H-indol-3-yl)methyl]-4-piperidinyl}-3,5-bis(methyloxy)benzamide 1206885-23-5 C25H31N3O3
4-methyl-N-{1-[(1-methyl-1-H-indol-3-yl)methyl]-4-piperidinyl}-3,5-bis(methyloxy)benzamide
—— (S)-2-amino-3-(benzyloxy)-N-(2,2-diethoxyethyl)-N-isopentylpropanamide 1222068-55-4 C21H36N2O4
(S)-2-amino-3-(benzyloxy)-N-(2,2-diethoxyethyl)-N-isopentylpropanamide
—— 3-(9-(1-(2-cyanoacetyl)azetidin-3-yl)-7-methyl-8-oxo-8,9-dihydro-7H-purin-2-yl)pyrazolo[1,5-a]pyridine-5-carbonitrile 1299417-08-5 C20H15N9O2
3-(9-(1-(2-cyanoacetyl)azetidin-3-yl)-7-methyl-8-oxo-8,9-dihydro-7H-purin-2-yl)pyrazolo[1,5-a]pyridine-5-carbonitrile
—— 2-(trifluoromethyl)-1,4,5,6-tetrahydropyrimidin-5-ol hydrochloride 1030379-87-3 C5H7F3N2O*ClH
2-(trifluoromethyl)-1,4,5,6-tetrahydropyrimidin-5-ol hydrochloride
—— N-[6-(2-trifluoromethylphenyl)pyrimidin-4-yl]methanesulfonamide 1207723-44-1 C12H10F3N3O2S
N-[6-(2-trifluoromethylphenyl)pyrimidin-4-yl]methanesulfonamide
—— 4-[2-(2-Aminoethyl)-6-oxo-3,4-dihydropyrazino[1,2-b]indazol-6-ium-1-yl]benzonitrile;2,2,2-trifluoroacetate 1202797-07-6 C2F3O2*C19H18N5O
4-[2-(2-Aminoethyl)-6-oxo-3,4-dihydropyrazino[1,2-b]indazol-6-ium-1-yl]benzonitrile;2,2,2-trifluoroacetate
—— 4-((S)-3-(2-trifluoromethylbenzenesulfonyl)pyrrolidin-1-yl)-6,7-dihydro-5H-cyclopentapyrimidine-2-carbonitrile 1374674-88-0 C19H17F3N4O2S
4-((S)-3-(2-trifluoromethylbenzenesulfonyl)pyrrolidin-1-yl)-6,7-dihydro-5H-cyclopentapyrimidine-2-carbonitrile
—— [(1S,2R,5S)-2-ethenyl-2-methyl-5-prop-1-en-2-ylcyclopentyl]oxy-tri(propan-2-yl)silane 1372714-18-5 C20H38OSi
[(1S,2R,5S)-2-ethenyl-2-methyl-5-prop-1-en-2-ylcyclopentyl]oxy-tri(propan-2-yl)silane
—— N-(5-(4-(3-(trifluoromethoxy)benzyloxy)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide 1206101-10-1 C24H19F3N4O3
N-(5-(4-(3-(trifluoromethoxy)benzyloxy)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide
—— 4-[5-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamino]-N-methyl-benzamide 1206195-06-3 C21H19N5O2
4-[5-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamino]-N-methyl-benzamide
—— [N-(5-chloro1,3-benzoxazol-2-yl)-N-{[4-(2-fluorobenzyloxy)]-3-methoxybenzyl}]propane-1,3-diamine hydrochloride 1206542-77-9 C25H25ClFN3O3*ClH
[N-(5-chloro1,3-benzoxazol-2-yl)-N-{[4-(2-fluorobenzyloxy)]-3-methoxybenzyl}]propane-1,3-diamine hydrochloride
—— furan-2-sulfonic acid [3-(4-pyridin-4-yl-1H-pyrazol-3-yl)-phenyl]-amide 1206833-72-8 C18H14N4O3S
furan-2-sulfonic acid [3-(4-pyridin-4-yl-1H-pyrazol-3-yl)-phenyl]-amide
—— 6-Methyl-4-oxo-4H-thiochromene-2-carboxylic acid ethyl ester 105508-64-3 C13H12O3S
6-Methyl-4-oxo-4H-thiochromene-2-carboxylic acid ethyl ester
—— 1-(6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-c]pyridazin-3-yl)-N<sup>3</sup>-(6-(3-piperidin-1-yl-(E)-propenyl)pyridin-3-yl)-1H-1,2,4-triazole-3,5-diamine 1037626-15-5 C28H31N9
1-(6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-c]pyridazin-3-yl)-N<sup>3</sup>-(6-(3-piperidin-1-yl-(E)-propenyl)pyridin-3-yl)-1H-1,2,4-triazole-3,5-diamine
—— 1-(3-fluoro-4-nitro-phenoxy)-cyclopropanecarboxylic acid tert-butyl ester 1219496-39-5 C14H16FNO5
1-(3-fluoro-4-nitro-phenoxy)-cyclopropanecarboxylic acid tert-butyl ester
—— 8-[2,6-Dichloro-3-(N-acetyl-N-methylamino)benzyloxy]-3-iodo-2-methylimidazo[1,2,a]pyridine 160643-85-6 C18H16Cl2IN3O2
8-[2,6-Dichloro-3-(N-acetyl-N-methylamino)benzyloxy]-3-iodo-2-methylimidazo[1,2,a]pyridine
—— 2-[{2-amino-6-[5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl}(2-fluoro-phenyl)amino]ethanol 1374420-38-8 C23H21FN8O
2-[{2-amino-6-[5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl}(2-fluoro-phenyl)amino]ethanol
—— (R)-4-(3-(1H-pyrazol-1-yl)phenylamino)-2-(4-methyl-1-(methylamino)-1-oxopentan-2-ylamino)-6-oxo-1,6-dihydropyrimidine-5-carboxamide 1374159-78-0 C21H26N8O3
(R)-4-(3-(1H-pyrazol-1-yl)phenylamino)-2-(4-methyl-1-(methylamino)-1-oxopentan-2-ylamino)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
—— (S)-4-fluoro-N-(1-(3-hydroxyazetidin-1-yl)pentan-2-yl)-N,3-di-methylbenzamide 1380101-06-3 C17H25FN2O2
(S)-4-fluoro-N-(1-(3-hydroxyazetidin-1-yl)pentan-2-yl)-N,3-di-methylbenzamide
—— ethyl (Z)-3-ethylidene-2-methyl-4-oxocyclohex-1-ene-1-carboxylate 1247042-25-6 C12H16O3
ethyl (Z)-3-ethylidene-2-methyl-4-oxocyclohex-1-ene-1-carboxylate
—— N-[4.3]paracyclophan-6-yl-acetamide 114619-54-4 C21H25NO
N-[4.3]paracyclophan-6-yl-acetamide