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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-{[(3r,4r)-4-(2-{[2,2-Difluoro-2-(4-Fluorophenyl)ethyl]amino}ethoxy)pyrrolidin-3-Yl]methyl}-4-Methylpyridin-2-Amine 1237495-37-2 C21H27F3N4O
6-{[(3r,4r)-4-(2-{[2,2-Difluoro-2-(4-Fluorophenyl)ethyl]amino}ethoxy)pyrrolidin-3-Yl]methyl}-4-Methylpyridin-2-Amine
—— (3R,7aR)-5'-bromo-6-(4-methylbenzyl)-1H-spiro[imidazo[1,5-c]thiazole-3,3'-indoline]-2',5,7(6H,7aH)-trione 1254366-85-2 C20H16BrN3O3S
(3R,7aR)-5'-bromo-6-(4-methylbenzyl)-1H-spiro[imidazo[1,5-c]thiazole-3,3'-indoline]-2',5,7(6H,7aH)-trione
—— 2-(2-chlorophenyl)-5-(cyclohexylmethyl)-4-methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione 1217798-80-5 C20H22ClN3O2
2-(2-chlorophenyl)-5-(cyclohexylmethyl)-4-methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione
—— (E)-3-(1-(3-(2-chlorophenyl)propyl)-2-oxo-1,2-dihydropyridin-3-yl)-N-hydroxyacrylamide 1257335-18-4 C17H17ClN2O3
(E)-3-(1-(3-(2-chlorophenyl)propyl)-2-oxo-1,2-dihydropyridin-3-yl)-N-hydroxyacrylamide
—— N-(4-methylpyridin-2-yl)-3-(trifluoromethyl)quinoxalin-2-amine 1258454-19-1 C15H11F3N4
N-(4-methylpyridin-2-yl)-3-(trifluoromethyl)quinoxalin-2-amine
—— 2-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-6-N-[(2S)-1-hydroxybutan-2-yl]pyridine-2,6-dicarboxamide 1038406-28-8 C19H21N5O3S
2-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-6-N-[(2S)-1-hydroxybutan-2-yl]pyridine-2,6-dicarboxamide
—— ethyl 2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-methylpiperidin-1-yl]-4-[5-(piperazin-1-yl)pyrazin-2-yl]-1,3-thiazole-5-carboxylate 1229572-77-3 C26H32Cl2N8O3S
ethyl 2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-methylpiperidin-1-yl]-4-[5-(piperazin-1-yl)pyrazin-2-yl]-1,3-thiazole-5-carboxylate
—— 3-(1,3-benzothiazol-2-yl)-2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)propanenitrile 1056889-26-9 C21H17N3OS
3-(1,3-benzothiazol-2-yl)-2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)propanenitrile
—— {4-[8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxalin-2-yl]-2-methyl-phenyl}-(4-methyl-piperazin-1-yl)-methanone 1092499-37-0 C32H33F2N5O2
{4-[8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxalin-2-yl]-2-methyl-phenyl}-(4-methyl-piperazin-1-yl)-methanone
—— 1-(4-(4-(4-chloro-3-methylphenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)prop-2-en-1-one 1092364-62-9 C24H25ClN4O3
1-(4-(4-(4-chloro-3-methylphenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)prop-2-en-1-one
—— (6,7-dimethoxy-2-oxo-1,2,3,4-tetrahydro-[3]quinolyl)-acetic acid 105911-84-0 C13H15NO5
(6,7-dimethoxy-2-oxo-1,2,3,4-tetrahydro-[3]quinolyl)-acetic acid
—— tert-butyl 1'-methyl-2'-oxo-1',2',3,6-tetrahydro-4,4'-bipyridine-1(2H)-carboxylate 1233524-68-9 C16H22N2O3
tert-butyl 1'-methyl-2'-oxo-1',2',3,6-tetrahydro-4,4'-bipyridine-1(2H)-carboxylate
—— ((R)-5-oxotetrahydrofuran-2-yl)methyl 4-((S)-2-((E)-3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)phenylcarbamate 1094104-93-4 C31H28ClN7O6
((R)-5-oxotetrahydrofuran-2-yl)methyl 4-((S)-2-((E)-3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)phenylcarbamate
—— 5-aminocarbonyl-N4-(1,2,2,6,6-pentamethylpiperidin-4-yl)-N2-{3-[5-(2,2,2-trifluoroethyl)thio]-1H-tetrazol-1-yl}phenyl-2,4-pyrimidinediamine 1349483-02-8 C24H31F3N10OS
5-aminocarbonyl-N4-(1,2,2,6,6-pentamethylpiperidin-4-yl)-N2-{3-[5-(2,2,2-trifluoroethyl)thio]-1H-tetrazol-1-yl}phenyl-2,4-pyrimidinediamine
—— 6-(furan-2-yl)-N-(1,3,4-thiadiazol-2-yl)imidazo[1,2-a]pyridine-2-carboxamide 1186087-83-1 C14H9N5O2S
6-(furan-2-yl)-N-(1,3,4-thiadiazol-2-yl)imidazo[1,2-a]pyridine-2-carboxamide
—— 3-hydroxy-3-(3-(2-hydroxy-2-propylpentylthio)phenyl)propanenitrile 1215078-58-2 C17H25NO2S
3-hydroxy-3-(3-(2-hydroxy-2-propylpentylthio)phenyl)propanenitrile
—— 2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-6-methoxy-4-methyl-quinoline-3-carboxamide 1242553-95-2 C21H21FN2O2S
2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-6-methoxy-4-methyl-quinoline-3-carboxamide
—— 2-[4-(5-Bromo-1-benzofuran-3-yl)pyrazol-1-yl]pyridine 1260488-43-4 C16H10BrN3O
2-[4-(5-Bromo-1-benzofuran-3-yl)pyrazol-1-yl]pyridine
—— (S)-4-tert-butyl-3-[(1S,5S)-3,4-dimethyl-2-oxo-5-propylcyclopent-3-enecarbonyl]oxazolidin-2-one 1252612-34-2 C18H27NO4
(S)-4-tert-butyl-3-[(1S,5S)-3,4-dimethyl-2-oxo-5-propylcyclopent-3-enecarbonyl]oxazolidin-2-one
—— 2-ethoxycarbonyl-1-phenyl-3-formylamino-1H-naphtho-[2,1-b]pyran 1258277-78-9 C23H19NO4
2-ethoxycarbonyl-1-phenyl-3-formylamino-1H-naphtho-[2,1-b]pyran
—— 2-[4-[[4-butyl-2-{2-(5-ethylpyridin-2-yl)ethyl}-6-oxo-1,6-dihydropyrimidin-5-yl]methyl]-2,6-dipropylphenoxy]-2-phenylacetic acid 1256779-83-5 C38H47N3O4
2-[4-[[4-butyl-2-{2-(5-ethylpyridin-2-yl)ethyl}-6-oxo-1,6-dihydropyrimidin-5-yl]methyl]-2,6-dipropylphenoxy]-2-phenylacetic acid
—— 3-[(S)-4-(3-chlorobenzoyl)morpholin-3-ylmethyl]-1-methyl-1H-indole-5-carboxylic acid dimethylamide 1258967-99-5 C24H26ClN3O3
3-[(S)-4-(3-chlorobenzoyl)morpholin-3-ylmethyl]-1-methyl-1H-indole-5-carboxylic acid dimethylamide
—— 3-(4-isopropylthiazol-2-yl)-6-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole 1257424-31-9 C18H21N5O3S2
3-(4-isopropylthiazol-2-yl)-6-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (2S)-N-[3-(1-hydroxy-2-methylpropan-2-yl)-1,2-oxazol-5-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]azetidine-2-carboxamide 1258443-23-0 C17H19F3N4O3
(2S)-N-[3-(1-hydroxy-2-methylpropan-2-yl)-1,2-oxazol-5-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]azetidine-2-carboxamide
—— acetic acid (4S)-11-(2-{dimethyl-[(3-phenylureido)-methyl]-silanyl}-ethyl)-4-ethyl-3,13-dioxo-3,4,12,13-tetrahydro-1H-2-oxa-6,12a-diaza-dibenzo[b,h]fluoren-4-yl ester 1142937-24-3 C34H36N4O6Si
acetic acid (4S)-11-(2-{dimethyl-[(3-phenylureido)-methyl]-silanyl}-ethyl)-4-ethyl-3,13-dioxo-3,4,12,13-tetrahydro-1H-2-oxa-6,12a-diaza-dibenzo[b,h]fluoren-4-yl ester
—— 4-chloro-5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid (5-isopropyl-isoxazol-3-yl)-amide 1229452-88-3 C21H19ClN6O3
4-chloro-5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid (5-isopropyl-isoxazol-3-yl)-amide
—— 2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)-3-phenylpropanenitrile 1056889-33-8 C20H18N2O
2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)-3-phenylpropanenitrile
—— (Z)-ethyl 3-(6,6-dimethyl-4-oxo-2-((2-oxo-5-(phenylsulfonamido)indolin-3-ylidene)methyl)-4,5,6,7-tetrahydro-1H-indol-3-yl)propanoate 1235459-08-1 C30H31N3O6S
(Z)-ethyl 3-(6,6-dimethyl-4-oxo-2-((2-oxo-5-(phenylsulfonamido)indolin-3-ylidene)methyl)-4,5,6,7-tetrahydro-1H-indol-3-yl)propanoate
—— [4-(2-ethylpyrimidin-5-yloxy)benzyl]methylamine 1030379-91-9 C14H17N3O
[4-(2-ethylpyrimidin-5-yloxy)benzyl]methylamine
—— sodium [(3S)-6-{[(3S)-7-(2-ethyl-1H-benzimidazol-1-yl)-2,3-dihydro-1-benzofuran-3-yl]amino}-2,3-dihydro-1-benzofuran-3-yl]acetate 1258396-01-8 C27H24N3O4*Na
sodium [(3S)-6-{[(3S)-7-(2-ethyl-1H-benzimidazol-1-yl)-2,3-dihydro-1-benzofuran-3-yl]amino}-2,3-dihydro-1-benzofuran-3-yl]acetate
—— 1-(3-fluoro-5-(6-fluoronaphthalen-2-yl)pyridin-4-yl)ethanol 1308668-40-7 C17H13F2NO
1-(3-fluoro-5-(6-fluoronaphthalen-2-yl)pyridin-4-yl)ethanol
—— (4-(4-chlorophenoxy)piperidin-1-yl)(6-(piperidin-1-yl)pyridin-3-yl)methanone 1304782-57-7 C22H26ClN3O2
(4-(4-chlorophenoxy)piperidin-1-yl)(6-(piperidin-1-yl)pyridin-3-yl)methanone
—— 4-fluoro-3-[[2-[[3-[(2S)-1-methoxypropan-2-yl]oxy-5-(4-methylsulfonylphenoxy)benzoyl]amino]-1,3-thiazol-5-yl]oxy]benzoic acid 1093121-01-7 C28H25FN2O9S2
4-fluoro-3-[[2-[[3-[(2S)-1-methoxypropan-2-yl]oxy-5-(4-methylsulfonylphenoxy)benzoyl]amino]-1,3-thiazol-5-yl]oxy]benzoic acid
—— (E)-3-(5-chloro-2-tetrazol-1-ylphenyl)-N-[(S)-1-(1H-indazol-6-ylcarbamoyl)-2-phenylethyl]acrylamide 1094103-65-7 C26H21ClN8O2
(E)-3-(5-chloro-2-tetrazol-1-ylphenyl)-N-[(S)-1-(1H-indazol-6-ylcarbamoyl)-2-phenylethyl]acrylamide
—— 2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-[2-(trifluoromethyl)phenyl]propanenitrile 1056889-57-6 C22H19F3N2O
2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-[2-(trifluoromethyl)phenyl]propanenitrile
—— N-[2-[3-(dimethylamino)prop-1-ynyl]-5-hydroxy-4-methylphenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide 1233529-47-9 C22H22F3N3O4
N-[2-[3-(dimethylamino)prop-1-ynyl]-5-hydroxy-4-methylphenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
—— p-Tolylsulfonsaeure-<methoxy-diphenyl-phosphoranyliden>-amid 112656-09-4 C20H20NO3PS
p-Tolylsulfonsaeure-<methoxy-diphenyl-phosphoranyliden>-amid
—— [10-Oxo-9-(2,4,6-triethylphenyl)-3-oxaspiro[5.5]undec-8-en-8-yl] 2,2-dimethylpropanoate 1058731-33-1 C27H38O4
[10-Oxo-9-(2,4,6-triethylphenyl)-3-oxaspiro[5.5]undec-8-en-8-yl] 2,2-dimethylpropanoate
—— N-{3-[6-tert-butyl-5-methoxy-8-(6-methyl-2-oxo-1,2-dihydro-pyridin-3-yl)-quinolin-3-yl]-propyl}-methanesulfonamide 1257831-22-3 C24H31N3O4S
N-{3-[6-tert-butyl-5-methoxy-8-(6-methyl-2-oxo-1,2-dihydro-pyridin-3-yl)-quinolin-3-yl]-propyl}-methanesulfonamide
—— 3-methyl-8-(2-methylamino-pyrimidin-5-yl)-1-(5-methyl-pyridin-3-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one 1257430-18-4 C22H19N7O
3-methyl-8-(2-methylamino-pyrimidin-5-yl)-1-(5-methyl-pyridin-3-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one
—— quinolin-6-yl-(5-trifluoromethyl-pyridin-2-yl)-amine 1258420-63-1 C15H10F3N3
quinolin-6-yl-(5-trifluoromethyl-pyridin-2-yl)-amine
—— 4-iodo-5-phenyl-2,3-dihydroselenopheno[2,3-b]selenophene 1256937-55-9 C12H9ISe2
4-iodo-5-phenyl-2,3-dihydroselenopheno[2,3-b]selenophene
—— N-(2-(5-chloro-2-(1-methyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)phenyl)methanesulfonamide 1258943-91-7 C15H16ClN7O2S
N-(2-(5-chloro-2-(1-methyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)phenyl)methanesulfonamide
—— 7-(3-chloro-benzenesulfonyl)-2-cyclohexyl-1,3,7-triaza-spiro[4.5]dec-1-en-4-one 1253915-61-5 C19H24ClN3O3S
7-(3-chloro-benzenesulfonyl)-2-cyclohexyl-1,3,7-triaza-spiro[4.5]dec-1-en-4-one
—— 9-cyclopentyl-2-{[4-(1,1-dioxidothiomorpholin-4-yl)-phenyl]-amino}-7-methyl-7,9-dihydro-8H-purin-8-one 1124329-21-0 C21H26N6O3S
9-cyclopentyl-2-{[4-(1,1-dioxidothiomorpholin-4-yl)-phenyl]-amino}-7-methyl-7,9-dihydro-8H-purin-8-one
—— 2-(tert-butoxy)-2-[3-(4-carbamoylphenyl)-2-(3,4-dihydro-2H-1-benzopyran-6-yl)-6-(trifluoromethyl)phenyl]acetic acid 1596341-26-2 C29H28F3NO5
2-(tert-butoxy)-2-[3-(4-carbamoylphenyl)-2-(3,4-dihydro-2H-1-benzopyran-6-yl)-6-(trifluoromethyl)phenyl]acetic acid
—— 2,3-dichloro-N-(3-(1-(trifluoromethyl)cyclopropyl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)propyl)benzamide 1600497-33-3 C19H15Cl2F6N3O
2,3-dichloro-N-(3-(1-(trifluoromethyl)cyclopropyl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)propyl)benzamide
—— N-((1S,5S)-5-((4-aminophenylsulfonyl)(3-fluoropropyl)amino)-1-ethyl-6-hydroxyhexyl)-Nα-methoxycarbonyl-β-phenyl-L-phenylalaninamide 1138083-62-1 C34H45FN4O6S
N-((1S,5S)-5-((4-aminophenylsulfonyl)(3-fluoropropyl)amino)-1-ethyl-6-hydroxyhexyl)-Nα-methoxycarbonyl-β-phenyl-L-phenylalaninamide
—— 1-[5-fluoro-2-(methylsulfonyl)benzoyl]-4-(1-methyl-1-([3-(trifluoromethoxy)phenyl]sulfonyl)ethyl)piperidine 1138328-40-1 C23H25F4NO6S2
1-[5-fluoro-2-(methylsulfonyl)benzoyl]-4-(1-methyl-1-([3-(trifluoromethoxy)phenyl]sulfonyl)ethyl)piperidine
—— 3-[9-(3-Methylbutan-2-yl)-2-morpholin-4-ylpurin-6-yl]phenol 1138158-80-1 C20H25N5O2
3-[9-(3-Methylbutan-2-yl)-2-morpholin-4-ylpurin-6-yl]phenol