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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-propyl-7-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[4.4]nonane-1-carboxamide 1263773-43-8 C17H24N6O
N-propyl-7-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[4.4]nonane-1-carboxamide
—— (5-phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)thiophen-2-ylmethylamine 1206206-06-5 C15H12N4S2
(5-phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)thiophen-2-ylmethylamine
—— 9-(4-fluorophenyl)-N-(5-(1-piperazinyl)-2-pyridinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine 1169692-10-7 C24H21FN8
9-(4-fluorophenyl)-N-(5-(1-piperazinyl)-2-pyridinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine
—— 1-[2-(Pyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-3-amine 1697038-41-7 C8H15N5
1-[2-(Pyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-3-amine
—— cleromyrine 126594-35-2 C30H44N6O6
cleromyrine
—— 4-Amino-7-methyl-2H-pyrido<1,2-a>pyrimidin-2-one hydrochloride 132371-17-6 C9H9N3O*ClH
4-Amino-7-methyl-2H-pyrido<1,2-a>pyrimidin-2-one hydrochloride
—— US8653087, III-410 1213246-97-9 C25H22F3N7O3
US8653087, III-410
—— US8653087, III-393 1213246-80-0 C23H18F4N8O2
US8653087, III-393
—— tert-butyl N-[(2S)-1-[(2S,4R)-4-[4-(but-3-enylcarbamoyl)-1-propan-2-ylbenzimidazol-2-yl]oxy-2-[[(1R,2R)-1-[(1-but-3-enylcyclopropyl)sulfonylcarbamoyl]-2-ethylcyclopropyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate 1365749-34-3 C44H65N7O9S
tert-butyl N-[(2S)-1-[(2S,4R)-4-[4-(but-3-enylcarbamoyl)-1-propan-2-ylbenzimidazol-2-yl]oxy-2-[[(1R,2R)-1-[(1-but-3-enylcyclopropyl)sulfonylcarbamoyl]-2-ethylcyclopropyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
—— tert-butyl 4-(2-(piperazin-1-yl)ethyl)piperidine-1-carboxylate 198627-75-7 C16H31N3O2
tert-butyl 4-(2-(piperazin-1-yl)ethyl)piperidine-1-carboxylate
—— (4,4-Dimethyl-2-triethylstannylpent-1-en-3-yl)-triethylstannane 135753-19-4 C19H42Sn2
(4,4-Dimethyl-2-triethylstannylpent-1-en-3-yl)-triethylstannane
—— ethyl 3-chloro-2-ethoxycarbonylmethyl-4,6-bis(methoxymethoxy)benzoate 1181236-18-9 C17H23ClO8
ethyl 3-chloro-2-ethoxycarbonylmethyl-4,6-bis(methoxymethoxy)benzoate
—— Ethyl 4,5-dimethyl-6-(5-thiophen-2-ylthiophen-2-yl)phosphinine-2-carboxylate 1292834-42-4 C18H17O2PS2
Ethyl 4,5-dimethyl-6-(5-thiophen-2-ylthiophen-2-yl)phosphinine-2-carboxylate
—— Tert-butyl 4-[benzyl-[2-(1-methylindol-3-yl)ethyl]carbamoyl]-2-oxo-4-prop-2-enyl-3,1-benzoxazine-1-carboxylate 1080409-47-7 C35H37N3O5
Tert-butyl 4-[benzyl-[2-(1-methylindol-3-yl)ethyl]carbamoyl]-2-oxo-4-prop-2-enyl-3,1-benzoxazine-1-carboxylate
—— 1-tetradecyl-1-(3-iodopropargyl)-piperidinium n-butylsulfonate 149964-52-3 C4H9O3S*C22H41IN
1-tetradecyl-1-(3-iodopropargyl)-piperidinium n-butylsulfonate
—— 2-(4-methoxyanilino)-N-methyl-2-naphthalen-2-ylacetamide 1154423-57-0 C20H20N2O2
2-(4-methoxyanilino)-N-methyl-2-naphthalen-2-ylacetamide
—— 6,7-Dichloro-2-pentylsulfonyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one 112588-25-7 C10H11Cl2N3O3S2
6,7-Dichloro-2-pentylsulfonyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 6-(6-chloropyrazolo[1,5-a]pyridin-3-yl)-N-[(3R,5R)-5-methylpyrrolidin-3-yl]pyrazin-2-amine 1207850-85-8 C16H17ClN6
6-(6-chloropyrazolo[1,5-a]pyridin-3-yl)-N-[(3R,5R)-5-methylpyrrolidin-3-yl]pyrazin-2-amine
—— tert-butyl 2-[3-({4-[4-amino-2-(2-methoxyethyl)-1H-imidazo[4,5-c]quinolin-1-yl]butylamino}methyl)phenoxy]acetate 1310696-89-9 C30H39N5O4
tert-butyl 2-[3-({4-[4-amino-2-(2-methoxyethyl)-1H-imidazo[4,5-c]quinolin-1-yl]butylamino}methyl)phenoxy]acetate
—— [5-(3-chloro-4-fluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-(2-phenoxyethyl)amine 1206203-31-7 C18H14ClFN4OS
[5-(3-chloro-4-fluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-(2-phenoxyethyl)amine
—— 4-[(1S)-1-[[1-[(2-phenyl-1,3-oxazol-4-yl)methyl]indole-7-carbonyl]amino]ethyl]benzoic acid 1196045-44-9 C28H23N3O4
4-[(1S)-1-[[1-[(2-phenyl-1,3-oxazol-4-yl)methyl]indole-7-carbonyl]amino]ethyl]benzoic acid
—— 1-(4-chloro-1,3-benzothiazol-2-yl)-2-(4-fluorophenyl)-4-hydroxy-3-(2-phenoxyacetyl)-2H-pyrrol-5-one 1071950-85-0 C25H16ClFN2O4S
1-(4-chloro-1,3-benzothiazol-2-yl)-2-(4-fluorophenyl)-4-hydroxy-3-(2-phenoxyacetyl)-2H-pyrrol-5-one
—— 2,2-Difluoro-2-(pyrazin-2-yl)acetic acid 1342462-39-8 C6H4F2N2O2
2,2-Difluoro-2-(pyrazin-2-yl)acetic acid
—— 3-(3-Ethyl-1,2,4-oxadiazol-5-yl)cyclopentanamine 1481234-07-4 C9H15N3O
3-(3-Ethyl-1,2,4-oxadiazol-5-yl)cyclopentanamine
—— [(1R,3S,5R,6S,8R,10S,12R,14S,15R,17S)-14-hydroxy-15-(methoxymethyl)-14-methyl-6-(phenylmethoxymethyl)-2,7,11,16-tetraoxatetracyclo[8.8.0.03,8.012,17]octadecan-5-yl] acetate 1174701-26-8 C27H38O9
[(1R,3S,5R,6S,8R,10S,12R,14S,15R,17S)-14-hydroxy-15-(methoxymethyl)-14-methyl-6-(phenylmethoxymethyl)-2,7,11,16-tetraoxatetracyclo[8.8.0.03,8.012,17]octadecan-5-yl] acetate
—— phenyl (E)-3-ethoxy-2-(2-oxaspiro[4.5]dec-3-ylidene)butanoate 1005737-86-9 C21H28O4
phenyl (E)-3-ethoxy-2-(2-oxaspiro[4.5]dec-3-ylidene)butanoate
—— t-Butyl 3-[1-[5-(tetrahydropyran-2-yl)oxy-n-pentyl]oxy-4-(4-N,N-dimethylaminocarbonylbutanamido)benzen-2-yl]propionate 134577-77-8 C30H48N2O7
t-Butyl 3-[1-[5-(tetrahydropyran-2-yl)oxy-n-pentyl]oxy-4-(4-N,N-dimethylaminocarbonylbutanamido)benzen-2-yl]propionate
—— tert-butyl 3-(4-chloro-3-{[(2S,3R)-4,4,4-trifluoro-2-(4-isopropylphenyl)-3-methylbutanoyl]-amino}phenyl)propanoate 1297550-42-5 C27H33ClF3NO3
tert-butyl 3-(4-chloro-3-{[(2S,3R)-4,4,4-trifluoro-2-(4-isopropylphenyl)-3-methylbutanoyl]-amino}phenyl)propanoate
—— 4-(4-methoxybenzyloxy)-6-(2-phenyloxazol-5-yl)-2-(4-trifluoromethylthiazol-2-yl)pyrimidine 1251166-55-8 C25H17F3N4O3S
4-(4-methoxybenzyloxy)-6-(2-phenyloxazol-5-yl)-2-(4-trifluoromethylthiazol-2-yl)pyrimidine
—— (3R)-1-[6-[[8-(3-hydroxypropyl)-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl]amino]pyridazin-3-yl]pyrrolidin-3-ol 1169697-12-4 C20H22N8O2
(3R)-1-[6-[[8-(3-hydroxypropyl)-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl]amino]pyridazin-3-yl]pyrrolidin-3-ol
—— 9-cyclopentyl-N-(6-(4-(2-(methyloxy)ethyl)-1-piperazinyl)-3-pyridazinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine 1169694-37-4 C25H31N9O
9-cyclopentyl-N-(6-(4-(2-(methyloxy)ethyl)-1-piperazinyl)-3-pyridazinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine
—— (3R)-1-[6-[[8-[(2R)-1-hydroxypropan-2-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl]amino]pyridazin-3-yl]pyrrolidin-3-ol 1169697-50-0 C20H22N8O2
(3R)-1-[6-[[8-[(2R)-1-hydroxypropan-2-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl]amino]pyridazin-3-yl]pyrrolidin-3-ol
—— 1-[(8S)-4-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-8-(4-chlorophenyl)-1,4-diazocan-1-yl]-2-methoxyethanone 1207511-15-6 C30H38ClF2N3O3
1-[(8S)-4-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-8-(4-chlorophenyl)-1,4-diazocan-1-yl]-2-methoxyethanone
—— 1-(4-chloro-1,3-benzothiazol-2-yl)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-2H-pyrrol-5-one 1071952-33-4 C25H17ClN2O6S
1-(4-chloro-1,3-benzothiazol-2-yl)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-2H-pyrrol-5-one
—— [5-(3-chloro-4-fluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-(4-methoxybenzyl)-amine 1137143-80-6 C18H14ClFN4OS
[5-(3-chloro-4-fluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-(4-methoxybenzyl)-amine
—— 4-fluoro-N-[3-(4-pyridin-4-yl-1H-pyrazol-3-yl)-phenyl]-benzenesulfonamide 1206833-52-4 C20H15FN4O2S
4-fluoro-N-[3-(4-pyridin-4-yl-1H-pyrazol-3-yl)-phenyl]-benzenesulfonamide
—— (3S)-1-[6-[(8-cyclopentyl-10-fluoro-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl)amino]pyridazin-3-yl]pyrrolidin-3-ol 1169696-69-8 C22H23FN8O
(3S)-1-[6-[(8-cyclopentyl-10-fluoro-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl)amino]pyridazin-3-yl]pyrrolidin-3-ol
—— 2-azido-1-[4-(3-(6-methoxybenzothiazol)-2-yl[1,2,4]oxadiazol-5-yl)piperid-1-yl]ethanone 1001467-74-8 C17H17N7O3S
2-azido-1-[4-(3-(6-methoxybenzothiazol)-2-yl[1,2,4]oxadiazol-5-yl)piperid-1-yl]ethanone
—— propane-1-sulfonic acid {3-[4-(1-ethyl-piperidin-4-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl]-2,4-difluoro-phenyl}-amide 1309433-14-4 C23H28F2N6O3S
propane-1-sulfonic acid {3-[4-(1-ethyl-piperidin-4-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl]-2,4-difluoro-phenyl}-amide
—— 1-(2',3',5'-tri-O-acetyl-α-D-lyxofuranosyl)uracil 107271-83-0 C15H18N2O9
1-(2',3',5'-tri-O-acetyl-α-D-lyxofuranosyl)uracil
—— methyl 3-(4-(2-((tert-butoxycarbonyl)amino)ethyl)phenyl)-5,7-dimethylbenzo[b]thiophene-2-carboxylate 1270930-50-1 C25H29NO4S
methyl 3-(4-(2-((tert-butoxycarbonyl)amino)ethyl)phenyl)-5,7-dimethylbenzo[b]thiophene-2-carboxylate
—— 2-(6-(benzyloxy)-2',4',6'-trimethyl-2-oxo-2,3,4,5-tetrahydro-[1,1'-biphenyl]-4-yl)propanal 1612216-88-2 C25H28O3
2-(6-(benzyloxy)-2',4',6'-trimethyl-2-oxo-2,3,4,5-tetrahydro-[1,1'-biphenyl]-4-yl)propanal
—— ethyl 4-(5-(4-chlorophenyl)-1-(N,N-dimethylsulfamoyl)imidazol-4-yl)benzoate 1609648-96-5 C20H20ClN3O4S
ethyl 4-(5-(4-chlorophenyl)-1-(N,N-dimethylsulfamoyl)imidazol-4-yl)benzoate
—— 3,3,3-trifluoro-2-hydroxy-2-(5-benzyloxyindol-3-yl)propionic acid ethyl ester 1374603-33-4 C20H18F3NO4
3,3,3-trifluoro-2-hydroxy-2-(5-benzyloxyindol-3-yl)propionic acid ethyl ester
—— 6-p-tolyl-2-tosyl-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine 1440216-51-2 C21H20N2O2S
6-p-tolyl-2-tosyl-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine
—— 2-[3-[tert-butyl(dimethyl)silyl]oxy-2-oxo-1H-indol-3-yl]acetaldehyde 1251936-68-1 C16H23NO3Si
2-[3-[tert-butyl(dimethyl)silyl]oxy-2-oxo-1H-indol-3-yl]acetaldehyde
—— benzyl N-[(1R,2R)-2-(3-methylbutylamino)cyclohexyl]carbamate 1304774-67-1 C19H30N2O2
benzyl N-[(1R,2R)-2-(3-methylbutylamino)cyclohexyl]carbamate
—— N-cyclohexyl-N-(n-butyl)-p-toluenesulfonamide 1234690-99-3 C17H27NO2S
N-cyclohexyl-N-(n-butyl)-p-toluenesulfonamide
—— 2-benzyl-1,2-dihydropyrrolo[3,4-b]carbazol-3(5H)-one 1309385-82-7 C21H16N2O
2-benzyl-1,2-dihydropyrrolo[3,4-b]carbazol-3(5H)-one
—— Heptacyclo[22.8.2.03,30.06,19.07,12.013,18.022,27]tetratriaconta-1,3(30),6(19),7,9,11,13,15,17,22(27),23,25,31-tridecaen-20-yn-4-one 1207872-63-6 C34H24O
Heptacyclo[22.8.2.03,30.06,19.07,12.013,18.022,27]tetratriaconta-1,3(30),6(19),7,9,11,13,15,17,22(27),23,25,31-tridecaen-20-yn-4-one