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—— (7R,8aS)-7-[(4-cyclopropylpyrimidin-2-yl)oxy]-2-{[3-(trifluoromethyl)-phenyl]sulfonyl}octahydropyrrolo[1,2-a]pyrazine 1429197-07-8 C21H23F3N4O3S
(7R,8aS)-7-[(4-cyclopropylpyrimidin-2-yl)oxy]-2-{[3-(trifluoromethyl)-phenyl]sulfonyl}octahydropyrrolo[1,2-a]pyrazine
—— 23-N-tert-butyl-6-(4-fluorophenyl)-5-N-methyl-11,20-bis(methylsulfonyl)-7-oxa-11,20-diazatetracyclo[19.3.1.02,10.04,8]pentacosa-1(24),2(10),3,5,8,21(25),22-heptaene-5,23-dicarboxamide 1620064-02-9 C37H45FN4O7S2
23-N-tert-butyl-6-(4-fluorophenyl)-5-N-methyl-11,20-bis(methylsulfonyl)-7-oxa-11,20-diazatetracyclo[19.3.1.02,10.04,8]pentacosa-1(24),2(10),3,5,8,21(25),22-heptaene-5,23-dicarboxamide
—— 5-bromo-N<sup>4</sup>-[(4-methylthiazol-5-yl)methyl]-2-(1H-pyrazolo[4,3-b]pyridin-1-yl)pyrimidine-4,6-diamine 1620909-92-3 C15H13BrN8S
5-bromo-N<sup>4</sup>-[(4-methylthiazol-5-yl)methyl]-2-(1H-pyrazolo[4,3-b]pyridin-1-yl)pyrimidine-4,6-diamine
—— (S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(4-(N-methaneylaminosulfonyl)phenylsulfonylamino)ethanoyloxy)ethyl)pyridine-1-oxide 1428849-24-4 C27H27Cl2F2N3O9S2
(S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(4-(N-methaneylaminosulfonyl)phenylsulfonylamino)ethanoyloxy)ethyl)pyridine-1-oxide
—— N-[2-(7-dodecoxy-1H-indol-3-yl)ethyl]acetamide 1432472-93-9 C24H38N2O2
N-[2-(7-dodecoxy-1H-indol-3-yl)ethyl]acetamide
—— ethyl (tert-butoxycarbonylamino)-3-(2,2-dimethyl-4-oxo-4H-1,3-dioxin-6-yl)propanoate 1173933-65-7 C16H25NO7
ethyl (tert-butoxycarbonylamino)-3-(2,2-dimethyl-4-oxo-4H-1,3-dioxin-6-yl)propanoate
—— N-(3-fluorophenyl)-2-(3-(7-(4-(4-methylpiperazine-1-carbonyl)phenyl)quinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 1186390-12-4 C31H29FN8O2
N-(3-fluorophenyl)-2-(3-(7-(4-(4-methylpiperazine-1-carbonyl)phenyl)quinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide
—— 4-(6-(cyclohexylamino)pyridin-3-yl)-N-(3-methyl-4-(1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-3-yl)phenyl)pyrimidin-2-amine 1182183-41-0 C32H43N7
4-(6-(cyclohexylamino)pyridin-3-yl)-N-(3-methyl-4-(1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-3-yl)phenyl)pyrimidin-2-amine
—— N-(4-trifluoromethoxybenzyl)-4-[4-(1H-benzotriazol-5-ylcarbamoyl)thiazol-2-yl]piperidine-1-carboxamide 1141395-33-6 C24H22F3N7O3S
N-(4-trifluoromethoxybenzyl)-4-[4-(1H-benzotriazol-5-ylcarbamoyl)thiazol-2-yl]piperidine-1-carboxamide
—— (2-cyclopropyl-benzo[4,5]thieno[2,3-d]pyrimidin-4-yl)-(3-methoxy-phenyl)-amine 1182278-69-8 C20H17N3OS
(2-cyclopropyl-benzo[4,5]thieno[2,3-d]pyrimidin-4-yl)-(3-methoxy-phenyl)-amine
—— (4-{6-[(1S)-1-tert-butoxycarbonylamino-2-(1-methyl-5-methylsulfinyl-1H-pyrazol-3-yl)-ethyl]-3-oxo-2,3-dihydro-pyridazin-4-yl}-phenyl)-carbamic acid methyl ester 1187649-17-7 C24H30N6O6S
(4-{6-[(1S)-1-tert-butoxycarbonylamino-2-(1-methyl-5-methylsulfinyl-1H-pyrazol-3-yl)-ethyl]-3-oxo-2,3-dihydro-pyridazin-4-yl}-phenyl)-carbamic acid methyl ester
—— (4bR,4'S,8aS,9R)-11-(2-fluoroethyl)-8a-hydroxy-3-methoxy-5,7,8,8a,9,10-hexahydrospiro[9,4b-(epiminoethano)phenanthrene-6,4'-imidazolidine]-2',5'-dione 1613736-13-2 C21H26FN3O4
(4bR,4'S,8aS,9R)-11-(2-fluoroethyl)-8a-hydroxy-3-methoxy-5,7,8,8a,9,10-hexahydrospiro[9,4b-(epiminoethano)phenanthrene-6,4'-imidazolidine]-2',5'-dione
—— thiophene-2-carboxylic acid [3-(quinolin-2-ylcarbamoyl)-phenyl]-amide 1185402-89-4 C21H15N3O2S
thiophene-2-carboxylic acid [3-(quinolin-2-ylcarbamoyl)-phenyl]-amide
—— 3-(5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl)-2-quinoxalinamine 1186469-50-0 C16H10FN5O
3-(5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl)-2-quinoxalinamine
—— (E)-N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-3-(3-methoxyphenyl)acrylamide 1185582-51-7 C34H42N6O3
(E)-N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-3-(3-methoxyphenyl)acrylamide
—— ((1S,6S)-6-Methyl-cyclohex-3-enyl)-acetic acid 116996-50-0 C9H14O2
((1S,6S)-6-Methyl-cyclohex-3-enyl)-acetic acid
—— 3-(prop-2-ynyloxy)deca-1,9-diene 1071478-35-7 C13H20O
3-(prop-2-ynyloxy)deca-1,9-diene
—— —— 1402921-96-3 C9H14O2
—— (Z)-4-((4-oxo-3-((trimethylsilyl)methyl)cyclopent-2-en-1-ylidene)(trimethylsilyl)methyl)benzaldehyde 1422954-47-9 C20H28O2Si2
(Z)-4-((4-oxo-3-((trimethylsilyl)methyl)cyclopent-2-en-1-ylidene)(trimethylsilyl)methyl)benzaldehyde
—— —— 1070974-37-6 C22H18ClF3N4O3S
—— —— 1067657-02-6 C36H32Cl2N8O2
—— —— 1067656-81-8 C36H34Cl2N8O
—— tert-butyl N-[2-(1-hydroxy-2-methylpropyl)pyridin-3-yl]carbamate 1309885-87-7 C14H22N2O3
tert-butyl N-[2-(1-hydroxy-2-methylpropyl)pyridin-3-yl]carbamate
—— N-[(1-cyclohexyltetrazol-5-yl)-(2-nitrophenyl)methyl]propan-1-amine 1369847-25-5 C17H24N6O2
N-[(1-cyclohexyltetrazol-5-yl)-(2-nitrophenyl)methyl]propan-1-amine
—— 3-bromo-4-ethyl-2H-benzo[h]chromene 1191065-36-7 C15H13BrO
3-bromo-4-ethyl-2H-benzo[h]chromene
—— 2-(6,6-Dimethyl-2-oxooct-7-enyl)benzaldehyde 1377152-10-7 C17H22O2
2-(6,6-Dimethyl-2-oxooct-7-enyl)benzaldehyde
—— 1,2,4,5-Tetrakis(4-tert-butylphenyl)-3,6-bis(4-phenylphenyl)benzene 1602577-12-7 C70H70
1,2,4,5-Tetrakis(4-tert-butylphenyl)-3,6-bis(4-phenylphenyl)benzene
—— (R)-2-(1-(4-methoxyphenyl)-2-nitroethyl)-1H-indole 1156494-03-9 C17H16N2O3
(R)-2-(1-(4-methoxyphenyl)-2-nitroethyl)-1H-indole
—— 1,2-dihydro-5,7-dimethoxy-2-(2-methylallyl)naphthalene 1361106-45-7 C16H20O2
1,2-dihydro-5,7-dimethoxy-2-(2-methylallyl)naphthalene
—— (2R,6S,8R,9R,11R)-2,11-bis(iodomethyl)-8,9-diphenyl-1,7,10-trioxaspiro[5.7]tridecane 1263204-00-7 C24H28I2O3
(2R,6S,8R,9R,11R)-2,11-bis(iodomethyl)-8,9-diphenyl-1,7,10-trioxaspiro[5.7]tridecane
—— —— 1092554-18-1 C32H37N6O7*I
—— —— 1092554-03-4 C31H30N5O8*Cl
—— (S)-N-<(1,1-dimethylethoxy)carbonyl>-L-valyl-N-<3,3-difluoro-2,4-dioxo-1-<2-oxo-2-(phenylmethoxy)ethyl>-4-(1-pyrrolidinyl)butyl>-L-alaninimide 145452-66-0 C30H42F2N4O8
(S)-N-<(1,1-dimethylethoxy)carbonyl>-L-valyl-N-<3,3-difluoro-2,4-dioxo-1-<2-oxo-2-(phenylmethoxy)ethyl>-4-(1-pyrrolidinyl)butyl>-L-alaninimide
—— (1S,6S,9R,13R,14S,15S,17R,19S)-15-[tert-butyl(dimethyl)silyl]oxy-6,13,19-trimethyl-11-methylidene-9-propyl-14-triethylsilyloxy-8,20-dioxabicyclo[15.2.1]icosan-7-one 1359738-91-2 C37H72O5Si2
(1S,6S,9R,13R,14S,15S,17R,19S)-15-[tert-butyl(dimethyl)silyl]oxy-6,13,19-trimethyl-11-methylidene-9-propyl-14-triethylsilyloxy-8,20-dioxabicyclo[15.2.1]icosan-7-one
—— 3-((trimethylsilylmethyloxy)methyl)cyclopentan-1-one 1448675-32-8 C10H20O2Si
3-((trimethylsilylmethyloxy)methyl)cyclopentan-1-one
—— (4S)-N-benzyl-2-diazo-3-oxo-N-phenyl-5-phenylmethoxy-4-(tritylamino)pentanamide 1007843-14-2 C44H38N4O3
(4S)-N-benzyl-2-diazo-3-oxo-N-phenyl-5-phenylmethoxy-4-(tritylamino)pentanamide
—— 5-Methoxy-1-(4-methylphenyl)sulfonyl-2-(2,2,2-trifluoroethyl)-2,3-dihydroindole 1609653-22-6 C18H18F3NO3S
5-Methoxy-1-(4-methylphenyl)sulfonyl-2-(2,2,2-trifluoroethyl)-2,3-dihydroindole
—— 6-Ethyl-5-[(1-methylpiperidin-2-yl)methylamino]-3-(3-methylsulfonylanilino)pyrazine-2-carboxamide 1254050-01-5 C21H30N6O3S
6-Ethyl-5-[(1-methylpiperidin-2-yl)methylamino]-3-(3-methylsulfonylanilino)pyrazine-2-carboxamide
—— US8653087, III-6 1213242-87-5 C27H25ClF3N7O2
US8653087, III-6
—— 3-[1-[4-[2-(Dimethylamino)ethoxy]-2,3-difluorophenyl]tetrazol-5-yl]-5-(4-methoxyphenyl)pyridin-2-amine 1224210-89-2 C23H23F2N7O2
3-[1-[4-[2-(Dimethylamino)ethoxy]-2,3-difluorophenyl]tetrazol-5-yl]-5-(4-methoxyphenyl)pyridin-2-amine
—— methyl N-[(1R)-2-oxo-1-phenyl-2-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-phenyl-2-(piperidine-1-carbonylamino)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]ethyl]carbamate 1228965-71-6 C52H53N9O5
methyl N-[(1R)-2-oxo-1-phenyl-2-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-phenyl-2-(piperidine-1-carbonylamino)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]ethyl]carbamate
—— 4-[4-(3-Propan-2-yl-3-azabicyclo[3.1.0]hexan-1-yl)phenyl]morpholine 1259554-94-3 C18H26N2O
4-[4-(3-Propan-2-yl-3-azabicyclo[3.1.0]hexan-1-yl)phenyl]morpholine
—— 2-(4-acetamidophenyl)-N-[2-[2,4-dichloro-N-methyl-3-[[2-methyl-4-(pyridin-2-ylmethoxy)quinolin-8-yl]oxymethyl]anilino]-2-oxoethyl]acetamide 1360587-13-8 C36H33Cl2N5O5
2-(4-acetamidophenyl)-N-[2-[2,4-dichloro-N-methyl-3-[[2-methyl-4-(pyridin-2-ylmethoxy)quinolin-8-yl]oxymethyl]anilino]-2-oxoethyl]acetamide
—— 3-[4-(1-Amino-4-hydroxy-9,10-dioxo-9,10-dihydro-anthracen-2-yloxy)-phenyl]-propionic acid 1-methyl-2-phenoxy-ethyl ester 16472-15-4 C32H27NO7
3-[4-(1-Amino-4-hydroxy-9,10-dioxo-9,10-dihydro-anthracen-2-yloxy)-phenyl]-propionic acid 1-methyl-2-phenoxy-ethyl ester
—— methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-(dimethylamino)-2-phenylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1228966-80-0 C45H50N8O4
methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-(dimethylamino)-2-phenylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 7-(4-chlorophenyl)-2-((S)-1-piperidin-4-ylpyrrolidine-2-carbonyl)-1,3,4,5,10,11a-hexahydro-2H-2,4a,10-triazadibenzo[a,d]cycloheptene-11-one 1262131-32-7 C28H34ClN5O2
7-(4-chlorophenyl)-2-((S)-1-piperidin-4-ylpyrrolidine-2-carbonyl)-1,3,4,5,10,11a-hexahydro-2H-2,4a,10-triazadibenzo[a,d]cycloheptene-11-one
—— 1-Triphenylsilyl-1-buten 18751-16-1 C22H22Si
1-Triphenylsilyl-1-buten
—— (3R,4S)-3-(2-methoxyphenyl)-4-nitro-3,4-dihydronaphthalene-2-carbaldehyde 1185744-37-9 C18H15NO4
(3R,4S)-3-(2-methoxyphenyl)-4-nitro-3,4-dihydronaphthalene-2-carbaldehyde
—— Hexafluor-1-iod-cyclobutanol 1651-62-3 C4HF6IO
Hexafluor-1-iod-cyclobutanol
—— [(2R,3S)-3-methylhept-6-en-2-yl] (2E,4R)-4,8-dimethyl-7-oxo-4-triethylsilyloxynona-2,8-dienoate 1417908-58-7 C25H44O4Si
[(2R,3S)-3-methylhept-6-en-2-yl] (2E,4R)-4,8-dimethyl-7-oxo-4-triethylsilyloxynona-2,8-dienoate