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中文名称 英文名称 CAS号 化学式 结构式图片
—— [1,2,4]triazolo[1,5-a]pyridine-7-sulfonyl chloride 1431877-58-5 C6H4ClN3O2S
[1,2,4]triazolo[1,5-a]pyridine-7-sulfonyl chloride
—— 3-chloro-6-(5-fluoro-3'-nitrobiphenyl-2-yloxy)-[1,2,4]triazolo[4,3-b]pyridazine 1429026-46-9 C17H9ClFN5O3
3-chloro-6-(5-fluoro-3'-nitrobiphenyl-2-yloxy)-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-[9-(3,5-dichlorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-3,3-dimethyl-6-oxohexanoic acid 1354803-27-2 C25H27Cl2N3O3
6-[9-(3,5-dichlorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-3,3-dimethyl-6-oxohexanoic acid
—— 6-((2R)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-5-fluoro-2-(quinolin-6-ylamino)nicotinamide 1354246-21-1 C24H21FN6O2
6-((2R)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-5-fluoro-2-(quinolin-6-ylamino)nicotinamide
—— 1-(4-methoxyphenoxy)-2-[1-(phenylsulfanyl)cyclopropyl]-2-propanol 448960-37-0 C19H22O3S
1-(4-methoxyphenoxy)-2-[1-(phenylsulfanyl)cyclopropyl]-2-propanol
—— ethyl 2-((4-bromo-2-fluorophenyl)amino)-6-oxo-1,4,5,6-tetrahydrocyclopenta[b]pyrrole-3-carboxylate 1370189-26-6 C16H14BrFN2O3
ethyl 2-((4-bromo-2-fluorophenyl)amino)-6-oxo-1,4,5,6-tetrahydrocyclopenta[b]pyrrole-3-carboxylate
—— 1-(2-fluoroethyl)-3-{4-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one 1093978-84-7 C25H25FN6O2
1-(2-fluoroethyl)-3-{4-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one
—— N-{3-fluoro-4-[1-methyl-3-(trifluoromethyl)pyrazol-5-yl]phenyl}(4-methyl(1,2,3-thiadiazol-5-yl))carboxamide 1431386-07-0 C15H11F4N5OS
N-{3-fluoro-4-[1-methyl-3-(trifluoromethyl)pyrazol-5-yl]phenyl}(4-methyl(1,2,3-thiadiazol-5-yl))carboxamide
—— (S)-3-(2,5-dichloropyrimidin-4-yl)-4-isopropyloxazolidin-2-one 1429181-02-1 C10H11Cl2N3O2
(S)-3-(2,5-dichloropyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— 1-Acetyl-3,3-dipropyl-azetidin 91369-91-4 C11H21NO
1-Acetyl-3,3-dipropyl-azetidin
—— 4-[(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzoyl)amino]-L-phenylalanine 1021943-15-6 C31H37N7O5
4-[(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzoyl)amino]-L-phenylalanine
—— (S)-3-(5-(4-chlorophenyl)-1,1-dioxo-4-(3-(pyrazin-2-yloxy)phenyl)-1,2,5-thiadiazolidin-2-yl)propane-1-sulfonamide 1035488-49-3 C21H22ClN5O5S2
(S)-3-(5-(4-chlorophenyl)-1,1-dioxo-4-(3-(pyrazin-2-yloxy)phenyl)-1,2,5-thiadiazolidin-2-yl)propane-1-sulfonamide
—— Methyl 2-[5-chloro-4-[[2-methyl-4-(2-methylpyrazol-3-yl)quinolin-8-yl]oxymethyl]pyridin-3-yl]sulfanylpropanoate 1064669-42-6 C24H23ClN4O3S
Methyl 2-[5-chloro-4-[[2-methyl-4-(2-methylpyrazol-3-yl)quinolin-8-yl]oxymethyl]pyridin-3-yl]sulfanylpropanoate
—— N'-[3,5-dichloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-2-yl]butane-1,4-diamine 1064668-64-9 C23H24Cl2N6O
N'-[3,5-dichloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-2-yl]butane-1,4-diamine
—— (S)-2-amino-N-{3-[4-(2-trifluoromethyl-phenylamino)-benzylcarbamoyl]-tetrahydro-furan-3-yl}-isonicotinamide 1242452-32-9 C25H24F3N5O3
(S)-2-amino-N-{3-[4-(2-trifluoromethyl-phenylamino)-benzylcarbamoyl]-tetrahydro-furan-3-yl}-isonicotinamide
—— methyl N-[3-[3-chloro-6-[[cyclopropyl(morpholine-2-carbonyl)amino]methyl]indol-1-yl]propyl]carbamate 1093081-33-4 C22H29ClN4O4
methyl N-[3-[3-chloro-6-[[cyclopropyl(morpholine-2-carbonyl)amino]methyl]indol-1-yl]propyl]carbamate
—— N-(2-aminophenyl)-4-{3-cyano-5-[(4-pyridin-4-ylpiperidin-1-yl)methyl]pyridin-2-yl}benzamide 1027973-38-1 C30H28N6O
N-(2-aminophenyl)-4-{3-cyano-5-[(4-pyridin-4-ylpiperidin-1-yl)methyl]pyridin-2-yl}benzamide
—— (S,E)-N-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)-3-cyano-7-(tetrahydrofuran-3-yl-oxy)quinolin-6-yl)-4-(dimethylamino)-but-2-enamide 1351941-89-3 C33H31ClFN5O4
(S,E)-N-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)-3-cyano-7-(tetrahydrofuran-3-yl-oxy)quinolin-6-yl)-4-(dimethylamino)-but-2-enamide
—— N-((6-(7-(4-(5-chloro-1H-benzo[d]imidazol-2-ylamino)-2-fluorophenoxy)thieno[3,2-b]pyridin-2-yl)pyridin-3-yl)methyl)-2-hydroxy-N-(2-methoxyethyl)acetamide 1429307-59-4 C31H26ClFN6O4S
N-((6-(7-(4-(5-chloro-1H-benzo[d]imidazol-2-ylamino)-2-fluorophenoxy)thieno[3,2-b]pyridin-2-yl)pyridin-3-yl)methyl)-2-hydroxy-N-(2-methoxyethyl)acetamide
—— N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-1-(2-propoxyethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429314-46-4 C19H24Cl2N2O4
N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-1-(2-propoxyethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— tert-butyl 4-[5-amino-2-chloro-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-4-yl]piperazine-1-carboxylate 1352625-54-7 C18H29ClN6O3
tert-butyl 4-[5-amino-2-chloro-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-4-yl]piperazine-1-carboxylate
—— N-(3-methoxy-benzyl)-5-(1-oxo-1,2,5,6,7,8-hexahydro-isoquinolin-4-yl)-nicotinamide 872176-29-9 C23H23N3O3
N-(3-methoxy-benzyl)-5-(1-oxo-1,2,5,6,7,8-hexahydro-isoquinolin-4-yl)-nicotinamide
—— 2-oxo-2-[4-(trifluoromethoxy)phenyl]ethyl 2-{3-[(tert-butylsulfinyl)amino]oxetan-3-yl}butanoate 1432024-02-6 C20H26F3NO6S
2-oxo-2-[4-(trifluoromethoxy)phenyl]ethyl 2-{3-[(tert-butylsulfinyl)amino]oxetan-3-yl}butanoate
—— 3-(2-amino-5-methyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)-4-chlorobenzonitrile 1431469-81-6 C14H9ClN4OS
3-(2-amino-5-methyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)-4-chlorobenzonitrile
—— 1-[(2,2-difluorocyclopropyl)methyl]-5-[5-(1-hydroxy-1-methylethyl)phenyl]-3-methyl-1,3-dihydro-1H-imidazo[4,5-b]pyridin-2-one 1352421-17-0 C20H21F2N3O2
1-[(2,2-difluorocyclopropyl)methyl]-5-[5-(1-hydroxy-1-methylethyl)phenyl]-3-methyl-1,3-dihydro-1H-imidazo[4,5-b]pyridin-2-one
—— 6-[8-(imidazo[1,2-a]pyrazin-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3-[5-methyl-1-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylmethyl)-1H-pyrazol-4-yl]pyridine-2-carboxylic acid tert-butyl ester 1430847-17-8 C41H46N8O3
6-[8-(imidazo[1,2-a]pyrazin-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3-[5-methyl-1-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylmethyl)-1H-pyrazol-4-yl]pyridine-2-carboxylic acid tert-butyl ester
—— 2-[4-[5-Amino-6-[5-[4-[3-(dimethylamino)azetidin-1-yl]phenyl]-1,3,4-oxadiazol-2-yl]pyrazin-2-yl]pyridin-2-yl]-2-methylpropanenitrile 1402390-26-4 C26H27N9O
2-[4-[5-Amino-6-[5-[4-[3-(dimethylamino)azetidin-1-yl]phenyl]-1,3,4-oxadiazol-2-yl]pyrazin-2-yl]pyridin-2-yl]-2-methylpropanenitrile
—— N-(6-(pyrrolidin-1-yl)pyridin-2-yl)-6-(2-(trifluoromethyl)phenyl)-[1,2,4]triazolo[4,3-b]pyridazine-3-carboxamide 1431643-39-8 C22H18F3N7O
N-(6-(pyrrolidin-1-yl)pyridin-2-yl)-6-(2-(trifluoromethyl)phenyl)-[1,2,4]triazolo[4,3-b]pyridazine-3-carboxamide
—— (1R,3S,4S)-N-[(1S)-2-[4-(4-chloro-3-cyanophenyl)phenyl]-1-cyanoethyl]-2-azabicyclo[2.2.1]heptane-3-carboxamide 1428665-32-0 C23H21ClN4O
(1R,3S,4S)-N-[(1S)-2-[4-(4-chloro-3-cyanophenyl)phenyl]-1-cyanoethyl]-2-azabicyclo[2.2.1]heptane-3-carboxamide
—— N-(adamantan-1-ylmethyl)-2-[2-(4-cyclobutylpiperazin-1-yl)-2-oxoethyl]imidazo[1,2-a]pyridine-5-carboxamide 1031831-46-5 C29H39N5O2
N-(adamantan-1-ylmethyl)-2-[2-(4-cyclobutylpiperazin-1-yl)-2-oxoethyl]imidazo[1,2-a]pyridine-5-carboxamide
—— 2-[9-Hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxy-1-piperidin-1-ylethanone 1220964-42-0 C21H20F3NO3
2-[9-Hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxy-1-piperidin-1-ylethanone
—— N-[(1-methyl-1H-benzimidazol-2-yl)methyl]-5H-spiro[benzo[h]quinazoline-6,4-piperidin]-2-amine 1234353-62-8 C25H26N6
N-[(1-methyl-1H-benzimidazol-2-yl)methyl]-5H-spiro[benzo[h]quinazoline-6,4-piperidin]-2-amine
—— N-[[6-bromo-1-(3-methoxypropyl)indol-3-yl]methyl]cyclopropanamine 1093085-28-9 C16H21BrN2O
N-[[6-bromo-1-(3-methoxypropyl)indol-3-yl]methyl]cyclopropanamine
—— 9-{2-[((1R,2S)-1-amino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-nonanoic acid methyl ester 1051391-63-9 C23H33N3O6S
9-{2-[((1R,2S)-1-amino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-nonanoic acid methyl ester
—— 2,4-difluoro-N-(6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-yl)benzenesulfonamide 1234373-84-2 C16H14F2N4O2S
2,4-difluoro-N-(6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-yl)benzenesulfonamide
—— 3,4-dichloro-N-[1-[3-ethyl-2-(4-methoxyphenoxy)pyridin-4-yl]ethyl]benzenesulfonamide 1110733-48-6 C22H22Cl2N2O4S
3,4-dichloro-N-[1-[3-ethyl-2-(4-methoxyphenoxy)pyridin-4-yl]ethyl]benzenesulfonamide
—— 4-(((4S,5S)-3-(4-chlorophenyl)-4-(3-methoxyphenyl)-2-oxooxazolidin-5-yl)methyl)-1-(6-methoxypyridin-3-yl)piperazin-2-one 1035486-30-6 C27H27ClN4O5
4-(((4S,5S)-3-(4-chlorophenyl)-4-(3-methoxyphenyl)-2-oxooxazolidin-5-yl)methyl)-1-(6-methoxypyridin-3-yl)piperazin-2-one
—— Triethyl(((4R, 5S)-5-methylnon-1-en-4-yl)oxy)silane 1337552-62-1 C16H34OSi
Triethyl(((4R, 5S)-5-methylnon-1-en-4-yl)oxy)silane
—— (2R,3S)-ethyl 1-((S)-2-(3-carbamoylphenylamino)-2-(4-fluoro-3-methoxyphenyl)acetyl)-2-(2-(cyclopropylsulfonyl)phenyl)pyrrolidine-3-carboxylate 960229-89-4 C32H34FN3O7S
(2R,3S)-ethyl 1-((S)-2-(3-carbamoylphenylamino)-2-(4-fluoro-3-methoxyphenyl)acetyl)-2-(2-(cyclopropylsulfonyl)phenyl)pyrrolidine-3-carboxylate
—— (3,4-dichlorobenzyl)-(8-methanesulfonyl-2-methylquinolin-4-yl)-amine 1121528-71-9 C18H16Cl2N2O2S
(3,4-dichlorobenzyl)-(8-methanesulfonyl-2-methylquinolin-4-yl)-amine
—— N-(2-hydroxyethyl)-2-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxy-N-methylacetamide 1220964-50-0 C19H18F3NO4
N-(2-hydroxyethyl)-2-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxy-N-methylacetamide
—— 2-[5-chloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-3-yl]sulfanyl-N,N-dimethylacetamide 1064669-58-4 C23H22ClN5O2S
2-[5-chloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-3-yl]sulfanyl-N,N-dimethylacetamide
—— 2,6-difluoro-N-(6-(4-(4-fluorophenyl)-1-(1-(3,3,3-trifluoropropanoyl)piperidin-4-yl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide 1615721-67-9 C29H22F6N8O2
2,6-difluoro-N-(6-(4-(4-fluorophenyl)-1-(1-(3,3,3-trifluoropropanoyl)piperidin-4-yl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide
—— 2-[2-(tert-butyldiphenylsilyloxy)ethyl]tetrahydrofuran-3-ol 1290051-40-9 C22H30O3Si
2-[2-(tert-butyldiphenylsilyloxy)ethyl]tetrahydrofuran-3-ol
—— (2S)-N-cyclopropyl-N-[1-(4-methyl-2-methylaminopentanoyl)-piperidin-4-yl]-3-difluoromethoxybenzenesulfonamide 884308-38-7 C22H33F2N3O4S
(2S)-N-cyclopropyl-N-[1-(4-methyl-2-methylaminopentanoyl)-piperidin-4-yl]-3-difluoromethoxybenzenesulfonamide
—— 2,3-dihydro-3,3-dimethyl-1H-naphtho<2,1-b>pyran-1-acetic acid 155222-11-0 C17H18O3
2,3-dihydro-3,3-dimethyl-1H-naphtho<2,1-b>pyran-1-acetic acid
—— (S)-8-{2-[((1R,2S)-1-tert-butoxycarbonylamino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-2-cyclopentyloxycarbonylamino-octanoic acid methyl ester 1051393-38-4 C33H48N4O10S
(S)-8-{2-[((1R,2S)-1-tert-butoxycarbonylamino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-2-cyclopentyloxycarbonylamino-octanoic acid methyl ester
—— [1-[9-Hydroxy-9-(trifluoromethyl)fluorene-2-carbonyl]azetidin-3-yl]-piperidin-1-ylmethanone 1220962-83-3 C24H23F3N2O3
[1-[9-Hydroxy-9-(trifluoromethyl)fluorene-2-carbonyl]azetidin-3-yl]-piperidin-1-ylmethanone
—— (4S,5S)-3-(4-chlorophenyl)-5-((4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl)methyl)-4-(3-methoxyphenyl)oxazolidin-2-one 1035488-88-0 C26H29ClN4O3
(4S,5S)-3-(4-chlorophenyl)-5-((4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl)methyl)-4-(3-methoxyphenyl)oxazolidin-2-one
—— 2-(4-(2-(benzyloxy)ethoxy)phenyl)-2-bromo-1-(4-methoxyphenyl)ethanone 951745-47-4 C24H23BrO4
2-(4-(2-(benzyloxy)ethoxy)phenyl)-2-bromo-1-(4-methoxyphenyl)ethanone