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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[(5-methoxy-2,3-dihydro-1H-pyrrolo[2,3-c]pyridin-1-yl)carbonyl]-8-methyl-1-(tetrahydrofuran-3-yl)imidazo[1,5-a]quinoxalin-4(5H)-one 1365032-81-0 C24H23N5O4
7-[(5-methoxy-2,3-dihydro-1H-pyrrolo[2,3-c]pyridin-1-yl)carbonyl]-8-methyl-1-(tetrahydrofuran-3-yl)imidazo[1,5-a]quinoxalin-4(5H)-one
—— 5-(4-chloro-phenoxy)-4-(4-chloro-phenyl)-2-methyl-thiazole 107519-61-9 C16H11Cl2NOS
5-(4-chloro-phenoxy)-4-(4-chloro-phenyl)-2-methyl-thiazole
—— (2,3-Dichloro-propionyl)-carbamic acid 2,4-dichloro-phenyl ester 58414-51-0 C10H7Cl4NO3
(2,3-Dichloro-propionyl)-carbamic acid 2,4-dichloro-phenyl ester
—— 2,7-bis-(2-pentylamino-ethyl)-benzo[<i>lmn</i>][3,8]phenanthroline-1,3,6,8-tetraone 3718-50-1 C28H36N4O4
2,7-bis-(2-pentylamino-ethyl)-benzo[<i>lmn</i>][3,8]phenanthroline-1,3,6,8-tetraone
—— 1-(4-chloro-phenyl)-3-(5-methyl-benzooxazol-2-yl)-thiourea 967-92-0 C15H12ClN3OS
1-(4-chloro-phenyl)-3-(5-methyl-benzooxazol-2-yl)-thiourea
—— 1-(5-methyl-benzooxazol-2-yl)-3-phenyl-urea 965-13-9 C15H13N3O2
1-(5-methyl-benzooxazol-2-yl)-3-phenyl-urea
—— Heptanethioic acid S-[2-((R)-17-hydroxy-10,13-dimethyl-3,11-dioxo-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl)-2-oxo-ethyl] ester 55561-01-8 C28H40O5S
Heptanethioic acid S-[2-((R)-17-hydroxy-10,13-dimethyl-3,11-dioxo-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl)-2-oxo-ethyl] ester
—— 4-Fluoro-thiobenzoic acid S-[2-((11S,17R)-11,17-dihydroxy-10,13-dimethyl-3-oxo-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-3H-cyclopenta[a]phenanthren-17-yl)-2-oxo-ethyl] ester 55560-92-4 C28H31FO5S
4-Fluoro-thiobenzoic acid S-[2-((11S,17R)-11,17-dihydroxy-10,13-dimethyl-3-oxo-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-3H-cyclopenta[a]phenanthren-17-yl)-2-oxo-ethyl] ester
—— methyl (R,S)-2,3,4,5-tetrahydro-8-[[[2-(1-methyl-1H-imidazol-4-yl)ethyl]amino]carbonyl]-3-oxo-4-(2-phenylethyl)-1H-1,4-benzodiazepine-2-acetate 1246556-57-9 C27H31N5O4
methyl (R,S)-2,3,4,5-tetrahydro-8-[[[2-(1-methyl-1H-imidazol-4-yl)ethyl]amino]carbonyl]-3-oxo-4-(2-phenylethyl)-1H-1,4-benzodiazepine-2-acetate
—— —— 53670-61-4 C20H39N3O4
—— α,α,α',α'-Tetrakis-(4-hydroxy-3,5-di-(2-ethylhexyl)-phenyl)-p-xylene 51866-59-2 C96H154O4
α,α,α',α'-Tetrakis-(4-hydroxy-3,5-di-(2-ethylhexyl)-phenyl)-p-xylene
—— (R)-(5-(5-(5-chloro-6-isopropoxypyridin-3-yl)-thiazol-2-yl)-4-methyl-indan-1-yl)acetonitrile 856168-97-3 C23H22ClN3OS
(R)-(5-(5-(5-chloro-6-isopropoxypyridin-3-yl)-thiazol-2-yl)-4-methyl-indan-1-yl)acetonitrile
—— US10280167, Example 60 1434587-73-1 C21H22N8O
US10280167, Example 60
—— (7R)-8-cyclohexyl-5-(3-fluoro-4-methoxyphenyl)-2-(1H-indazol-5-ylamino)-7-methyl-7,8-dihydropteridin-6(5H)-one 1435455-60-9 C27H28FN7O2
(7R)-8-cyclohexyl-5-(3-fluoro-4-methoxyphenyl)-2-(1H-indazol-5-ylamino)-7-methyl-7,8-dihydropteridin-6(5H)-one
—— 9-nitro-4-tosyl-3,4,5,6-tetrahydro-2H-imidazo[2,1-b][1,3,6]oxadiazocine 1437119-27-1 C14H16N4O5S
9-nitro-4-tosyl-3,4,5,6-tetrahydro-2H-imidazo[2,1-b][1,3,6]oxadiazocine
—— benzyl 7-iodo-8-amino-4-benzyloxy-quinoline-2-carboxylate 495410-09-8 C24H19IN2O3
benzyl 7-iodo-8-amino-4-benzyloxy-quinoline-2-carboxylate
—— N-cyclopropyl-4-(4-{[2-(4-sulfamoylphenyl)ethyl]amino}imidazo[1,2-a]quinoxalin-1-yl)benzamide 1254193-78-6 C28H26N6O3S
N-cyclopropyl-4-(4-{[2-(4-sulfamoylphenyl)ethyl]amino}imidazo[1,2-a]quinoxalin-1-yl)benzamide
—— 3-bromo-8-cyano-4-hydroxy-quinoline-2-carboxylic acid 495409-65-9 C11H5BrN2O3
3-bromo-8-cyano-4-hydroxy-quinoline-2-carboxylic acid
—— 2-((6R,12aR)-6-benzo[1,3]dioxol-5-yl-1,4-dioxo-1,2,3,4,6,7,12,12a-octahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-3-yl)-N-(2-pyrrolidin-1-yl-ethyl)acetamide 395665-73-3 C29H31N5O5
2-((6R,12aR)-6-benzo[1,3]dioxol-5-yl-1,4-dioxo-1,2,3,4,6,7,12,12a-octahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-3-yl)-N-(2-pyrrolidin-1-yl-ethyl)acetamide
—— 6-(acetoxymethyl)-1,4-diaza-1'-benzyl-4-benzyloxycarbonyl-7-oxaspiro[bicyclo[4.3.0]nonane-8,4'-piperidin]-2-one 318988-45-3 C28H33N3O6
6-(acetoxymethyl)-1,4-diaza-1'-benzyl-4-benzyloxycarbonyl-7-oxaspiro[bicyclo[4.3.0]nonane-8,4'-piperidin]-2-one
—— (S)-4-(5-aminothiazolo[5,4-d]pyrimidin-7-yl)-N-(4-carbamoylphenyl)-3-methyl-piperazine-1-carboxamide 1435955-20-6 C18H20N8O2S
(S)-4-(5-aminothiazolo[5,4-d]pyrimidin-7-yl)-N-(4-carbamoylphenyl)-3-methyl-piperazine-1-carboxamide
—— tert-butyl 1-(4-(2-(ethylamino)-6-phenyl-5H-pyrrolo[3,2-d]pyrimidin-5-yl)phenyl)cyclobutylcarbamate 1439396-46-9 C29H33N5O2
tert-butyl 1-(4-(2-(ethylamino)-6-phenyl-5H-pyrrolo[3,2-d]pyrimidin-5-yl)phenyl)cyclobutylcarbamate
—— —— 1192317-67-1 C34H26F6N2O6S
—— —— 1609392-05-3 C19H20N6O3S
—— —— 1312421-03-6 C19H14F2N2O2
—— —— 1254313-09-1 C28H21Cl2F9N2O3
—— O-(6-Chlor-2-pyridinyl)-O-methylphenylphosphonothioat 57864-25-2 C12H11ClNO2PS
O-(6-Chlor-2-pyridinyl)-O-methylphenylphosphonothioat
—— (7R,17R)-17-Ethynyl-7-hydroxymethyl-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol 54502-78-2 C21H26O3
(7R,17R)-17-Ethynyl-7-hydroxymethyl-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol
—— 1-(5-methyl-1-pyridin-2-yl-1<i>H</i>-pyrazol-4-yl)-3-(4-<i>o</i>-tolyl-piperazin-1-yl)-propan-1-one 10050-02-9 C23H27N5O
1-(5-methyl-1-pyridin-2-yl-1<i>H</i>-pyrazol-4-yl)-3-(4-<i>o</i>-tolyl-piperazin-1-yl)-propan-1-one
—— (3aS,5R,6S,7R,7aR)-3-(3,4-Dichloro-phenyl)-5-hydroxymethyl-3,3a,5,6,7,7a-hexahydro-pyrano[2,3-d]imidazole-6,7-diol 25473-79-4 C13H14Cl2N2O4
(3aS,5R,6S,7R,7aR)-3-(3,4-Dichloro-phenyl)-5-hydroxymethyl-3,3a,5,6,7,7a-hexahydro-pyrano[2,3-d]imidazole-6,7-diol
—— 2-(3,4-dichloro-<i>trans</i>-styryl)-1-hexyl-pyridinium; bromide 110533-46-5 Br*C19H22Cl2N
2-(3,4-dichloro-<i>trans</i>-styryl)-1-hexyl-pyridinium; bromide
—— 3α,7α,23-trihydroxy-6α-ethyl-23(S)-methyl-24-nor-5β-cholan-23-sulfate sodium salt 1207065-06-2 C26H45O6S*Na
3α,7α,23-trihydroxy-6α-ethyl-23(S)-methyl-24-nor-5β-cholan-23-sulfate sodium salt
—— 1-morpholin-4-yl-3-prop-2-ynyloxy-propan-2-ol 23452-58-6 C10H17NO3
1-morpholin-4-yl-3-prop-2-ynyloxy-propan-2-ol
—— 17-allyl-4,5α-epoxy-3-methoxy-6α-(toluene-4-sulfonyloxy)-morphin-7-ene 883195-59-3 C27H29NO5S
17-allyl-4,5α-epoxy-3-methoxy-6α-(toluene-4-sulfonyloxy)-morphin-7-ene
—— 5-bromo-2-(1H-indazol-1-yl)-N<sup>4</sup>-[(2-methylthiazol-4-yl)methyl]pyrimidine-4,6-diamine 1620909-04-7 C16H14BrN7S
5-bromo-2-(1H-indazol-1-yl)-N<sup>4</sup>-[(2-methylthiazol-4-yl)methyl]pyrimidine-4,6-diamine
—— 3-[(adamantan-1-ylmethyl)amino]pyridine-4-carboxylic acid 1616265-98-5 C17H22N2O2
3-[(adamantan-1-ylmethyl)amino]pyridine-4-carboxylic acid
—— 4-[(1E,3E,5E)-6-(2-benzofuranyl)hexa-1,3,5-trienyl]-5-hydroxy-2(5H)-furanone 958300-57-7 C18H14O4
4-[(1E,3E,5E)-6-(2-benzofuranyl)hexa-1,3,5-trienyl]-5-hydroxy-2(5H)-furanone
—— PG2159 857467-01-7 C7H14NO8S*Na
PG2159
—— 8,8'-methylenebis(1-isopropyl-3-methylchromeno[4,3-c]pyrazol-4(1H)-one) 1000808-93-4 C29H28N4O4
8,8'-methylenebis(1-isopropyl-3-methylchromeno[4,3-c]pyrazol-4(1H)-one)
—— 1-(6-fluoro-3-(4-(cyclobutylcarbonyl)piperazine-1-carbonyl)benzyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione 1432671-29-8 C25H29FN4O4
1-(6-fluoro-3-(4-(cyclobutylcarbonyl)piperazine-1-carbonyl)benzyl)-5,6,7,8-tetrahydroquinazoline-2,4(1H,3H)-dione
—— 1-cyclopropyl-4-oxo-7-(3-{[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-6-yl)-oxazolidin-5-ylmethyl]-amino}-azetidin-1-yl)-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 1434079-93-2 C26H25N7O7
1-cyclopropyl-4-oxo-7-(3-{[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-6-yl)-oxazolidin-5-ylmethyl]-amino}-azetidin-1-yl)-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid
—— 6-chloro-2-(4-difluoropiperidin-1-yl)-8-methyl-4-phenylquinoline-3-carboxylic acid 1433902-08-9 C22H19ClF2N2O2
6-chloro-2-(4-difluoropiperidin-1-yl)-8-methyl-4-phenylquinoline-3-carboxylic acid
—— 9-nitro-4-((5-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-yl)methyl)-3,4,5,6-tetrahydro-2H-imidazo[2,1-b][1,3,6]oxadiazocine 1437123-74-4 C17H15F3N6O5
9-nitro-4-((5-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-yl)methyl)-3,4,5,6-tetrahydro-2H-imidazo[2,1-b][1,3,6]oxadiazocine
—— 4-(4-chloro-2-(imidazolo[1,2-a]pyridin-5-yl)phenoxy)-2,5-difluoro-N-(5-(methylthio)-1,3,4-thiadiazol-2-yl)benzenesulfonamide 1432913-21-7 C22H14ClF2N5O3S3
4-(4-chloro-2-(imidazolo[1,2-a]pyridin-5-yl)phenoxy)-2,5-difluoro-N-(5-(methylthio)-1,3,4-thiadiazol-2-yl)benzenesulfonamide
—— 4-(5-(1-methyl-2-oxopyrrolidine-3-carbonyl)pyridin-3-yl)benzaldehyde 1434288-79-5 C18H16N2O3
4-(5-(1-methyl-2-oxopyrrolidine-3-carbonyl)pyridin-3-yl)benzaldehyde
—— (S)-N1-(2-pyridin-4-yl-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-yl)propane-1,2-diamine 1438879-97-0 C18H21N5S
(S)-N1-(2-pyridin-4-yl-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-yl)propane-1,2-diamine
—— (8S,11S,14S,22S,25S,28S,31S)-14,28-dibenzyl-10,24-bis[(2S)-3-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-12,15,26,29-tetraoxo-2-oxa-5,6,7,10,13,16,19,20,21,24,27,30-dodecazahexacyclo[31.2.2.14,7.18,11.118,21.122,25]hentetraconta-1(36),4(41),5,18(39),19,33(37),34-heptaene-31-carboxylic acid 1434125-45-7 C61H80N16O11
(8S,11S,14S,22S,25S,28S,31S)-14,28-dibenzyl-10,24-bis[(2S)-3-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-12,15,26,29-tetraoxo-2-oxa-5,6,7,10,13,16,19,20,21,24,27,30-dodecazahexacyclo[31.2.2.14,7.18,11.118,21.122,25]hentetraconta-1(36),4(41),5,18(39),19,33(37),34-heptaene-31-carboxylic acid
—— 6-(4-fluorophenyl)-N-methyl-2-(2-methyl-5-{[2-(pyridin-2-yl)propan-2-yl]carbamoyl}phenyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide 1438844-32-6 C29H26FN5O2S
6-(4-fluorophenyl)-N-methyl-2-(2-methyl-5-{[2-(pyridin-2-yl)propan-2-yl]carbamoyl}phenyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
—— 2-[2-(3,4-difluorophenyl)sulfonylethylthio]-N-(2-thienylmethyl)-nicotinamide 1134168-89-0 C19H16F2N2O3S3
2-[2-(3,4-difluorophenyl)sulfonylethylthio]-N-(2-thienylmethyl)-nicotinamide
—— 4-chloro-N-{(3S)-1-[4-(2-naphthyl)pyrimidin-2-yl]pyrrolidin-3-yl}benzamide 1123233-16-8 C25H21ClN4O
4-chloro-N-{(3S)-1-[4-(2-naphthyl)pyrimidin-2-yl]pyrrolidin-3-yl}benzamide