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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-{5-[(1R)-1-cyclopropyl-1-{5-[1-(2-methoxyethyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}ethyl]pyridin-2-yl} pyrimidin-2-amine 1369483-96-4 C22H24N8O2
5-{5-[(1R)-1-cyclopropyl-1-{5-[1-(2-methoxyethyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}ethyl]pyridin-2-yl} pyrimidin-2-amine
—— 3-{2-[methyl(methylsulfonyl)amino]phenyl}-11-oxo-N-(4-pyrrolidin-1-ylbutyl)-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepine-7-carboxamide 1372590-13-0 C30H35N5O4S
3-{2-[methyl(methylsulfonyl)amino]phenyl}-11-oxo-N-(4-pyrrolidin-1-ylbutyl)-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepine-7-carboxamide
—— 5-((7,7-dimethyl-5-oxo-5,6,7,8-tetrahydroquinolin-3-yl)ethynyl)nicotinonitrile 1373336-37-8 C19H15N3O
5-((7,7-dimethyl-5-oxo-5,6,7,8-tetrahydroquinolin-3-yl)ethynyl)nicotinonitrile
—— {4-[2-((S)-2-amino-4,5-dihydro-oxazol-4-yl)-ethyl]-phenyl}-(2-methyl-pyrimidin-4-yl)-amine 1374037-85-0 C16H19N5O
{4-[2-((S)-2-amino-4,5-dihydro-oxazol-4-yl)-ethyl]-phenyl}-(2-methyl-pyrimidin-4-yl)-amine
—— 3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)urea 1227093-64-2 C11H16N4O
3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)urea
—— {5-[(1-Butyl-1,2,3,4-tetrahydro-6-quinolyl)methylidene]-4-oxo-2-thioxothiazolidin-3-yl}acetic acid 313479-28-6 C19H22N2O3S2
{5-[(1-Butyl-1,2,3,4-tetrahydro-6-quinolyl)methylidene]-4-oxo-2-thioxothiazolidin-3-yl}acetic acid
—— {4-[2-(4-chloro-phenyl)-2H-pyrazol-3-yl]-pyridin-2-yl}-urea 1375499-88-9 C15H12ClN5O
{4-[2-(4-chloro-phenyl)-2H-pyrazol-3-yl]-pyridin-2-yl}-urea
—— 5-[5-[1-[(2,6-difluorophenyl)methyl]-(3R)-piperidinyl]-1H-1,2,4-triazol-3-yl]-3-[3,5-dimethyl-4-isoxazolyl]-1H-indazole 1374352-21-2 C26H25F2N7O
5-[5-[1-[(2,6-difluorophenyl)methyl]-(3R)-piperidinyl]-1H-1,2,4-triazol-3-yl]-3-[3,5-dimethyl-4-isoxazolyl]-1H-indazole
—— 4-(4-acryloylamino-2-methylbenzenesulfonyl)piperazine-1-carboxylic acid tert-butyl ester 1306722-12-2 C19H27N3O5S
4-(4-acryloylamino-2-methylbenzenesulfonyl)piperazine-1-carboxylic acid tert-butyl ester
—— 1-[5-[7-(4-ethoxy-2-pyridyl)-2-(ethylcarbamoylamino)-1,3-benzothiazol-5-yl]pyrimidin-2-yl]-4-methyl-piperidine-4-carboxylic acid 1372545-57-7 C28H31N7O4S
1-[5-[7-(4-ethoxy-2-pyridyl)-2-(ethylcarbamoylamino)-1,3-benzothiazol-5-yl]pyrimidin-2-yl]-4-methyl-piperidine-4-carboxylic acid
—— tert-butyl 1-(4-(3-Iodoimidazo[1,2-a]pyridin-2-yl)phenyl)cyclobutylcarbamate 1357270-57-5 C22H24IN3O2
tert-butyl 1-(4-(3-Iodoimidazo[1,2-a]pyridin-2-yl)phenyl)cyclobutylcarbamate
—— tert-butyl 3-[[(1S)-1-phenylethyl]-[2-[[(1S)-1-phenylethyl]-[3-[[(1S)-1-phenylethyl]-[2-[[(1S)-1-phenylethyl]amino]acetyl]amino]propanoyl]amino]acetyl]amino]propanoate 1356571-54-4 C46H58N4O5
tert-butyl 3-[[(1S)-1-phenylethyl]-[2-[[(1S)-1-phenylethyl]-[3-[[(1S)-1-phenylethyl]-[2-[[(1S)-1-phenylethyl]amino]acetyl]amino]propanoyl]amino]acetyl]amino]propanoate
—— (E)-4-{[(1E)-2-(4-chlorophenoxy)-N-cyano-2-methylpropanimidoyl]amino}adamantane-1-carboxamide 1252789-57-3 C22H27ClN4O2
(E)-4-{[(1E)-2-(4-chlorophenoxy)-N-cyano-2-methylpropanimidoyl]amino}adamantane-1-carboxamide
—— 5-Methoxy-1-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-pyrrolo[2,3-C]pyridine 1310705-10-2 C15H21BN2O3
5-Methoxy-1-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-pyrrolo[2,3-C]pyridine
—— 3-(2-Methoxyphenyl)-2-phenyl-5-phenylmethoxy-1-benzofuran 1203470-13-6 C28H22O3
3-(2-Methoxyphenyl)-2-phenyl-5-phenylmethoxy-1-benzofuran
—— (4S)-benzyl 2,4-di(furan-2-yl)pyrrolidine-1-carboxylate 1094497-93-4 C20H19NO4
(4S)-benzyl 2,4-di(furan-2-yl)pyrrolidine-1-carboxylate
—— 3,4,5-trimethoxy-N-(3-{2-[methyl(methylsulfonyl)amino]phenyl}-11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepin-8-yl)benzamide 1372590-82-3 C31H30N4O7S
3,4,5-trimethoxy-N-(3-{2-[methyl(methylsulfonyl)amino]phenyl}-11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepin-8-yl)benzamide
—— (2R)-1-(1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)tetrahydro-1H-pyrrolo[2,3-c]pyridine-6(2H,7H,7aH)-yl)-2-(3-chlorophenylamino)pentan-1-one 1374239-96-9 C24H29ClN6O
(2R)-1-(1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)tetrahydro-1H-pyrrolo[2,3-c]pyridine-6(2H,7H,7aH)-yl)-2-(3-chlorophenylamino)pentan-1-one
—— 7,7-dimethyl-1'-(pyridin-3-ylmethyl)-2,3,7,8-tetrahydrospiro[[1,4]dioxino[2,3-g]chromene-9,3'-indolin]-2'-one 1373240-54-0 C26H24N2O4
7,7-dimethyl-1'-(pyridin-3-ylmethyl)-2,3,7,8-tetrahydrospiro[[1,4]dioxino[2,3-g]chromene-9,3'-indolin]-2'-one
—— Ethyl 2-chloro-3-(2,4-dichlorophenyl)-3-oxopropanoate 1358761-51-9 C11H9Cl3O3
Ethyl 2-chloro-3-(2,4-dichlorophenyl)-3-oxopropanoate
—— methyl N-[(2S)-1-[(2S)-2-[5-chloro-4-[4-[4-[2-[(3S)-2-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-3,4-dihydropyrazol-3-yl]-1H-imidazol-5-yl]phenyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1373165-58-2 C39H46ClN9O6
methyl N-[(2S)-1-[(2S)-2-[5-chloro-4-[4-[4-[2-[(3S)-2-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-3,4-dihydropyrazol-3-yl]-1H-imidazol-5-yl]phenyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— N-[3-(1H-imidazol-1-yl)propyl]-3-{[4-({2-[methyl(methylsulfonyl)amino]benzyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamide 1372262-73-1 C28H31N9O3S
N-[3-(1H-imidazol-1-yl)propyl]-3-{[4-({2-[methyl(methylsulfonyl)amino]benzyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamide
—— 2-phenyl-6-({3-[1-(1H-pyrrol-2-ylcarbonyl)piperidin-4-yl]azetidin-1-yl}carbonyl)-1,3-benzoxazole 1373356-12-7 C27H26N4O3
2-phenyl-6-({3-[1-(1H-pyrrol-2-ylcarbonyl)piperidin-4-yl]azetidin-1-yl}carbonyl)-1,3-benzoxazole
—— N-[2-(1H-imidazol-1-yl)ethyl]-6-{4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-1-yl}pyridine-2-carboxamide 1373268-82-6 C24H37N7O
N-[2-(1H-imidazol-1-yl)ethyl]-6-{4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-1-yl}pyridine-2-carboxamide
—— 3-Methoxy-1-(3-methylphenyl)butan-2-amine 1519392-36-9 C12H19NO
3-Methoxy-1-(3-methylphenyl)butan-2-amine
—— N-{2-[4-(heptyloxy)phenyl]ethyl}-β-alanine trifluoroacetate 847581-63-9 C2HF3O2*C18H29NO3
N-{2-[4-(heptyloxy)phenyl]ethyl}-β-alanine trifluoroacetate
—— [1-(2-Chlorophenyl)-2-nitroethyl] thiocyanate 1116691-37-2 C9H7ClN2O2S
[1-(2-Chlorophenyl)-2-nitroethyl] thiocyanate
—— N-((5-(2-methylthiazol-5-yl)thiophen-2-yl)methyl)adamantan-1-amine 1443122-96-0 C19H24N2S2
N-((5-(2-methylthiazol-5-yl)thiophen-2-yl)methyl)adamantan-1-amine
—— ethyl 4-(acetylamino)-2-(4-methylphenyl)-1,3-thiazole-5-carboxylate 1445752-63-5 C15H16N2O3S
ethyl 4-(acetylamino)-2-(4-methylphenyl)-1,3-thiazole-5-carboxylate
—— N<sup>2</sup>,N<sup>2</sup>,N<sup>5</sup>,N<sup>5</sup>-tetraethyl-1-(4-fluorophenyl)-3,4-dihydroxy-1H-pyrrole-2,5-dicarboxamide 1443052-68-3 C20H26FN3O4
N<sup>2</sup>,N<sup>2</sup>,N<sup>5</sup>,N<sup>5</sup>-tetraethyl-1-(4-fluorophenyl)-3,4-dihydroxy-1H-pyrrole-2,5-dicarboxamide
—— (S)-2-(2-(1-benzyl-2-methyl-1H-indol-3-yl)acetamido)-N-(6-methoxypyridin-3-yl)-N-methyl-3-phenylpropanamide 1375275-54-9 C34H34N4O3
(S)-2-(2-(1-benzyl-2-methyl-1H-indol-3-yl)acetamido)-N-(6-methoxypyridin-3-yl)-N-methyl-3-phenylpropanamide
—— {4-[2-(3-fluoro-phenyl)-2-hydroxy-ethyl]-pyridin-2-yl}-urea 1375500-16-5 C14H14FN3O2
{4-[2-(3-fluoro-phenyl)-2-hydroxy-ethyl]-pyridin-2-yl}-urea
—— {[8-(2-chlorophenyl)-6-hydroxy[1,2,4]triazolo[1,5-a]pyridine-5-carbonyl]amino}acetic acid 1262132-51-3 C15H11ClN4O4
{[8-(2-chlorophenyl)-6-hydroxy[1,2,4]triazolo[1,5-a]pyridine-5-carbonyl]amino}acetic acid
—— N-[2-(2,6-dichlorophenyl)-2H-pyrazolo[4,3-c]pyridin-4-yl]-2-methoxy-pyrimidine-4,6-diamine 1378037-64-9 C17H13Cl2N7O
N-[2-(2,6-dichlorophenyl)-2H-pyrazolo[4,3-c]pyridin-4-yl]-2-methoxy-pyrimidine-4,6-diamine
—— 1-(2-methyl-cyclohexyl)-5-oxo-pyrrolidine-3-carboxylic acid methyl ester 1377615-28-5 C13H21NO3
1-(2-methyl-cyclohexyl)-5-oxo-pyrrolidine-3-carboxylic acid methyl ester
—— N-(cyclopropylmethyl)-N-[4-(5-fluoropyridin-3-yl)-2-methylimidazol-1-yl]-2,2-dimethyl-3-methylsulfanylpropanamide 1374355-87-9 C19H25FN4OS
N-(cyclopropylmethyl)-N-[4-(5-fluoropyridin-3-yl)-2-methylimidazol-1-yl]-2,2-dimethyl-3-methylsulfanylpropanamide
—— 2-(2-bromo-phenyl)-1-(2,6-dimethoxy-phenyl)-ethanone 872990-83-5 C16H15BrO3
2-(2-bromo-phenyl)-1-(2,6-dimethoxy-phenyl)-ethanone
—— [2-(1,2,3-benzothiadiazol-7-yl)cyclopropyl]methanol 1079993-62-6 C10H10N2OS
[2-(1,2,3-benzothiadiazol-7-yl)cyclopropyl]methanol
—— 1-methyl-2-phenyl-2-chloromercuriovinyl acetate 56955-02-3 C11H11ClHgO2
1-methyl-2-phenyl-2-chloromercuriovinyl acetate
—— methyl 4-[(2,3-dihydro-1H-inden-1-yl)oxy]-3,5-difluorobenzenepropanoate 691899-42-0 C19H18F2O3
methyl 4-[(2,3-dihydro-1H-inden-1-yl)oxy]-3,5-difluorobenzenepropanoate
—— 3beta,14-di-(ethoxymethoxy)-17beta-phenyl-5beta,14beta-androstane 150667-53-1 C31H48O4
3beta,14-di-(ethoxymethoxy)-17beta-phenyl-5beta,14beta-androstane
—— 2-[1-(4-Fluorophenyl)-4-(3-methoxyphenyl)imidazol-2-yl]-1-[4-(4-methoxypyridin-2-yl)piperazin-1-yl]ethanone 1443769-81-0 C28H28FN5O3
2-[1-(4-Fluorophenyl)-4-(3-methoxyphenyl)imidazol-2-yl]-1-[4-(4-methoxypyridin-2-yl)piperazin-1-yl]ethanone
—— cyclobutyl (2S)-2-[[(4-bromophenoxy)-[[(2R,4R)-4-(5-methyl-2,4-dioxo-pyrimidin-1-yl)-1,3-dioxolan-2-yl]methoxy]phosphoryl]amino]propanoate 1142818-12-9 C22H27BrN3O9P
cyclobutyl (2S)-2-[[(4-bromophenoxy)-[[(2R,4R)-4-(5-methyl-2,4-dioxo-pyrimidin-1-yl)-1,3-dioxolan-2-yl]methoxy]phosphoryl]amino]propanoate
—— N-(2-methoxyethyl)-4-({4-[({2-[methyl(methylsulfonyl)amino]pyridin-3-yl}amino)methyl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide 1372263-56-3 C24H28N8O4S
N-(2-methoxyethyl)-4-({4-[({2-[methyl(methylsulfonyl)amino]pyridin-3-yl}amino)methyl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide
—— N-(4'-methoxyphenyl)-3-propionamido-4-methoxybenzamide 1131314-55-0 C18H20N2O4
N-(4'-methoxyphenyl)-3-propionamido-4-methoxybenzamide
—— 3-{[4-({2-[methyl(methylsulfonyl)amino]benzyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino}-N-(1-methylpiperidin-4-yl)benzamide 1372262-61-7 C28H34N8O3S
3-{[4-({2-[methyl(methylsulfonyl)amino]benzyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino}-N-(1-methylpiperidin-4-yl)benzamide
—— methyl N-[(2S)-1-[(2S)-2-[5-[6-(3,4-difluorophenyl)-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1370468-55-5 C49H53F2N9O7
methyl N-[(2S)-1-[(2S)-2-[5-[6-(3,4-difluorophenyl)-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 5-amino-1-ethyl-8-(2-furyl)-3-[2-[4-[4-(2-methoxyethoxy)phenyl]piperazin-1-yl]ethyl]-[1,2,4]triazolo[5,1-f]purin-2-one 1367366-13-9 C27H33N9O4
5-amino-1-ethyl-8-(2-furyl)-3-[2-[4-[4-(2-methoxyethoxy)phenyl]piperazin-1-yl]ethyl]-[1,2,4]triazolo[5,1-f]purin-2-one
—— 2-((1H-indol-3-yl)methyl)-9-(6-methoxypyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-1-one 1373767-77-1 C23H27N5O2
2-((1H-indol-3-yl)methyl)-9-(6-methoxypyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-1-one
—— 5-o-tolyl-2,3-dihydrothieno[3,2-c]pyridin-4(5H)-one 1359984-38-5 C14H13NOS
5-o-tolyl-2,3-dihydrothieno[3,2-c]pyridin-4(5H)-one