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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 11-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]undecanoic acid —— C33H38FN5O4S2
11-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]undecanoic acid
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-heptyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H34FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-heptyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-[4-[7-(3-Methylphenyl)-5-phenylpyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]propan-1-ol —— C26H29N5O
3-[4-[7-(3-Methylphenyl)-5-phenylpyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]propan-1-ol
—— 3-[2-(3,4-Dimethoxyphenyl)ethyl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C33H32FN5O4S2
3-[2-(3,4-Dimethoxyphenyl)ethyl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 4-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid —— C26H24FN5O4S2
4-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid
—— 3-(1,1-Dioxothiolan-3-yl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H26FN5O4S3
3-(1,1-Dioxothiolan-3-yl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 11-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]undecanoic acid —— C34H40FN5O4S2
11-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]undecanoic acid
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(3-methoxypropyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28FN5O3S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(3-methoxypropyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-(1,3-Benzodioxol-5-ylmethyl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H24FN5O4S2
3-(1,3-Benzodioxol-5-ylmethyl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-Dodecyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C35H44FN5O2S2
3-Dodecyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-Cyclohexyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H30FN5O2S2
3-Cyclohexyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C31H28FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid —— C26H24FN5O4S2
3-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C31H28FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C31H28FN5O3S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-heptyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H32FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-heptyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C31H36FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H26FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H26FN5O3S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 6-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C28H28FN5O4S2
6-[5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 1-[4-[5-Phenyl-7-[3-(trifluoromethyl)phenyl]pyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanone —— C25H22F3N5O
1-[4-[5-Phenyl-7-[3-(trifluoromethyl)phenyl]pyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanone
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-hexyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H30FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-hexyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H34FN5O2S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 4-[4-[(2-Chlorophenyl)methyl]piperazin-1-yl]-5-phenyl-7-[3-(trifluoromethyl)phenyl]pyrrolo[2,3-d]pyrimidine —— C30H25ClF3N5
4-[4-[(2-Chlorophenyl)methyl]piperazin-1-yl]-5-phenyl-7-[3-(trifluoromethyl)phenyl]pyrrolo[2,3-d]pyrimidine
—— 3-Benzyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H24FN5O2S2
3-Benzyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-(2-Ethylhexyl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H34FN5O2S2
3-(2-Ethylhexyl)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-[(4-Fluorophenyl)methyl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H23F2N5O2S2
3-[(4-Fluorophenyl)methyl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 7-(4-Bromophenyl)-4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-5-phenylpyrrolo[2,3-d]pyrimidine —— C29H25BrClN5
7-(4-Bromophenyl)-4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-5-phenylpyrrolo[2,3-d]pyrimidine
—— 5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(oxolan-2-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H26FN5O3S2
5-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-(oxolan-2-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 3-Benzyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H26FN5O2S2
3-Benzyl-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 1-(3-chloropropylsulfonyl)-4-[[(2S)-oxolan-2-yl]methyl]piperazine —— C12H23ClN2O3S
1-(3-chloropropylsulfonyl)-4-[[(2S)-oxolan-2-yl]methyl]piperazine
—— (8aR)-2-(1H-pyrazol-4-ylsulfonyl)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C10H16N4O2S
(8aR)-2-(1H-pyrazol-4-ylsulfonyl)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— (8aR)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C12H20N4O2S
(8aR)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— 1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]butane-1,3-dione —— C13H22N2O3
1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]butane-1,3-dione
—— 1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]butane-1,3-dione —— C13H22N2O3
1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]butane-1,3-dione
—— (1S,2S)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H18N2O3
(1S,2S)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1S,2R)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H18N2O3
(1S,2R)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1R,2S)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H18N2O3
(1R,2S)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1S,2S)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H16N2O3
(1S,2S)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1R,2S)-2-[4-(3-methylbutyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid —— C14H24N2O3
(1R,2S)-2-[4-(3-methylbutyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid
—— (1R,2R)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H18N2O3
(1R,2R)-2-(4-cyclopropylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1S,2S)-2-[4-(3-methylbutyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid —— C14H24N2O3
(1S,2S)-2-[4-(3-methylbutyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid
—— (1R,2S)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H16N2O3
(1R,2S)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1R,2R)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid —— C12H16N2O3
(1R,2R)-2-(4-prop-2-ynylpiperazine-1-carbonyl)cyclopropane-1-carboxylic acid
—— (1S,2S)-2-[4-(dimethylcarbamoyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid —— C12H19N3O4
(1S,2S)-2-[4-(dimethylcarbamoyl)piperazine-1-carbonyl]cyclopropane-1-carboxylic acid
—— 1-[4-(4-Fluorophenyl)piperazin-1-yl]-3,3-dimethylbutan-1-one —— C16H23FN2O
1-[4-(4-Fluorophenyl)piperazin-1-yl]-3,3-dimethylbutan-1-one
—— 1-[4-(4-Fluorophenyl)piperazin-1-yl]-2,2-dimethylbutan-1-one —— C16H23FN2O
1-[4-(4-Fluorophenyl)piperazin-1-yl]-2,2-dimethylbutan-1-one
—— (2S)-2-bromo-3-methyl-1-[4-(3-methylbutyl)piperazin-1-yl]butan-1-one —— C14H27BrN2O
(2S)-2-bromo-3-methyl-1-[4-(3-methylbutyl)piperazin-1-yl]butan-1-one
—— 4-[(2R)-2-bromo-3-methylbutanoyl]-N,N-dimethylpiperazine-1-carboxamide —— C12H22BrN3O2
4-[(2R)-2-bromo-3-methylbutanoyl]-N,N-dimethylpiperazine-1-carboxamide
—— 4-[(2S)-2-bromo-3-methylbutanoyl]-N,N-dimethylpiperazine-1-carboxamide —— C12H22BrN3O2
4-[(2S)-2-bromo-3-methylbutanoyl]-N,N-dimethylpiperazine-1-carboxamide