| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | ((1R,3s,5S)-3-(7-amino-6-(methylsulfonyl)-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)(1H-tetrazol-5-yl)methanone | 1319250-33-3 | C27H26N10O3S |
| —— | (trans)-8-({[6-(2-oxo-1(2H)-pyridinyl)-3-pyridazinyl]amino}methyl)-3-(3-pyridazinyl)-1-oxa-3-azaspiro[4.5]decan-2-one hydrochloride | 1177268-11-9 | C22H23N7O3*ClH |
| —— | (trans)-8-{[(6-{[(3-methyl-3-oxetanyl)methyl]oxy}-3-pyridazinyl)amino]methyl}-3-(3-pyridazinyl)-oxa-3-azaspiro[4.5]decan-2-one | 1177267-56-9 | C22H28N6O4 |
| —— | 1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone | 1319249-71-2 | C27H27N11O2 |
| —— | (trans)-8-[({6-[3-(trifluoromethyl)phenyl]-3-pyridazinyl}amino)methyl]-1-oxa-3-azaspiro[4.5]decan-2-one | 1177269-38-3 | C20H21F3N4O2 |
| —— | 1112121-24-0 | C22H16F2N2O5 | |
| —— | 3-hydroxy-4-(1-tert-butyl-5-hydroxy-3-isopropylpyrazol-4-yl)cyclobutene-1,2-dione | 856006-84-3 | C14H20N2O4 |
| —— | 6(R)-1-[3-[4-(4-fluorophenyl)-4-cyanopiperidin-1-yl]propyl-aminocarbonyl]-6-(3,4-difluorophenyl)piperidin-2-one | 353745-35-4 | C27H29F3N4O2 |
| —— | N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-2-(diethylamino)thieno[3,2-c]pyridine-6-carboxamide | 478151-64-3 | C19H26N4OS |
| —— | 6-(4-Sulfamylphenyl)-3(2H)pyridazinon | 54558-14-4 | C10H9N3O3S |
| —— | 3-[4-[5-[2-(6-Aminopyridin-3-yl)ethynyl]-6-ethylpyrimidin-4-yl]piperazin-1-yl]-3-oxopropanenitrile | 1321872-37-0 | C20H21N7O |
| —— | (-)-(3R)-1-(2-fluorobenzyl)-N-(9-chloro-3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N-isobutylpyrrolidine-3-carboxamide | 1233924-32-7 | C26H32ClFN2O3 |
| —— | 3(S)-9-(2,3-Dihydro-1H-pyrrolo[2,3-b]pyridin-6-yl)-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid | 351446-55-4 | C21H28N4O2 |
| —— | 2-(1-(4-((2S)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-2-ylmethoxy)benzoyl)-5-trifluoromethyl-2-methylindol-3-yl)acetic acid | 502606-53-3 | C29H25F3N2O5 |
| —— | tetrazolo[1,5-a][1,4]benzodiazepine | 68751-41-7 | C10H11N5 |
| —— | 2-(3-chloro-4-hydroxyphenyl)-3-hydroxy-6-methyl-8-(4-pyridinyl)-4H-chromen-4-one | 372103-33-8 | C21H14ClNO4 |
| —— | 6-fluoro-3-(4-isoquinolin-6-yltriazol-1-yl)-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one | 1231190-47-8 | C23H17F4N5O |
| —— | 2-[[3-methyl-4-(2,2,3,3,4,4,5,5-octafluoropentoxy)pyridin-2-yl]methylsulfinyl]-1H-benzimidazole | 132332-11-7 | C19H15F8N3O2S |
| —— | 1-(4-chloro-2,2-dimethyl-7-propoxychromen-6-yl)propan-1-ol | 132477-87-3 | C17H23ClO3 |
| —— | N-[5-(1-benzofuran-2-carbonyl)-3-(3-chlorophenyl)-1,3,4-thiadiazol-2-ylidene]benzamide | 131187-77-4 | C24H14ClN3O3S |
| —— | (1R,2R,3S,6R,7S,8S)-1,8-diphenyl-15λ6-thiapentacyclo[6.6.1.13,6.02,7.09,14]hexadeca-9,11,13-triene 15,15-dioxide | 134268-68-1 | C27H24O2S |
| —— | 3-nitrodithieno<3,4-b:3',4'-d>pyridine | 132491-69-1 | C9H4N2O2S2 |
| —— | 2-[6-amino-5-(hydroxymethyl)-4-(3-piperidinyl)-2-pyridinyl]-3-(cyclopropylmethoxy)phenol | 406208-26-2 | C21H27N3O3 |
| —— | 3-chloro-4-fluoro-N-[2-[3-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroquinolin-8-yl]benzamide | 1227054-33-2 | C23H17ClF4N2O |
| —— | N-hydroxy-5-[(3-methyl-1-benzofuran-2-yl)carbonyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide | 1338562-93-8 | C18H18N4O4 |
| —— | N-[2-(2,2-difluoro-1,3-benzodioxol-5-yl)-5,6,7,8-tetrahydroquinolin-8-yl]pyrazine-2-carboxamide | 1227054-63-8 | C21H16F2N4O3 |
| —— | 8-(1,3-thiazol-4-yl)spiro[2,4-dihydrochromene-3,4'-5H-1,3-oxazole]-2'-amine | 1221162-57-7 | C14H13N3O2S |
| —— | 5-(<2H3>methylthio)thiophen-3(2H)-one | 142820-65-3 | C5H6OS2 |
| —— | 1-benzyl-3-(1,1-dioxido-4H-pyrido[3,2-e][1,2,4]thiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinone | 686265-90-7 | C22H16N4O4S |
| —— | 4-Phenyl-1-[2-hydroxy-3-(1-allyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yloxy)propyl]-1-methylpiperidiniumiodide | 78484-04-5 | C27H35N2O3*I |
| —— | 1-Methyl-3-benzyl-4-(methylamino)-uracil | 66400-22-4 | C13H15N3O2 |
| —— | 6-fluoro-N-((1R,2S)-2-methylcyclohexyl)-1H-indole-2-carboxamide | 1578260-95-3 | C16H19FN2O |
| —— | US10138229, Example 106 | 1558037-37-8 | C23H27N5O3 |
| —— | 3-[2-[4-(1H-indol-3-yl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrimido[2,1-b]benzothiazol-4-one | 86487-74-3 | C26H26N4OS |
| —— | 2-[5-(5-carbamimidoyl-1H-benzimidazol-2-yl)-3'-aminosulfonyl-6-hydroxy-biphenyl-3-yl]acetic acid | 731015-19-3 | C22H19N5O5S |
| —— | 6,11-dihydro-6-methyl-5H-pyrimido[4,5-b][1,5]benzodiazepin-5-one | 78438-72-9 | C12H10N4O |
| —— | 6-[2-tert-Butyl-5-(4-fluorophenyl)pyrimidin-4(3H)-ylidene]cyclohexa-2,4-dien-1-one | 923594-31-4 | C20H19FN2O |
| —— | 1-(3-chlorophenyl)-3-methyl-5-methylsulfanyl-4H-imidazo[4,5-c]pyrazole | 251989-23-8 | C12H11ClN4S |
| —— | 7-methoxy-3-(4-methoxyphenyl)-5-methyl-8-propoxy-1H-quinolin-4-one | 1228466-76-9 | C21H23NO4 |
| —— | (3RS)-3-(tert-butyl-diphenyl-silanyloxy)-4,4-dimethyl-1-(5-phenylethynyl-pyridin-2-yl)-pyrrolidin-2-one | 1338492-70-8 | C35H36N2O2Si |
| —— | (S)-5-amino-2-(2,6-difluorophenyl)-N-(1-methyl-5-(tetrahydrofuran-3-yloxy)-1H-pyrazol-4-yl)thiazole-4-carboxamide | 1338717-05-7 | C18H17F2N5O3S |
| —— | 8-chloro-7-iodo-3,4-dihydro-1H-1-benzazepine-2,5-dione | 1228960-87-9 | C10H7ClINO2 |
| —— | 3-(7-chloro-1,1-dioxo-1,4-dihydrobenzo[1,2,4]thiadiazin-3-yl)-4-hydroxy-1-(3-methylbutyl)-1H-quinolin-2-one | 477930-96-4 | C21H20ClN3O4S |
| —— | {2-amino-6-[2-(3,4-dimethylpiperazine-1-sulfonyl)-4,5-difluorophenyl]quinazolin-4-yl}-(1,3-dihydroisoindol-2-yl)methanone | 1229293-04-2 | C29H28F2N6O3S |
| —— | 5-amino-N-(5-(4-(aminomethyl)piperidin-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(3-fluorophenyl)thiazole-4-carboxamide | 1338717-17-1 | C20H24FN7OS |
| —— | tert-butyI 3-(3-methyl-1,2,4-oxadiazoI-5-yI)-3-(tetrahydro-2H-pyran-2-yloxy)piperidine-1-carboxylate | 1243307-48-3 | C18H29N3O5 |
| —— | 3-amino-6-(3-isopropyl-phenyl)-pyridine-2-carboxylic acid ((S)-3-amino-3,4,5,6-tetrahydro-2H-[1,4']bipyridinyl-3'-yl)-amide | 1052709-92-8 | C25H30N6O |
| —— | 2-{(E)-2-[2-cyclobutylmethoxy-3-(difluoromethoxy)phenyl]vinyl}-3-[4-(trifluoromethoxy)phenyl]-3H-imidazo[4,5-b]pyridine | 1233449-36-9 | C27H22F5N3O3 |
| —— | 5-benzyl-5,6-dihydro-4H-benzo[de][2,6]naphthyridin-9-ol | 1589471-12-4 | C18H16N2O |
| —— | 8-O-tert-butyl 4-O-(2-phenylethyl) 11-thiophen-2-yl-2,3,6,7,9,10-hexahydro-[1,4]oxazino[3,2-h][3]benzazepine-4,8-dicarboxylate | 1334435-15-2 | C30H34N2O5S |