| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 2-butyl-7-chloro-5-({[2-chloro-4-(trifluoromethyl)pyridin-3-yl]methyl}amino)-2,3-dihydro-1H-isoindol-1-one | 1338467-60-9 | C19H18Cl2F3N3O |
| —— | 6-[4-(3-Pyridylmethylenamino)phenyl]-5-methyl-4,5-dihydro-1,2,4-triazin-3(2H)-one | 95104-76-0 | C16H15N5O |
| —— | N-(4-(4-(3-(3-tert-butyl-1-(4-methoxyphenyl)-1H-pyrazol-5-yl)ureido)-2,3-dichlorophenoxy)pyridin-2-yl)-2-methoxyacetamide | 1337931-07-3 | C29H30Cl2N6O5 |
| —— | 5-methoxyindol-2-yl 3-carboxy-2-pyridyl ketone | 120943-86-4 | C16H12N2O4 |
| —— | 5-fluoro-4-methyl-2-[1-(4-piperidin-4-yl-butyl)-1H-indol-6-yl]-1H-benzoimidazole | 1161425-14-4 | C25H29FN4 |
| —— | 5-hydroxy-3,4-dihydro-1H-2-benzopyran-1-one | 1823935-63-2 | C9H8O3 |
| —— | 6-{(3R,4R,5S)-4-[4-((R)-2-ethoxy-propoxymethyl)-phenyl]-5-pyrrolidin-1-ylmethyl-piperidin-3-yloxymethyl}-4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazine | 1160437-74-0 | C35H53N3O5 |
| —— | 5-chloro-N-methyl-6-({4-[(1-methyl-1H-pyrazol-3-yl)amino]quinazolin-6-yl}oxy)-N-(2-pyrrolidin-1-ylethyl)nicotinamide | 1154578-80-9 | C25H27ClN8O2 |
| —— | [3,2-b]indole oleanolic acid 28-O-[β-D-arabinopyranosyl] ester | 1084776-39-5 | C41H57NO6 |
| —— | 1-[5-(2,5-Difluorophenyl)spiro[1,3,4-thiadiazole-2,4'-2,3-dihydrochromene]-3-yl]propan-1-one | 1146208-98-1 | C19H16F2N2O2S |
| —— | (5-(Difluoromethyl)-6-fluoropyridin-3-yl)boronic acid | 1366482-38-3 | C6H5BF3NO2 |
| —— | 5,6-dihydro-4-ethylamino-6,6-dimethyl-4H-thieno[2,3-b]thiopyran-2-sulfonamide | 122028-31-3 | C11H18N2O2S3 |
| —— | 2-Methyl-5-(3-methyl-thioureido)-1,2,4-thiadiazolin-3-thion | 125039-68-1 | C5H8N4S3 |
| —— | 5-(3-Methylimidazo[1,2-a]pyrimidin-2-yl)-3-methyl-2-benzothiazolinone | 94704-31-1 | C15H12N4OS |
| —— | 2-((E)-2-Furan-2-yl-vinyl)-5,5,8a-trimethyl-6,7,8,8a-tetrahydro-5H-chromene | 125811-98-5 | C18H22O2 |
| —— | 2-hydroxymethyl-5,8-dihydro-[1,2,4]triazolo[1,2-<i>a</i>]pyridazine-1,3-dione | 39793-55-0 | C7H9N3O3 |
| —— | 5.5-Ethylendioxy-2-isopropyl-pentan-1-ol | 60796-16-9 | C10H20O3 |
| —— | ((1R,3s,5S)-3-(7-amino-6-(methylsulfonyl)-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)(1H-tetrazol-5-yl)methanone | 1319250-33-3 | C27H26N10O3S |
| —— | (trans)-8-({[6-(2-oxo-1(2H)-pyridinyl)-3-pyridazinyl]amino}methyl)-3-(3-pyridazinyl)-1-oxa-3-azaspiro[4.5]decan-2-one hydrochloride | 1177268-11-9 | C22H23N7O3*ClH |
| —— | (trans)-8-{[(6-{[(3-methyl-3-oxetanyl)methyl]oxy}-3-pyridazinyl)amino]methyl}-3-(3-pyridazinyl)-oxa-3-azaspiro[4.5]decan-2-one | 1177267-56-9 | C22H28N6O4 |
| —— | 1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone | 1319249-71-2 | C27H27N11O2 |
| —— | (trans)-8-[({6-[3-(trifluoromethyl)phenyl]-3-pyridazinyl}amino)methyl]-1-oxa-3-azaspiro[4.5]decan-2-one | 1177269-38-3 | C20H21F3N4O2 |
| —— | 1112121-24-0 | C22H16F2N2O5 | |
| —— | 3-hydroxy-4-(1-tert-butyl-5-hydroxy-3-isopropylpyrazol-4-yl)cyclobutene-1,2-dione | 856006-84-3 | C14H20N2O4 |
| —— | 6(R)-1-[3-[4-(4-fluorophenyl)-4-cyanopiperidin-1-yl]propyl-aminocarbonyl]-6-(3,4-difluorophenyl)piperidin-2-one | 353745-35-4 | C27H29F3N4O2 |
| —— | N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-2-(diethylamino)thieno[3,2-c]pyridine-6-carboxamide | 478151-64-3 | C19H26N4OS |
| —— | 6-(4-Sulfamylphenyl)-3(2H)pyridazinon | 54558-14-4 | C10H9N3O3S |
| —— | 3-[4-[5-[2-(6-Aminopyridin-3-yl)ethynyl]-6-ethylpyrimidin-4-yl]piperazin-1-yl]-3-oxopropanenitrile | 1321872-37-0 | C20H21N7O |
| —— | (-)-(3R)-1-(2-fluorobenzyl)-N-(9-chloro-3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N-isobutylpyrrolidine-3-carboxamide | 1233924-32-7 | C26H32ClFN2O3 |
| —— | 3(S)-9-(2,3-Dihydro-1H-pyrrolo[2,3-b]pyridin-6-yl)-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid | 351446-55-4 | C21H28N4O2 |
| —— | 2-(1-(4-((2S)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-2-ylmethoxy)benzoyl)-5-trifluoromethyl-2-methylindol-3-yl)acetic acid | 502606-53-3 | C29H25F3N2O5 |
| —— | tetrazolo[1,5-a][1,4]benzodiazepine | 68751-41-7 | C10H11N5 |
| —— | 2-(3-chloro-4-hydroxyphenyl)-3-hydroxy-6-methyl-8-(4-pyridinyl)-4H-chromen-4-one | 372103-33-8 | C21H14ClNO4 |
| —— | 6-fluoro-3-(4-isoquinolin-6-yltriazol-1-yl)-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one | 1231190-47-8 | C23H17F4N5O |
| —— | 2-[[3-methyl-4-(2,2,3,3,4,4,5,5-octafluoropentoxy)pyridin-2-yl]methylsulfinyl]-1H-benzimidazole | 132332-11-7 | C19H15F8N3O2S |
| —— | 1-(4-chloro-2,2-dimethyl-7-propoxychromen-6-yl)propan-1-ol | 132477-87-3 | C17H23ClO3 |
| —— | N-[5-(1-benzofuran-2-carbonyl)-3-(3-chlorophenyl)-1,3,4-thiadiazol-2-ylidene]benzamide | 131187-77-4 | C24H14ClN3O3S |
| —— | (1R,2R,3S,6R,7S,8S)-1,8-diphenyl-15λ6-thiapentacyclo[6.6.1.13,6.02,7.09,14]hexadeca-9,11,13-triene 15,15-dioxide | 134268-68-1 | C27H24O2S |
| —— | 3-nitrodithieno<3,4-b:3',4'-d>pyridine | 132491-69-1 | C9H4N2O2S2 |
| —— | 2-[6-amino-5-(hydroxymethyl)-4-(3-piperidinyl)-2-pyridinyl]-3-(cyclopropylmethoxy)phenol | 406208-26-2 | C21H27N3O3 |
| —— | 3-chloro-4-fluoro-N-[2-[3-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroquinolin-8-yl]benzamide | 1227054-33-2 | C23H17ClF4N2O |
| —— | N-hydroxy-5-[(3-methyl-1-benzofuran-2-yl)carbonyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide | 1338562-93-8 | C18H18N4O4 |
| —— | N-[2-(2,2-difluoro-1,3-benzodioxol-5-yl)-5,6,7,8-tetrahydroquinolin-8-yl]pyrazine-2-carboxamide | 1227054-63-8 | C21H16F2N4O3 |
| —— | 8-(1,3-thiazol-4-yl)spiro[2,4-dihydrochromene-3,4'-5H-1,3-oxazole]-2'-amine | 1221162-57-7 | C14H13N3O2S |
| —— | 5-(<2H3>methylthio)thiophen-3(2H)-one | 142820-65-3 | C5H6OS2 |
| —— | 1-benzyl-3-(1,1-dioxido-4H-pyrido[3,2-e][1,2,4]thiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinone | 686265-90-7 | C22H16N4O4S |
| —— | 4-Phenyl-1-[2-hydroxy-3-(1-allyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yloxy)propyl]-1-methylpiperidiniumiodide | 78484-04-5 | C27H35N2O3*I |
| —— | 1-Methyl-3-benzyl-4-(methylamino)-uracil | 66400-22-4 | C13H15N3O2 |
| —— | 6-fluoro-N-((1R,2S)-2-methylcyclohexyl)-1H-indole-2-carboxamide | 1578260-95-3 | C16H19FN2O |
| —— | US10138229, Example 106 | 1558037-37-8 | C23H27N5O3 |