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中文名称 英文名称 CAS号 化学式 结构式图片
—— <1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-3-N-allylthymine>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide) 142102-81-6 C27H47N3O8SSi2
<1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-3-N-allylthymine>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide)
—— 3,5-di-O-benzoyl-1,2-O-isopropylidene-3-C-methyl-D-ribofuranose 16831-88-2 C23H24O7
3,5-di-O-benzoyl-1,2-O-isopropylidene-3-C-methyl-D-ribofuranose
—— Propan-2-yl 2,2-dimethyl-1,3-oxazolidine-3-carbodithioate 1158215-00-9 C9H17NOS2
Propan-2-yl 2,2-dimethyl-1,3-oxazolidine-3-carbodithioate
—— 5-bromo-1,1-dioxo-2-quinolin-4-ylmethyl-1,2-dihydro-1-benzo[d]-isothiazol-3-one 1202040-92-3 C17H11BrN2O3S
5-bromo-1,1-dioxo-2-quinolin-4-ylmethyl-1,2-dihydro-1-benzo[d]-isothiazol-3-one
—— 3-(1-aminoethyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one 1548340-99-3 C16H17N3O
3-(1-aminoethyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one
—— benzaldehyde 2-methyl-4-phenylthiosemicarbazone 137609-50-8 C15H15N3S
benzaldehyde 2-methyl-4-phenylthiosemicarbazone
—— (R)-((3aR,5R,6S,7R,7aR)-6,7-bis(benzyloxy)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)(1,3-dithian-2-yl)methanol 1374768-27-0 C27H34N2O4S3
(R)-((3aR,5R,6S,7R,7aR)-6,7-bis(benzyloxy)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)(1,3-dithian-2-yl)methanol
—— <1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-3-N-(3-methyl-2-butenyl)thymine>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide) 142102-82-7 C29H51N3O8SSi2
<1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-3-N-(3-methyl-2-butenyl)thymine>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide)
—— [(5R,6R,8R,9R)-9-(tert-Butyl-dimethyl-silanyloxy)-6-(tert-butyl-dimethyl-silanyloxymethyl)-8-(5-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-2,2-dioxo-1,7-dioxa-2λ<sup>6</sup>-thia-spiro[4.4]non-3-en-4-ylamino]-acetic acid methyl ester 1053258-63-1 C27H47N3O10SSi2
[(5R,6R,8R,9R)-9-(tert-Butyl-dimethyl-silanyloxy)-6-(tert-butyl-dimethyl-silanyloxymethyl)-8-(5-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-2,2-dioxo-1,7-dioxa-2λ<sup>6</sup>-thia-spiro[4.4]non-3-en-4-ylamino]-acetic acid methyl ester
—— <1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-4-(bromomethyl)-1,2,3-triazole>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide) 160261-71-2 C22H41BrN4O6SSi2
<1-<2',5'-bis-O-(tert-butyldimethylsilyl)-β-D-ribofuranosyl>-4-(bromomethyl)-1,2,3-triazole>-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide)
—— 4-(2-chloro-4-cyanophenoxy)-N-(quinolinylmethyl)-benzenesulfonamide 1416568-23-4 C23H16ClN3O3S
4-(2-chloro-4-cyanophenoxy)-N-(quinolinylmethyl)-benzenesulfonamide
—— 1-{4-[(2,4-dichlorophenyl)diazenyl]-5-hydroxy-3-methyl-1H-pyrazol-1-yl}-2-(naphthalen-2-yloxy)ethanone 1217526-80-1 C22H16Cl2N4O3
1-{4-[(2,4-dichlorophenyl)diazenyl]-5-hydroxy-3-methyl-1H-pyrazol-1-yl}-2-(naphthalen-2-yloxy)ethanone
—— (3aR,7aR)-N-[(R)-(4-bromophenyl)-(1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine 1281868-07-2 C23H37BrN3OPS2
(3aR,7aR)-N-[(R)-(4-bromophenyl)-(1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine
—— (3aR,7aR)-N-[(R)-1,3-dithian-2-yl-(4-phenylmethoxyphenyl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine 1281868-12-9 C30H44N3O2PS2
(3aR,7aR)-N-[(R)-1,3-dithian-2-yl-(4-phenylmethoxyphenyl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine
—— 3-(1,3-dithian-2-ylidene)-N-methyl-2-phenyl-N-tosylbutanamide 1433278-70-6 C22H25NO3S3
3-(1,3-dithian-2-ylidene)-N-methyl-2-phenyl-N-tosylbutanamide
—— 2-[(5,7-difluoro-6-quinolinyl)methyl]isoindoline-1,3-dione 1268261-16-0 C18H10F2N2O2
2-[(5,7-difluoro-6-quinolinyl)methyl]isoindoline-1,3-dione
—— N-(4-quinolinylmethyl)-5-[5-(trifluoromethyl)-3-isoxazolyl]-2-thiophene sulfonamide 1616291-09-8 C18H12F3N3O3S2
N-(4-quinolinylmethyl)-5-[5-(trifluoromethyl)-3-isoxazolyl]-2-thiophene sulfonamide
—— 6-tert-butyl-N-(quinolin-4-ylmethyl)-2,3-dihydrobenzo[b][1,4]dioxine-2-carboxamide 1173003-71-8 C23H24N2O3
6-tert-butyl-N-(quinolin-4-ylmethyl)-2,3-dihydrobenzo[b][1,4]dioxine-2-carboxamide
—— 4-(2-chloro-4-cyanophenoxy)benzenesulfonyl chloride 1416569-28-2 C13H7Cl2NO3S
4-(2-chloro-4-cyanophenoxy)benzenesulfonyl chloride
—— 2-(1-Methylindazol-3-yl)-1,3-thiazole 1345965-53-8 C11H9N3S
2-(1-Methylindazol-3-yl)-1,3-thiazole
—— N-methyl-N-[(E)-2-phenyl-2-(trimethylsilyl)ethenyl]-p-toluenesulfonamide 1026133-68-5 C19H25NO2SSi
N-methyl-N-[(E)-2-phenyl-2-(trimethylsilyl)ethenyl]-p-toluenesulfonamide
—— 2-bromo-6-(1H-imidazol-1-yl)-7-methyl-7H-indeno[2,1-c]quinolin-7-yl pentanoate 1293989-06-6 C25H22BrN3O2
2-bromo-6-(1H-imidazol-1-yl)-7-methyl-7H-indeno[2,1-c]quinolin-7-yl pentanoate
—— 4-(1-Morpholinyl)-5,6,7,8-tetrahydro-3-phenyl-2H-1-benzopyran-2-one 105850-01-9 C19H21NO3
4-(1-Morpholinyl)-5,6,7,8-tetrahydro-3-phenyl-2H-1-benzopyran-2-one
—— (3aR,7aR)-N-[(R)-1,3-dithian-2-yl-(4-methylphenyl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine 1281868-03-8 C24H40N3OPS2
(3aR,7aR)-N-[(R)-1,3-dithian-2-yl-(4-methylphenyl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine
—— (3aR,7aR)-N-[(R)-(4-chlorophenyl)-(2-methyl-1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine 1281868-06-1 C24H39ClN3OPS2
(3aR,7aR)-N-[(R)-(4-chlorophenyl)-(2-methyl-1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine
—— (3aR,7aR)-N-[(R)-(4-chlorophenyl)-(1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine 1281868-05-0 C23H37ClN3OPS2
(3aR,7aR)-N-[(R)-(4-chlorophenyl)-(1,3-dithian-2-yl)methyl]-2-oxo-1,3-di(propan-2-yl)-3a,4,5,6,7,7a-hexahydrobenzo[d][1,3,2]diazaphosphol-2-amine
—— mono-Moxonidine fumarate 1008754-17-3 C4H4O4*C9H12ClN5O
mono-Moxonidine fumarate
—— 1-(1-((5,7-difluoroquinolin-6-yl)methyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)ethanone 1268261-21-7 C16H10F2N6O
1-(1-((5,7-difluoroquinolin-6-yl)methyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)ethanone
—— 3-(1,1-difluoroethyl)-6-methoxypyridazine 1591829-38-7 C7H8F2N2O
3-(1,1-difluoroethyl)-6-methoxypyridazine
—— (3S,5S)-5-[[tert-butyl(dimethyl)silyl]oxymethyl]-3-hydroxyoxolan-2-one 145024-94-8 C11H22O4Si
(3S,5S)-5-[[tert-butyl(dimethyl)silyl]oxymethyl]-3-hydroxyoxolan-2-one
—— 3-chloro-5-((4-(1,1-difluoroethyl)-1-((6-(1,1-difluoroethyl)-3-oxo-2,3-dihydropyridazin-4-yl)methyl)-6-oxo-1,6-dihydropyrimidin-5-yl)oxy)benzonitrile 1591826-86-6 C20H14ClF4N5O3
3-chloro-5-((4-(1,1-difluoroethyl)-1-((6-(1,1-difluoroethyl)-3-oxo-2,3-dihydropyridazin-4-yl)methyl)-6-oxo-1,6-dihydropyrimidin-5-yl)oxy)benzonitrile
—— 6-bromo-N<sup>2</sup>-((5,7-difluoroquinolin-6-yl)methyl)pyrazine-2,3-diamine 1268261-18-2 C14H10BrF2N5
6-bromo-N<sup>2</sup>-((5,7-difluoroquinolin-6-yl)methyl)pyrazine-2,3-diamine
—— 5-N-acetyl-2,3,5,8-tetradeoxy-2,3-difluoro-D-erythro-β-L-manno-non-2-ulopyranosonic acid 1437796-26-3 C11H17F2NO7
5-N-acetyl-2,3,5,8-tetradeoxy-2,3-difluoro-D-erythro-β-L-manno-non-2-ulopyranosonic acid
—— 4-amino-6-(1-(8-methyl-1-oxo-2-phenyl-1,2-dihydropyrrolo[1,2-a] pyrazin-3-yl)ethylamino)pyrimidine-5-carbonitrile 1548334-82-2 C21H19N7O
4-amino-6-(1-(8-methyl-1-oxo-2-phenyl-1,2-dihydropyrrolo[1,2-a] pyrazin-3-yl)ethylamino)pyrimidine-5-carbonitrile
—— (E)-1-(1-((5,7-difluoroquinolin-6-yl)methyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)ethanone O-2-hydroxyethyl oxime 1268260-60-1 C18H15F2N7O2
(E)-1-(1-((5,7-difluoroquinolin-6-yl)methyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)ethanone O-2-hydroxyethyl oxime
—— 4-[8-(4-hydroxymethylphenyl)-5-oxo-7-thioxo-6-azaspiro[3.4]oct-6-yl]-2-trifluoromethylbenzonitrile 1025810-19-8 C21H16F3N3O2S
4-[8-(4-hydroxymethylphenyl)-5-oxo-7-thioxo-6-azaspiro[3.4]oct-6-yl]-2-trifluoromethylbenzonitrile
—— 2-((3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)acetonitrile 1374768-42-9 C24H27N3O3S
2-((3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)acetonitrile
—— (3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-5-(2-fluoroethyl)-N,N-dimethyl-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-amine 1374768-44-1 C24H29FN2O3S
(3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-5-(2-fluoroethyl)-N,N-dimethyl-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-amine
—— (5,7-difluoroquinolin-6-yl)methanol 1268261-15-9 C10H7F2NO
(5,7-difluoroquinolin-6-yl)methanol
—— tert-butyl (3aR,5R,6S,7R,7aR)-5-(1-hydroxyethyl)-6,7-bis(4-methoxybenzyloxy)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-yl(propyl)carbamate 1374662-34-6 C32H44N2O8S
tert-butyl (3aR,5R,6S,7R,7aR)-5-(1-hydroxyethyl)-6,7-bis(4-methoxybenzyloxy)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-yl(propyl)carbamate
—— 4-azido-6-(methoxymethyl)-1-methyl-2-(2,2,2-trifluoroethyl)-1,2,3,4-tetrahydroisoquinoline 1610345-80-6 C14H17F3N4O
4-azido-6-(methoxymethyl)-1-methyl-2-(2,2,2-trifluoroethyl)-1,2,3,4-tetrahydroisoquinoline
—— 3-(1-azidoethyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one 1548340-93-7 C16H15N5O
3-(1-azidoethyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one
—— ((3aR,5R,6S,7R,7aR)-2-(azetidin-1-yl)-6,7-dihydroxy-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)methyl 4-methylbenzenesulfonate 1374966-61-6 C17H22N2O6S2
((3aR,5R,6S,7R,7aR)-2-(azetidin-1-yl)-6,7-dihydroxy-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)methyl 4-methylbenzenesulfonate
—— (3aR,5R,6S,7R,7aR)-2-(dimethylamino)-5-(2,2,2-trifluoroethyl)-5,6,7,7a-tetrahydro-3aH-pyrano [3,2-d] thiazole-6,7-diol 1374768-51-0 C10H15F3N2O3S
(3aR,5R,6S,7R,7aR)-2-(dimethylamino)-5-(2,2,2-trifluoroethyl)-5,6,7,7a-tetrahydro-3aH-pyrano [3,2-d] thiazole-6,7-diol
—— 3-(((tert-butyldimethylsilyl)oxy)methyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one 1548340-65-3 C21H28N2O2Si
3-(((tert-butyldimethylsilyl)oxy)methyl)-8-methyl-2-phenylpyrrolo[1,2-a]pyrazin-1(2H)-one
—— (3aR,5R,6S,7R,7aR)-2-(azetidin-1-yl)-5-((cyclopentylamino)methyl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol 1374966-62-7 C15H25N3O3S
(3aR,5R,6S,7R,7aR)-2-(azetidin-1-yl)-5-((cyclopentylamino)methyl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol
—— (3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-5-(2,2-difluoroethyl)-N,N-dimethyl-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-amine 1374768-46-3 C24H28F2N2O3S
(3aR,5R,6R,7R,7aR)-6,7-bis(benzyloxy)-5-(2,2-difluoroethyl)-N,N-dimethyl-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-2-amine
—— 3-(((tert-butyldimethylsilyl)oxy)methyl)-8-methylpyrrolo[1,2-a]pyrazin-1(2H)-one 1548340-60-8 C15H24N2O2Si
3-(((tert-butyldimethylsilyl)oxy)methyl)-8-methylpyrrolo[1,2-a]pyrazin-1(2H)-one
—— methyl 5-tert-butylbenzo[b]thiophene-2-carboxylate 126231-20-7 C14H16O2S
methyl 5-tert-butylbenzo[b]thiophene-2-carboxylate
—— (3aR,5R,6S,7R,7aR)-5-(2,2-difluoroethyl)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol 1374768-47-4 C10H16F2N2O3S
(3aR,5R,6S,7R,7aR)-5-(2,2-difluoroethyl)-2-(dimethylamino)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazole-6,7-diol