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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 7-(3-{1-[(2,2-difluorocyclopropyl)methyl]-3-methyl-2,2-dioxido-1,3-dihydro[1,2,5]thiadiazolo[3,4-b]pyridin-5-yl}-4-methylbenzyl)-2,7-diazaspiro[3.5]nonane-2-carboxylate 1333264-52-0 C30H39F2N5O4S
tert-butyl 7-(3-{1-[(2,2-difluorocyclopropyl)methyl]-3-methyl-2,2-dioxido-1,3-dihydro[1,2,5]thiadiazolo[3,4-b]pyridin-5-yl}-4-methylbenzyl)-2,7-diazaspiro[3.5]nonane-2-carboxylate
—— N-(2,6-diethylphenyl)-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydroisoxazolo[4,3-h]quinazoline-3-carboxamide 1356410-25-7 C31H35N7O2
N-(2,6-diethylphenyl)-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydroisoxazolo[4,3-h]quinazoline-3-carboxamide
—— 3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid [(R)-1-(2-methoxy-phenyl)-ethyl]-amide 1352433-58-9 C16H15N3O3S
3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid [(R)-1-(2-methoxy-phenyl)-ethyl]-amide
—— Methyl 2-[4-(4-fluoro-3-methylphenyl)-2-propan-2-ylimidazol-1-yl]acetate 1443143-29-0 C16H19FN2O2
Methyl 2-[4-(4-fluoro-3-methylphenyl)-2-propan-2-ylimidazol-1-yl]acetate
—— (2-(aminomethyl)-7,8-dihydro-2H-1,6,9-trioxa-9a-borabenzo[cd]azulene-8,8-diyl)dimethanol hydrochloride 1444766-42-0 C12H16BNO5*ClH
(2-(aminomethyl)-7,8-dihydro-2H-1,6,9-trioxa-9a-borabenzo[cd]azulene-8,8-diyl)dimethanol hydrochloride
—— 2-(5-hydroxy-2,4,6,7-tetramethyl-2,3-dihydro-benzo[1,2-b]furan-2-yl)ethyl 2-(6-methoxy-2-naphthyl)propionate 180344-50-7 C28H32O5
2-(5-hydroxy-2,4,6,7-tetramethyl-2,3-dihydro-benzo[1,2-b]furan-2-yl)ethyl 2-(6-methoxy-2-naphthyl)propionate
—— N-[1-[(2,6-difluorophenyl)methyl]-3(R)-piperidinyl]-1,4,6,7-tetrahydro-3-(2-methyl-4-pyridinyl)-5H-pyrazolo[4,3-c]pyridine-5-carboxamide 1366051-57-1 C25H28F2N6O
N-[1-[(2,6-difluorophenyl)methyl]-3(R)-piperidinyl]-1,4,6,7-tetrahydro-3-(2-methyl-4-pyridinyl)-5H-pyrazolo[4,3-c]pyridine-5-carboxamide
—— 4'-(cyclopropylmethoxy)-3'-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)biphenyl-3-carbonitrile 1446235-96-6 C25H21N3O2
4'-(cyclopropylmethoxy)-3'-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)biphenyl-3-carbonitrile
—— (S)-(5-methyl-2-(pyrimidin-2-yl)phenyl)(6-(((6-methyl-4-(trifluoromethyl)pyridin-2-yl)amino)methyl)-5-azaspiro[2.4]heptan-5-yl)methanone 1445595-47-0 C26H26F3N5O
(S)-(5-methyl-2-(pyrimidin-2-yl)phenyl)(6-(((6-methyl-4-(trifluoromethyl)pyridin-2-yl)amino)methyl)-5-azaspiro[2.4]heptan-5-yl)methanone
—— US9598416, Example 60 1443617-19-3 C23H27N5O2S
US9598416, Example 60
—— (4-Chloro-3-methylphenyl)-[4-[1-(3-chlorophenyl)-1,2,4-triazole-3-carbonyl]-3,3-dimethylpiperazin-1-yl]methanone 1443756-44-2 C23H23Cl2N5O2
(4-Chloro-3-methylphenyl)-[4-[1-(3-chlorophenyl)-1,2,4-triazole-3-carbonyl]-3,3-dimethylpiperazin-1-yl]methanone
—— {(S)-3-[4-(6-ethanesulfinyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-(tetrahydro-pyran-4-yl)-methanone 1445999-22-3 C25H31N3O5S
{(S)-3-[4-(6-ethanesulfinyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-(tetrahydro-pyran-4-yl)-methanone
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate 1428666-49-2 C27H28F3N3O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— 1-(3-fluoro-4-(5-(4-isopropoxyphenyl)thiazol-2-yl)benzyl)azetidine-3-carboxylic acid 1444255-82-6 C23H23FN2O3S
1-(3-fluoro-4-(5-(4-isopropoxyphenyl)thiazol-2-yl)benzyl)azetidine-3-carboxylic acid
—— 7-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-3-(3-methylimidazo[2,1-b][1,3]thiazol-6-yl)-2H-chromen-2-one 1446329-17-4 C21H22N4O2S
7-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-3-(3-methylimidazo[2,1-b][1,3]thiazol-6-yl)-2H-chromen-2-one
—— 1-(2-hydroxyethyl)-6-(4-fluorophenyl)-3-{4-[(1H-2-methylimidazo[4.5-c]pyrid-1-yl)methyl]benzoyl}indole 1237798-58-1 C31H25FN4O2
1-(2-hydroxyethyl)-6-(4-fluorophenyl)-3-{4-[(1H-2-methylimidazo[4.5-c]pyrid-1-yl)methyl]benzoyl}indole
—— 5-methanesulfonyl-benzoimidazol-2-yl chloride 1075753-35-3 C8H7ClN2O2S
5-methanesulfonyl-benzoimidazol-2-yl chloride
—— Acetic acid (2R,3S,4R,5R,6R)-3-acetoxy-2-acetoxymethyl-6-(2-acetylamino-6-oxo-1,6-dihydro-purin-9-yl)-5-(2,2,2-trifluoro-acetylamino)-tetrahydro-pyran-4-yl ester 189829-34-3 C21H23F3N6O10
Acetic acid (2R,3S,4R,5R,6R)-3-acetoxy-2-acetoxymethyl-6-(2-acetylamino-6-oxo-1,6-dihydro-purin-9-yl)-5-(2,2,2-trifluoro-acetylamino)-tetrahydro-pyran-4-yl ester
—— p-Aminophenyl 3-O-methoxycarbonylmethyl-α-D-mannopyranoside 183880-49-1 C15H21NO8
p-Aminophenyl 3-O-methoxycarbonylmethyl-α-D-mannopyranoside
—— N-{4-[butyl(methyl)carbamoyl]phenyl}-1,3-dihydro-2H-isoindole-2-carboxamide 1375546-30-7 C21H25N3O2
N-{4-[butyl(methyl)carbamoyl]phenyl}-1,3-dihydro-2H-isoindole-2-carboxamide
—— N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1-methyl-1H-imidazole-2-carboxamide 1005781-33-8 C21H19N7O3
N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1-methyl-1H-imidazole-2-carboxamide
—— 7-Oxa-15-acetoaza-dispiro-<5.2;5.1>pentadecan 101086-27-5 C15H25NO2
7-Oxa-15-acetoaza-dispiro-<5.2;5.1>pentadecan
—— 3β-Acetoxy-11α,23-dibrom-22α,25a-spirosten-(5)-on-(12) 117875-95-3 C29H40Br2O5
3β-Acetoxy-11α,23-dibrom-22α,25a-spirosten-(5)-on-(12)
—— 6-formyl-7-methoxy-1,2,3,11a-tetrahydropyrrolo<1,2-b><2>benzazepin-5-one 123267-49-2 C15H15NO3
6-formyl-7-methoxy-1,2,3,11a-tetrahydropyrrolo<1,2-b><2>benzazepin-5-one
—— methyl 17β-hydroxy-12-methoxy-4α,17α-dimethyl-18-nor-5α-androsta-8,11,13-triene-4β-carboxylate 132055-22-2 C23H32O4
methyl 17β-hydroxy-12-methoxy-4α,17α-dimethyl-18-nor-5α-androsta-8,11,13-triene-4β-carboxylate
—— —— 1365992-38-6 C27H25Cl2N7O4S
—— (+/-)-cis-2-(6-(((tert-butyldimethylsilyl)oxy)methyl)-4-methylenetetrahydro-2H-pyran-2-yl)acetaldehyde 1346851-74-8 C15H28O3Si
(+/-)-cis-2-(6-(((tert-butyldimethylsilyl)oxy)methyl)-4-methylenetetrahydro-2H-pyran-2-yl)acetaldehyde
—— benzyl 6-methyl-1-oxo-2,3-dihydro-1H-indene-2-carboxylate 1360817-55-5 C18H16O3
benzyl 6-methyl-1-oxo-2,3-dihydro-1H-indene-2-carboxylate
—— ethyl (Z)-3-propyl-3-heptenoate 141017-55-2 C12H22O2
ethyl (Z)-3-propyl-3-heptenoate
—— (E)-6-chloro-2-methyl-4-(2-(4-methylbenzylidene)hydrazinyl)quinoline 1610053-97-8 C18H16ClN3
(E)-6-chloro-2-methyl-4-(2-(4-methylbenzylidene)hydrazinyl)quinoline
—— 4-(5-{4-Fluorophenylmethyl}fur-2-yl)-3-butyn-2-ol 154355-84-7 C15H13FO2
4-(5-{4-Fluorophenylmethyl}fur-2-yl)-3-butyn-2-ol
—— 3-(3-{2-[4-(2-aminopyrimidin-5-yl)phenyl]-3-methylbutan-2-yl}-1,2,4-oxadiazol-5-yl)-6-methylpyridin-2-ol 1360550-45-3 C23H24N6O2
3-(3-{2-[4-(2-aminopyrimidin-5-yl)phenyl]-3-methylbutan-2-yl}-1,2,4-oxadiazol-5-yl)-6-methylpyridin-2-ol
—— 5-(7-fluoro-3-methyl-1-benzothien-2-yl)-8-methyl-1,9-dihydro-2H-[1,3]oxazolo[4,5-h][2,3]benzodiazepin-2-one 1398497-08-9 C20H14FN3O2S
5-(7-fluoro-3-methyl-1-benzothien-2-yl)-8-methyl-1,9-dihydro-2H-[1,3]oxazolo[4,5-h][2,3]benzodiazepin-2-one
—— 3-(2-methanesulfonyl-ethyl)-8-methoxy-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamine 1022953-10-1 C14H22N2O3S
3-(2-methanesulfonyl-ethyl)-8-methoxy-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamine
—— 6-(3-fluorophenyl)-N-[1-(6-methyl-2-piperidin-1-ylpyrimidin-4-yl)piperidin-4-yl]nicotinamide 1033838-28-6 C27H31FN6O
6-(3-fluorophenyl)-N-[1-(6-methyl-2-piperidin-1-ylpyrimidin-4-yl)piperidin-4-yl]nicotinamide
—— 6-[[6-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethylamino]pyrimidin-4-yl]amino]pyridine-2-carboxylic acid 1093166-48-3 C22H21FN6O2
6-[[6-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethylamino]pyrimidin-4-yl]amino]pyridine-2-carboxylic acid
—— 1,2-dibromo-1-(4-cyanophenyl)-2-(5,6,7,8-tetrahydro-3-methoxy-5,5,8,8-tetramethyl-2-naphthyl)ethane 131776-71-1 C24H27Br2NO
1,2-dibromo-1-(4-cyanophenyl)-2-(5,6,7,8-tetrahydro-3-methoxy-5,5,8,8-tetramethyl-2-naphthyl)ethane
—— 1,4,6,7-tetrahydro-3-imidazo[1,2-a]pyridin-6-yl-N-[1-(1-naphthalenylmethyl)-3(R)-piperidinyl]-5H-pyrazolo[4,3-c]pyridine-5-carboxamide 1366051-91-3 C30H31N7O
1,4,6,7-tetrahydro-3-imidazo[1,2-a]pyridin-6-yl-N-[1-(1-naphthalenylmethyl)-3(R)-piperidinyl]-5H-pyrazolo[4,3-c]pyridine-5-carboxamide
—— {(S)-3-[5-fluoro-4-(6-methanesulfonyl-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}(tetrahydro-pyran-4-yl)-methanone 1446001-58-6 C25H30FN3O6S
{(S)-3-[5-fluoro-4-(6-methanesulfonyl-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}(tetrahydro-pyran-4-yl)-methanone
—— 4-{2-[(1-acetylpiperidin-4-yl)oxy]-5-(ethylsulfonyl)phenyl}-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1446235-37-5 C23H27N3O5S
4-{2-[(1-acetylpiperidin-4-yl)oxy]-5-(ethylsulfonyl)phenyl}-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— N-((3,4-dihydro-2H-pyran-6-yl)methyl)-2-iodobenzamide 1359180-10-1 C13H14INO2
N-((3,4-dihydro-2H-pyran-6-yl)methyl)-2-iodobenzamide
—— [3-[5-fluoro-2-((R)-3-phenylbutyryl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-4-(2,2,2-trifluoroethoxy)phenyl]acetic acid 1445888-02-7 C29H27F4NO4
[3-[5-fluoro-2-((R)-3-phenylbutyryl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-4-(2,2,2-trifluoroethoxy)phenyl]acetic acid
—— 2,2,2-trifluoro-1-(trifluoromethyl)ethyl 4-(4'-chlorobiphenyl-3-yloxy)piperidine-1-carboxylate 1352010-55-9 C21H18ClF6NO3
2,2,2-trifluoro-1-(trifluoromethyl)ethyl 4-(4'-chlorobiphenyl-3-yloxy)piperidine-1-carboxylate
—— 5-{(R)-3-[(3,4-difluoro-benzoylamino)-methyl]-pyrrolidin-1-yl}-quinazoline-8-carboxylic acid amide 1445783-13-0 C21H19F2N5O2
5-{(R)-3-[(3,4-difluoro-benzoylamino)-methyl]-pyrrolidin-1-yl}-quinazoline-8-carboxylic acid amide
—— 2-methoxy-5-{6-[(S)-1-(thiazole-5-carbonyl)-pyrrolidin-3-yloxy]-2,3-dihydro-benzo[1,4]oxazin-4-yl}-nicotinonitrile 1446000-51-6 C23H21N5O4S
2-methoxy-5-{6-[(S)-1-(thiazole-5-carbonyl)-pyrrolidin-3-yloxy]-2,3-dihydro-benzo[1,4]oxazin-4-yl}-nicotinonitrile
—— N-(2-chloro-4-((3-(3-ethoxypropoxy)benzyl)oxy)benzyl)cyclopropanamine 1443057-94-0 C22H28ClNO3
N-(2-chloro-4-((3-(3-ethoxypropoxy)benzyl)oxy)benzyl)cyclopropanamine
—— 3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid(2-isopropoxy-pyridin-3-ylmethyl)-amide 1352434-14-0 C16H16N4O3S
3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid(2-isopropoxy-pyridin-3-ylmethyl)-amide
—— N-[(1S)-1-[4-[1-(4-ethoxyphenyl)azetidin-3-yl]oxyphenyl]ethyl]-1,2-thiazole-5-carboxamide 1443669-93-9 C23H25N3O3S
N-[(1S)-1-[4-[1-(4-ethoxyphenyl)azetidin-3-yl]oxyphenyl]ethyl]-1,2-thiazole-5-carboxamide
—— 3-hydroxy-8-methoxy-1,9-dimethyl-11-oxo-4-(pyrimidin-2-ylaminomethyl)-11H-dibenzo[b,e][1,4]dioxepine-6-carboxylic acid 1089142-39-1 C22H19N3O7
3-hydroxy-8-methoxy-1,9-dimethyl-11-oxo-4-(pyrimidin-2-ylaminomethyl)-11H-dibenzo[b,e][1,4]dioxepine-6-carboxylic acid
—— (2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-methylphenyl)pyrimidin-2-yl]phenyl]propanoic acid 1443790-09-7 C31H31N3O3
(2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-methylphenyl)pyrimidin-2-yl]phenyl]propanoic acid