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中文名称 英文名称 CAS号 化学式 结构式图片
—— (methylthio)methyl 2-(5-(5-(3-(methylsulfonyl)phenyl)-1H-pyrrol-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)acetate 1454288-86-8 C19H18F3N3O4S2
(methylthio)methyl 2-(5-(5-(3-(methylsulfonyl)phenyl)-1H-pyrrol-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)acetate
—— —— 1159349-38-8 C94H124N4O8Zn
—— (R)-5-(benzo[d]thiazol-2-yl)-6-(piperidin-3-ylamino)-2-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)pyrimidin-4(3H)-one 1433159-57-9 C26H34N6O2S
(R)-5-(benzo[d]thiazol-2-yl)-6-(piperidin-3-ylamino)-2-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)pyrimidin-4(3H)-one
—— 2-(4-(4-(diethylamino)phenyl)-6-(4-methoxyphenyl)pyridin-2-yl)phenol 1428735-98-1 C28H28N2O2
2-(4-(4-(diethylamino)phenyl)-6-(4-methoxyphenyl)pyridin-2-yl)phenol
—— (R)-5-(1,3-benzothiazol-2-yl)-2-(1-cyclobutylpiperidin-4-yl)-6-[(piperidin-3-yl)amino]-3,4-dihydropyrimidin-4-one 1433159-31-9 C25H32N6OS
(R)-5-(1,3-benzothiazol-2-yl)-2-(1-cyclobutylpiperidin-4-yl)-6-[(piperidin-3-yl)amino]-3,4-dihydropyrimidin-4-one
—— tert-butyl N-[2-[4-[3-(1H-benzimidazol-2-yl)-4-fluorophenyl]piperazin-1-yl]-2-oxoethyl]carbamate 1160831-86-6 C24H28FN5O3
tert-butyl N-[2-[4-[3-(1H-benzimidazol-2-yl)-4-fluorophenyl]piperazin-1-yl]-2-oxoethyl]carbamate
—— Tert-butyl 4-[3-[[6-(1-oxo-3,4-dihydroisoquinolin-2-yl)pyridine-2-carbonyl]amino]pyridin-4-yl]piperazine-1-carboxylate 1107625-91-1 C29H32N6O4
Tert-butyl 4-[3-[[6-(1-oxo-3,4-dihydroisoquinolin-2-yl)pyridine-2-carbonyl]amino]pyridin-4-yl]piperazine-1-carboxylate
—— 5-(3-butyl-5-methyl-isoxazol-4-ylmethoxy)-2H-pyrazole-3-carboxylic acid N',N'-dimethyl-hydrazide 1254964-76-5 C15H23N5O3
5-(3-butyl-5-methyl-isoxazol-4-ylmethoxy)-2H-pyrazole-3-carboxylic acid N',N'-dimethyl-hydrazide
—— 4-[3-[1-(difluoromethyl)benzimidazol-2-yl]phenyl]-N,N-dimethylpiperazine-1-carboxamide 1160831-46-8 C21H23F2N5O
4-[3-[1-(difluoromethyl)benzimidazol-2-yl]phenyl]-N,N-dimethylpiperazine-1-carboxamide
—— 2-(1-amino-cyclobutylmethyl)-8-(5-methoxy-pyridin-3-yl)-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam 1105657-72-4 C23H22N4O2
2-(1-amino-cyclobutylmethyl)-8-(5-methoxy-pyridin-3-yl)-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam
—— (6S,9aS)-8-(1,3-benzothiazol-4-ylmethyl)-N-benzyl-6-[(2,4-dioxopyrimidin-1-yl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1145673-13-7 C30H30N8O5S
(6S,9aS)-8-(1,3-benzothiazol-4-ylmethyl)-N-benzyl-6-[(2,4-dioxopyrimidin-1-yl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide
—— 4-(5-propan-2-yl-1H-pyrazol-4-yl)-N-(4-pyrrolidin-1-ylbutyl)pyridin-2-amine 1160103-67-2 C19H29N5
4-(5-propan-2-yl-1H-pyrazol-4-yl)-N-(4-pyrrolidin-1-ylbutyl)pyridin-2-amine
—— 2-(1-amino-cyclopropylmethyl)-8-[3-methoxy-4-(2-methoxy-ethoxy)-phenyl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam 1105657-34-8 C26H27N3O4
2-(1-amino-cyclopropylmethyl)-8-[3-methoxy-4-(2-methoxy-ethoxy)-phenyl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam
—— 3-(3-chloro-4-isopropoxy-phenyl)-5-cyclohexyl-[1,2,4]oxadiazole 1035213-10-5 C17H21ClN2O2
3-(3-chloro-4-isopropoxy-phenyl)-5-cyclohexyl-[1,2,4]oxadiazole
—— (2R)-N-(5-chloropyrazin-2-yl)-2-(3-cyclopropyl-4-cyclopropylsulfonylphenyl)-3-[(1R)-3-hydroxycyclopentyl]propanamide 1174230-61-5 C24H28ClN3O4S
(2R)-N-(5-chloropyrazin-2-yl)-2-(3-cyclopropyl-4-cyclopropylsulfonylphenyl)-3-[(1R)-3-hydroxycyclopentyl]propanamide
—— 2-[2-(3-fluorophenyl)ethylamino]-N-(4-piperazin-1-ylpyridin-3-yl)pyrimidine-4-carboxamide 1107624-24-7 C22H24FN7O
2-[2-(3-fluorophenyl)ethylamino]-N-(4-piperazin-1-ylpyridin-3-yl)pyrimidine-4-carboxamide
—— (6S,9aS)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-8-[[6-(propylamino)-1-benzothiophen-3-yl]methyl]-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1145673-92-2 C36H40N6O4S
(6S,9aS)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-8-[[6-(propylamino)-1-benzothiophen-3-yl]methyl]-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide
—— Ethyl 1-[4-[2-[[4-[cyclohexyl(methyl)carbamoyl]-2-methylphenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylate 1423071-85-5 C34H43N3O4S
Ethyl 1-[4-[2-[[4-[cyclohexyl(methyl)carbamoyl]-2-methylphenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— 1-(2-methyl-5-thiazolylmethyl)-2-(nitromethylene)tetrahydropyrimidine 105843-31-0 C10H14N4O2S
1-(2-methyl-5-thiazolylmethyl)-2-(nitromethylene)tetrahydropyrimidine
—— 2-[5-Butan-2-yl-3-(4-fluoro-3-methylphenyl)-1,2,4-triazol-1-yl]-1-[4-(6-methoxypyrimidin-4-yl)piperazin-1-yl]ethanone 1447725-27-0 C24H30FN7O2
2-[5-Butan-2-yl-3-(4-fluoro-3-methylphenyl)-1,2,4-triazol-1-yl]-1-[4-(6-methoxypyrimidin-4-yl)piperazin-1-yl]ethanone
—— 2-[[[9-Cyclohexyl-2-(2-hydroxypropylamino)purin-6-yl]amino]methyl]-6-methoxyphenol 1257695-31-0 C22H30N6O3
2-[[[9-Cyclohexyl-2-(2-hydroxypropylamino)purin-6-yl]amino]methyl]-6-methoxyphenol
—— 2-[5-Cyclohexyl-3-(3-methoxyphenyl)-1,2,4-triazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone 1447724-77-7 C26H32N6O2
2-[5-Cyclohexyl-3-(3-methoxyphenyl)-1,2,4-triazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone
—— 1-{(R)-4-[4-(1H-benzoimidazol-2-yl)-2-trifluoromethyl-thiazol-5-yl]-2-methyl-piperazin-1-yl}-2-pyrazolo[3,4-b]pyridin-2-yl-ethanone 1449367-60-5 C24H21F3N8OS
1-{(R)-4-[4-(1H-benzoimidazol-2-yl)-2-trifluoromethyl-thiazol-5-yl]-2-methyl-piperazin-1-yl}-2-pyrazolo[3,4-b]pyridin-2-yl-ethanone
—— 3,4-dihydro-1H-pyrrolo[2,1-c][1,4]oxazine-6,8-dicarboxylic acid 8-[((R)-1-phenylpropyl)amide] 6-[((R)-1-pyridin-2-ylpropyl)amide] 1449137-79-4 C26H30N4O3
3,4-dihydro-1H-pyrrolo[2,1-c][1,4]oxazine-6,8-dicarboxylic acid 8-[((R)-1-phenylpropyl)amide] 6-[((R)-1-pyridin-2-ylpropyl)amide]
—— N-cyclohexyl-2-(2-methylphenyl)-2-[N-(2-thiophen-2-ylacetyl)-3-(trifluoromethyl)anilino]acetamide 1355325-19-7 C28H29F3N2O2S
N-cyclohexyl-2-(2-methylphenyl)-2-[N-(2-thiophen-2-ylacetyl)-3-(trifluoromethyl)anilino]acetamide
—— 5-(5-(6-(benzo[d]thiazol-6-ylamino)-4-(isopropylamino)pyridin-3-yl)-1,3,4-oxadiazol-2-yl)-N-cyclopropyl-2-fluorobenzenesulfonamide 1447225-51-5 C26H24FN7O3S2
5-(5-(6-(benzo[d]thiazol-6-ylamino)-4-(isopropylamino)pyridin-3-yl)-1,3,4-oxadiazol-2-yl)-N-cyclopropyl-2-fluorobenzenesulfonamide
—— 1-(4-(2-fluorophenyl)-6-(5-fluoropyridin-3-ylamino)-1,3,5-triazin-2-ylamino)-2-methylpropan-2-ol 1446506-00-8 C18H18F2N6O
1-(4-(2-fluorophenyl)-6-(5-fluoropyridin-3-ylamino)-1,3,5-triazin-2-ylamino)-2-methylpropan-2-ol
—— (4-fluoro-3-methoxyphenyl)(oxo)acetic acid 1081764-19-3 C9H7FO4
(4-fluoro-3-methoxyphenyl)(oxo)acetic acid
—— 2-bromo-1-cyclobutyl-1H-imidazole-4-carboxylic acid ethyl ester 1448870-30-1 C10H13BrN2O2
2-bromo-1-cyclobutyl-1H-imidazole-4-carboxylic acid ethyl ester
—— 4-Thiazolemethanol, 2-(difluoromethyl)- 1447915-01-6 C5H5F2NOS
4-Thiazolemethanol, 2-(difluoromethyl)-
—— 4-chloro-2-(4-chloro-1H-pyrazol-1-yl)benzaldehyde 1446818-99-0 C10H6Cl2N2O
4-chloro-2-(4-chloro-1H-pyrazol-1-yl)benzaldehyde
—— N-cyclohexyl-2-(3-fluoro-N-[2-(2-fluorophenoxy)acetyl]anilino)-2-(2-methylphenyl)acetamide 1355327-18-2 C29H30F2N2O3
N-cyclohexyl-2-(3-fluoro-N-[2-(2-fluorophenoxy)acetyl]anilino)-2-(2-methylphenyl)acetamide
—— 4-[2-(2,4-dichlorophenoxy)phenylsulfamoyl]-N-{2-oxo-2-[4-(2-oxo-2-pyrrolidin-1-ylethyl)piperazin-1-yl]ethyl}benzamide 1032611-87-2 C31H33Cl2N5O6S
4-[2-(2,4-dichlorophenoxy)phenylsulfamoyl]-N-{2-oxo-2-[4-(2-oxo-2-pyrrolidin-1-ylethyl)piperazin-1-yl]ethyl}benzamide
—— 9-(4-(2-aminopropyl)phenyl)-8-hydroxy-6-methylthieno[2,3-c]quinolin-4(5H)-one hydrochloride 1338544-81-2 C21H20N2O2S*ClH
9-(4-(2-aminopropyl)phenyl)-8-hydroxy-6-methylthieno[2,3-c]quinolin-4(5H)-one hydrochloride
—— (3S)-N-{1-[(1-methyl-3-phenyl-1H-indazol-5-yl)carbonyl]azetidin-3-yl}-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine 1373525-24-6 C26H26N6O2S
(3S)-N-{1-[(1-methyl-3-phenyl-1H-indazol-5-yl)carbonyl]azetidin-3-yl}-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine
—— (3S)-N-(1-{[3-(4-fluorophenyl)-1-methyl-1H-indazol-5-yl]carbonyl}azetidin-3-yl)-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine 1373525-29-1 C26H25FN6O2S
(3S)-N-(1-{[3-(4-fluorophenyl)-1-methyl-1H-indazol-5-yl]carbonyl}azetidin-3-yl)-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine
—— (R)-2-hydroxy-4-phenyl-N-((R)-1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)butanamide 1257117-37-5 C19H21F3N2O3
(R)-2-hydroxy-4-phenyl-N-((R)-1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)butanamide
—— 2-methoxy-4-methyl-6-morpholin-4-yl-N-[[4-(trifluoromethyl)-phenyl]-methyl]-pyridine-3-carboxylic acid amide 1373486-93-1 C20H22F3N3O3
2-methoxy-4-methyl-6-morpholin-4-yl-N-[[4-(trifluoromethyl)-phenyl]-methyl]-pyridine-3-carboxylic acid amide
—— 5-[(4-(5-methylthien)-2-yl)2-trifluoromethylphenyl]-5-phenyl-3,4-dihydroxy-2(5H)-furanone 1098479-00-5 C22H15F3O4S
5-[(4-(5-methylthien)-2-yl)2-trifluoromethylphenyl]-5-phenyl-3,4-dihydroxy-2(5H)-furanone
—— 5-[(4-(5-methylpyrid)-2-yl)2-cyclohexylphenyl]-5-(4-nitrophenyl)-3,4-dihydroxy-2(5H)-furanone 1098479-73-2 C28H26N2O6
5-[(4-(5-methylpyrid)-2-yl)2-cyclohexylphenyl]-5-(4-nitrophenyl)-3,4-dihydroxy-2(5H)-furanone
—— (S)-ethyl 2-(6-cyano-3-methyl-1-(trifluoromethylsulfonyloxy)naphthalen-2-yl)-2-(tert-pentyloxy)acetate 1447070-96-3 C22H24F3NO6S
(S)-ethyl 2-(6-cyano-3-methyl-1-(trifluoromethylsulfonyloxy)naphthalen-2-yl)-2-(tert-pentyloxy)acetate
—— (4-((2',6'-dimethyl-4'-(3-methylsulfonyl)propoxy-[1,1'-biphenyl]-3-yl)methoxy)phenyl)carbamic acid tert-butyl ester 1372195-14-6 C30H37NO6S
(4-((2',6'-dimethyl-4'-(3-methylsulfonyl)propoxy-[1,1'-biphenyl]-3-yl)methoxy)phenyl)carbamic acid tert-butyl ester
—— 6-(6-chloropyridin-2-yl)-N<sup>2</sup>-(3,5-difluorophenyl)-N<sup>4</sup>-isopropyl-1,3,5-triazine-2,4-diamine 1446501-64-9 C17H15ClF2N6
6-(6-chloropyridin-2-yl)-N<sup>2</sup>-(3,5-difluorophenyl)-N<sup>4</sup>-isopropyl-1,3,5-triazine-2,4-diamine
—— (E)-3-(5-(2-cyclo-hexylvinyl)furan-2-yl)-3-hydroxypropanenitrile 1448434-07-8 C15H19NO2
(E)-3-(5-(2-cyclo-hexylvinyl)furan-2-yl)-3-hydroxypropanenitrile
—— (S)-N-((S)-1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(3-(difluoromethoxy)phenyl)-5-oxopyrrolidine-2-carboxamide 1448347-54-3 C30H24ClF4N5O4
(S)-N-((S)-1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(3-(difluoromethoxy)phenyl)-5-oxopyrrolidine-2-carboxamide
—— N-[2-(4-morpholin-4-ylpiperidin-1-yl)-2-oxoethyl]-4-(2-phenoxyphenylsulfamoyl)benzamide 1032612-77-3 C30H34N4O6S
N-[2-(4-morpholin-4-ylpiperidin-1-yl)-2-oxoethyl]-4-(2-phenoxyphenylsulfamoyl)benzamide
—— N<sup>2</sup>-(cyclopropylmethyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine 1446503-07-6 C18H18N6
N<sup>2</sup>-(cyclopropylmethyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine
—— 4,6-dichloro-2-methylsulfanylpyrimidine-5-carboxylic acid (2-hydroxy-2-methylpropyl)(tetrahydropyran-4-yl)amide 1448988-06-4 C15H21Cl2N3O3S
4,6-dichloro-2-methylsulfanylpyrimidine-5-carboxylic acid (2-hydroxy-2-methylpropyl)(tetrahydropyran-4-yl)amide
—— 6-fluoro-8-((S)-3-methoxy-pyrrolidin-1-yl)-imidazo[1,2-a]pyridine-2-carboxylic acid [5-(3-chloro-5-fluoro-phenyl)-1H-benzoimidazol-2-yl]-amide 1254168-90-5 C26H21ClF2N6O2
6-fluoro-8-((S)-3-methoxy-pyrrolidin-1-yl)-imidazo[1,2-a]pyridine-2-carboxylic acid [5-(3-chloro-5-fluoro-phenyl)-1H-benzoimidazol-2-yl]-amide
—— N-((2R,6S,13aS,14aR,16aS,Z)-2-(7-fluoro-3-methylquinoxalin-2-yloxy)-14a-(1-methylcyclopropylsulfonylcarbamoyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecin-6-yl)thiazole-4-carboxamide 1352300-97-0 C35H40FN7O7S2
N-((2R,6S,13aS,14aR,16aS,Z)-2-(7-fluoro-3-methylquinoxalin-2-yloxy)-14a-(1-methylcyclopropylsulfonylcarbamoyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecin-6-yl)thiazole-4-carboxamide