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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(7-chloroquinazolin-4-yl)-7-(2-methyl-1H-benzimidazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1256945-42-2 C25H20ClN5O
4-(7-chloroquinazolin-4-yl)-7-(2-methyl-1H-benzimidazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 4-(2-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenylamino)pyrimidin-4-yl)-2-(pyrrolidin-1-yl)benzonitrile 1128095-38-4 C24H22N8
4-(2-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenylamino)pyrimidin-4-yl)-2-(pyrrolidin-1-yl)benzonitrile
—— 6-{[6-amino-9-(2-{1-[(2-methoxyethoxy)acetyl]piperidin-4-yl}ethyl)-9H-purin-8-yl]thio}-1,3-benzodioxole-5-carbonitrile 1156465-49-4 C25H29N7O5S
6-{[6-amino-9-(2-{1-[(2-methoxyethoxy)acetyl]piperidin-4-yl}ethyl)-9H-purin-8-yl]thio}-1,3-benzodioxole-5-carbonitrile
—— 5-hexyl-3-[3-(trifluoromethyl)benzyl]-1,3-oxazolidin-2-one 1174338-27-2 C17H22F3NO2
5-hexyl-3-[3-(trifluoromethyl)benzyl]-1,3-oxazolidin-2-one
—— 4-N-[2-(dimethylamino)ethyl]-3-methylsulfanyl-6-N-(4-morpholin-4-ylphenyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 1037477-99-8 C20H28N8OS
4-N-[2-(dimethylamino)ethyl]-3-methylsulfanyl-6-N-(4-morpholin-4-ylphenyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
—— [1-[4-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperidin-4-yl]methanol 1037476-92-8 C21H27N7O3S
[1-[4-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperidin-4-yl]methanol
—— N-(4-(2-methyl-2H-tetrazol-5-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine 1128096-69-4 C22H22N8O
N-(4-(2-methyl-2H-tetrazol-5-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine
—— 8-N-(1-adamantylmethyl)-3-N-[(2S)-1-hydroxybutan-2-yl]-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide 1038388-40-7 C28H34N4O3S
8-N-(1-adamantylmethyl)-3-N-[(2S)-1-hydroxybutan-2-yl]-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide
—— (2R)-2-[2-(cyclopentyloxy)-5-({6-[2-fluoro-1-(fluoromethyl)ethoxy]-1-(1-formylpiperidin-4-yl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl}methyl)phenoxy]-N-phenylpropanamide 1162652-52-9 C38H42F2N4O7
(2R)-2-[2-(cyclopentyloxy)-5-({6-[2-fluoro-1-(fluoromethyl)ethoxy]-1-(1-formylpiperidin-4-yl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl}methyl)phenoxy]-N-phenylpropanamide
—— methyl 3-(2-isobutanoyloxy-4-methoxyphenyl)propanoate 117285-72-0 C15H20O5
methyl 3-(2-isobutanoyloxy-4-methoxyphenyl)propanoate
—— —— 1396812-96-6 C24H28BrNOS
—— 1-ethynyl-2-((2-methoxyphenyl)ethynyl)benzene 1289154-70-6 C17H12O
1-ethynyl-2-((2-methoxyphenyl)ethynyl)benzene
—— (2R,3R,4R,5S,6S)-2-(acetoxymethyl)-6-(5-(4-((E)-3,3-dimethyl-4-((2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)amino)-4-oxobut-1-en-1-yl)-2-methylbenzyl)-4-isopropyl-2-methoxyphenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate 1240305-05-8 C47H65N3O12
(2R,3R,4R,5S,6S)-2-(acetoxymethyl)-6-(5-(4-((E)-3,3-dimethyl-4-((2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)amino)-4-oxobut-1-en-1-yl)-2-methylbenzyl)-4-isopropyl-2-methoxyphenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate
—— 1-((2R,4S,5R)-5-((bis(4-methoxyphenyl)(phenyl)methoxy)methyl)-4-((3-((2R,3S,5R)-3-hydroxy-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)propyl)thio)tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione 158944-93-5 C43H48N4O10S
1-((2R,4S,5R)-5-((bis(4-methoxyphenyl)(phenyl)methoxy)methyl)-4-((3-((2R,3S,5R)-3-hydroxy-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)propyl)thio)tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
—— [((t-Bu)2C24H28N6S2(Me)6)Ni2(μ-O2CCCH)]ClO4 1258236-78-0 C41H65N6Ni2O2S2*ClO4
[((t-Bu)2C24H28N6S2(Me)6)Ni2(μ-O2CCCH)]ClO4
—— 5,6-dimethyl-2-(3-methylphenyl)thieno[2,3-d]pyrimidin-4-amine 1239906-89-8 C15H15N3S
5,6-dimethyl-2-(3-methylphenyl)thieno[2,3-d]pyrimidin-4-amine
—— methyl-succinic acid bis-(N,N'-diethyl ureide) 101082-94-4 C15H28N4O4
methyl-succinic acid bis-(N,N'-diethyl ureide)
—— 3-ethoxy-4-((3-ethyl-1,1-dimethyl-1,3-dihydro-2H-benzo[e]indol-2-ylidene)methyl)cyclobut-3-ene-1,2-dione 1242756-96-2 C23H23NO3
3-ethoxy-4-((3-ethyl-1,1-dimethyl-1,3-dihydro-2H-benzo[e]indol-2-ylidene)methyl)cyclobut-3-ene-1,2-dione
—— 3-(m-tolyl)isoquinolin-1(2H)-one 194292-26-7 C16H13NO
3-(m-tolyl)isoquinolin-1(2H)-one
—— methyl (Z)-2-acetamido-3-(m-tolyl)acrylate 1155818-37-3 C13H15NO3
methyl (Z)-2-acetamido-3-(m-tolyl)acrylate
—— diethyl 2-(((4-(hydroxymethyl)phenyl)amino)methylene)malonate 1020068-93-2 C15H19NO5
diethyl 2-(((4-(hydroxymethyl)phenyl)amino)methylene)malonate
—— 4-phenyl-1-(1-phenylethyl)-1H-pyrrole-2,3-dicarboxylic acid dimethyl ester 1314975-87-5 C22H21NO4
4-phenyl-1-(1-phenylethyl)-1H-pyrrole-2,3-dicarboxylic acid dimethyl ester
—— 5-bromo-6-(2-chlorovinyl)benzo[d][1,3]dioxole 1001099-67-7 C9H6BrClO2
5-bromo-6-(2-chlorovinyl)benzo[d][1,3]dioxole
—— 3-tert.-Butyl-1,5-diphenyl-verdazyl 15145-49-0 C18H21N4
3-tert.-Butyl-1,5-diphenyl-verdazyl
—— 4-({6-[2-fluoro-1-(fluoromethyl)ethoxy]-1-(1-formylpiperidin-4-yl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl}methyl)biphenyl-2-carbonitrile 1162650-22-7 C31H28F2N4O4
4-({6-[2-fluoro-1-(fluoromethyl)ethoxy]-1-(1-formylpiperidin-4-yl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl}methyl)biphenyl-2-carbonitrile
—— 2-(2-fluorophenyl)-5-(4-(2-morpholinoethoxy)phenyl)oxazole-4-carboxamide 1082441-19-7 C22H22FN3O4
2-(2-fluorophenyl)-5-(4-(2-morpholinoethoxy)phenyl)oxazole-4-carboxamide
—— 6-bromo-3-(3,4-dimethoxybenzyl)-1-[1-(hydroxyacetyl)piperidin-3-yl]quinazoline-2,4(1H,3H)-dione 1140590-20-0 C24H26BrN3O6
6-bromo-3-(3,4-dimethoxybenzyl)-1-[1-(hydroxyacetyl)piperidin-3-yl]quinazoline-2,4(1H,3H)-dione
—— N-[5-(3,5-difluorobenzyl)-1H-indazol-3-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}-2-(tetrahydro-2H-pyran-4-ylamino)benzamide 1108744-01-9 C31H35F2N5O3
N-[5-(3,5-difluorobenzyl)-1H-indazol-3-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}-2-(tetrahydro-2H-pyran-4-ylamino)benzamide
—— 3-(2-tert-butylphenoxy)-1-(3-phenylpropanoyl)azetidine 1146957-78-9 C22H27NO2
3-(2-tert-butylphenoxy)-1-(3-phenylpropanoyl)azetidine
—— N-(3-cyclopentyl-2-phenylpropyl)-1-pyrimidin-2-yl-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1104271-29-5 C23H24F3N5O
N-(3-cyclopentyl-2-phenylpropyl)-1-pyrimidin-2-yl-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— N-cyclohexyl-2-(2,6-difluorophenyl)-5-(trifluoromethyl)imidazo[1,2-a]pyridin-3-amine 1152030-68-6 C20H18F5N3
N-cyclohexyl-2-(2,6-difluorophenyl)-5-(trifluoromethyl)imidazo[1,2-a]pyridin-3-amine
—— 1-(4-amino-5-methylpyrimidin-2-yl)-N-{[1-(4-fluorophenyl)cyclohexyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1104270-83-8 C23H24F4N6O
1-(4-amino-5-methylpyrimidin-2-yl)-N-{[1-(4-fluorophenyl)cyclohexyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— [(S)-1-(4-{(R)-3-[1-(5-chloropyrimidin-2-yl)piperidin-4-yl]butoxy}phenyl)-2-(3,3-difluoropyrrolidin-1-yl)-2-oxoethyl]carbamic acid tert-butyl ester 1131872-78-0 C30H40ClF2N5O4
[(S)-1-(4-{(R)-3-[1-(5-chloropyrimidin-2-yl)piperidin-4-yl]butoxy}phenyl)-2-(3,3-difluoropyrrolidin-1-yl)-2-oxoethyl]carbamic acid tert-butyl ester
—— 6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-phenylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine 1256952-67-6 C29H29N7OS
6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-phenylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine
—— 2-[[3-methylsulfanyl-6-(4-morpholin-4-ylanilino)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino]ethanol 1037474-70-6 C18H23N7O2S
2-[[3-methylsulfanyl-6-(4-morpholin-4-ylanilino)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino]ethanol
—— {5-(2-methoxy-phenyl)-7-methyl-2-[(pyridin-3-ylmethyl)-amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}-thiophen-2-yl-methanone 1131991-59-7 C25H21N5O2S
{5-(2-methoxy-phenyl)-7-methyl-2-[(pyridin-3-ylmethyl)-amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}-thiophen-2-yl-methanone
—— (3R,4S)-1-((2-(1H-indol-3-yl)-9-methyl-6-morpholino-9H-purin-8-yl)methyl)-3-fluoro-N,N-dimethylpiperidin-4-amine 1257306-86-7 C26H33FN8O
(3R,4S)-1-((2-(1H-indol-3-yl)-9-methyl-6-morpholino-9H-purin-8-yl)methyl)-3-fluoro-N,N-dimethylpiperidin-4-amine
—— (2R,4S)-ethyl 5-(biphenyl-4-yl)-4-(2,4-difluoro-3-hydroxybenzamido)-2-methylpentanoate 1257266-06-0 C27H27F2NO4
(2R,4S)-ethyl 5-(biphenyl-4-yl)-4-(2,4-difluoro-3-hydroxybenzamido)-2-methylpentanoate
—— 5-(3,5-Dimethyl-4-isoxazolyl)-3-fluoro-2-hydroxybenzaldehyde 1093118-31-0 C12H10FNO3
5-(3,5-Dimethyl-4-isoxazolyl)-3-fluoro-2-hydroxybenzaldehyde
—— 1-(6-azetidin-1-yl-2-methyl-pyridin-3-yl)-8-(5-ethoxy-6-methoxymethyl-pyridin-3-yl)-3-methyl-1,3-dihydro-imidazo[4,5-c]quinolin-2-one 1257430-40-2 C29H30N6O3
1-(6-azetidin-1-yl-2-methyl-pyridin-3-yl)-8-(5-ethoxy-6-methoxymethyl-pyridin-3-yl)-3-methyl-1,3-dihydro-imidazo[4,5-c]quinolin-2-one
—— N-methyl-N-pyridin-3-yl-6-(2,4-dichlorophenoxy)-nicotinamide 1246663-31-9 C18H13Cl2N3O2
N-methyl-N-pyridin-3-yl-6-(2,4-dichlorophenoxy)-nicotinamide
—— (2S,3R)-3-(3-carboxy-propionylamino)-4-(3'-chloro-biphenyl-4-yl)-2-methoxybutyric acid methyl ester 1375592-65-6 C22H24ClNO6
(2S,3R)-3-(3-carboxy-propionylamino)-4-(3'-chloro-biphenyl-4-yl)-2-methoxybutyric acid methyl ester
—— 3-chloro-5-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)pyridin-2-amine 1251158-96-9 C24H23ClFN3O4S
3-chloro-5-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)pyridin-2-amine
—— N-methyl-N-pyridin-3-yl-4-(trifluoromethoxy)benzamide 1246664-89-0 C14H11F3N2O2
N-methyl-N-pyridin-3-yl-4-(trifluoromethoxy)benzamide
—— (R)-ethyl 4-(3'-chlorobiphenyl-4-yl)-3-(3-hydroxy-1H-pyrazole-5-carboxamido)butanoate 1257444-20-4 C22H22ClN3O4
(R)-ethyl 4-(3'-chlorobiphenyl-4-yl)-3-(3-hydroxy-1H-pyrazole-5-carboxamido)butanoate
—— N-(4-{5-[1-(2-fluorophenyl)-5-pyridin-4-yl-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}benzyl)-2-methylalanine 1166831-42-0 C26H22FN7O3
N-(4-{5-[1-(2-fluorophenyl)-5-pyridin-4-yl-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}benzyl)-2-methylalanine
—— 5-(4-(piperazin-1-yl)phenyl)-2-(pyridin-3-ylamino)oxazole-4-carboxamide 1082443-20-6 C19H20N6O2
5-(4-(piperazin-1-yl)phenyl)-2-(pyridin-3-ylamino)oxazole-4-carboxamide
—— (S)-cyclopropanecarboxylic acid {3-[3-fluoro-4-(4-[1,2,4]triazol-1-ylmethyl-[1,2,3]triazol-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-amide 1087353-49-8 C19H19FN8O3
(S)-cyclopropanecarboxylic acid {3-[3-fluoro-4-(4-[1,2,4]triazol-1-ylmethyl-[1,2,3]triazol-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-amide
—— N-methyl-3-(2-methylpropanoylamino)-N-pyridin-3-ylbenzamide 1246665-04-2 C17H19N3O2
N-methyl-3-(2-methylpropanoylamino)-N-pyridin-3-ylbenzamide
—— N-((9-methyl-2-(2-methyl-1H-benzo[d]imidazol-1-yl)-6-morpholino-9H-purin-8-yl)methyl)-1-phenylethanamine 1257380-92-9 C27H30N8O
N-((9-methyl-2-(2-methyl-1H-benzo[d]imidazol-1-yl)-6-morpholino-9H-purin-8-yl)methyl)-1-phenylethanamine