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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-cyclooctyl-1-phenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one 1056634-07-1 C19H22N4O
5-cyclooctyl-1-phenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one
—— N-(benzo[b]thiophen-2-yl)-N-(2-methyl-benzyl)-benzenesulfonamide 1104622-00-5 C22H19NO2S2
N-(benzo[b]thiophen-2-yl)-N-(2-methyl-benzyl)-benzenesulfonamide
—— 1,3-dihydro-1,3-diimino-4,7-bis(hexyloxy)isoindole 162898-83-1 C20H31N3O2
1,3-dihydro-1,3-diimino-4,7-bis(hexyloxy)isoindole
—— 2-(α-Hydroxy-isopropyl)-7-methoxy-1-methyl-1,2,3,4,9,10-hexahydro-phenanthren 102020-81-5 C19H26O2
2-(α-Hydroxy-isopropyl)-7-methoxy-1-methyl-1,2,3,4,9,10-hexahydro-phenanthren
—— 4-Hydroxy-benzoesaeure-(4-hydroxy-phenyl)-(4-hydroxy-benzyl)-amid 102079-16-3 C20H17NO4
4-Hydroxy-benzoesaeure-(4-hydroxy-phenyl)-(4-hydroxy-benzyl)-amid
—— N-(3-methyl-benzo[b]thiophen-2-yl)-N-(4-trifluoromethyl-benzyl)-4-carboxy-benzenesulfonamide 1104625-86-6 C24H18F3NO4S2
N-(3-methyl-benzo[b]thiophen-2-yl)-N-(4-trifluoromethyl-benzyl)-4-carboxy-benzenesulfonamide
—— N-(3-fluoro-propyl)-N-(3-methyl-benzo[b]thiophen-2-yl)-3,4-difluoro-benzenesulfonamide 1104622-93-6 C18H16F3NO2S2
N-(3-fluoro-propyl)-N-(3-methyl-benzo[b]thiophen-2-yl)-3,4-difluoro-benzenesulfonamide
—— 2-amino-8-(2-aminopyrimidin-5-yl)-7-methoxy-6-[2-methyl-5-(3-trifluoromethylbenzamide)phenyl]quinazoline 1191929-63-1 C28H22F3N7O2
2-amino-8-(2-aminopyrimidin-5-yl)-7-methoxy-6-[2-methyl-5-(3-trifluoromethylbenzamide)phenyl]quinazoline
—— 5-(3,5-dichlorophenylsulphonylamino)naphthalene-1-carboxylic acid 2-aminocarbonylbenzylamide 1192207-85-4 C25H19Cl2N3O4S
5-(3,5-dichlorophenylsulphonylamino)naphthalene-1-carboxylic acid 2-aminocarbonylbenzylamide
—— N-(3-(1-hydroxyethyl)benzo[b]thiophen-2-yl)-N-(3,3,3-trifluoro-propyl)-ethanesulfonamide 1104625-38-8 C15H18F3NO3S2
N-(3-(1-hydroxyethyl)benzo[b]thiophen-2-yl)-N-(3,3,3-trifluoro-propyl)-ethanesulfonamide
—— (Z)-methyl 2-(2-bromo-4-fluorophenyl)-3-((1-(tetrahydro-2H-pyran-4-yl)ethyl)amino)but-2-enoate 1450658-72-6 C18H23BrFNO3
(Z)-methyl 2-(2-bromo-4-fluorophenyl)-3-((1-(tetrahydro-2H-pyran-4-yl)ethyl)amino)but-2-enoate
—— N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-(1-(1-(ethylsulfonyl)piperidin-4-yl)ethyl)-2-methyl-1H-indole-3-carboxamide 1450656-15-1 C27H36N4O4S
N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-(1-(1-(ethylsulfonyl)piperidin-4-yl)ethyl)-2-methyl-1H-indole-3-carboxamide
—— 2-(chloromethyl)-4-(trifluoromethyl)thiophene 1643965-96-1 C6H4ClF3S
2-(chloromethyl)-4-(trifluoromethyl)thiophene
—— Tert-butyl 4-[4-[[5-[(2,6-difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-2-fluorophenyl]piperazine-1-carboxylate 1453212-49-1 C28H32F3N5O5
Tert-butyl 4-[4-[[5-[(2,6-difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-2-fluorophenyl]piperazine-1-carboxylate
—— N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-methyl-2-oxo-1,2-dihydropyridin-4-yl)ethyl)-1H-indole-3-carboxamide 1450653-51-6 C26H28N4O3
N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-methyl-2-oxo-1,2-dihydropyridin-4-yl)ethyl)-1H-indole-3-carboxamide
—— 1H-Indazole-3,5-diamine, 7-fluoro- 1352393-91-9 C7H7FN4
1H-Indazole-3,5-diamine, 7-fluoro-
—— 2-(2,6-dichloro-phenylamino)-6-chloro-1H-benzimidazol-5-carboxylic acid (3-chloro-phenyl)amide 1219118-93-0 C20H12Cl4N4O
2-(2,6-dichloro-phenylamino)-6-chloro-1H-benzimidazol-5-carboxylic acid (3-chloro-phenyl)amide
—— 5-bromo-2-(3,3-difluoropyrrolidin-1-yl)aniline 1644453-93-9 C10H11BrF2N2
5-bromo-2-(3,3-difluoropyrrolidin-1-yl)aniline
—— 4-Benzyl-2-(2-nitrophenyl)-4,5-dihydro-1,3-thiazole 1312996-45-4 C16H14N2O2S
4-Benzyl-2-(2-nitrophenyl)-4,5-dihydro-1,3-thiazole
—— (2-methyl-1-propylindol-3-yl)-(5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)methanone 1328169-86-3 C20H20N2OS
(2-methyl-1-propylindol-3-yl)-(5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)methanone
—— 6-(2-methoxypyridin-4-yl)-5-phenyl-1,2,4-triazin-3-amine 1321513-57-8 C15H13N5O
6-(2-methoxypyridin-4-yl)-5-phenyl-1,2,4-triazin-3-amine
—— 3-(2-chloro-phenoxy)-2-(4-chloro-phenyl)-6,7,8,9-tetrahydro-2H-pyrazolo[4,3-c]quinoline 1117954-20-7 C22H17Cl2N3O
3-(2-chloro-phenoxy)-2-(4-chloro-phenyl)-6,7,8,9-tetrahydro-2H-pyrazolo[4,3-c]quinoline
—— (R)-5-(1-(tert-butyldimethylsilyloxy)-2-(3-((4-(2-isopropylthiazole-4-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl)methyl)phenethylamino)ethyl)-8-hydroxyquinolin-2(1H)-one 1179336-75-4 C41H57N5O5SSi
(R)-5-(1-(tert-butyldimethylsilyloxy)-2-(3-((4-(2-isopropylthiazole-4-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl)methyl)phenethylamino)ethyl)-8-hydroxyquinolin-2(1H)-one
—— 1-[3-(3-amino-1,1-difluoropropyl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]cyclopropane-1-carbonitrile 1160502-06-6 C19H17F2N5
1-[3-(3-amino-1,1-difluoropropyl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]cyclopropane-1-carbonitrile
—— Methyl 2-[4-[4-(6-carbamoyl-3,5-dimethylpyrazin-2-yl)-3-methylphenyl]phenyl]acetate 1166830-72-3 C23H23N3O3
Methyl 2-[4-[4-(6-carbamoyl-3,5-dimethylpyrazin-2-yl)-3-methylphenyl]phenyl]acetate
—— 5-tert-butyl 2-ethyl 3-{[(4-methoxyphenyl)acetyl]amino}-6,6-dimethylpyrrolo[3,4-c]pyrazole-2,5(4H,6H)-dicarboxylate 1041015-83-1 C24H32N4O6
5-tert-butyl 2-ethyl 3-{[(4-methoxyphenyl)acetyl]amino}-6,6-dimethylpyrrolo[3,4-c]pyrazole-2,5(4H,6H)-dicarboxylate
—— 3-(4-(1-(2-cyano-1-cyclopentylethyl)-1H-pyrazol-4-yl)pyrimidin-2-ylamino)-N-(pyridin-3-ylmethyl)benzamide 1153939-62-8 C28H28N8O
3-(4-(1-(2-cyano-1-cyclopentylethyl)-1H-pyrazol-4-yl)pyrimidin-2-ylamino)-N-(pyridin-3-ylmethyl)benzamide
—— 1,1-Dimethylethyl N-methyl-N-[cis-3-[(1-methylethyl)amino]cyclobutyl]carbamate 1033718-23-8 C13H26N2O2
1,1-Dimethylethyl N-methyl-N-[cis-3-[(1-methylethyl)amino]cyclobutyl]carbamate
—— 2-(4-fluorophenyl)-N-(3-methyl-1H-indazol-5-yl)-2-oxo-N-[2-(6-trifluoromethylpyridin-3-yl)ethyl]acetamide 1201196-62-4 C24H18F4N4O2
2-(4-fluorophenyl)-N-(3-methyl-1H-indazol-5-yl)-2-oxo-N-[2-(6-trifluoromethylpyridin-3-yl)ethyl]acetamide
—— 5-phenyl-6-[3-(propan-2-yl)phenyl]-1,2,4-triazin-3-amine 1321513-13-6 C18H18N4
5-phenyl-6-[3-(propan-2-yl)phenyl]-1,2,4-triazin-3-amine
—— 4-iodo-5-(4-methoxytetrahydropyran-4-yl)-2-(methylthio)thiazole 1270931-19-5 C10H14INO2S2
4-iodo-5-(4-methoxytetrahydropyran-4-yl)-2-(methylthio)thiazole
—— 2-[(7R)-1,3-dichloro-7-[(4-fluorophenyl)sulfonyl-methylamino]-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetic acid 1268339-78-1 C21H19Cl2FN2O4S
2-[(7R)-1,3-dichloro-7-[(4-fluorophenyl)sulfonyl-methylamino]-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetic acid
—— (E)-3-[3-chloro-5-methyl-4-({5-[(4-methylbenzyl)oxy]pyridin-2-yl}oxy)phenyl]-1-(4-{4-[2-(4-ethoxyphenoxy)ethoxy]benzyl}piperazin-1-yl)prop-2-en-1-one 1322780-34-6 C44H46ClN3O6
(E)-3-[3-chloro-5-methyl-4-({5-[(4-methylbenzyl)oxy]pyridin-2-yl}oxy)phenyl]-1-(4-{4-[2-(4-ethoxyphenoxy)ethoxy]benzyl}piperazin-1-yl)prop-2-en-1-one
—— (4R)-4-[[7-(3-chloro-4-methoxyphenyl)-1,6-naphthyridin-5-yl]oxymethyl]pyrrolidin-2-one 1319738-52-7 C20H18ClN3O3
(4R)-4-[[7-(3-chloro-4-methoxyphenyl)-1,6-naphthyridin-5-yl]oxymethyl]pyrrolidin-2-one
—— (E)-1-(4-(7-methoxyfuro[2,3-b]quinolin-4-ylamino)phenyl)ethanone O-4-morpholinobutyl oxime 1310569-97-1 C28H32N4O4
(E)-1-(4-(7-methoxyfuro[2,3-b]quinolin-4-ylamino)phenyl)ethanone O-4-morpholinobutyl oxime
—— 5-(4-chlorobenzyl)-2-(4-methoxyphenyl)-1,2,4,5,6,7-hexahydro-3H-pyrazolo[4,3-c]pyridin-3-one 1331732-73-0 C20H20ClN3O2
5-(4-chlorobenzyl)-2-(4-methoxyphenyl)-1,2,4,5,6,7-hexahydro-3H-pyrazolo[4,3-c]pyridin-3-one
—— 2-Benzyl-1,3-benzoxazol-6-amine 1152529-22-0 C14H12N2O
2-Benzyl-1,3-benzoxazol-6-amine
—— 6-(3-methoxypiperidin-1-yl)-5-phenyl-1,2,4-triazin-3-amine 1321516-21-5 C15H19N5O
6-(3-methoxypiperidin-1-yl)-5-phenyl-1,2,4-triazin-3-amine
—— 6-methyl-3-(pyrimidin-5-ylamino)-pyrazine-2-carboxylic acid [2-(2-hydroxy-ethyl)-5-pyridin-2-yl-2H-pyrazol-3-yl]-amide 1316121-21-7 C20H19N9O2
6-methyl-3-(pyrimidin-5-ylamino)-pyrazine-2-carboxylic acid [2-(2-hydroxy-ethyl)-5-pyridin-2-yl-2H-pyrazol-3-yl]-amide
—— (R)-3-(cyclopentylmethyl)-4-(cyclopropyl(4-(2,5-dichlorophenyl)thiazol-2-yl)amino)-4-oxobutanoic acid 1229363-81-8 C22H24Cl2N2O3S
(R)-3-(cyclopentylmethyl)-4-(cyclopropyl(4-(2,5-dichlorophenyl)thiazol-2-yl)amino)-4-oxobutanoic acid
—— [4-[5-[2-(6-Aminopyridin-3-yl)ethynyl]-6-ethylpyrimidin-4-yl]-2-chlorophenyl]-[4-(2-hydroxycyclopentyl)piperazin-1-yl]methanone 1321612-51-4 C29H31ClN6O2
[4-[5-[2-(6-Aminopyridin-3-yl)ethynyl]-6-ethylpyrimidin-4-yl]-2-chlorophenyl]-[4-(2-hydroxycyclopentyl)piperazin-1-yl]methanone
—— (1R,3S,5R,6R,7R)-1-(hydroxymethyl)-8-azabicyclo[3.2.1]octane-3,6,7-triol hydrochloride 1301611-62-0 C8H15NO4*ClH
(1R,3S,5R,6R,7R)-1-(hydroxymethyl)-8-azabicyclo[3.2.1]octane-3,6,7-triol hydrochloride
—— (R,S)-2-amino-N-(2-methoxypyridin-3-yl)-2-phenyl-N-[2-(4-trifluoromethylphenyl)ethyl]acetamide 1201195-23-4 C23H22F3N3O2
(R,S)-2-amino-N-(2-methoxypyridin-3-yl)-2-phenyl-N-[2-(4-trifluoromethylphenyl)ethyl]acetamide
—— N-(2-t-butoxycarbonylaminophenyl)-4-[3-(3-methylisoxazol-5-yl)-1-[3-(morpholin-4-yl)propyl]ureidomethyl]benzamide 1034495-90-3 C31H40N6O6
N-(2-t-butoxycarbonylaminophenyl)-4-[3-(3-methylisoxazol-5-yl)-1-[3-(morpholin-4-yl)propyl]ureidomethyl]benzamide
—— (E)-3-{4'-(trifluoromethoxy)-4-[4-(trifluoromethyl)benzyloxy]biphenyl-3-yl}propenoic acid 1018958-89-8 C24H16F6O4
(E)-3-{4'-(trifluoromethoxy)-4-[4-(trifluoromethyl)benzyloxy]biphenyl-3-yl}propenoic acid
—— (3S,5S)-1-{[(5R,6S)-5,6-bis(4-chlorophenyl)-3-isopropyl-6-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl]carbonyl}-N,N-dimethyl-5-(morpholin-4-ylcarbonyl)pyrrolidin-3-amine 1033708-31-4 C33H39Cl2N5O3S
(3S,5S)-1-{[(5R,6S)-5,6-bis(4-chlorophenyl)-3-isopropyl-6-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl]carbonyl}-N,N-dimethyl-5-(morpholin-4-ylcarbonyl)pyrrolidin-3-amine
—— (4S)-4-{[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]amino}-1-[(2R)-2-{[(2S)-1-ethoxy-1-oxo-4-phenylbutan-2-yl]amino}butanoyl]-L-proline 1321614-82-7 C31H39F3N4O6
(4S)-4-{[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]amino}-1-[(2R)-2-{[(2S)-1-ethoxy-1-oxo-4-phenylbutan-2-yl]amino}butanoyl]-L-proline
—— 2-(6-(2-chloro-4-(methylsulfonyl)benzyl)-2,5-dimethyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid 1179808-76-4 C18H18ClNO4S2
2-(6-(2-chloro-4-(methylsulfonyl)benzyl)-2,5-dimethyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
—— N-[5-(5-bromo-2-methoxybenzenesulfonyl)-2-methoxyphenyl]-N-(3-fluoropiperidin-4-yl)amine hydrochloride 1335405-57-6 C19H22BrFN2O4S*ClH
N-[5-(5-bromo-2-methoxybenzenesulfonyl)-2-methoxyphenyl]-N-(3-fluoropiperidin-4-yl)amine hydrochloride
—— 4-(2-fluoro-5-methylphenylamino)-7-methoxy-6-(4-methylpiperazin-1-yl)cinnoline-3-carboxamide 1041852-69-0 C22H25FN6O2
4-(2-fluoro-5-methylphenylamino)-7-methoxy-6-(4-methylpiperazin-1-yl)cinnoline-3-carboxamide