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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(1,1-Dimethyl-2-methylene-pentyl)-4-phenyl-[1,2,4]triazolidine-3,5-dione 133305-02-9 C16H21N3O2
1-(1,1-Dimethyl-2-methylene-pentyl)-4-phenyl-[1,2,4]triazolidine-3,5-dione
—— 2,8-dimethoxycarbonyl-1,4-dihydro-4-oxoquinoline 14195-43-8 C13H11NO5
2,8-dimethoxycarbonyl-1,4-dihydro-4-oxoquinoline
—— ((R)-1-{trans-(1S,2S)-1-[4-(3,5-dimethyl-[1,2,4]triazol-4-yl)phenoxy]indan-2-yl}piperidin-3-yl)-(3,3,3-trifluoropropyl)amine 1215271-26-3 C27H32F3N5O
((R)-1-{trans-(1S,2S)-1-[4-(3,5-dimethyl-[1,2,4]triazol-4-yl)phenoxy]indan-2-yl}piperidin-3-yl)-(3,3,3-trifluoropropyl)amine
—— Ethyl 4-isopropyl-2-(4-fluorophenyl)pyrrole-3-carboxylate 139993-92-3 C16H18FNO2
Ethyl 4-isopropyl-2-(4-fluorophenyl)pyrrole-3-carboxylate
—— Propan-2-yl 4-[5-methyl-6-(1-methylsulfonylpiperidin-4-yl)sulfanylpyrimidin-4-yl]oxypiperidine-1-carboxylate 1233081-45-2 C20H32N4O5S2
Propan-2-yl 4-[5-methyl-6-(1-methylsulfonylpiperidin-4-yl)sulfanylpyrimidin-4-yl]oxypiperidine-1-carboxylate
—— 1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2-[(E)-2-(2-cyclopentyloxy-3-methoxyphenyl)vinyl]-1H-benzimidazole 1233448-64-0 C27H23ClF3N3O2
1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2-[(E)-2-(2-cyclopentyloxy-3-methoxyphenyl)vinyl]-1H-benzimidazole
—— methyl 6-O-acetyl-4-O-benzyl-2,3-anhydro-α-L-gulopyranoside 1219031-07-8 C16H20O6
methyl 6-O-acetyl-4-O-benzyl-2,3-anhydro-α-L-gulopyranoside
—— 4-[5-(8-bromo-3-methyl-2-oxo-2,3-dihydro-imidazo[4,5-c]quinolin-1-yl)-6-methoxy-pyridin-2-yl]-piperazine-1-carboxylic acid tert-butyl ester 1257431-18-7 C26H29BrN6O4
4-[5-(8-bromo-3-methyl-2-oxo-2,3-dihydro-imidazo[4,5-c]quinolin-1-yl)-6-methoxy-pyridin-2-yl]-piperazine-1-carboxylic acid tert-butyl ester
—— 2-chloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)-6-(trifluoromethyl)benzamide 1258295-46-3 C17H13ClF3N3O2
2-chloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)-6-(trifluoromethyl)benzamide
—— 4-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)-5-fluoro-2-methoxy-N-(3-morpholin-4-ylpropyl)benzamide 1084952-73-7 C27H27F4N7O3
4-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)-5-fluoro-2-methoxy-N-(3-morpholin-4-ylpropyl)benzamide
—— 4-(6-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}pyrazolo[1,5-a]pyrimidin-3-yl)-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide 1109281-96-0 C23H23F3N6O2S
4-(6-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}pyrazolo[1,5-a]pyrimidin-3-yl)-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide
—— (2Z,5E)-2-amino-6-(4-chloro-2-fluoro-3-methoxyphenyl)-4-oxo-hexa-2,5-dienoic acid ethyl ester 1257337-07-7 C15H15ClFNO4
(2Z,5E)-2-amino-6-(4-chloro-2-fluoro-3-methoxyphenyl)-4-oxo-hexa-2,5-dienoic acid ethyl ester
—— N-[(3S,4S)-4-hydroxy-1,1-dioxidotetrahydro-3-thienyl]-4-[6-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide 1109283-61-5 C19H18N6O4S2
N-[(3S,4S)-4-hydroxy-1,1-dioxidotetrahydro-3-thienyl]-4-[6-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide
—— (S)-4-[4-((S)-2-Azido-2-methoxycarbonyl-ethyl)-1-benzyl-1H-imidazol-2-yl]-2-tert-butoxycarbonylamino-butyric acid benzyl ester 138629-35-3 C30H36N6O6
(S)-4-[4-((S)-2-Azido-2-methoxycarbonyl-ethyl)-1-benzyl-1H-imidazol-2-yl]-2-tert-butoxycarbonylamino-butyric acid benzyl ester
—— (N-Boc-L-Val-L-Pro-OMe)-ZnI 1196065-20-9 C16H27N2O5*IZn
(N-Boc-L-Val-L-Pro-OMe)-ZnI
—— OsCl(η(5)-indenyl)(triphenylphosphine)2 176037-97-1 C45H37ClOsP2
OsCl(η(5)-indenyl)(triphenylphosphine)2
—— methyl ((R)-(((1R,2S,5R)-2-isopropyl-5-methylcyclohexyl)oxy)(phenyl)phosphoryl)-L-phenylalaninate 1228361-72-5 C26H36NO4P
methyl ((R)-(((1R,2S,5R)-2-isopropyl-5-methylcyclohexyl)oxy)(phenyl)phosphoryl)-L-phenylalaninate
—— (S)-2-amino-3-(1H-indol-3-yl)-N-[2-(4-sulfamoyl-phenyl)-ethyl]-propionamide 1258783-91-3 C19H22N4O3S
(S)-2-amino-3-(1H-indol-3-yl)-N-[2-(4-sulfamoyl-phenyl)-ethyl]-propionamide
—— 9-Phenylaethinyl-xanthydrol 111561-35-4 C21H14O2
9-Phenylaethinyl-xanthydrol
—— 3-(3-isopropoxyphenyl)-6-(3-oxo-3-{4-[2-oxo-2-(1-pyrrolidinyl)ethyl]piperazino}propyl)-1,2,4-triazin-5(2H)-one 1107695-15-7 C25H34N6O4
3-(3-isopropoxyphenyl)-6-(3-oxo-3-{4-[2-oxo-2-(1-pyrrolidinyl)ethyl]piperazino}propyl)-1,2,4-triazin-5(2H)-one
—— N-(4-trifluoromethoxybenzyl)-N-pyridin-3-yl-6-[(4,6-dimethyl-pyrimidin-2-yl)sulfanyl]-nicotinamide 1246664-55-0 C25H20F3N5O2S
N-(4-trifluoromethoxybenzyl)-N-pyridin-3-yl-6-[(4,6-dimethyl-pyrimidin-2-yl)sulfanyl]-nicotinamide
—— 4-(2-(2-(azetidin-1-yl)-1H-benzo[d]imidazol-1-yl)-8-((4-tert-butylpiperazin-1-yl)methyl)-9-methyl-9H-purin-6-yl)morpholine 1257382-69-6 C29H40N10O
4-(2-(2-(azetidin-1-yl)-1H-benzo[d]imidazol-1-yl)-8-((4-tert-butylpiperazin-1-yl)methyl)-9-methyl-9H-purin-6-yl)morpholine
—— 2,2,2-trifluoro-1-(4-{[7-(1H-indazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}phenyl)ethanol 1251151-37-7 C25H20F3N3O3
2,2,2-trifluoro-1-(4-{[7-(1H-indazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}phenyl)ethanol
—— 4-[5-(3-methyl-1H-pyrazolo[4,3-c]pyridin-4-ylamino)-pyridin-3-yl]-benzonitrile 1246346-54-2 C19H14N6
4-[5-(3-methyl-1H-pyrazolo[4,3-c]pyridin-4-ylamino)-pyridin-3-yl]-benzonitrile
—— 6-(4-(2,6-dichlorobenzamido)pyridin-2-ylamino)nicotinamide 1258293-83-2 C18H13Cl2N5O2
6-(4-(2,6-dichlorobenzamido)pyridin-2-ylamino)nicotinamide
—— (4-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)phenyl)-(4-pyridin-4-ylmethylpiperazin-1-yl)methanone 1084952-51-1 C29H25F3N8O
(4-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)phenyl)-(4-pyridin-4-ylmethylpiperazin-1-yl)methanone
—— N-(benzo[d][1,3]dioxol-5-yl)-1-((5-ethyl-1,3,4-oxadiazol-2-yl)methyl)-1H-indazole-3-carboxamide 1190098-59-9 C20H17N5O4
N-(benzo[d][1,3]dioxol-5-yl)-1-((5-ethyl-1,3,4-oxadiazol-2-yl)methyl)-1H-indazole-3-carboxamide
—— 4-({4-[(3-chlorophenyl)sulfonyl]-2-methylphenyl}carbonyl)-7-(2-methyl-1H-benzimidazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251153-87-3 C31H26ClN3O4S
4-({4-[(3-chlorophenyl)sulfonyl]-2-methylphenyl}carbonyl)-7-(2-methyl-1H-benzimidazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— [4-(4-methyl-piperazin-1-yl)-phenyl]-(3-methyl-1H-pyrazolo[4,3-c]pyridin-4-yl)-amine 1246346-80-4 C18H22N6
[4-(4-methyl-piperazin-1-yl)-phenyl]-(3-methyl-1H-pyrazolo[4,3-c]pyridin-4-yl)-amine
—— 3-methyl-8-(2-methylamino-pyrimidin-5-yl)-1-(3-methyl-pyridin-2-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one 1257428-95-7 C22H19N7O
3-methyl-8-(2-methylamino-pyrimidin-5-yl)-1-(3-methyl-pyridin-2-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one
—— (1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (6-methanesulfonyl-2-methyl-pyridin-3-yl)-amide 1268879-03-3 C21H18F2N4O3S
(1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (6-methanesulfonyl-2-methyl-pyridin-3-yl)-amide
—— 3-isopropyl-3-(3-methoxyphenyl)-1-{2-[[2-(4-methoxyphenyl)ethyl](methyl)amino]ethyl}piperidin-2-one 1219625-44-1 C27H38N2O3
3-isopropyl-3-(3-methoxyphenyl)-1-{2-[[2-(4-methoxyphenyl)ethyl](methyl)amino]ethyl}piperidin-2-one
—— N-methyl-N-(3-{[2-(1-methyl-2-oxo-2,3-dihydro-1H-indol-5-ylamino)-[1,2,4]triazolo[1,5-a]pyridin-8-ylamino]methyl}pyridin-2-yl)methanesulfonamide 1257706-06-1 C23H24N8O3S
N-methyl-N-(3-{[2-(1-methyl-2-oxo-2,3-dihydro-1H-indol-5-ylamino)-[1,2,4]triazolo[1,5-a]pyridin-8-ylamino]methyl}pyridin-2-yl)methanesulfonamide
—— (S)-N-(6-(5-cyanopyrazin-2-ylamino)-4-(piperidin-3-ylamino)pyridin-3-yl)-2-(dimethylamino)acetamide 1137476-43-7 C19H25N9O
(S)-N-(6-(5-cyanopyrazin-2-ylamino)-4-(piperidin-3-ylamino)pyridin-3-yl)-2-(dimethylamino)acetamide
—— 2-[6-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrimidin-4-yl]-4-imidazol-1-yl-1H-pyrazol-3-one 1154029-85-2 C15H17N7O2
2-[6-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrimidin-4-yl]-4-imidazol-1-yl-1H-pyrazol-3-one
—— N,N,N,-trimethyl-N-<3-(6,6-dimethylbicyclo<3.1.1>hept-2-en-2yl)-1-methylallyl>ammonium iodide 111735-66-1 C16H28N*I
N,N,N,-trimethyl-N-<3-(6,6-dimethylbicyclo<3.1.1>hept-2-en-2yl)-1-methylallyl>ammonium iodide
—— 2-(3-(4-(3-chlorophenyl)piperazino)propoxy)benzaldehyde 103076-63-7 C20H23ClN2O2
2-(3-(4-(3-chlorophenyl)piperazino)propoxy)benzaldehyde
—— 2-[7-(4-Tert-butylpiperidin-1-yl)-5-methyl-2-phenylpyrazolo[1,5-a]pyrimidin-6-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid 1451006-45-3 C28H38N4O3
2-[7-(4-Tert-butylpiperidin-1-yl)-5-methyl-2-phenylpyrazolo[1,5-a]pyrimidin-6-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid
—— 10-ethoxy-25-fluoro-14-methoxy-N-methyl-20-(trifluoromethyl)-9-oxa-4,5,16,18,22,28-hexaaza-10-phosphapentacyclo[21.2.2.2(12,15).1(2,5).1(17,21)]hentriaconta-1(25),2(31),3,12,14,17(28),18,20,23,26,29-undecaene-24-carboxamide 10-oxide 1380305-10-1 C29H30F4N7O5P
10-ethoxy-25-fluoro-14-methoxy-N-methyl-20-(trifluoromethyl)-9-oxa-4,5,16,18,22,28-hexaaza-10-phosphapentacyclo[21.2.2.2(12,15).1(2,5).1(17,21)]hentriaconta-1(25),2(31),3,12,14,17(28),18,20,23,26,29-undecaene-24-carboxamide 10-oxide
—— 2-amino-N-[6-[2-(3,5-dimethylphenyl)ethynyl]pyridin-2-yl]propanamide 1452572-81-4 C18H19N3O
2-amino-N-[6-[2-(3,5-dimethylphenyl)ethynyl]pyridin-2-yl]propanamide
—— 3-(3-hydroxypiperidin-1-yl)sulfonyl-N-(3-pyridin-4-ylphenyl)benzamide 1445785-13-6 C23H23N3O4S
3-(3-hydroxypiperidin-1-yl)sulfonyl-N-(3-pyridin-4-ylphenyl)benzamide
—— ethyl 4-methyl-3-oxo-2-[(3,4,5-trifluorophenyl)methyl]pentanoate 1370227-71-6 C15H17F3O3
ethyl 4-methyl-3-oxo-2-[(3,4,5-trifluorophenyl)methyl]pentanoate
—— N-[(9S,11R)-14,20-dioxo-7-oxa-13,16,19,23-tetraazatetracyclo[19.3.1.1<sup>2</sup>'<sup>6</sup>.0<sup>9</sup>'<sup>13</sup>]hexacosa-1(25),2(26),3,5,21,23-hexaen-11-yl]-2-(2-naphthyl)acetamide 1460306-03-9 C33H33N5O4
N-[(9S,11R)-14,20-dioxo-7-oxa-13,16,19,23-tetraazatetracyclo[19.3.1.1<sup>2</sup>'<sup>6</sup>.0<sup>9</sup>'<sup>13</sup>]hexacosa-1(25),2(26),3,5,21,23-hexaen-11-yl]-2-(2-naphthyl)acetamide
—— 2,2,10,10-tetraethyl-6,7-dihydro-1H-pyrimido[1,2,3-ij][1,8]naphthyridine-1,3,9,11(2H,5H,10H)-tetraone 1039339-72-4 C19H26N2O4
2,2,10,10-tetraethyl-6,7-dihydro-1H-pyrimido[1,2,3-ij][1,8]naphthyridine-1,3,9,11(2H,5H,10H)-tetraone
—— 7-Benzoyl-9,10-dimethyl-indolo[1,2-a]quinoline-8,11-dione 108562-27-2 C25H17NO3
7-Benzoyl-9,10-dimethyl-indolo[1,2-a]quinoline-8,11-dione
—— 2-(tert-Butyl-dimethyl-silanyloxy)-8,8-dichloro-1-methyl-bicyclo[4.2.0]octan-7-one 108694-61-7 C15H26Cl2O2Si
2-(tert-Butyl-dimethyl-silanyloxy)-8,8-dichloro-1-methyl-bicyclo[4.2.0]octan-7-one
—— (R)-ethyl 1-(1-(di-tert-butoxyphosphoryloxy)butan-2-yl)-6-(6-(3-ethylureido)-4-(4-(trifluoromethyl)thiazol-2-yl)pyridin-3-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate 1258213-45-4 C36H45F3N5O8PS
(R)-ethyl 1-(1-(di-tert-butoxyphosphoryloxy)butan-2-yl)-6-(6-(3-ethylureido)-4-(4-(trifluoromethyl)thiazol-2-yl)pyridin-3-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate
—— N-[3-[[[2-[4-[4-(dimethylamino)piperidine-1-carbonyl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-N-methylmethanesulfonamide 1160213-60-4 C28H35F3N8O4S
N-[3-[[[2-[4-[4-(dimethylamino)piperidine-1-carbonyl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-N-methylmethanesulfonamide
—— 4-(6-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-3-yl)-N-[4-(trifluoromethyl)phenyl]thiophene-2-carboxamide 1109282-72-5 C23H14F3N5OS
4-(6-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-3-yl)-N-[4-(trifluoromethyl)phenyl]thiophene-2-carboxamide
—— 4-chloro-2-fluoro-5-[(7-quinolin-3-yl-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl)carbonyl]benzenesulfonamide 1251164-49-4 C25H19ClFN3O4S
4-chloro-2-fluoro-5-[(7-quinolin-3-yl-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl)carbonyl]benzenesulfonamide