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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[1-[(4-methoxy-2,6-dimethyl-phenyl)sulfonyl]-piperidin-2-yl]-methoxy]-1-[4-(2-pyrrolidin-1-yl-ethoxy)-4-[4-(trifluoromethyl)-phenyl]-piperidin-1-yl]-ethanone 1191239-66-3 C35H48F3N3O6S
2-[[1-[(4-methoxy-2,6-dimethyl-phenyl)sulfonyl]-piperidin-2-yl]-methoxy]-1-[4-(2-pyrrolidin-1-yl-ethoxy)-4-[4-(trifluoromethyl)-phenyl]-piperidin-1-yl]-ethanone
—— N-(2-t-butoxycarbonylaminophenyl)-5-[3-propargyl-1-(2-dimethylaminoethyl)ureidomethyl]pyridine-2-carboxylic acid amide 1064004-54-1 C26H34N6O4
N-(2-t-butoxycarbonylaminophenyl)-5-[3-propargyl-1-(2-dimethylaminoethyl)ureidomethyl]pyridine-2-carboxylic acid amide
—— 5-(benzo[d][1,3]dioxol-5-yl)-3-((5-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)pyridin-3-yl)methyl)-5-methylimidazolidine-2,4-dione 1198165-05-7 C29H25F6N3O6
5-(benzo[d][1,3]dioxol-5-yl)-3-((5-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)pyridin-3-yl)methyl)-5-methylimidazolidine-2,4-dione
—— 5-(benzo[d][1,3]dioxol-5-yl)-3-(3-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)phenethyl)-5-methylimidazolidine-2,4-dione 1198164-61-2 C31H28F6N2O6
5-(benzo[d][1,3]dioxol-5-yl)-3-(3-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)phenethyl)-5-methylimidazolidine-2,4-dione
—— dimethyl 2-((E)-4-acetoxyhept-2-enyl)-2-allylmalonate 1262125-37-0 C17H26O6
dimethyl 2-((E)-4-acetoxyhept-2-enyl)-2-allylmalonate
—— (R)-4-D-5-phenyl-3-(1-phenylethyl)oxazol-2(3H)-one 1259119-21-5 C17H15NO2
(R)-4-D-5-phenyl-3-(1-phenylethyl)oxazol-2(3H)-one
—— —— 1071836-45-7 C21H17ClN2O6
—— N-(5-(4-(4-amino-5-cyanopyrimidin-2-yl)-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-chloropyridin-3-yl)methanesulfonamide 1379580-15-0 C21H20ClN7O3S
N-(5-(4-(4-amino-5-cyanopyrimidin-2-yl)-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-chloropyridin-3-yl)methanesulfonamide
—— {(S)-2-[5-(5-methoxy-2-methylphenyl)-[1,2,4]oxadiazol-3-yl]pyrrolidin-1-yl}-(5-methyl-2-[1,2,3]triazol-2-ylphenyl)methanone 1597524-57-6 C24H24N6O3
{(S)-2-[5-(5-methoxy-2-methylphenyl)-[1,2,4]oxadiazol-3-yl]pyrrolidin-1-yl}-(5-methyl-2-[1,2,3]triazol-2-ylphenyl)methanone
—— (R)-5-amino-3-(5-amino-2-fluorophenyl)-6,6-dimethyl-3-(trifluoromethyl)-3,6-dihydro-2H-1,4-thiazine 1,1-dioxide 1600506-43-1 C13H15F4N3O2S
(R)-5-amino-3-(5-amino-2-fluorophenyl)-6,6-dimethyl-3-(trifluoromethyl)-3,6-dihydro-2H-1,4-thiazine 1,1-dioxide
—— 4-((3S,4S)-1-(5-cyanopyrimidin-2-yl)-4-methylpyrrolidin-3-ylamino)-6-(1-ethyl-1H-pyrazol-4-yl)pyrrolo[1,2-b]pyridazine-3-carboxamide 1400578-49-5 C23H24N10O
4-((3S,4S)-1-(5-cyanopyrimidin-2-yl)-4-methylpyrrolidin-3-ylamino)-6-(1-ethyl-1H-pyrazol-4-yl)pyrrolo[1,2-b]pyridazine-3-carboxamide
—— 2-(2,4-dimethyl-6-oxo-1,6-dihydro-pyrimidin-5-yl)-<i>N</i>-phenethyl-acetamide 14356-71-9 C16H19N3O2
2-(2,4-dimethyl-6-oxo-1,6-dihydro-pyrimidin-5-yl)-<i>N</i>-phenethyl-acetamide
—— 2-(2-Naphthyl)-5-acetyl-4,5,6,7 tetrahydro furo[3,2-c]pyridine 104916-30-5 C19H17NO2
2-(2-Naphthyl)-5-acetyl-4,5,6,7 tetrahydro furo[3,2-c]pyridine
—— N-(2-aminoethyl)-1-(4-chlorophenyl)-9H-pyrido[3,4-b]indole-3-carboxamide 1401863-53-3 C20H17ClN4O
N-(2-aminoethyl)-1-(4-chlorophenyl)-9H-pyrido[3,4-b]indole-3-carboxamide
—— 4-methyl-5-(1-methylethyl)-6-[9-methyl-7-pyridin-3-yl-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]pyrimidin-2-amine 1379579-80-2 C23H27N5O
4-methyl-5-(1-methylethyl)-6-[9-methyl-7-pyridin-3-yl-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]pyrimidin-2-amine
—— methyl 3-((4-((S)-1-((S)-6-(2-hydroxy-2-methylpropyl)-2-oxo-6-phenyl-1,3-oxazinan-3-yl)ethyl)phenyl)ethynyl)-3-(methoxycarbonyloxy)azetidine-1-carboxylate 1259034-65-5 C31H36N2O8
methyl 3-((4-((S)-1-((S)-6-(2-hydroxy-2-methylpropyl)-2-oxo-6-phenyl-1,3-oxazinan-3-yl)ethyl)phenyl)ethynyl)-3-(methoxycarbonyloxy)azetidine-1-carboxylate
—— 4-[[1-[4-ethyl-phenylsulfonyl]-5-(trifluoromethyl)-1H-indol-2-yl]methyl]benzoic acid 1274941-39-7 C25H20F3NO4S
4-[[1-[4-ethyl-phenylsulfonyl]-5-(trifluoromethyl)-1H-indol-2-yl]methyl]benzoic acid
—— (R)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)propan-2-yl)-2-(1-methyl-1H-pyrazol-4-yl)thiazole-4-carboxamide 1297541-28-6 C21H18ClN7OS
(R)-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)propan-2-yl)-2-(1-methyl-1H-pyrazol-4-yl)thiazole-4-carboxamide
—— 3-amino-6-(2,6-difluoro-4-(3-methoxyoxetan-3-yl)phenyl)-5-fluoropicolinic acid 1395994-28-1 C16H13F3N2O4
3-amino-6-(2,6-difluoro-4-(3-methoxyoxetan-3-yl)phenyl)-5-fluoropicolinic acid
—— 5-((S)-3-acetylamino-2-hydroxypropyl)-3-chloro-3',6'-dihydro-2'H[2,4']bipyridinyl-1'-carboxylic acid (3-chloro-4-trifluoromethylphenyl)amide 1353526-97-2 C23H23Cl2F3N4O3
5-((S)-3-acetylamino-2-hydroxypropyl)-3-chloro-3',6'-dihydro-2'H[2,4']bipyridinyl-1'-carboxylic acid (3-chloro-4-trifluoromethylphenyl)amide
—— 4-{[(4-methyl-2-pyridinyl)methyl]oxy}-3-(1,2,3,4-tetrahydro-7-isoquinolinyl)benzonitrile 1398695-68-5 C23H21N3O
4-{[(4-methyl-2-pyridinyl)methyl]oxy}-3-(1,2,3,4-tetrahydro-7-isoquinolinyl)benzonitrile
—— [4-(2-chloro-phenyl)-pyridin-3-yl]-isopropyl-amine 1395415-95-8 C14H15ClN2
[4-(2-chloro-phenyl)-pyridin-3-yl]-isopropyl-amine
—— 2-Methoxy-1,4-oxathian-S-oxid 1140523-69-8 C5H10O3S
2-Methoxy-1,4-oxathian-S-oxid
—— N-(2-hexylaminoethyl)-N-hexyl-5-isoquinolinesulfonamide 111541-24-3 C23H37N3O2S
N-(2-hexylaminoethyl)-N-hexyl-5-isoquinolinesulfonamide
—— N-[1-[2-(2-methoxyphenyl)ethyl]azepan-3-yl]-3-pyridin-4-yl-1H-indazole-5-carboxamide 1353250-87-9 C28H31N5O2
N-[1-[2-(2-methoxyphenyl)ethyl]azepan-3-yl]-3-pyridin-4-yl-1H-indazole-5-carboxamide
—— 2-((R)-3-benzhydryloxypyrrolidin-1-ylmethyl)isonicotinic acid 1351373-24-4 C24H24N2O3
2-((R)-3-benzhydryloxypyrrolidin-1-ylmethyl)isonicotinic acid
—— 2-fluoro-8-(4-fluorophenyl)-9-[6-(methyl{3-[(6,6,6-trifluorohexyl)sulphonyl]propyl}amino)hexyl]-6,7-dihydro-5H-benzo[7]annulen-3-ol 1353007-98-3 C33H44F5NO3S
2-fluoro-8-(4-fluorophenyl)-9-[6-(methyl{3-[(6,6,6-trifluorohexyl)sulphonyl]propyl}amino)hexyl]-6,7-dihydro-5H-benzo[7]annulen-3-ol
—— N-(2-{6-[2-imino-3-(1H-indol-4-ylme thyl)-7-methyl-2,3-dihydro-benzoimidazol-1-yl]-pyridazin-3-yl}-4-methoxy-phenyl)-acetamide 1352873-62-1 C30H27N7O2
N-(2-{6-[2-imino-3-(1H-indol-4-ylme thyl)-7-methyl-2,3-dihydro-benzoimidazol-1-yl]-pyridazin-3-yl}-4-methoxy-phenyl)-acetamide
—— 3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid 2-difluoromethoxy-benzylamide 1352433-44-3 C15H11F2N3O3S
3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid 2-difluoromethoxy-benzylamide
—— US10485800, Cmpd ID GY 1351476-92-0 C30H31N5O2
US10485800, Cmpd ID GY
—— 7-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-1,3-dihydro-2H-imidazo[4,5-c]-1,6-naphthyridin-2-one 1300737-07-8 C21H17N5O2
7-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-1,3-dihydro-2H-imidazo[4,5-c]-1,6-naphthyridin-2-one
—— 1-ethyl-3,3,5-trimethyl-7-((N-(2-methylpyridin-3-ylmethyl)-N-(2-(7-oxo-7H-thieno[2,3-c]pyridin-6-yl)ethyl)amino)methyl)-1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione 1266560-50-2 C31H35N5O3S
1-ethyl-3,3,5-trimethyl-7-((N-(2-methylpyridin-3-ylmethyl)-N-(2-(7-oxo-7H-thieno[2,3-c]pyridin-6-yl)ethyl)amino)methyl)-1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione
—— 1-(4-Fluoro-phenyl)-2-methyl-5-(4-pyrrol-1-yl-phenyl)-1H-pyrrole-3-carboxylic acid ethyl ester 131721-70-5 C24H21FN2O2
1-(4-Fluoro-phenyl)-2-methyl-5-(4-pyrrol-1-yl-phenyl)-1H-pyrrole-3-carboxylic acid ethyl ester
—— 17β-acetoxy-3-methoxy-estra-1,3,5(10)-trien-16-one 111186-56-2 C21H26O4
17β-acetoxy-3-methoxy-estra-1,3,5(10)-trien-16-one
—— 1,14-dithio-2,13-dithia-tetradecanedioic acid <i>O</i>,<i>O</i>'-diethyl ester 111412-14-7 C16H30O2S4
1,14-dithio-2,13-dithia-tetradecanedioic acid <i>O</i>,<i>O</i>'-diethyl ester
—— N-(2-methylaminoethyl)-N-methyl-5-isoquinolinesulfonamide 111541-20-9 C13H17N3O2S
N-(2-methylaminoethyl)-N-methyl-5-isoquinolinesulfonamide
—— N-Acetyl-N-[3-(2,5-dihydroxy-4-methyl-phenyl)-propyl]-acetamide 121746-36-9 C14H19NO4
N-Acetyl-N-[3-(2,5-dihydroxy-4-methyl-phenyl)-propyl]-acetamide
—— (2R,4S)-5-(3'-chlorobiphenyl-4-yl)-2-methyl-4-(2H-tetrazole-5-carbonylamino)pentanoic acid 1257266-26-4 C20H20ClN5O3
(2R,4S)-5-(3'-chlorobiphenyl-4-yl)-2-methyl-4-(2H-tetrazole-5-carbonylamino)pentanoic acid
—— 6-(2,6-difluoro-4-(2-hydroxypropan-2-yl)phenyl)-N-(4-((1R,3R,4R,5S)-3,4-dihydroxy-4,5-dimethylcyclohexyl)pyridin-3-yl)-5-fluoropicolinamide 1395278-58-6 C28H30F3N3O4
6-(2,6-difluoro-4-(2-hydroxypropan-2-yl)phenyl)-N-(4-((1R,3R,4R,5S)-3,4-dihydroxy-4,5-dimethylcyclohexyl)pyridin-3-yl)-5-fluoropicolinamide
—— rac-1,4-dioxan-2-yl-acetic acid benzyl ester 1394037-03-6 C13H16O4
rac-1,4-dioxan-2-yl-acetic acid benzyl ester
—— 3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid 4-isopropoxy-benzylamide 1352433-47-6 C17H17N3O3S
3-oxo-3H-isothiazolo[5,4-b]pyridine-2-carboxylic acid 4-isopropoxy-benzylamide
—— N-(4-methylphenyl)sulfonyl-6-tributylstannyl-3,4-dihydro-2H-pyran-5-carboxamide 124647-34-3 C25H41NO4SSn
N-(4-methylphenyl)sulfonyl-6-tributylstannyl-3,4-dihydro-2H-pyran-5-carboxamide
—— 3-(3-Chloro-phenyl)-5-hydroxy-1,3-dihydro-anthra[1,2-d]imidazole-2,6,11-trione 126359-33-9 C21H11ClN2O4
3-(3-Chloro-phenyl)-5-hydroxy-1,3-dihydro-anthra[1,2-d]imidazole-2,6,11-trione
—— 6,6-dichloro-5-(4-methylphenyl)-3-phenyl-2,5-dihydrooxepin-7-one 124558-55-0 C19H16Cl2O2
6,6-dichloro-5-(4-methylphenyl)-3-phenyl-2,5-dihydrooxepin-7-one
—— benzyl 3-O-(4-methoxybenzyl)-2,6-dideoxy-2-iodo-α-L-talopyranoside 119746-63-3 C21H25IO5
benzyl 3-O-(4-methoxybenzyl)-2,6-dideoxy-2-iodo-α-L-talopyranoside
—— ((E)-2-Oxo-hept-3-enyl)-phosphonic acid diethyl ester 123269-15-8 C11H21O4P
((E)-2-Oxo-hept-3-enyl)-phosphonic acid diethyl ester
—— 3-Chloro-6-[(5-chloro-2-methoxyphenyl)methyl]pyridazine 120129-87-5 C12H10Cl2N2O
3-Chloro-6-[(5-chloro-2-methoxyphenyl)methyl]pyridazine
—— 2-[3-(Oxiran-2-yl)propyl]phenol 123999-65-5 C11H14O2
2-[3-(Oxiran-2-yl)propyl]phenol
—— 4-[3-(2-chloro-benzyl)-2-imino-2,3-dihydrobenzoimidazol-1-yl]biphenyl-3-ylamine 1352872-55-9 C26H21ClN4
4-[3-(2-chloro-benzyl)-2-imino-2,3-dihydrobenzoimidazol-1-yl]biphenyl-3-ylamine
—— (S)-5-(5-amino-2-fluoro-phenyl)-2,5-dimethyl-2,5,6,7-tetrahydro-[1,4]thiazepin-3-ylamine 1396787-92-0 C13H18FN3S
(S)-5-(5-amino-2-fluoro-phenyl)-2,5-dimethyl-2,5,6,7-tetrahydro-[1,4]thiazepin-3-ylamine