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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(5-fluorothiazol-2-yl)-2-(4-(1,1-dioxotetrahydrothiopyran-4-ylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-cyclohexylpropanamide 1036208-26-0 C23H30FN3O6S3
N-(5-fluorothiazol-2-yl)-2-(4-(1,1-dioxotetrahydrothiopyran-4-ylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-cyclohexylpropanamide
—— (S)-N-(5-chlorothiazol-2-yl)-2-(4-(furan-2-ylmethylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide 1036207-86-9 C22H24ClN3O6S2
(S)-N-(5-chlorothiazol-2-yl)-2-(4-(furan-2-ylmethylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide
—— (RS)-1-(2,2-Diethoxyethyl)-3-((4-methylphenyl)aminocarbonylmethyl)-3-(N'-(2-methylphenyl)ureido)indolin-2-one 159883-10-0 C31H36N4O5
(RS)-1-(2,2-Diethoxyethyl)-3-((4-methylphenyl)aminocarbonylmethyl)-3-(N'-(2-methylphenyl)ureido)indolin-2-one
—— 1-cyclopropyl-N-{3-[1-(3-cyanophenyl)-2,2,2-trifluoro-ethoxy]quinoxalin-2-yl}methanesulfonamide 1226506-11-1 C21H17F3N4O3S
1-cyclopropyl-N-{3-[1-(3-cyanophenyl)-2,2,2-trifluoro-ethoxy]quinoxalin-2-yl}methanesulfonamide
—— 2-chloro-5-(2-fluoro-3-pyridinyl)phenyl 5-thio-β-D-xylopyranoside 1011721-51-9 C16H15ClFNO4S
2-chloro-5-(2-fluoro-3-pyridinyl)phenyl 5-thio-β-D-xylopyranoside
—— 3-azido-1-(octahydroisoquinolin-2-yl)propan-1-one 1257992-55-4 C12H20N4O
3-azido-1-(octahydroisoquinolin-2-yl)propan-1-one
—— 4-[(1R)-1-[(3R,5R)-4-[2-chloro-4-(2-hydroxyethoxy)phenyl]-3-(4-chlorophenyl)-5-methylpiperazin-1-yl]ethyl]benzonitrile 1097206-88-6 C28H29Cl2N3O2
4-[(1R)-1-[(3R,5R)-4-[2-chloro-4-(2-hydroxyethoxy)phenyl]-3-(4-chlorophenyl)-5-methylpiperazin-1-yl]ethyl]benzonitrile
—— (R)-2-(4-acetylpiperazin-1-yl)-4-(1-(2-fluoro-3-(trifluoromethyl)phenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one 1079656-91-9 C24H28F4N6O2
(R)-2-(4-acetylpiperazin-1-yl)-4-(1-(2-fluoro-3-(trifluoromethyl)phenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one
—— 3-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-1-(propan-2-yloxymethyl)-1-[4-(trifluoromethyl)phenyl]urea 1138592-33-2 C20H19F9N4O4
3-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-1-(propan-2-yloxymethyl)-1-[4-(trifluoromethyl)phenyl]urea
—— methyl-{5'-[(2-phenyl-5-trifluoromethyl-oxazole-4-carbonyl)-amino]-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-yl}-carbamic acid 2,2-dimethyl-propyl ester 1085838-33-0 C28H32F3N5O4
methyl-{5'-[(2-phenyl-5-trifluoromethyl-oxazole-4-carbonyl)-amino]-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-yl}-carbamic acid 2,2-dimethyl-propyl ester
—— 3-biphenyl-3-yl-6-(1-methyl-piperidin-3-yloxy)-imidazo[1,2-b]pyridazine 1000155-39-4 C24H24N4O
3-biphenyl-3-yl-6-(1-methyl-piperidin-3-yloxy)-imidazo[1,2-b]pyridazine
—— 4-(3,4-Difluoroanilino)thieno[3,2-c]quinoline-7-carboxylic acid 1009825-23-3 C18H10F2N2O2S
4-(3,4-Difluoroanilino)thieno[3,2-c]quinoline-7-carboxylic acid
—— (R)-2-(4-acetylpiperazin-1-yl)-4-(1-(4-(cyclopropylmethoxy)-3-fluorophenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one 1079659-45-2 C27H35FN6O3
(R)-2-(4-acetylpiperazin-1-yl)-4-(1-(4-(cyclopropylmethoxy)-3-fluorophenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one
—— 7-methyl-5-oxo-2-(pyrazin-2-ylmethylamino)-N-(2-pyrrolidin-1-ylethyl)benzimidazolo[1,2-a][1,8]naphthyridine-6-carboxamide 1138544-55-4 C27H28N8O2
7-methyl-5-oxo-2-(pyrazin-2-ylmethylamino)-N-(2-pyrrolidin-1-ylethyl)benzimidazolo[1,2-a][1,8]naphthyridine-6-carboxamide
—— 3-[6-(3-chlorophenoxy)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopentylbenzamide 1000158-05-3 C24H21ClN4O2
3-[6-(3-chlorophenoxy)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopentylbenzamide
—— 1-Methyl-2,7-dioxo-3-(5-phenyl-[1,3,4]thiadiazol-2-yl)-1,2,4,7-tetrahydro-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid ethyl ester 133389-62-5 C18H15N5O4S
1-Methyl-2,7-dioxo-3-(5-phenyl-[1,3,4]thiadiazol-2-yl)-1,2,4,7-tetrahydro-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid ethyl ester
—— N-((1-(2-methoxyphenyl)cyclopropyl)methyl)-1-((7-oxo-2-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methoxy)cyclohexanecarboxamide 1227416-90-1 C30H33N5O4
N-((1-(2-methoxyphenyl)cyclopropyl)methyl)-1-((7-oxo-2-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methoxy)cyclohexanecarboxamide
—— 5-(1-methyl-1H-pyrazol-4-yl)-2-[7-(2,3,6-trifluorobenzyl)imidazo[1,5-b]pyridazin-5-yl]pyrimidin-4-amine 1337564-36-9 C21H15F3N8
5-(1-methyl-1H-pyrazol-4-yl)-2-[7-(2,3,6-trifluorobenzyl)imidazo[1,5-b]pyridazin-5-yl]pyrimidin-4-amine
—— (3R,3aR,6R,7R,9aS,9bR)-6-Hydroxymethyl-3-methoxy-6,9a-dimethyl-dodecahydro-naphtho[1,2-c]furan-7-ol 109873-69-0 C16H28O4
(3R,3aR,6R,7R,9aS,9bR)-6-Hydroxymethyl-3-methoxy-6,9a-dimethyl-dodecahydro-naphtho[1,2-c]furan-7-ol
—— (1R,2R,9R)-2,10,10-Trimethyl-5-[1-methyl-prop-(Z)-ylidene]-3-oxa-6-aza-tricyclo[7.1.1.0<sup>2,7</sup>]undec-6-en-4-one 134639-28-4 C16H23NO2
(1R,2R,9R)-2,10,10-Trimethyl-5-[1-methyl-prop-(Z)-ylidene]-3-oxa-6-aza-tricyclo[7.1.1.0<sup>2,7</sup>]undec-6-en-4-one
—— (R,S)-2,2,3,3-tetramethyl-10-methylthio-1,4,6-trioxaspiro<4.5>decane 129917-68-6 C12H22O3S
(R,S)-2,2,3,3-tetramethyl-10-methylthio-1,4,6-trioxaspiro<4.5>decane
—— methyl 4-deoxy-2,3-O-isopropylidene-4-(trifluoroacetamido)-β-D-ribopyranoside 104575-46-4 C11H16F3NO5
methyl 4-deoxy-2,3-O-isopropylidene-4-(trifluoroacetamido)-β-D-ribopyranoside
—— 4-Tert-butyl-2-[[11,17,23-tritert-butyl-4-[(5-tert-butyl-2-hydroxyphenyl)methylideneamino]-25,26,27,28-tetrapropoxy-5-pentacyclo[19.3.1.13,7.19,13.115,19]octacosa-1(24),3(28),4,6,9,11,13(27),15(26),16,18,21(25),22-dodecaenyl]iminomethyl]phenol 1190216-09-1 C74H98N2O6
4-Tert-butyl-2-[[11,17,23-tritert-butyl-4-[(5-tert-butyl-2-hydroxyphenyl)methylideneamino]-25,26,27,28-tetrapropoxy-5-pentacyclo[19.3.1.13,7.19,13.115,19]octacosa-1(24),3(28),4,6,9,11,13(27),15(26),16,18,21(25),22-dodecaenyl]iminomethyl]phenol
—— 98.4-cyclopropyl-N-{2-hydroxymethyl-3-[1-methyl-6-oxo-5-(pyrazin-2-ylamino)-1,6-dihydro-pyridin-3-yl]-phenyl}-benzamide 1147530-50-4 C27H25N5O3
98.4-cyclopropyl-N-{2-hydroxymethyl-3-[1-methyl-6-oxo-5-(pyrazin-2-ylamino)-1,6-dihydro-pyridin-3-yl]-phenyl}-benzamide
—— acetic acid (2S,4S)-4-[2-(6-carbamoyl-5-methyl-thieno[2,3-d]pyrimidin-4-ylamino)-5-fluoro-phenoxy]-pyrrolidin-2-ylmethyl ester hydrochloride 1332713-27-5 C21H22FN5O4S*ClH
acetic acid (2S,4S)-4-[2-(6-carbamoyl-5-methyl-thieno[2,3-d]pyrimidin-4-ylamino)-5-fluoro-phenoxy]-pyrrolidin-2-ylmethyl ester hydrochloride
—— N-ethyl-N'-[1-imidazol-1-yl-1-(2-methylphenyl)methylidene]-N-(4-trifluoromethylbenzyl)hydrazine 1094022-80-6 C21H21F3N4
N-ethyl-N'-[1-imidazol-1-yl-1-(2-methylphenyl)methylidene]-N-(4-trifluoromethylbenzyl)hydrazine
—— 1,3-Dimethyl-2,3-dihydro-1H-indole-2-carboxylic acid ethyl ester 108797-72-4 C13H17NO2
1,3-Dimethyl-2,3-dihydro-1H-indole-2-carboxylic acid ethyl ester
—— 1,1,1,3,3,3-Hexafluoro-2-[4-[[6-fluoro-2-[2-[[4-(trifluoromethoxy)phenyl]methylidene]hydrazinyl]pyrimidin-4-yl]amino]phenyl]propan-2-ol 1138152-91-6 C21H13F10N5O2
1,1,1,3,3,3-Hexafluoro-2-[4-[[6-fluoro-2-[2-[[4-(trifluoromethoxy)phenyl]methylidene]hydrazinyl]pyrimidin-4-yl]amino]phenyl]propan-2-ol
—— (2R)-N-(2-carbamoyl-6-methylphenyl)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide 1140490-88-5 C23H25ClN6O2
(2R)-N-(2-carbamoyl-6-methylphenyl)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide
—— ethyl (2S)-2-[[2-(cyclopropylsulfonylamino)acetyl]amino]-3-(furan-2-yl)propanoate 1061647-74-2 C14H20N2O6S
ethyl (2S)-2-[[2-(cyclopropylsulfonylamino)acetyl]amino]-3-(furan-2-yl)propanoate
—— 3-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-1-(3,4-dichlorophenyl)-1-methylurea 1138593-04-0 C16H12Cl2F6N4O3
3-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-1-(3,4-dichlorophenyl)-1-methylurea
—— (S)-tert-butyl 3-methyl-4-(1-phenylpyrido[3,4-d]pyridazin-4-yl)piperazine-1-carboxylate 1133749-17-3 C23H27N5O2
(S)-tert-butyl 3-methyl-4-(1-phenylpyrido[3,4-d]pyridazin-4-yl)piperazine-1-carboxylate
—— (S)-3-cyclohexyl-2-(4-(furan-2-ylmethylcarbamothioyl)-2-oxopiperazin-1-yl)-N-(thiazol-2-yl)propanamide 1061645-12-2 C22H29N5O3S2
(S)-3-cyclohexyl-2-(4-(furan-2-ylmethylcarbamothioyl)-2-oxopiperazin-1-yl)-N-(thiazol-2-yl)propanamide
—— tert-butyl(dimethyl){[4-(S-methylsulfonimidoyl)benzyl]oxy}silane 1027730-47-7 C14H25NO2SSi
tert-butyl(dimethyl){[4-(S-methylsulfonimidoyl)benzyl]oxy}silane
—— (E)-1-((4-methoxyphenyl)sulfonyl)-N-(4-(phenyldiazenyl)phenyl)piperidine-4-carboxamide 1007004-96-7 C25H26N4O4S
(E)-1-((4-methoxyphenyl)sulfonyl)-N-(4-(phenyldiazenyl)phenyl)piperidine-4-carboxamide
—— 3,7-Dimethyl-1-(m-tolyloxycarbonylmethyl)-xanthin 19410-34-5 C16H16N4O4
3,7-Dimethyl-1-(m-tolyloxycarbonylmethyl)-xanthin
—— thiazol-5-ylmethyl 2-piperidin-4-ylethylcarbamate hydrochloride 1206673-63-3 C12H19N3O2S*ClH
thiazol-5-ylmethyl 2-piperidin-4-ylethylcarbamate hydrochloride
—— N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-2-phenoxy-acetamide trifluoroacetate 1146700-42-6 C2HF3O2*C24H31N3O2
N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-2-phenoxy-acetamide trifluoroacetate
—— —— 1620158-79-3 C7H4FIO
—— 2-(1-((6-chloropyridin-3-yl)methyl)-8-nitro-5-oxo-1,2,3,5,6,7-hexahydroimidazo[1,2-a]pyridin-6-yl)-N,N-diethylacetamide 1568939-10-5 C19H24ClN5O4
2-(1-((6-chloropyridin-3-yl)methyl)-8-nitro-5-oxo-1,2,3,5,6,7-hexahydroimidazo[1,2-a]pyridin-6-yl)-N,N-diethylacetamide
—— tert-butyl (2S)-2-[5-[4-[4-[2-[(4S,7R,10Z)-7-(methoxycarbonylamino)-6-oxo-1-oxa-5-azacyclododec-10-en-4-yl]-1H-imidazol-5-yl]phenyl]phenyl]-1H-imidazol-2-yl]pyrrolidine-1-carboxylate 1360164-18-6 C39H47N7O6
tert-butyl (2S)-2-[5-[4-[4-[2-[(4S,7R,10Z)-7-(methoxycarbonylamino)-6-oxo-1-oxa-5-azacyclododec-10-en-4-yl]-1H-imidazol-5-yl]phenyl]phenyl]-1H-imidazol-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl 4-((3-methoxyphenyl)sulfonyl)-4,6,6a,7,9,10-hexahydro-8H-pyrazino[1,2-a]pyrrolo[4,3,2-de]quinoline-8-carboxylate 1613592-98-5 C25H29N3O5S
tert-butyl 4-((3-methoxyphenyl)sulfonyl)-4,6,6a,7,9,10-hexahydro-8H-pyrazino[1,2-a]pyrrolo[4,3,2-de]quinoline-8-carboxylate
—— (2R)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]-N-[(4R)-8-fluoro-3,4-dihydro-1H-isochromen-4-yl]pyrrolidine-1-carboxamide 1140489-90-2 C24H25ClFN5O2
(2R)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]-N-[(4R)-8-fluoro-3,4-dihydro-1H-isochromen-4-yl]pyrrolidine-1-carboxamide
—— N-[5-(1-{3-[4-(1-benzyl-1H-tetrazol-5-yl)-piperidin-1-yl]-2-hydroxy-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide 1048034-54-3 C36H46F3N9O4S
N-[5-(1-{3-[4-(1-benzyl-1H-tetrazol-5-yl)-piperidin-1-yl]-2-hydroxy-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide
—— N-(2-methyl-5-{[(1-methylpropyl)amino]methyl}phenyl)-4-[(4-phenylquinazolin-2-yl)amino]benzamide 1059733-98-0 C33H33N5O
N-(2-methyl-5-{[(1-methylpropyl)amino]methyl}phenyl)-4-[(4-phenylquinazolin-2-yl)amino]benzamide
—— 4-chloro-N-[3-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-benzamide trifluoroacetate 1146700-91-5 C2HF3O2*C23H28ClN3O
4-chloro-N-[3-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-benzamide trifluoroacetate
—— 4-[2-(3-methyl-butylamino)purin-9-yl]benzamide 1332368-99-6 C17H20N6O
4-[2-(3-methyl-butylamino)purin-9-yl]benzamide
—— N-{2-[4-hydroxy-1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]cyclohexanecarboxamide 1226998-00-0 C35H43N5O3
N-{2-[4-hydroxy-1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]cyclohexanecarboxamide
—— 8-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]amino]-α,α-dimethyl-6-(trifluoromethaneyl)-imidazolo[1,2-a]pyridine-2-methanol 1232037-97-6 C22H22F3N5O2
8-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]amino]-α,α-dimethyl-6-(trifluoromethaneyl)-imidazolo[1,2-a]pyridine-2-methanol
—— N,N-diethyl-N'-benz[c]acridin-7-yl-pentanediyldiamine 103042-66-6 C26H31N3
N,N-diethyl-N'-benz[c]acridin-7-yl-pentanediyldiamine