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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(R)-3-(6-chloro-benzooxazol-2-ylamino)-pyrrolidin-1-yl]-(2-methoxy-5-methyl-phenyl)-methanone 1163121-25-2 C20H20ClN3O3
[(R)-3-(6-chloro-benzooxazol-2-ylamino)-pyrrolidin-1-yl]-(2-methoxy-5-methyl-phenyl)-methanone
—— 3,7-dimethyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide 1075710-71-2 C27H26N2O2
3,7-dimethyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide
—— 4-(carboxyphenylmethoxy)-5,7-dichloronaphthalene-2-carboxylic acid 1257342-60-1 C19H12Cl2O5
4-(carboxyphenylmethoxy)-5,7-dichloronaphthalene-2-carboxylic acid
—— 1-[(3,4-difluorophenyl)methyl]-N-[3-[3-[(1-methylpiperidin-4-yl)amino]quinoxalin-6-yl]prop-2-ynyl]-6-oxopyrimidine-5-carboxamide 1345437-98-0 C29H27F2N7O2
1-[(3,4-difluorophenyl)methyl]-N-[3-[3-[(1-methylpiperidin-4-yl)amino]quinoxalin-6-yl]prop-2-ynyl]-6-oxopyrimidine-5-carboxamide
—— N-(4-fluoro-3-(trifluoromethyl)phenyl)-4-methyl-3-(3-(pyridin-3-yl)acrylamido)benzamide 1255702-51-2 C23H17F4N3O2
N-(4-fluoro-3-(trifluoromethyl)phenyl)-4-methyl-3-(3-(pyridin-3-yl)acrylamido)benzamide
—— [(R)-3-(6-chloro-quinoxalin-2-ylamino)-pyrrolidin-1-yl]-(2-trifluoromethyl-phenyl)-methanone 1163122-76-6 C20H16ClF3N4O
[(R)-3-(6-chloro-quinoxalin-2-ylamino)-pyrrolidin-1-yl]-(2-trifluoromethyl-phenyl)-methanone
—— 4,5-dichloro-N-(2-sulfamoylphenyl)thiophene-2-sulfonamide 1161944-08-6 C10H8Cl2N2O4S3
4,5-dichloro-N-(2-sulfamoylphenyl)thiophene-2-sulfonamide
—— N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)phenyl]-6-methylpyridine-3-carboxamide 1092393-38-8 C24H21N5O3
N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)phenyl]-6-methylpyridine-3-carboxamide
—— 1-[5-(2-methyl-thiazol-4-yl)-thien-2-yl]carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan] 1159092-57-5 C22H23N3O2S2
1-[5-(2-methyl-thiazol-4-yl)-thien-2-yl]carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan]
—— 4-(3-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)isoquinolin-1-yl)benzoic acid 1152274-12-8 C27H18F2N2O5
4-(3-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)isoquinolin-1-yl)benzoic acid
—— 4-(aminocarbonyl)-3-[(1,2-dimethylpropyl)amino]benzoic acid 1149385-35-2 C13H18N2O3
4-(aminocarbonyl)-3-[(1,2-dimethylpropyl)amino]benzoic acid
—— 4-((R)-3-(8-methoxy-2-oxo-1,4-dihydro-2H-2λ5-benzo[d][1,3,2]oxazaphosphinin-2-yl)-2-((6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl)amino)propionyl)piperazine-1-carboxylic acid butyl ester 1159501-49-1 C36H46N7O8P
4-((R)-3-(8-methoxy-2-oxo-1,4-dihydro-2H-2λ5-benzo[d][1,3,2]oxazaphosphinin-2-yl)-2-((6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl)amino)propionyl)piperazine-1-carboxylic acid butyl ester
—— tert-butyl 4-(5-(5-chloro-3-(4-cyanophenoxy)pyridin-2-ylamino)-1,2,4-thiadiazol-3-yl)piperidine-1-carboxylate 1065604-39-8 C24H25ClN6O3S
tert-butyl 4-(5-(5-chloro-3-(4-cyanophenoxy)pyridin-2-ylamino)-1,2,4-thiadiazol-3-yl)piperidine-1-carboxylate
—— (1R,2S)-N-[4-(difluoromethyl)pyridin-2-yl]-2-[(2,4-dimethylpyrimidin-5-yl)oxymethyl]-2-phenylcyclopropane-1-carboxamide 1369763-18-7 C23H22F2N4O2
(1R,2S)-N-[4-(difluoromethyl)pyridin-2-yl]-2-[(2,4-dimethylpyrimidin-5-yl)oxymethyl]-2-phenylcyclopropane-1-carboxamide
—— (4-cyclopropylidene-3,5-dimethylcyclohexyl)benzene 1235836-79-9 C15H18
(4-cyclopropylidene-3,5-dimethylcyclohexyl)benzene
—— (R)-2-tert-butylmethylphosphino-3-(di-tert-butylphosphino)quinoxaline 1372791-52-0 C21H34N2P2
(R)-2-tert-butylmethylphosphino-3-(di-tert-butylphosphino)quinoxaline
—— 4,4-dimethyl-11-methoxy-7-nitro-1,2,3,4-tetrahydro-1,4-diazepino<5,6,7-kl>acridinium chloride 142181-64-4 C18H19N4O3*Cl
4,4-dimethyl-11-methoxy-7-nitro-1,2,3,4-tetrahydro-1,4-diazepino<5,6,7-kl>acridinium chloride
—— 5-(2,5-dichlorophenyl)-2-({6-(pyrrolidin-1-ylmethyl)pyridin-2-yl}amino)thiophene-3-carboxamide 1093872-16-2 C21H20Cl2N4OS
5-(2,5-dichlorophenyl)-2-({6-(pyrrolidin-1-ylmethyl)pyridin-2-yl}amino)thiophene-3-carboxamide
—— 6-(2,2-Bis-methylsulfanyl-vinyl)-4-(4-chloro-phenyl)-2-oxo-1,2-dihydro-pyridine-3-carbonitrile 114577-57-0 C16H13ClN2OS2
6-(2,2-Bis-methylsulfanyl-vinyl)-4-(4-chloro-phenyl)-2-oxo-1,2-dihydro-pyridine-3-carbonitrile
—— 4-[1'-(5-cyano-1,3-thiazol-2-yl)-4,4'-bipiperidin-1-yl]pyrimidine-2-carbonitrile 1039743-05-9 C19H21N7S
4-[1'-(5-cyano-1,3-thiazol-2-yl)-4,4'-bipiperidin-1-yl]pyrimidine-2-carbonitrile
—— 4-(aminocarbonyl)-2-chloro-5-(pentan-3-ylamino)benzoic acid 1149386-42-4 C13H17ClN2O3
4-(aminocarbonyl)-2-chloro-5-(pentan-3-ylamino)benzoic acid
—— N-(3,4-dimethylisoxazol-5-yl)-4-(2-phenylpyridin-4-yl)piperazine-1-carboxamide 1143578-18-0 C21H23N5O2
N-(3,4-dimethylisoxazol-5-yl)-4-(2-phenylpyridin-4-yl)piperazine-1-carboxamide
—— [(μ-4,4'-C6F4C6F4)(Au(C.tplbond.NC6H4O(CH2)3CH3-p))2] 189288-42-4 C34H26Au2F8N2O2
[(μ-4,4'-C6F4C6F4)(Au(C.tplbond.NC6H4O(CH2)3CH3-p))2]
—— 3,4,6-tris(t-butylthio)-3-methylthiothieno<3,4-c>thiophen-1(3H)-one 134541-67-6 C19H30OS5
3,4,6-tris(t-butylthio)-3-methylthiothieno<3,4-c>thiophen-1(3H)-one
—— 1-(1,3-benzodioxol-5-yl)ethylidenehydrazine 1257974-55-2 C9H10N2O2
1-(1,3-benzodioxol-5-yl)ethylidenehydrazine
—— 3-benzylidene-2-methyl-6-nitro-isoindolin-1-one 146748-07-4 C16H12N2O3
3-benzylidene-2-methyl-6-nitro-isoindolin-1-one
—— 5-{[7-isopropyl-6-(2-methyl-2H-pyrazol-3-yl)-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl]-methanesulfonyl-amino}-5-oxo-pentanoic acid ethyl ester 1350740-84-9 C23H29N5O7S
5-{[7-isopropyl-6-(2-methyl-2H-pyrazol-3-yl)-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl]-methanesulfonyl-amino}-5-oxo-pentanoic acid ethyl ester
—— US10202379, Reference Example 230 1370239-62-5 C26H27N3O5
US10202379, Reference Example 230
—— 9-Fluoro-5-ethyl-8-(1-piperazinyl)-6,7-dihydro-1,7-dioxo-1H, 5H-benzo[ij]quinolizine-2-carboxylic acid hydrochloride 108405-63-6 C19H20FN3O4*ClH
9-Fluoro-5-ethyl-8-(1-piperazinyl)-6,7-dihydro-1,7-dioxo-1H, 5H-benzo[ij]quinolizine-2-carboxylic acid hydrochloride
—— 5,9-dioxabicyclo[11.4.0]heptadeca-1(17),13,15-trien-2,11-diyne-6,8-dione 116510-14-6 C15H10O4
5,9-dioxabicyclo[11.4.0]heptadeca-1(17),13,15-trien-2,11-diyne-6,8-dione
—— 1-(7-Methyl-3-methylene-oct-6-enyl)-2-oxo-cyclopentanecarboxylic acid methyl ester 115395-40-9 C17H26O3
1-(7-Methyl-3-methylene-oct-6-enyl)-2-oxo-cyclopentanecarboxylic acid methyl ester
—— (1R,9S,12R)-5-(trifluoromethyl)tricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-12-amine 110267-95-3 C13H14F3N
(1R,9S,12R)-5-(trifluoromethyl)tricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-12-amine
—— (S)-2-{(1S,2S,3R)-3-[(S)-5-((R)-2-Benzyloxy-1-methyl-ethyl)-2-methyl-cyclopent-1-enylmethyl]-2-hydroxymethyl-3-methyl-cyclopentyl}-propan-1-ol 117152-40-6 C27H42O3
(S)-2-{(1S,2S,3R)-3-[(S)-5-((R)-2-Benzyloxy-1-methyl-ethyl)-2-methyl-cyclopent-1-enylmethyl]-2-hydroxymethyl-3-methyl-cyclopentyl}-propan-1-ol
—— (3S,4R)-4-benzyloxymethyl-3-hydroxyethyl-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylic acid tert-butyl ester 1037368-39-0 C27H35NO5
(3S,4R)-4-benzyloxymethyl-3-hydroxyethyl-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylic acid tert-butyl ester
—— 3-[N'-(4-Chloro-phenyl)-hydrazino]-3-methyl-butan-2-one 117609-34-4 C11H15ClN2O
3-[N'-(4-Chloro-phenyl)-hydrazino]-3-methyl-butan-2-one
—— 4,4,5,5-Tetramethyl-2-phenyl-4,5-dihydro-oxazole; compound with trifluoro-methanesulfonic acid 116935-12-7 CHF3O3S*C13H17NO
4,4,5,5-Tetramethyl-2-phenyl-4,5-dihydro-oxazole; compound with trifluoro-methanesulfonic acid
—— 3-[4-(Trifluoromethyl)piperidin-1-yl]cyclobutan-1-amine 1517845-90-7 C10H17F3N2
3-[4-(Trifluoromethyl)piperidin-1-yl]cyclobutan-1-amine
—— US10202379, Reference Example 285 1370248-88-6 C16H14ClFO2S
US10202379, Reference Example 285
—— N-[2-(5-{[4-(ethylsulfonyl)piperazin-1-yl]methyl}-1,3-thiazol-2-yl)-1H-indol-7-yl]-N-isopropylthiophene-2-sulfonamide trifluoroacetate 1020360-91-1 C2HF3O2*C25H31N5O4S4
N-[2-(5-{[4-(ethylsulfonyl)piperazin-1-yl]methyl}-1,3-thiazol-2-yl)-1H-indol-7-yl]-N-isopropylthiophene-2-sulfonamide trifluoroacetate
—— 5,6,7-trideoxy-2,3-O-isopropylidene-4-O-methylsulphonyl-L-ribo-hept-6-enononitrile 115886-16-3 C11H17NO5S
5,6,7-trideoxy-2,3-O-isopropylidene-4-O-methylsulphonyl-L-ribo-hept-6-enononitrile
—— anhydro-1-methoxy-3-methyl-5-hydroxy-1,2,3-triazolium hydroxide 116932-94-6 C4H7N3O2
anhydro-1-methoxy-3-methyl-5-hydroxy-1,2,3-triazolium hydroxide
—— (5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-m-tolylamine 1032184-47-6 C14H16N4
(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-m-tolylamine
—— (1S)-(1,3,5/2,4,6)-5-O-(2,3,4,6-tetra-O-acetyl-β-D-glucopyranosyl)-2-acetoxy-6-acetoxymethyl-3,4-dibenzyloxy-N-<(1S)-(1,4,6/5)-4,5,6-tribenzyloxy-3-benzyloxymethylcyclohex-2-enyl>cyclohexylamine 114779-33-8 C74H83NO20
(1S)-(1,3,5/2,4,6)-5-O-(2,3,4,6-tetra-O-acetyl-β-D-glucopyranosyl)-2-acetoxy-6-acetoxymethyl-3,4-dibenzyloxy-N-<(1S)-(1,4,6/5)-4,5,6-tribenzyloxy-3-benzyloxymethylcyclohex-2-enyl>cyclohexylamine
—— (3aS)-7-hydroxy-3a-methyl-1-propan-2-yl-2,3,4,6,7,8-hexahydroazulen-5-one 117133-36-5 C14H22O2
(3aS)-7-hydroxy-3a-methyl-1-propan-2-yl-2,3,4,6,7,8-hexahydroazulen-5-one
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-3-hydroxy-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073444-72-0 C29H37N5O9
4-[(S)-4-carboxy-2-({4-[2-((S)-3-hydroxy-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 2-alpha-methylacetonyl 3-oxo 5-p-methoxyphenyl as.-triazine 113913-01-2 C14H15N3O3
2-alpha-methylacetonyl 3-oxo 5-p-methoxyphenyl as.-triazine
—— 2-(ethyl-methyl-amino)-1-[5-(2-fluoro-2-methyl-propyl)-2-methoxy-phenyl]-1-(4-thiazol-2-ylphenyl)ethanol 1097730-10-3 C25H31FN2O2S
2-(ethyl-methyl-amino)-1-[5-(2-fluoro-2-methyl-propyl)-2-methoxy-phenyl]-1-(4-thiazol-2-ylphenyl)ethanol
—— methyl O-(2,3,4-tri-O-acetyl-α-L-fucopyranosyl)-(1->3)-O-(2-acetamido-4,6-di-O-acetyl-2-deoxy-β-D-glucopyranosyl)-(1->3)-2,4,6-tri-O-acetyl-β-D-galactopyranoside 115944-98-4 C37H53NO23
methyl O-(2,3,4-tri-O-acetyl-α-L-fucopyranosyl)-(1->3)-O-(2-acetamido-4,6-di-O-acetyl-2-deoxy-β-D-glucopyranosyl)-(1->3)-2,4,6-tri-O-acetyl-β-D-galactopyranoside
—— 5-Amino-2-(1-bromo-2-oxo-2-phenyl-ethyl)-7-phenyl-7H-pyrano[2,3-d]thiazole-6-carbonitrile 112434-48-7 C21H14BrN3O2S
5-Amino-2-(1-bromo-2-oxo-2-phenyl-ethyl)-7-phenyl-7H-pyrano[2,3-d]thiazole-6-carbonitrile
—— 2-amino-3-methyl-5-[3-(1-methyl-1H-imidazol-4-yl)phenyl]-5-[4-(pentafluoro-λ6-sulfanyl)phenyl]-3,5-dihydro-4H-imidazol-4-one 1083179-72-9 C20H18F5N5OS
2-amino-3-methyl-5-[3-(1-methyl-1H-imidazol-4-yl)phenyl]-5-[4-(pentafluoro-λ6-sulfanyl)phenyl]-3,5-dihydro-4H-imidazol-4-one