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中文名称 英文名称 CAS号 化学式 结构式图片
—— 9-methyl-10H-phenothiazine-2-carboxylic acid 19693-22-2 C14H11NO2S
9-methyl-10H-phenothiazine-2-carboxylic acid
—— 1-(2-methoxybenzyl)-1H-pyrrolo[2,3-b]pyridine-5-carboxylic acid 1575392-74-3 C16H14N2O3
1-(2-methoxybenzyl)-1H-pyrrolo[2,3-b]pyridine-5-carboxylic acid
—— 5-Methyl-2-(2-oxo-propyl)-cyclopent-2-enone 117902-40-6 C9H12O2
5-Methyl-2-(2-oxo-propyl)-cyclopent-2-enone
—— (R,E)-1-((R)-2-((R)-1-(tert-butyldimethylsilyloxy)pent-4-enyl)cyclohexylidene)-1-[(S)-N-methyl-S-phenylsulfonimidoyl]hex-5-en-2-ol 1380215-64-4 C30H49NO3SSi
(R,E)-1-((R)-2-((R)-1-(tert-butyldimethylsilyloxy)pent-4-enyl)cyclohexylidene)-1-[(S)-N-methyl-S-phenylsulfonimidoyl]hex-5-en-2-ol
—— N-{9-[(2R,3R,4R,5R)-4-(tert-Butyl-dimethyl-silanyloxy)-5-(tert-butyl-dimethyl-silanyloxymethyl)-3-(3-hydroxy-propoxy)-tetrahydro-furan-2-yl]-6-oxo-6,9-dihydro-1H-purin-2-yl}-isobutyramide 192316-94-2 C29H53N5O7Si2
N-{9-[(2R,3R,4R,5R)-4-(tert-Butyl-dimethyl-silanyloxy)-5-(tert-butyl-dimethyl-silanyloxymethyl)-3-(3-hydroxy-propoxy)-tetrahydro-furan-2-yl]-6-oxo-6,9-dihydro-1H-purin-2-yl}-isobutyramide
—— 2,3,4-tri-O-benzyl-6,7,8,9-tetradeoxy-β-D-gluco-nonadi-6(E),8-enopyranose 1470226-44-8 C30H32O5
2,3,4-tri-O-benzyl-6,7,8,9-tetradeoxy-β-D-gluco-nonadi-6(E),8-enopyranose
—— 3-[3-({4-[3-cyano-4-(tetrahydro-2H-pyran-4-yloxy)phenyl]pyrimidin-2-yl}amino)phenyl]-1,1-dimethylurea 1292317-04-4 C25H26N6O3
3-[3-({4-[3-cyano-4-(tetrahydro-2H-pyran-4-yloxy)phenyl]pyrimidin-2-yl}amino)phenyl]-1,1-dimethylurea
—— 1-((1-(cyclopentylidenemethyl)cyclopropyl)ethynyl)-4-nitrobenzene 1233341-05-3 C17H17NO2
1-((1-(cyclopentylidenemethyl)cyclopropyl)ethynyl)-4-nitrobenzene
—— 1-(2-phenylethyl)-3-(6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-yl)urea 1234375-10-0 C19H21N5O
1-(2-phenylethyl)-3-(6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-yl)urea
—— 2-acetamido-3,4,6-tri-O-acetyl-2-deoxy-β-D-galactopyranosyl-(1->4)-6-O-acetyl-2,3-di-benzoyl-α-D-glucopyranosyl trichloroacetimidate 1246851-91-1 C38H41Cl3N2O17
2-acetamido-3,4,6-tri-O-acetyl-2-deoxy-β-D-galactopyranosyl-(1->4)-6-O-acetyl-2,3-di-benzoyl-α-D-glucopyranosyl trichloroacetimidate
—— (2S,3S)-2-(naphthalen-1-yl)-3,5,5-trimethylmorpholin-2-ol 1231951-81-7 C17H21NO2
(2S,3S)-2-(naphthalen-1-yl)-3,5,5-trimethylmorpholin-2-ol
—— tert-butyl (2S,4R)-4-fluoro-2-{[(6R)-6-methyl-4-(trlfluoroacetyl)-4,7-diazaspiro[2.5]oct-7-yl]carbonyl}pyrrolidine-1-carboxylate 1235576-52-9 C19H27F4N3O4
tert-butyl (2S,4R)-4-fluoro-2-{[(6R)-6-methyl-4-(trlfluoroacetyl)-4,7-diazaspiro[2.5]oct-7-yl]carbonyl}pyrrolidine-1-carboxylate
—— 4-{[(5Z)-5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl}benzoic acid 1373425-48-9 C27H17ClF3N3O4S
4-{[(5Z)-5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl}benzoic acid
—— (7S)-N-(6-fluoro-2-methyl-3-(5-((5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)amino)-6-oxo-1,6-dihydropyridazin-3-yl)phenyl)-7-hydroxy-3-thiatricyclo[6.2.1.0a(2,6)]undeca-2(6),4-diene-4-carboxamide 1227209-98-4 C29H30FN7O3S
(7S)-N-(6-fluoro-2-methyl-3-(5-((5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)amino)-6-oxo-1,6-dihydropyridazin-3-yl)phenyl)-7-hydroxy-3-thiatricyclo[6.2.1.0a(2,6)]undeca-2(6),4-diene-4-carboxamide
—— 3-(4-((5-chloro-3-hydroxy-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)-3-fluorophenyl)-2-methylpropanoic acid 1234842-48-8 C21H22ClFO5
3-(4-((5-chloro-3-hydroxy-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)-3-fluorophenyl)-2-methylpropanoic acid
—— 4-oxo-4-(1-(o-tolyl)-3,4-dihydro-1H-isoquinolin-2-yl)-N-[[2-(trifluoromethyl)-phenyl]methyl]butyric acid amide 1229515-29-0 C28H27F3N2O2
4-oxo-4-(1-(o-tolyl)-3,4-dihydro-1H-isoquinolin-2-yl)-N-[[2-(trifluoromethyl)-phenyl]methyl]butyric acid amide
—— N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(2,6-dimethyl-4-pyridinyl)-4-thiazolyl]methyl]-2-methoxy-acetamide 1309442-17-8 C20H28N4O3S
N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(2,6-dimethyl-4-pyridinyl)-4-thiazolyl]methyl]-2-methoxy-acetamide
—— 3-chloro-2-fluoro-N-(1-hydroxy-3,4-dihydro-1H-benzo[c][1,2]oxaborinin-7-yl)-benzamide 1335094-87-5 C15H12BClFNO3
3-chloro-2-fluoro-N-(1-hydroxy-3,4-dihydro-1H-benzo[c][1,2]oxaborinin-7-yl)-benzamide
—— 2-ethyl-N-((1-methyl-1H-indol-6-yl)methyl)imidazo[1,2-a]pyridine-3-carboxamide 1334716-94-7 C20H20N4O
2-ethyl-N-((1-methyl-1H-indol-6-yl)methyl)imidazo[1,2-a]pyridine-3-carboxamide
—— 5-{2-({4-[2-(2-aminoethoxy)ethoxy]-3-methoxyphenyl}amino)pyrimidin-4-yl}-2-({1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}oxy)benzonitrile 1292311-51-3 C30H36N6O6
5-{2-({4-[2-(2-aminoethoxy)ethoxy]-3-methoxyphenyl}amino)pyrimidin-4-yl}-2-({1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}oxy)benzonitrile
—— N-(2-fluoro-5-(5-((5-(((2-hydroxyethyl)amino)methyl)pyridin-2-yl)amino)-6-oxo-1,6-dihydropyridazin-3-yl)phenyl)-1-benzothiophene-2-carboxamide 1227207-66-0 C27H23FN6O3S
N-(2-fluoro-5-(5-((5-(((2-hydroxyethyl)amino)methyl)pyridin-2-yl)amino)-6-oxo-1,6-dihydropyridazin-3-yl)phenyl)-1-benzothiophene-2-carboxamide
—— 3-(4-(ethylamino)-2-(furan-2-yl)quinazolin-6-yl)prop-2-yn-1-ol 1235475-59-8 C17H15N3O2
3-(4-(ethylamino)-2-(furan-2-yl)quinazolin-6-yl)prop-2-yn-1-ol
—— N-(4-chlorophenyl)-6-fluoro-1-(6-(hydroxyamino)-6-oxohexyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide 1233375-84-2 C22H21ClFN3O4
N-(4-chlorophenyl)-6-fluoro-1-(6-(hydroxyamino)-6-oxohexyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide
—— N-((S)-1-((S)-3-hydroxypyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)-3-(2,4,5-trifluorophenyl)-6,7-dihydropyrano[4,3-c]pyrazole-1(4H)-carboxamide 1231908-57-8 C23H27F3N4O4
N-((S)-1-((S)-3-hydroxypyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)-3-(2,4,5-trifluorophenyl)-6,7-dihydropyrano[4,3-c]pyrazole-1(4H)-carboxamide
—— (S)-5,9-dimethyl-deca-1,2,8-triene 1228108-15-3 C12H20
(S)-5,9-dimethyl-deca-1,2,8-triene
—— 4-[[4-[Cyano-(4-methylphenyl)methyl]-5-methylpyrimidin-2-yl]amino]benzonitrile 1232185-42-0 C21H17N5
4-[[4-[Cyano-(4-methylphenyl)methyl]-5-methylpyrimidin-2-yl]amino]benzonitrile
—— 1-methyl-6-(4-(2-(1-((3-methylisoxazol-5-yl)methyl)piperidin-4-yl)ethoxy)-3-(trifluoromethyl)phenyl)-1H-imidazo[4,5-c]pyridine-4-carbonitrile 1235840-76-2 C27H27F3N6O2
1-methyl-6-(4-(2-(1-((3-methylisoxazol-5-yl)methyl)piperidin-4-yl)ethoxy)-3-(trifluoromethyl)phenyl)-1H-imidazo[4,5-c]pyridine-4-carbonitrile
—— N-[2-(4-chlorophenyl)ethyl]-6-(phenoxymethyl)pyridine-3-carboxamide 1350964-19-0 C21H19ClN2O2
N-[2-(4-chlorophenyl)ethyl]-6-(phenoxymethyl)pyridine-3-carboxamide
—— N-(5-methyl-1H-pyrazol-3-yl)-2-(4-((1-phenylcyclobutyl)carbonyl)-1-piperazinyl)-pyrrolo[2,1-f][1,2,4]triazine-4-amine 1221267-83-9 C25H28N8O
N-(5-methyl-1H-pyrazol-3-yl)-2-(4-((1-phenylcyclobutyl)carbonyl)-1-piperazinyl)-pyrrolo[2,1-f][1,2,4]triazine-4-amine
—— (5Z)-5-({1-[2,4-bis(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-3-hydroxy-1,3-thiazolidine-2,4-dione 1351569-80-6 C20H11F6N3O3S
(5Z)-5-({1-[2,4-bis(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-3-hydroxy-1,3-thiazolidine-2,4-dione
—— [3-methoxy-4-(4-methylamino-5-trifluoromethylpyrimidin-2-ylamino)phenyl]-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)methanone 1351761-60-8 C20H22F3N5O3
[3-methoxy-4-(4-methylamino-5-trifluoromethylpyrimidin-2-ylamino)phenyl]-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)methanone
—— 7-[(3,5-Dichlorophenyl)-[(3,5-difluoropyridin-2-yl)amino]methyl]quinolin-8-ol 1314513-80-8 C21H13Cl2F2N3O
7-[(3,5-Dichlorophenyl)-[(3,5-difluoropyridin-2-yl)amino]methyl]quinolin-8-ol
—— 2-(4-(3-methyl-2-phenylbutanoyl)-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)pyrrolo[2,1-f][1,2,4]triazine-4-amine 1221268-76-3 C25H30N8O
2-(4-(3-methyl-2-phenylbutanoyl)-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)pyrrolo[2,1-f][1,2,4]triazine-4-amine
—— 2-{(E)-2-[3-(difluoromethoxy)-2-(2,2-dimethylpropoxy)phenyl]vinyl}-N-[4-(trifluoro-methyl)-1,3-thiazol-2-yl]imidazo[1,2-a]pyridine-3-carboxamide 1228829-09-1 C26H23F5N4O3S
2-{(E)-2-[3-(difluoromethoxy)-2-(2,2-dimethylpropoxy)phenyl]vinyl}-N-[4-(trifluoro-methyl)-1,3-thiazol-2-yl]imidazo[1,2-a]pyridine-3-carboxamide
—— 5-(3-fluoro-phenyl)-1H-pyrazole-3-carboxylic acid {2-[4-(5-fluoro-2-trifluoromethyl-benzoyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1232027-98-3 C24H20F5N5O3
5-(3-fluoro-phenyl)-1H-pyrazole-3-carboxylic acid {2-[4-(5-fluoro-2-trifluoromethyl-benzoyl)-piperazin-1-yl]-2-oxo-ethyl}-amide
—— 2-ethoxy-N-(3-(4,5-diethyl-1,6-dihydro-6-oxopyrimidin-2-yl)-4-n-propoxyphenyl)benzamide 1229018-00-1 C26H31N3O4
2-ethoxy-N-(3-(4,5-diethyl-1,6-dihydro-6-oxopyrimidin-2-yl)-4-n-propoxyphenyl)benzamide
—— (5Z)-3-[2-(tert-butylamino)ethyl]-5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-1,3-thiazolidine-2,4-dione 1351565-80-4 C25H24ClF3N4O2S
(5Z)-3-[2-(tert-butylamino)ethyl]-5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-1,3-thiazolidine-2,4-dione
—— N-[4-cyclopentyl-5-hydroxy-2-(3-hydroxyprop-1-ynyl)phenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide 1233529-54-8 C24H23F3N2O5
N-[4-cyclopentyl-5-hydroxy-2-(3-hydroxyprop-1-ynyl)phenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
—— methyl (3R,8aR)-5-oxohexahydro-5H-[1,3]oxazolo[3,2-a]pyridin-3-carboxylate 1196714-44-9 C9H13NO4
methyl (3R,8aR)-5-oxohexahydro-5H-[1,3]oxazolo[3,2-a]pyridin-3-carboxylate
—— 4-(4-{[4'-chloro-4-(2-pyrrolidin-1-ylethoxy)-1,1'-biphenyl-2-yl]methyl}piperazin-1-yl)-N-({3-nitro-4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]phenyl}sulfonyl)-2-phenoxybenzamide 1228783-60-5 C48H53ClN6O8S
4-(4-{[4'-chloro-4-(2-pyrrolidin-1-ylethoxy)-1,1'-biphenyl-2-yl]methyl}piperazin-1-yl)-N-({3-nitro-4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]phenyl}sulfonyl)-2-phenoxybenzamide
—— N,N-dimethyl-4-(1H-pyrazol-4-yl)-N-(pyridin-2-yl)thiazole-2,5-diamine 1235312-63-6 C13H14N6S
N,N-dimethyl-4-(1H-pyrazol-4-yl)-N-(pyridin-2-yl)thiazole-2,5-diamine
—— 1-(6-(hydroxyamino)-6-oxohexyl)-6-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 1233375-60-4 C17H20N2O6
1-(6-(hydroxyamino)-6-oxohexyl)-6-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
—— 5-({3-[3-(4-isobutylphenyl)-1,2,4-oxadiazol-5-yl]-5-methyl-1H-pyrazol-1-yl}methyl)-N-methylpyridin-2-amine 1227298-06-7 C23H26N6O
5-({3-[3-(4-isobutylphenyl)-1,2,4-oxadiazol-5-yl]-5-methyl-1H-pyrazol-1-yl}methyl)-N-methylpyridin-2-amine
—— cyclopropyl-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid (2-cyano-1,2,2-trimethyl-ethyl)-amide 1350707-43-5 C16H19N5O
cyclopropyl-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid (2-cyano-1,2,2-trimethyl-ethyl)-amide
—— (2S)-4-amino-N-[(1R,2S,3R,4R,5S)-5-amino-3-[(2S,3R,4S,5R)-4-[(2R,3R,4R,5S,6S)-3-amino-6-(aminomethyl)-4,5-dihydroxyoxan-2-yl]oxy-3-hydroxy-5-(hydroxymethyl)oxolan-2-yl]oxy-4-[[(2R,3R,6S)-3-amino-6-(methylaminomethyl)-3,6-dihydro-2H-pyran-2-yl]oxy]-2-hydroxycyclohexyl]-2-hydroxybutanamide 1221493-71-5 C28H53N7O13
(2S)-4-amino-N-[(1R,2S,3R,4R,5S)-5-amino-3-[(2S,3R,4S,5R)-4-[(2R,3R,4R,5S,6S)-3-amino-6-(aminomethyl)-4,5-dihydroxyoxan-2-yl]oxy-3-hydroxy-5-(hydroxymethyl)oxolan-2-yl]oxy-4-[[(2R,3R,6S)-3-amino-6-(methylaminomethyl)-3,6-dihydro-2H-pyran-2-yl]oxy]-2-hydroxycyclohexyl]-2-hydroxybutanamide
—— 4-(4-(2-(5-((5-tert-butyloxazol-2-yl)methylthio)thiazol-2-ylamino)-2-oxoethyl)phenoxy)-N-hydroxy-N-methylbutanamide 1233699-83-6 C24H30N4O5S2
4-(4-(2-(5-((5-tert-butyloxazol-2-yl)methylthio)thiazol-2-ylamino)-2-oxoethyl)phenoxy)-N-hydroxy-N-methylbutanamide
—— 1-methyl-N-[(1R)-1-[5-[4-(trifluoromethyl)anilino]pyrazin-2-yl]ethyl]imidazo[4,5-c]pyridine-6-carboxamide 1234011-08-5 C21H18F3N7O
1-methyl-N-[(1R)-1-[5-[4-(trifluoromethyl)anilino]pyrazin-2-yl]ethyl]imidazo[4,5-c]pyridine-6-carboxamide
—— 2-phenyl-5-trifluoromethyl-oxazole-4-carboxylic acid [4-(3-cyclopropyl-[1,2,4]oxadiazol-5-yl)-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-5'-yl]-amide 1229419-09-3 C26H23F3N6O3
2-phenyl-5-trifluoromethyl-oxazole-4-carboxylic acid [4-(3-cyclopropyl-[1,2,4]oxadiazol-5-yl)-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-5'-yl]-amide
—— 3,4,5,6-tetrahydro-(4S,5S)-4,5-dihydroxy-2-[(2-phenyl)benzyl]-7-[(2-phenethyl)benzyl]-1,2,7-thiadiazepine 1,1-dioxide 1233878-58-4 C32H34N2O4S
3,4,5,6-tetrahydro-(4S,5S)-4,5-dihydroxy-2-[(2-phenyl)benzyl]-7-[(2-phenethyl)benzyl]-1,2,7-thiadiazepine 1,1-dioxide
—— (S)-(1-(3-(4-(pyridin-2-ylamino)phenoxy)pyrazin-2-yl)pyrrolidin-2-yl)methanol 1231921-41-7 C20H21N5O2
(S)-(1-(3-(4-(pyridin-2-ylamino)phenoxy)pyrazin-2-yl)pyrrolidin-2-yl)methanol