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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S,4S,7S,8R,9S,13R)-7-(furan-3-ylmethyl)-8-methyl-6,15-dioxatetracyclo[7.7.0.01,13.04,8]hexadec-11-ene-5,14-dione 1079220-32-8 C20H22O5
(1S,4S,7S,8R,9S,13R)-7-(furan-3-ylmethyl)-8-methyl-6,15-dioxatetracyclo[7.7.0.01,13.04,8]hexadec-11-ene-5,14-dione
—— [4-(6-methanesulfonyl-1H-indol-4-yl)-6-morpholin-4-yl-pyrimidin-2-yl]-(1,2,3,4-tetrahydro-isoquinolin-6-yl)-amine 1072084-60-6 C26H28N6O3S
[4-(6-methanesulfonyl-1H-indol-4-yl)-6-morpholin-4-yl-pyrimidin-2-yl]-(1,2,3,4-tetrahydro-isoquinolin-6-yl)-amine
—— (4-Bromo-3-methoxy-1,2-thiazol-5-yl)methanol 1955499-62-3 C5H6BrNO2S
(4-Bromo-3-methoxy-1,2-thiazol-5-yl)methanol
—— 2-chloro-6-[2-(4-methoxyphenyl)ethylamino]-9-cyclopentylpurine 1098626-03-9 C19H22ClN5O
2-chloro-6-[2-(4-methoxyphenyl)ethylamino]-9-cyclopentylpurine
—— 5-(4-Nitro-phenyl)-1,5-dihydro-pyrazolo[4,5-c]pyrazol-3-ol 125161-18-4 C10H7N5O3
5-(4-Nitro-phenyl)-1,5-dihydro-pyrazolo[4,5-c]pyrazol-3-ol
—— 4-Benzenesulfonyl-5-(4-chloro-phenyl)-3-p-tolyl-4,5-dihydro-isoxazole 122773-25-5 C22H18ClNO3S
4-Benzenesulfonyl-5-(4-chloro-phenyl)-3-p-tolyl-4,5-dihydro-isoxazole
—— 7-(4-tert-Butylphenyl)-9-methyl-3,8-dioxa-7-azabicyclo<4.2.1>nonan 127355-51-5 C17H25NO2
7-(4-tert-Butylphenyl)-9-methyl-3,8-dioxa-7-azabicyclo<4.2.1>nonan
—— [3-(3-chloro-phenyl)-3-(5-methyl-tetrazol-2-yl)-propyl]-dimethyl-amine 1198349-59-5 C13H18ClN5
[3-(3-chloro-phenyl)-3-(5-methyl-tetrazol-2-yl)-propyl]-dimethyl-amine
—— N-(2,6-diethylphenyl)-1-methyl-8-({1-[(2-piperidin-1-ylethyl)sulfonyl]piperidin-4-yl}amino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide 1202056-26-5 C33H46N8O3S
N-(2,6-diethylphenyl)-1-methyl-8-({1-[(2-piperidin-1-ylethyl)sulfonyl]piperidin-4-yl}amino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
—— 3-[[3-(5-Bromopyrimidin-2-yl)phenyl]methyl]-6-methyl-[1,2,4]triazolo[4,3-b]pyridazine 1201929-72-7 C17H13BrN6
3-[[3-(5-Bromopyrimidin-2-yl)phenyl]methyl]-6-methyl-[1,2,4]triazolo[4,3-b]pyridazine
—— methyl (2R)-2-(dimethylcarbamoyl)piperidine-1-carboxylate 1201156-73-1 C10H18N2O3
methyl (2R)-2-(dimethylcarbamoyl)piperidine-1-carboxylate
—— ethyl 4-(4-formyl-1-phenyl-1H-pyrazol-3-yl)-3,5-dimethyl-1H-pyrrole-2-carboxylate 1190975-82-6 C19H19N3O3
ethyl 4-(4-formyl-1-phenyl-1H-pyrazol-3-yl)-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-((R)-5-((E)-3,7-difluoro-6H-dibenzo[b,e]oxepin-11-ylidenemethyl)-1-(1-methyl-2-morpholin-4-yl-ethyl)-1,3-dihydro-benzoimidazol-2-ylidene)-cyanamide 1162263-71-9 C30H27F2N5O2
(E)-N-((R)-5-((E)-3,7-difluoro-6H-dibenzo[b,e]oxepin-11-ylidenemethyl)-1-(1-methyl-2-morpholin-4-yl-ethyl)-1,3-dihydro-benzoimidazol-2-ylidene)-cyanamide
—— Ethyl 2-cyclohexylimino-4-methyl-3-[(2,3,4-trihydroxyphenyl)methylideneamino]-1,3-thiazole-5-carboxylate 1459803-60-1 C20H25N3O5S
Ethyl 2-cyclohexylimino-4-methyl-3-[(2,3,4-trihydroxyphenyl)methylideneamino]-1,3-thiazole-5-carboxylate
—— ethyl 3-(4-chlorophenyl)-2-diazo-3-hydroxypropanoate 1118755-04-6 C11H11ClN2O3
ethyl 3-(4-chlorophenyl)-2-diazo-3-hydroxypropanoate
—— 4-[4-(2,6-difluorophenyl)pyrimidin-2-yl]-N-pyridazin-3-ylpiperazine-1-carboxamide 1143579-03-6 C19H17F2N7O
4-[4-(2,6-difluorophenyl)pyrimidin-2-yl]-N-pyridazin-3-ylpiperazine-1-carboxamide
—— (2-{1-[4-(1-methyl-piperidin-4-yl)-butyl]-1H-indol-4-yl}-1H-benzoimidazol-5-yl)-phenyl-methanone 1161424-93-6 C32H34N4O
(2-{1-[4-(1-methyl-piperidin-4-yl)-butyl]-1H-indol-4-yl}-1H-benzoimidazol-5-yl)-phenyl-methanone
—— (S)-3,5-dimethylbenzoic acid N-(1-tert-butylbutyl)-N'-(2-fluorobenzoyl)hydrazide 1093131-06-6 C24H31FN2O2
(S)-3,5-dimethylbenzoic acid N-(1-tert-butylbutyl)-N'-(2-fluorobenzoyl)hydrazide
—— 8-methoxy-3-methyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid methyl ester 1075715-14-8 C19H17NO4
8-methoxy-3-methyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid methyl ester
—— 5-fluoro-2-[[(E)-2-(4-methylsulfanylphenyl)ethenyl]sulfonylamino]-benzenesulfonamide 1161942-76-2 C15H15FN2O4S3
5-fluoro-2-[[(E)-2-(4-methylsulfanylphenyl)ethenyl]sulfonylamino]-benzenesulfonamide
—— (4S,5S)-4-hydroxy-5-[(3S)-4-methyl-1-(2-methyl-1,3-dioxolan-2-yl)pentan-3-yl]oxolan-2-one 1263400-96-9 C14H24O5
(4S,5S)-4-hydroxy-5-[(3S)-4-methyl-1-(2-methyl-1,3-dioxolan-2-yl)pentan-3-yl]oxolan-2-one
—— 3-formyl-4-(pyridin-3-yl)phenyl trifluoromethanesulfonate 1296208-53-1 C13H8F3NO4S
3-formyl-4-(pyridin-3-yl)phenyl trifluoromethanesulfonate
—— N-(3-(1-(6-aminopyrimidin-4-yl)-1H-indol-6-yl)phenyl)-5-(4-chlorophenyl)isoxazol-3-carboxamide 1298084-07-7 C28H19ClN6O2
N-(3-(1-(6-aminopyrimidin-4-yl)-1H-indol-6-yl)phenyl)-5-(4-chlorophenyl)isoxazol-3-carboxamide
—— methyl [(1S,2S)-2-(4-{[(2R)-2,4-dibenzylpiperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)cyclohexyl]carbamate 1083852-95-2 C36H41N5O3
methyl [(1S,2S)-2-(4-{[(2R)-2,4-dibenzylpiperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)cyclohexyl]carbamate
—— <4-Chlor-benzaldehyd>-2,4,6-trinitrophenylhydrazon 19258-59-4 C13H8ClN5O6
<4-Chlor-benzaldehyd>-2,4,6-trinitrophenylhydrazon
—— 1,2-bis-(4-methoxy-but-3-en-1-ynyl)-cyclohexane-1,2-diol 108774-48-7 C16H20O4
1,2-bis-(4-methoxy-but-3-en-1-ynyl)-cyclohexane-1,2-diol
—— 8-bromo-7-hydroxychromone 1313728-35-6 C9H5BrO3
8-bromo-7-hydroxychromone
—— methyl 2,2-dibenzyl-3-[4-(4-chlorophenyl)-4-fluoropiperidin-1-yl]propionate 1345610-73-2 C29H31ClFNO2
methyl 2,2-dibenzyl-3-[4-(4-chlorophenyl)-4-fluoropiperidin-1-yl]propionate
—— tert-butyl 4-[4-(2-bromo-5-carboxy-phenoxy)-pyrimidin-2-yl]-piperazine-1-carboxylate 1215031-01-8 C20H23BrN4O5
tert-butyl 4-[4-(2-bromo-5-carboxy-phenoxy)-pyrimidin-2-yl]-piperazine-1-carboxylate
—— tert-butyl (7-methyl-7-azabicyclo[2.2.1]heptan-1-yl)(phenyl)methylcarbamate 1236547-82-2 C19H28N2O2
tert-butyl (7-methyl-7-azabicyclo[2.2.1]heptan-1-yl)(phenyl)methylcarbamate
—— US10202379, Reference Example 390 1370241-22-7 C24H22ClN3O4
US10202379, Reference Example 390
—— 6-bromo-N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-[(1R)-1-methyl-2-(methyloxy)ethyl]-1H-indole-4-carboxamide 1346574-42-2 C22H26BrN3O3
6-bromo-N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-[(1R)-1-methyl-2-(methyloxy)ethyl]-1H-indole-4-carboxamide
—— tert-butyl 4-(2-(3-(4-methylphenylsulfonamido)cyclobutoxy)pyridin-3-yl)piperidine-1-carboxylate 1349185-44-9 C26H35N3O5S
tert-butyl 4-(2-(3-(4-methylphenylsulfonamido)cyclobutoxy)pyridin-3-yl)piperidine-1-carboxylate
—— 1-[(3,4-difluorophenyl)methyl]-6-oxo-N-[3-[3-[(3-pyrrolidin-1-ylcyclobutyl)amino]quinoxalin-6-yl]prop-2-ynyl]pyrimidine-5-carboxamide 1345438-20-1 C31H29F2N7O2
1-[(3,4-difluorophenyl)methyl]-6-oxo-N-[3-[3-[(3-pyrrolidin-1-ylcyclobutyl)amino]quinoxalin-6-yl]prop-2-ynyl]pyrimidine-5-carboxamide
—— 4-(benzylamino)-6-(4-(cyclopropyl(methyl)carbamoyl)-3-methylphenylamino)nicotinamide 1374214-32-0 C25H27N5O2
4-(benzylamino)-6-(4-(cyclopropyl(methyl)carbamoyl)-3-methylphenylamino)nicotinamide
—— 2-chloro-N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)phenyl]benzamide 1092393-03-7 C24H19ClN4O3
2-chloro-N-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)phenyl]benzamide
—— 4'-(2-(4-cyanophenylamino)-5-methyl-5H-pyrrolo[3,2-d]pyrimidin-4-yloxy)-N-cyclopropyl-3',5'-dimethylbiphenyl-4-carboxamide 1164099-97-1 C32H28N6O2
4'-(2-(4-cyanophenylamino)-5-methyl-5H-pyrrolo[3,2-d]pyrimidin-4-yloxy)-N-cyclopropyl-3',5'-dimethylbiphenyl-4-carboxamide
—— 2-[5-(2,6-Dimethoxyphenyl)-1-(2-methyl-4-nitrophenyl)-3-pyrazolylcarbonylamino]-2-adamantanecarboxylic acid 184165-23-9 C30H32N4O7
2-[5-(2,6-Dimethoxyphenyl)-1-(2-methyl-4-nitrophenyl)-3-pyrazolylcarbonylamino]-2-adamantanecarboxylic acid
—— (R)-2-((S)-2-amino-3-methylbutyryl)-7-(4-chloro-2-fluorophenyl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione 1262129-94-1 C23H24ClFN4O3
(R)-2-((S)-2-amino-3-methylbutyryl)-7-(4-chloro-2-fluorophenyl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione
—— 4-[(2R,3R)-2-amino-5-azaspiro[2.4]heptan-5-yl]-6-fluoro-N-methyl-2-(1,5-naphthyridin-3-yloxy)-9H-pyrimido[4,5-b]indol-8-amine 1400803-50-0 C25H23FN8O
4-[(2R,3R)-2-amino-5-azaspiro[2.4]heptan-5-yl]-6-fluoro-N-methyl-2-(1,5-naphthyridin-3-yloxy)-9H-pyrimido[4,5-b]indol-8-amine
—— 4-Pyrimidinecarbonitrile, 6-[(3-methoxypropyl)amino]- 1865214-56-7 C9H12N4O
4-Pyrimidinecarbonitrile, 6-[(3-methoxypropyl)amino]-
—— Decanal, 2-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-, (S)- 139427-51-3 C16H34O2Si
Decanal, 2-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-, (S)-
—— N-Methyl-N-(3-methylbutyl)-2-pyrrolidineacetamide 1247356-89-3 C12H24N2O
N-Methyl-N-(3-methylbutyl)-2-pyrrolidineacetamide
—— 5-chloro-4-(3-methylpyridin-2-yl)-2-[4-(methylsulfonyl)piperazin-1-yl]pyrimidine 1373614-44-8 C15H18ClN5O2S
5-chloro-4-(3-methylpyridin-2-yl)-2-[4-(methylsulfonyl)piperazin-1-yl]pyrimidine
—— N-(2,5-dimorpholinopyridin-3-yl)-5,7-difluoro-3-methyl-2-(pyridin-3-yl)quinolin-4-amine 1259441-94-5 C28H28F2N6O2
N-(2,5-dimorpholinopyridin-3-yl)-5,7-difluoro-3-methyl-2-(pyridin-3-yl)quinolin-4-amine
—— (2S)-2-amino-4-(4-(5-(methylsulfinyl)pyrimidin-2-ylamino)phenyl)butan-1-ol 1374038-52-4 C15H20N4O2S
(2S)-2-amino-4-(4-(5-(methylsulfinyl)pyrimidin-2-ylamino)phenyl)butan-1-ol
—— 7-(4-chloro-3,5-difluorophenyl)-2-(3,3-dimethylbutyryl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione 1262130-34-6 C24H24ClF2N3O3
7-(4-chloro-3,5-difluorophenyl)-2-(3,3-dimethylbutyryl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione
—— 2-(3,5-difluorophenyl)-N-[2-(4,4-difluoro-1-piperidyl)-6-(7,8-dihydro-5H-1,6-naphthyridin-6-yl)-4-methyl-3-pyridyl]-acetamide 1253378-39-0 C27H27F4N5O
2-(3,5-difluorophenyl)-N-[2-(4,4-difluoro-1-piperidyl)-6-(7,8-dihydro-5H-1,6-naphthyridin-6-yl)-4-methyl-3-pyridyl]-acetamide
—— tert-butyl 4-(5-(5-bromo-3-(2-methylpyridin-3-yloxy)pyridin-2-ylamino)-1,2,4-thiadiazol-3-yl)piperidine-1-carboxylate 1065609-02-0 C23H27BrN6O3S
tert-butyl 4-(5-(5-bromo-3-(2-methylpyridin-3-yloxy)pyridin-2-ylamino)-1,2,4-thiadiazol-3-yl)piperidine-1-carboxylate
—— N-[1-[2-(aminocarbonyl)-1,3-dioxolan-2-yl]-2-(4-fluorophenyl)ethyl]-2-[3-(2,4-dichlorophenyl)-1H-pyrazol-1-yl]nicotinamide 1166926-72-2 C27H22Cl2FN5O4
N-[1-[2-(aminocarbonyl)-1,3-dioxolan-2-yl]-2-(4-fluorophenyl)ethyl]-2-[3-(2,4-dichlorophenyl)-1H-pyrazol-1-yl]nicotinamide