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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2,4)-4-{[2-(3-chloro-6-methoxyquinolin-4-yl)ethyl]amino}-1-(3-phenylcyclobutyl)piperidine-2-carboxylic acid 1080635-81-9 C28H32ClN3O3
(2,4)-4-{[2-(3-chloro-6-methoxyquinolin-4-yl)ethyl]amino}-1-(3-phenylcyclobutyl)piperidine-2-carboxylic acid
—— N-(2,3-Dichlorophenyl)-4-[4-(1,1-dimethylethyl)phenyl]-4-methyl-2,5-dioxo-1-imidazolidineacetamide 1134600-67-1 C22H23Cl2N3O3
N-(2,3-Dichlorophenyl)-4-[4-(1,1-dimethylethyl)phenyl]-4-methyl-2,5-dioxo-1-imidazolidineacetamide
—— tert-butyl {1-[2-(7-cyano-4-methyl-2-oxoquinolin-1(2H)-yl)ethyl]piperidin-4-yl}carbamate 1033312-32-1 C23H30N4O3
tert-butyl {1-[2-(7-cyano-4-methyl-2-oxoquinolin-1(2H)-yl)ethyl]piperidin-4-yl}carbamate
—— 2-[(1S,3S)-1-methyl-1-(3-phenylsulfanylpropyl)-pyrrolidin-3-yl]-2,2-diphenylacetamide trifluoroacetate 1050644-28-4 C2F3O2*C28H33N2OS
2-[(1S,3S)-1-methyl-1-(3-phenylsulfanylpropyl)-pyrrolidin-3-yl]-2,2-diphenylacetamide trifluoroacetate
—— —— 1192564-86-5 C2HF3O2*C26H26ClF5N6O
—— —— 1195188-39-6 C22H24ClN5O
—— (1aS,3aR,6bR)-5-Methylsulphonyloxy-2-(1-methyl-1H-tetrazol-5-ylsulphanylacetyl)-1-oxo-1a,2,3,3a,4,6b-hexahydro-1H-2,6a-diazacyclobut[cd]indene-6-carboxylic acid sodium salt 170580-65-1 C14H15N6O7S2*Na
(1aS,3aR,6bR)-5-Methylsulphonyloxy-2-(1-methyl-1H-tetrazol-5-ylsulphanylacetyl)-1-oxo-1a,2,3,3a,4,6b-hexahydro-1H-2,6a-diazacyclobut[cd]indene-6-carboxylic acid sodium salt
—— 3-Butyl-5,6-dihydro-N-hydroxy-5-[2'-(1H-tetrazol-5-yl)[1.1'-biphenyl]-4-yl]triazolo[4,3-a]pyridin-8(7H)-imine 170837-13-5 C23H24N8O
3-Butyl-5,6-dihydro-N-hydroxy-5-[2'-(1H-tetrazol-5-yl)[1.1'-biphenyl]-4-yl]triazolo[4,3-a]pyridin-8(7H)-imine
—— —— 1072019-63-6 C9H6F6N2O2
—— —— 1072024-52-2 C12H11F7N2O3
—— —— 1094837-86-1 C29H30ClN3O4
—— N-(4-carbamimidoylbenzyl)-2-(1-isobutyl-2-methyl-6-oxo-4-phenyl-1,6-dihydro-pyrimidine-5-yl)-acetamide acetic acid salt 1037508-29-4 C2H4O2*C25H29N5O2
N-(4-carbamimidoylbenzyl)-2-(1-isobutyl-2-methyl-6-oxo-4-phenyl-1,6-dihydro-pyrimidine-5-yl)-acetamide acetic acid salt
—— 1-(2,2-dimethylpropyl)-6-[6-(4-fluorophenyl)-imidazo[2,1-b]thiazol-5-yl]-1H-benzoimidazol-2-ylamine 1029524-64-8 C23H22FN5S
1-(2,2-dimethylpropyl)-6-[6-(4-fluorophenyl)-imidazo[2,1-b]thiazol-5-yl]-1H-benzoimidazol-2-ylamine
—— —— 1033703-67-1 C24H26F2N4O
—— 4-[2-oxo-4-(2-pyridin-4-yl-ethylcarbamoyl)-pyrrolidin-1-yl]-piperidine-1-carboxylic acid 3,5-dichloro-benzyl ester 1248727-69-6 C25H28Cl2N4O4
4-[2-oxo-4-(2-pyridin-4-yl-ethylcarbamoyl)-pyrrolidin-1-yl]-piperidine-1-carboxylic acid 3,5-dichloro-benzyl ester
—— —— 1032464-40-6 C12H12FN3S
—— —— 1032047-99-6 C17H25N7O
—— —— 1059186-29-6 C15H12F4N2O4
—— —— 1059186-30-9 C16H18N2O4
—— —— 1072022-33-3 C12H12ClF5N2O4
—— —— 1072022-17-3 C12H10ClF5N2O2
—— —— 1033841-91-6 C24H28FN5O
—— —— 1070779-15-5 C17H23N3O4S
—— N-[(1S)-1-(4-{[6-(4-methylpyridin-3-yl)quinazolin-2-yl]amino}phenyl)ethyl]acetamide 1032574-23-4 C24H23N5O
N-[(1S)-1-(4-{[6-(4-methylpyridin-3-yl)quinazolin-2-yl]amino}phenyl)ethyl]acetamide
—— 3-(1-{6-[4-(4-amino-5-fluoro-pyrimidin-2-yloxy)-piperidin-1-yl]-pyrimidin-4-yl}-piperidin-4-yl)-phenol 1033834-70-6 C24H28FN7O2
3-(1-{6-[4-(4-amino-5-fluoro-pyrimidin-2-yloxy)-piperidin-1-yl]-pyrimidin-4-yl}-piperidin-4-yl)-phenol
—— 5-fluoro-2-{1-[6-(2-fluoro-6-methoxy-phenoxy)-pyrimidin-4-yl]-piperidin-4-yloxy}-pyrimidin-4-ylamine 1033834-23-9 C20H20F2N6O3
5-fluoro-2-{1-[6-(2-fluoro-6-methoxy-phenoxy)-pyrimidin-4-yl]-piperidin-4-yloxy}-pyrimidin-4-ylamine
—— 5-fluoro-2-{1-[6-(3-phenoxy-phenoxy)-pyrimidin-4-yl]-piperidin-4-yloxy}-pyrimidin-4-ylamine 1033833-93-0 C25H23FN6O3
5-fluoro-2-{1-[6-(3-phenoxy-phenoxy)-pyrimidin-4-yl]-piperidin-4-yloxy}-pyrimidin-4-ylamine
—— —— 1297597-53-5 C14H8Br3ClN2S
—— —— 1258285-20-9 C24H32N2O6S
—— 1-methyl-1H-imidazole-4-carboxylic acid (5-tert-butylamino-pentyl)-(3-phenoxy-benzyl)-amide 1031297-79-6 C27H36N4O2
1-methyl-1H-imidazole-4-carboxylic acid (5-tert-butylamino-pentyl)-(3-phenoxy-benzyl)-amide
—— 4-methyl-thiazole-5-carboxylic acid (4-amino-cyclohexyl)-[2-(3-chloro-phenyl)-ethyl]-amide 1031291-97-0 C19H24ClN3OS
4-methyl-thiazole-5-carboxylic acid (4-amino-cyclohexyl)-[2-(3-chloro-phenyl)-ethyl]-amide
—— —— 1094837-67-8 C33H35ClN2O6
—— 3-(2-fluoro-4-iodo-phenylamino)-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid cyclopropylmethoxy-amide monoformate 1030382-03-6 CH2O2*C18H16FIN4O2
3-(2-fluoro-4-iodo-phenylamino)-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid cyclopropylmethoxy-amide monoformate
—— 1-methyl-1H-imidazole-4-carboxylic acid (2-aza-bicyclo[3.3.1]non-6-yl)-[6-(3,4-dichloro-phenyl)-pyridin-2-ylmethyl]-amide 1031299-44-1 C25H27Cl2N5O
1-methyl-1H-imidazole-4-carboxylic acid (2-aza-bicyclo[3.3.1]non-6-yl)-[6-(3,4-dichloro-phenyl)-pyridin-2-ylmethyl]-amide
—— trans-((R)-3-hydroxypyrrolidin-1-yl)-[4-(4-indazol-1-ylpyrimidin-2-ylamino)-cyclohexyl]-methanone 1032452-25-7 C22H26N6O2
trans-((R)-3-hydroxypyrrolidin-1-yl)-[4-(4-indazol-1-ylpyrimidin-2-ylamino)-cyclohexyl]-methanone
—— —— 1029138-12-2 C18H21ClN2O
—— (2S,4S,5S)-5-amino-6-benzyloxy-4-hydroxy-2-isopropyl-hexanoic acid [(S)-1-(3,4-dichloro-benzylcarbamoyl)-2-methyl-propyl]-amide 1056671-52-3 C28H39Cl2N3O4
(2S,4S,5S)-5-amino-6-benzyloxy-4-hydroxy-2-isopropyl-hexanoic acid [(S)-1-(3,4-dichloro-benzylcarbamoyl)-2-methyl-propyl]-amide
—— ethyl (2S)-2-[[[(2R,3S,4R,5R)-4-cyano-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate 1491021-83-0 C22H27N4O9P
ethyl (2S)-2-[[[(2R,3S,4R,5R)-4-cyano-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
—— 2-hydroxypropyl {4-[1-ethyl-4-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl}carbamate 1144070-96-1 C23H28N6O4
2-hydroxypropyl {4-[1-ethyl-4-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl}carbamate
—— 2-[6-(2-imidazol-1-ylethyl)-3H-1,3-benzothiazol-2-ylidene]-2-[4-(trifluoromethyl)pyrimidin-2-yl]acetamide 1219483-06-3 C19H15F3N6OS
2-[6-(2-imidazol-1-ylethyl)-3H-1,3-benzothiazol-2-ylidene]-2-[4-(trifluoromethyl)pyrimidin-2-yl]acetamide
—— 4-[2-(2-cyclopropylethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine 1403988-09-9 C22H23FN4O3S
4-[2-(2-cyclopropylethoxy)-4-fluorophenyl]-N-{3-[(methylsulfonyl)methyl]phenyl}-1,3,5-triazin-2-amine
—— 1-[3-(4-carbamoylphenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid 1401320-96-4 C21H15N3O4
1-[3-(4-carbamoylphenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid
—— 5-cyclopropyl-1-(3,5-dimethylisoxazole-4-carbonyl)-2,3,5,6-tetrahydropyrido[2,3-b][1,5]diazocin-4(1H)-one 1307894-49-0 C18H20N4O3
5-cyclopropyl-1-(3,5-dimethylisoxazole-4-carbonyl)-2,3,5,6-tetrahydropyrido[2,3-b][1,5]diazocin-4(1H)-one
—— N-[[3-[[3-[(4-bromophenyl)carbamoyl]-4-(2,2-difluoroethoxy)phenyl]carbamoyl]-4-chlorophenyl]methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide 1294496-40-4 C29H24BrClF2N4O4S
N-[[3-[[3-[(4-bromophenyl)carbamoyl]-4-(2,2-difluoroethoxy)phenyl]carbamoyl]-4-chlorophenyl]methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
—— [({2-[(1-{5-[3-fluoro-4-(hydroxymethyl)phenyl]pyridin-2-yl}piperidin-4-yl)methyl]-5-hydroxy-6-methylpyrimidin-4-yl}carbonyl)amino]acetic acid 1296273-59-0 C26H28FN5O5
[({2-[(1-{5-[3-fluoro-4-(hydroxymethyl)phenyl]pyridin-2-yl}piperidin-4-yl)methyl]-5-hydroxy-6-methylpyrimidin-4-yl}carbonyl)amino]acetic acid
—— 6-(4-(1-aminocyclobutyl)phenyl)-1,3-dimethyl-5-phenylfuro[2,3-d]pyrimidine-2,4(1H,3H)-dione 1301610-04-7 C24H23N3O3
6-(4-(1-aminocyclobutyl)phenyl)-1,3-dimethyl-5-phenylfuro[2,3-d]pyrimidine-2,4(1H,3H)-dione
—— 1-methylsulfanyl-8,10,12,13-tetraoxapentacyclo[5.5.1.02,6.03,11.04,9]tridecane 136093-79-3 C10H12O4S
1-methylsulfanyl-8,10,12,13-tetraoxapentacyclo[5.5.1.02,6.03,11.04,9]tridecane
—— 3-(5-{[4-(1-methylethyl)phenyl]amino}-5-oxopentyl)-1-phenyl-1H-indole-5-carboxylic acid 1144523-36-3 C29H30N2O3
3-(5-{[4-(1-methylethyl)phenyl]amino}-5-oxopentyl)-1-phenyl-1H-indole-5-carboxylic acid
—— 6,9-dichloro-3-oxo-N-[4-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide 1067226-78-1 C17H11Cl2F3N2O3
6,9-dichloro-3-oxo-N-[4-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide
—— tert-butyl N-[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-[[(4S,5S,7S)-5-hydroxy-2,8-dimethyl-7-[[(2S,3S)-3-methyl-1-oxo-1-(pyridin-2-ylmethylamino)pentan-2-yl]carbamoyl]nonan-4-yl]amino]-3-[1-(4-methylphenyl)sulfonylimidazol-4-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]oxymethyl]pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]carbamate 112374-81-9 C65H89N9O11S
tert-butyl N-[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-[[(4S,5S,7S)-5-hydroxy-2,8-dimethyl-7-[[(2S,3S)-3-methyl-1-oxo-1-(pyridin-2-ylmethylamino)pentan-2-yl]carbamoyl]nonan-4-yl]amino]-3-[1-(4-methylphenyl)sulfonylimidazol-4-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]oxymethyl]pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]carbamate