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中文名称 英文名称 CAS号 化学式 结构式图片
—— —— 1607482-70-1 C17H10BrF3N2O
—— 3-(3-methoxy-5-(trifluoromethyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1604802-10-9 C13H10F3N5O
3-(3-methoxy-5-(trifluoromethyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— N-([cis-3-(2-benzofuryl)-3-methyl]cyclobutyl)-N-hydroxyurea 143588-76-5 C14H16N2O3
N-([cis-3-(2-benzofuryl)-3-methyl]cyclobutyl)-N-hydroxyurea
—— ethyl 3-[N-benzyl-2-[[1-(1-benzyl-5-fluoro-2-oxoindol-3-ylidene)-2-oxo-2-phenylethyl]amino]anilino]-2-cyanoprop-2-enoate 1391839-47-6 C42H33FN4O4
ethyl 3-[N-benzyl-2-[[1-(1-benzyl-5-fluoro-2-oxoindol-3-ylidene)-2-oxo-2-phenylethyl]amino]anilino]-2-cyanoprop-2-enoate
—— 2'-Deoxy-3'-O-[(1,1-dimethylethyl)dimethylsilyl]-N,5-dimethyl-cytidine 1569273-35-3 C17H31N3O4Si
2'-Deoxy-3'-O-[(1,1-dimethylethyl)dimethylsilyl]-N,5-dimethyl-cytidine
—— benzyl 2-diazo-5-methoxypentanoate 1352218-72-4 C13H16N2O3
benzyl 2-diazo-5-methoxypentanoate
—— 5,5'-methylenebis(2-(2-methoxyphenylamino)benzoic acid) 1056450-37-3 C29H26N2O6
5,5'-methylenebis(2-(2-methoxyphenylamino)benzoic acid)
—— (R)-(3,3-dimethyl-2,3-dihydro-1H-pyrrolo[3,2-b]pyridin-6-yl)-(3-fluoro-phenyl)-methanol 1605318-46-4 C16H17FN2O
(R)-(3,3-dimethyl-2,3-dihydro-1H-pyrrolo[3,2-b]pyridin-6-yl)-(3-fluoro-phenyl)-methanol
—— [4-Chloro-2-(dimethylamino)-3-phenylquinolin-6-yl](1-methyl-1H-imidazol-5-yl)pyridin-3-ylmethanol trifluoroacetate 1600563-92-5 C2HF3O2*C27H24ClN5O
[4-Chloro-2-(dimethylamino)-3-phenylquinolin-6-yl](1-methyl-1H-imidazol-5-yl)pyridin-3-ylmethanol trifluoroacetate
—— —— 1050329-33-3 C30H38O5S
—— N-[5-[2-(methoxymethyl)phenyl]pent-4-yn-2-yl]quinazolin-4-amine 1262027-49-5 C21H21N3O
N-[5-[2-(methoxymethyl)phenyl]pent-4-yn-2-yl]quinazolin-4-amine
—— 5-[2-cyclopropyl-8-(4-morpholinyl)imidazo[1,2-b]pyridazin-3-yl]-α,α-dimethyl-2-pyridineethanol 1298030-87-1 C22H27N5O2
5-[2-cyclopropyl-8-(4-morpholinyl)imidazo[1,2-b]pyridazin-3-yl]-α,α-dimethyl-2-pyridineethanol
—— (5S,6R,7R,8S)-5-{3-[4-(benzyl-ethyl-amino)-benzyl]-4-chloro-phenyl}-4-oxa-spiro[2.5]octane-6,7,8-triol 1290630-21-5 C29H32ClNO4
(5S,6R,7R,8S)-5-{3-[4-(benzyl-ethyl-amino)-benzyl]-4-chloro-phenyl}-4-oxa-spiro[2.5]octane-6,7,8-triol
—— 5'-O-acetyl-3-[3-[2-(2-methylbenzoyloxy)-4-pyridyloxycarbonyl]benzoyl]-3'-O-benzyl-2'-deoxy-5-fluorouridine 103767-04-0 C39H32FN3O11
5'-O-acetyl-3-[3-[2-(2-methylbenzoyloxy)-4-pyridyloxycarbonyl]benzoyl]-3'-O-benzyl-2'-deoxy-5-fluorouridine
—— 2-(4-pentafluoropropionylaminophenethyl)-6-(3,4-dimethoxyphenyl)-5-ethyl-2,3,4,5-tetrahydropyridazin-3-one 1230635-90-1 C25H26F5N3O4
2-(4-pentafluoropropionylaminophenethyl)-6-(3,4-dimethoxyphenyl)-5-ethyl-2,3,4,5-tetrahydropyridazin-3-one
—— rubiyunnanin G 1261030-08-3 C45H56N6O14
rubiyunnanin G
—— [4-(4',5'-difluoro-2'-methoxy-biphenyl-4-yloxymethyl)-indol-1-yl]-acetic acid 1298130-08-1 C24H19F2NO4
[4-(4',5'-difluoro-2'-methoxy-biphenyl-4-yloxymethyl)-indol-1-yl]-acetic acid
—— ({[2-({1-[4'-(1,1-difluoro-2-hydroxypropyl)biphenyl-4-yl]piperidin-4-yl}methyl)-5-hydroxy-6-methylpyrimidin-4-yl]carbonyl}amino)acetic acid 1296273-37-4 C29H32F2N4O5
({[2-({1-[4'-(1,1-difluoro-2-hydroxypropyl)biphenyl-4-yl]piperidin-4-yl}methyl)-5-hydroxy-6-methylpyrimidin-4-yl]carbonyl}amino)acetic acid
—— 2-{2-[(4aS,5R)-4a-ethyl-5-hydroxy-1-(pyridin-3-yl)-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-6-fluorobenzamide 1299473-28-1 C26H27FN4O2
2-{2-[(4aS,5R)-4a-ethyl-5-hydroxy-1-(pyridin-3-yl)-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-6-fluorobenzamide
—— 2-{2-[(4aR,5R)-4a-cyclopropyl-1-(4-fluorophenyl)-5-hydroxy-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-N-[1-(hydroxymethyl)cyclopropyl]benzamide 1299473-60-1 C32H34FN3O3
2-{2-[(4aR,5R)-4a-cyclopropyl-1-(4-fluorophenyl)-5-hydroxy-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-N-[1-(hydroxymethyl)cyclopropyl]benzamide
—— 5-(3,5-dimethylisoxazol-4-yl)-3-ethyl-1-(2-fluoro-4-hydroxyphenyl)-N'-hydroxy-1H-pyrazole-4-carboximidamide 1290138-04-3 C17H18FN5O3
5-(3,5-dimethylisoxazol-4-yl)-3-ethyl-1-(2-fluoro-4-hydroxyphenyl)-N'-hydroxy-1H-pyrazole-4-carboximidamide
—— (2S,3R,4R,5S,6R)-2-[3-(3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethyl)-4-fluoro-phenyl]-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol 1291094-11-5 C21H24FNO6
(2S,3R,4R,5S,6R)-2-[3-(3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethyl)-4-fluoro-phenyl]-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol
—— 4-Amino-2-[[2-(2-hydroxypropan-2-yl)phenyl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 1305262-90-1 C19H19N5O2
4-Amino-2-[[2-(2-hydroxypropan-2-yl)phenyl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one
—— 17-Methoxy-16-phenylmethoxy-21-[(4-propan-2-ylphenyl)methyl]-5,7-dioxa-13-azoniapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-1(13),2,4(8),9,14,16,18,20-octaene;chloride 1257844-18-0 C36H34NO4*Cl
17-Methoxy-16-phenylmethoxy-21-[(4-propan-2-ylphenyl)methyl]-5,7-dioxa-13-azoniapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-1(13),2,4(8),9,14,16,18,20-octaene;chloride
—— 2-chloro-N-(3-(3-(2-(2-methyl-l,2,3,4-tetrahydroisoquinolin-7-ylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)phenyl)benzamide 1301135-19-2 C34H28ClN7O
2-chloro-N-(3-(3-(2-(2-methyl-l,2,3,4-tetrahydroisoquinolin-7-ylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)phenyl)benzamide
—— Tucatinib hemiethanolate 1429755-56-5 C54H54N16O5
Tucatinib hemiethanolate
—— 4-hydroxy-6-methylenandrosta-1,4-diene-3,17-dione 115836-77-6 C20H24O3
4-hydroxy-6-methylenandrosta-1,4-diene-3,17-dione
—— 5-(2-amino-5-oxo-4-phenyl-5H-indeno[1,2-d]pyrimidin-9-yl)thiophene-2-carbonitrile 1297604-26-2 C22H12N4OS
5-(2-amino-5-oxo-4-phenyl-5H-indeno[1,2-d]pyrimidin-9-yl)thiophene-2-carbonitrile
—— 2-(4-amino-3,5-dichlorophenyl)-N-cyclopropyl-3-hydroxy-4-oxo-1H-quinoline-6-carboxamide 1259368-55-2 C19H15Cl2N3O3
2-(4-amino-3,5-dichlorophenyl)-N-cyclopropyl-3-hydroxy-4-oxo-1H-quinoline-6-carboxamide
—— 3-(4-tert-butylphenyl)-7-chloro-1,3-benzoxazine-2,4(3H)-dithione 1261228-20-9 C18H16ClNOS2
3-(4-tert-butylphenyl)-7-chloro-1,3-benzoxazine-2,4(3H)-dithione
—— 5-cyclopropyl-8-methoxy-1-(2-(3-methoxyphenyl)-2-oxoethyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307893-65-7 C23H26N2O4
5-cyclopropyl-8-methoxy-1-(2-(3-methoxyphenyl)-2-oxoethyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one
—— 2-chloro-N-(1-(1-methyl-1H-pyrazol-3-ylamino)-1,2-dioxoheptan-3-yl)-4-(pyridin-2-ylmethoxy)-3-(trifluoromethyl)benzamide 1259539-08-6 C25H25ClF3N5O4
2-chloro-N-(1-(1-methyl-1H-pyrazol-3-ylamino)-1,2-dioxoheptan-3-yl)-4-(pyridin-2-ylmethoxy)-3-(trifluoromethyl)benzamide
—— (E)-1-(4-bromophenyl)-2-[(4-bromophenyl)methylsulfanyl]-3-(4-hydroxy-3-methoxy-5-nitrophenyl)prop-2-en-1-one 1035199-06-4 C23H17Br2NO5S
(E)-1-(4-bromophenyl)-2-[(4-bromophenyl)methylsulfanyl]-3-(4-hydroxy-3-methoxy-5-nitrophenyl)prop-2-en-1-one
—— N-(2-glycinamido-2-deoxy-β-D-glucopyranosyl)-N-hexadecyl-octadecanoamide 113467-38-2 C42H83N3O6
N-(2-glycinamido-2-deoxy-β-D-glucopyranosyl)-N-hexadecyl-octadecanoamide
—— 2-(4-butyrylaminobenzyl)-6-(3-difluoromethoxy-4-methoxyphenyl)-5-ethyl-2,3,4,5-tetrahydropyridazin-3-one 1230636-47-1 C25H29F2N3O4
2-(4-butyrylaminobenzyl)-6-(3-difluoromethoxy-4-methoxyphenyl)-5-ethyl-2,3,4,5-tetrahydropyridazin-3-one
—— 4-acetylthio-6-methylenandrost-4-ene-3,17-dione 115837-17-7 C22H28O3S
4-acetylthio-6-methylenandrost-4-ene-3,17-dione
—— 4-methyl-2-{5-[4-methyl-1-(3,4,5-trifluoro-phenyl)-pentylamino]-4'-trifluoromethyl-biphenyl-3-yl}-pentanoic acid 1145691-52-6 C31H33F6NO2
4-methyl-2-{5-[4-methyl-1-(3,4,5-trifluoro-phenyl)-pentylamino]-4'-trifluoromethyl-biphenyl-3-yl}-pentanoic acid
—— 3-(6-hydroxy-hex-1-ynyl)-N-[(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-benzamide 1107005-96-8 C24H26N2O3
3-(6-hydroxy-hex-1-ynyl)-N-[(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-benzamide
—— 6-Bromo-8-[(1-methyl-4-phenylpiperidin-4-yl)methoxymethyl]quinoline 1100206-42-5 C23H25BrN2O
6-Bromo-8-[(1-methyl-4-phenylpiperidin-4-yl)methoxymethyl]quinoline
—— 1-[4-[3-[[4-[(3-chloro-2,4-difluoro-phenyl)-methyl-amino]pyrimidin-2-yl]amino]-5-methylsulfonyl-phenyl]piperazin-1-yl]ethanone 1051896-27-5 C24H25ClF2N6O3S
1-[4-[3-[[4-[(3-chloro-2,4-difluoro-phenyl)-methyl-amino]pyrimidin-2-yl]amino]-5-methylsulfonyl-phenyl]piperazin-1-yl]ethanone
—— N-[3-[(4-bromophenyl)carbamoyl]-4-(2,2-difluoroethoxy)phenyl]-2-chloro-5-[[(2-hydroxy-2-methylpropanoyl)amino]methyl]benzamide 1294496-44-8 C27H25BrClF2N3O5
N-[3-[(4-bromophenyl)carbamoyl]-4-(2,2-difluoroethoxy)phenyl]-2-chloro-5-[[(2-hydroxy-2-methylpropanoyl)amino]methyl]benzamide
—— (2R,3aS,3a1S,3a2S,5S,5aR,8aS,10aS)-2,5-dimethyldodecahydropyrene-1,8(3a1H,3a2H)-dione 106140-97-0 C18H26O2
(2R,3aS,3a1S,3a2S,5S,5aR,8aS,10aS)-2,5-dimethyldodecahydropyrene-1,8(3a1H,3a2H)-dione
—— (1R,6S)-2-[3-(2,4-dimethyl-benzenesulfonyl)-3,8-diaza-bicyclo[4.2.0]oct-8-yl]-quinoxaline 1295516-27-6 C22H24N4O2S
(1R,6S)-2-[3-(2,4-dimethyl-benzenesulfonyl)-3,8-diaza-bicyclo[4.2.0]oct-8-yl]-quinoxaline
—— (4S,5R)-5-[(2R)-3-(2,2-dimethyl-6-oxo-1,3-dioxin-4-yl)-2-methoxypropyl]-2,2-dimethyl-1,3-dioxolane-4-carbaldehyde 1262750-15-1 C16H24O7
(4S,5R)-5-[(2R)-3-(2,2-dimethyl-6-oxo-1,3-dioxin-4-yl)-2-methoxypropyl]-2,2-dimethyl-1,3-dioxolane-4-carbaldehyde
—— 2-amino-9-(4-methoxyphenyl)-4-phenylindeno[1,2-d]pyrimidin-5-one 1297599-72-4 C24H17N3O2
2-amino-9-(4-methoxyphenyl)-4-phenylindeno[1,2-d]pyrimidin-5-one
—— 4-(2-fluorobenzylamino)-6-(4-(2-oxopiperidin-1-yl)phenylamino)nicotinamide 1374211-06-9 C24H24FN5O2
4-(2-fluorobenzylamino)-6-(4-(2-oxopiperidin-1-yl)phenylamino)nicotinamide
—— 2-(4-chloro-2-fluoro-phenoxy)-2-(4-cyclopropane-sulfonyl-phenyl)-N-[1,3,4]thiadiazol-2-yl-acetamide 1143513-03-4 C19H15ClFN3O4S2
2-(4-chloro-2-fluoro-phenoxy)-2-(4-cyclopropane-sulfonyl-phenyl)-N-[1,3,4]thiadiazol-2-yl-acetamide
—— N-[(2'-chlorobiphenyl-4-yl)methyl]-N-[3-fluoro-5-(1H-tetrazol-5-yl)phenyl]propanamide 1262338-58-8 C23H19ClFN5O
N-[(2'-chlorobiphenyl-4-yl)methyl]-N-[3-fluoro-5-(1H-tetrazol-5-yl)phenyl]propanamide
—— [(1S,5S)-3-[(1R)-1-phenylethyl]-3-azabicyclo[3. 3. 0]oct-7-en-1-yl]carboxylic acid tert-butyl ester 1037367-95-5 C20H27NO2
[(1S,5S)-3-[(1R)-1-phenylethyl]-3-azabicyclo[3. 3. 0]oct-7-en-1-yl]carboxylic acid tert-butyl ester
—— 4-{3-isopropyl-4-(quinolin-3-yl)-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-{3-(methylthio)propylamino}benzonitrile 1260536-97-7 C29H28N6S
4-{3-isopropyl-4-(quinolin-3-yl)-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-{3-(methylthio)propylamino}benzonitrile