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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-chloro-2-[2-chloro-6-(methylsulfinyl)-4-(trifluoromethoxy)phenoxy]-7-(1-ethylpropyl)-1-methyl-1H-benzimidazole 1022249-34-8 C21H21Cl2F3N2O3S
4-chloro-2-[2-chloro-6-(methylsulfinyl)-4-(trifluoromethoxy)phenoxy]-7-(1-ethylpropyl)-1-methyl-1H-benzimidazole
—— 6-amino-2-butoxy-9-{3-[(4-isopropoxybenzyl)(3-morpholin-4-ylpropyl)amino]propyl}-7,9-dihydro-8H-purin-8-one 1033003-42-7 C29H45N7O4
6-amino-2-butoxy-9-{3-[(4-isopropoxybenzyl)(3-morpholin-4-ylpropyl)amino]propyl}-7,9-dihydro-8H-purin-8-one
—— 1-[2-(1-benzenesulfonyl-piperidin-3-yl)-acetylamino]-piperidine-3-carboxylic acid methyl ester 1040878-71-4 C20H29N3O5S
1-[2-(1-benzenesulfonyl-piperidin-3-yl)-acetylamino]-piperidine-3-carboxylic acid methyl ester
—— 1-(3-chlorophenyl)-3-(4-bromophenyl)pyrrole-2,5-dione 1032508-24-9 C16H9BrClNO2
1-(3-chlorophenyl)-3-(4-bromophenyl)pyrrole-2,5-dione
—— N-(2-ethylphenyl)-4-(4-methyl-6-((4-(morpholine-4-carbonyl)phenyl)amino)-5-oxo-4,5-dihydropyrazin-2-yl)indoline-1-carboxamide 1622173-17-4 C33H34N6O4
N-(2-ethylphenyl)-4-(4-methyl-6-((4-(morpholine-4-carbonyl)phenyl)amino)-5-oxo-4,5-dihydropyrazin-2-yl)indoline-1-carboxamide
—— N-(4-(2-hydroxyamino-2-oxo-1-phenylethyl)phenyl)-2-methylbenzamide 1070678-85-1 C22H20N2O3
N-(4-(2-hydroxyamino-2-oxo-1-phenylethyl)phenyl)-2-methylbenzamide
—— (2S,3S,4R)-(3,4-isopropylidenedioxy-1-(1'S,2'S,3'S,4'S,5'R)-5'-hydroxymethyl-2',3',4'-tribenzyloxycyclohexylaminooctadecan-2-yl)hexacosanamide 1245916-78-2 C75H124N2O7
(2S,3S,4R)-(3,4-isopropylidenedioxy-1-(1'S,2'S,3'S,4'S,5'R)-5'-hydroxymethyl-2',3',4'-tribenzyloxycyclohexylaminooctadecan-2-yl)hexacosanamide
—— tert-butyl [tert-butoxycarbonyl(6-{[4-(1-butylcyclopropyl)benzyl](pyridin-4-ylsulfonyl)aminomethyl}pyridin-2-yl)amino]acetate 1313216-80-6 C36H48N4O6S
tert-butyl [tert-butoxycarbonyl(6-{[4-(1-butylcyclopropyl)benzyl](pyridin-4-ylsulfonyl)aminomethyl}pyridin-2-yl)amino]acetate
—— tert-butyl N-[(2S)-1-{3-[(4-chloro-3-fluorophenyl)amino]-2-(3-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}-1-oxo-3-(4-propanamidophenyl)propan-2-yl]carbamate 1261112-39-3 C35H37ClF2N6O4
tert-butyl N-[(2S)-1-{3-[(4-chloro-3-fluorophenyl)amino]-2-(3-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}-1-oxo-3-(4-propanamidophenyl)propan-2-yl]carbamate
—— 6-[3-Fluoro-4-[2-(pteridin-4-ylamino)ethyl]phenoxy]pyridine-3-carbonitrile 1268608-33-8 C20H14FN7O
6-[3-Fluoro-4-[2-(pteridin-4-ylamino)ethyl]phenoxy]pyridine-3-carbonitrile
—— tert-butyl N-[3-[cyclohexyl(phenyl)methyl]-2-methyl-4-oxoquinazolin-6-yl]carbamate 1197003-97-6 C27H33N3O3
tert-butyl N-[3-[cyclohexyl(phenyl)methyl]-2-methyl-4-oxoquinazolin-6-yl]carbamate
—— tert-butyl 4-[4-bromo-3-(trifluoromethyl)phenyl]piperazine-1-carboxylate 1197294-00-0 C16H20BrF3N2O2
tert-butyl 4-[4-bromo-3-(trifluoromethyl)phenyl]piperazine-1-carboxylate
—— 6-chloro-2-(4-(2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl)phenyl)-1-methyl-1H-benzoimidazole 1038842-07-7 C23H15Cl2FN4
6-chloro-2-(4-(2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl)phenyl)-1-methyl-1H-benzoimidazole
—— 6-(2,6-dichlorophenyl)-8-methoxy-2-(3-methoxyphenylamino)-pyrido[2,3-d]pyrimidin-7-one 1021302-47-5 C21H16Cl2N4O3
6-(2,6-dichlorophenyl)-8-methoxy-2-(3-methoxyphenylamino)-pyrido[2,3-d]pyrimidin-7-one
—— N-(2-hydroxy-2-phenylethyl)-2'-methylspiro[cyclohexane-1,9'-thioxanthene]-3'-sulfonamide 10',10'-dioxide 1027347-44-9 C27H29NO5S2
N-(2-hydroxy-2-phenylethyl)-2'-methylspiro[cyclohexane-1,9'-thioxanthene]-3'-sulfonamide 10',10'-dioxide
—— 4-fluoro-1'-(1-naphthoyl)-3H-spiro[2-benzofuran-1,4'-piperidine] 1034352-67-4 C23H20FNO2
4-fluoro-1'-(1-naphthoyl)-3H-spiro[2-benzofuran-1,4'-piperidine]
—— (E)-1-(4-chlorophenyl)-2-(4-methylphenylsulfenyl)-3-(4-phenoxyphenyl)prop-2-en-1-one 1035198-20-9 C28H21ClO2S
(E)-1-(4-chlorophenyl)-2-(4-methylphenylsulfenyl)-3-(4-phenoxyphenyl)prop-2-en-1-one
—— 3-{[4-({[4-bromo-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]methyl}benzoic acid 1027009-01-3 C20H20BrF3N2O4S
3-{[4-({[4-bromo-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]methyl}benzoic acid
—— N-[(1R,2S)-1-[1-(6-fluoropyridin-3-yl)indazol-5-yl]oxy-1-phenyl-propan-2-yl]cyclopropanesulfonamide 1028458-67-4 C24H23FN4O3S
N-[(1R,2S)-1-[1-(6-fluoropyridin-3-yl)indazol-5-yl]oxy-1-phenyl-propan-2-yl]cyclopropanesulfonamide
—— 1-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-(3-(hydroxymethyl)phenoxy)propan-2-ol 1041191-01-8 C27H29FN4O3S
1-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-(3-(hydroxymethyl)phenoxy)propan-2-ol
—— 4-[(4-Chlorophenyl)methyl]-2-({(2R)-1-[(2-oxo-3-piperidinyl)methyl]-2-pyrrolidinyl}methyl)-1(2H)-phthalazinone 1035040-75-5 C26H29ClN4O2
4-[(4-Chlorophenyl)methyl]-2-({(2R)-1-[(2-oxo-3-piperidinyl)methyl]-2-pyrrolidinyl}methyl)-1(2H)-phthalazinone
—— N-(2-hydroxy-3-(piperidin-1-yl)propyl)-2-methyl-7-[1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide 1032267-30-3 C26H32N4O3
N-(2-hydroxy-3-(piperidin-1-yl)propyl)-2-methyl-7-[1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
—— 6-(3-hydroxyphenyl)-1-(piperidin-1-ylcarbonyl)-2-naphthol 1041113-83-0 C22H21NO3
6-(3-hydroxyphenyl)-1-(piperidin-1-ylcarbonyl)-2-naphthol
—— 2-((1-(mesitylsulfonyl)piperidin-2-yl)methoxy)-1-(4-(pyrrolidin-1-yl)piperidin-1-yl)-ethanone 1018820-33-1 C26H41N3O4S
2-((1-(mesitylsulfonyl)piperidin-2-yl)methoxy)-1-(4-(pyrrolidin-1-yl)piperidin-1-yl)-ethanone
—— (R)-tert-butyl 2-acetoxy-2-((R)-4-(2-methyl-3-oxoisoindolin-5-yl)-3-oxomorpholin-2-yl)acetate 1228774-23-9 C21H26N2O7
(R)-tert-butyl 2-acetoxy-2-((R)-4-(2-methyl-3-oxoisoindolin-5-yl)-3-oxomorpholin-2-yl)acetate
—— 1-(4-methoxy-phenylethynyl)-5H-benzo[c][1,8]naphthyridin-6-one 1186375-86-9 C21H14N2O2
1-(4-methoxy-phenylethynyl)-5H-benzo[c][1,8]naphthyridin-6-one
—— 3-(3-amino-propyl)-5-(indan-5-ylcarbamoyl)-1H-indole-2-carboxylic acid 1055251-46-1 C22H23N3O3
3-(3-amino-propyl)-5-(indan-5-ylcarbamoyl)-1H-indole-2-carboxylic acid
—— 2-Benzyl-1-propyl-8-[3-(thiazol-2-ylaminomethyl)-adamantan-1-yl]-1,7-dihydro-purin-6-one 1303955-51-2 C29H34N6OS
2-Benzyl-1-propyl-8-[3-(thiazol-2-ylaminomethyl)-adamantan-1-yl]-1,7-dihydro-purin-6-one
—— (+/-)-4-[(4-Chlorophenyl)phenylmethoxy]-1-piperidineheptanoic acid hydrochloride 133016-17-8 C25H32ClNO3*ClH
(+/-)-4-[(4-Chlorophenyl)phenylmethoxy]-1-piperidineheptanoic acid hydrochloride
—— 3,6-Bis-dimethylamino-9-phenyl-acridan 16292-10-7 C23H25N3
3,6-Bis-dimethylamino-9-phenyl-acridan
—— (4-chloro-3-trifluoromethyl-phenyl)-(3H-imidazol-4-ylmethyl)-isopropyl-amine 1020814-73-6 C14H15ClF3N3
(4-chloro-3-trifluoromethyl-phenyl)-(3H-imidazol-4-ylmethyl)-isopropyl-amine
—— 3-(4-fluorophenyl)-7-(2-fluorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 1621966-98-0 C18H10F2N2OS
3-(4-fluorophenyl)-7-(2-fluorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one
—— 3,5-dimethyl-4-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-pyrazole-1-carboxylic acid 4-chlorobenzylamide 1029046-65-8 C21H20ClN5O
3,5-dimethyl-4-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-pyrazole-1-carboxylic acid 4-chlorobenzylamide
—— 5-(5-{2-[[3-(dimethylamino)propyl](methyl)amino]-4-pyridinyl}-1H-benzimidazol-1-yl)-3-({(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}oxy)-2-thiophenecarboxamide 1032198-58-5 C32H33F3N6O2S
5-(5-{2-[[3-(dimethylamino)propyl](methyl)amino]-4-pyridinyl}-1H-benzimidazol-1-yl)-3-({(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}oxy)-2-thiophenecarboxamide
—— N-(2-((2-((4-oxocyclohexyl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)prop-1-ene-2-sulfonamide 1621999-07-2 C20H22F3N5O3S
N-(2-((2-((4-oxocyclohexyl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)prop-1-ene-2-sulfonamide
—— N-(4-chlorobenzyl)-N-methyl-4,5,6,7-tetrahydrobenzo[d]thiazole-7-carboxamide 1620877-97-5 C16H17ClN2OS
N-(4-chlorobenzyl)-N-methyl-4,5,6,7-tetrahydrobenzo[d]thiazole-7-carboxamide
—— 6-(2,4-difluorophenyl)-5-(3-(1-methylcyclopropyl)-[1,2,4]triazolo[4,3-a]pyridin-6-yl)imidazo[2,1-b]oxazole 1029525-68-5 C21H15F2N5O
6-(2,4-difluorophenyl)-5-(3-(1-methylcyclopropyl)-[1,2,4]triazolo[4,3-a]pyridin-6-yl)imidazo[2,1-b]oxazole
—— <6,8,9,11-2H4>-2,3-dihydro-1H-benzo<c>pyrazolo<1,2-a>cinnoline 124522-41-4 C15H14N2
<6,8,9,11-2H4>-2,3-dihydro-1H-benzo<c>pyrazolo<1,2-a>cinnoline
—— 2-(trifluoromethyl)-1,3-benzoxazol-5-amine 122139-97-3 C8H5F3N2O
2-(trifluoromethyl)-1,3-benzoxazol-5-amine
—— 2-chloro-4,6-difluoro-5-trifluoromethoxybenzoic acid 1027182-16-6 C8H2ClF5O3
2-chloro-4,6-difluoro-5-trifluoromethoxybenzoic acid
—— [1,3,3,8-Tetramethyl-5-oxo-bicyclo[4.2.0]oct-(7E)-ylidene]-acetic acid ethyl ester 125041-75-0 C16H24O3
[1,3,3,8-Tetramethyl-5-oxo-bicyclo[4.2.0]oct-(7E)-ylidene]-acetic acid ethyl ester
—— 4-(4-bromo-2-oxopyridin-1(2H)-yl)-2-methyl-2-(methylsulfonyl)-N-(tetrahydro-2H-pyran-2-yloxy)butanamide 1312478-62-8 C16H23BrN2O6S
4-(4-bromo-2-oxopyridin-1(2H)-yl)-2-methyl-2-(methylsulfonyl)-N-(tetrahydro-2H-pyran-2-yloxy)butanamide
—— 6-amino-5-[1-(2,6-dichloro-3-fluoro-phenyl)-ethoxy]-pyridazine-3-carboxyIic acid methylamide 1040376-95-1 C14H13Cl2FN4O2
6-amino-5-[1-(2,6-dichloro-3-fluoro-phenyl)-ethoxy]-pyridazine-3-carboxyIic acid methylamide
—— N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-2-oxo-3-pentyl-2,3-dihydro-1H-benzimidazole-1-carboxamide 1012880-92-0 C20H30N4O2
N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-2-oxo-3-pentyl-2,3-dihydro-1H-benzimidazole-1-carboxamide
—— 1-(4-{2-[5-(4,6-dimethyl-pyrimidine-5-carbonyl)-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl]-ethyl}-4-phenyl-piperidin-1-yl)-2-methyl-propan-1-one 1014700-91-4 C30H41N5O2
1-(4-{2-[5-(4,6-dimethyl-pyrimidine-5-carbonyl)-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl]-ethyl}-4-phenyl-piperidin-1-yl)-2-methyl-propan-1-one
—— 4-{[(4-(2,2,2-trifluoroethyl-amino)-6-carbamoylphenyl)-pyrido[3,2-d]pyrimidin-2-ylamino]-methyl}-benzenesulfonamide 1036736-55-6 C23H20F3N7O3S
4-{[(4-(2,2,2-trifluoroethyl-amino)-6-carbamoylphenyl)-pyrido[3,2-d]pyrimidin-2-ylamino]-methyl}-benzenesulfonamide
—— 4-(4-morpholino-6-((4-N-methylsulfonylpiperazin-1-yl)methyl)thieno[3,2-d]pyrimidin-2-yl)pyridin-2-amine 1032756-11-8 C21H27N7O3S2
4-(4-morpholino-6-((4-N-methylsulfonylpiperazin-1-yl)methyl)thieno[3,2-d]pyrimidin-2-yl)pyridin-2-amine
—— 8-tert-butyl-3-[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-7,8-dihydro-3H-[1,3]oxazino[6,5-g][1,2,3]benzotriazine-4,9-dione 1039453-35-4 C17H20N8O3
8-tert-butyl-3-[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-7,8-dihydro-3H-[1,3]oxazino[6,5-g][1,2,3]benzotriazine-4,9-dione
—— 3-Bromo-5-methoxy-anthra[1,9-cd]isoxazol-6-one 127727-69-9 C15H8BrNO3
3-Bromo-5-methoxy-anthra[1,9-cd]isoxazol-6-one
—— [3-(1,3,3-trimethyl-1,2,3,4-tetrahydro-quinolin-4-yl)-3H-imidazol-4-yl]-methanol 1034193-38-8 C16H21N3O
[3-(1,3,3-trimethyl-1,2,3,4-tetrahydro-quinolin-4-yl)-3H-imidazol-4-yl]-methanol