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中文名称 英文名称 CAS号 化学式 结构式图片
—— benzyl [1-(2-methoxyphenyl)-2-oxo-2-(phenylmethoxycarbonylamino)ethyl] carbonate 144220-12-2 C25H23NO7
benzyl [1-(2-methoxyphenyl)-2-oxo-2-(phenylmethoxycarbonylamino)ethyl] carbonate
—— (3-acetoxy-4-acetyl-5-methoxy-phenyl)-(tetra-<i>O</i>-acetyl-β-D-glucopyranoside) 135650-52-1 C25H30O14
(3-acetoxy-4-acetyl-5-methoxy-phenyl)-(tetra-<i>O</i>-acetyl-β-D-glucopyranoside)
—— 1-(3,4-dimethoxy-6-methyl-2,5-benzoquinonyl)-2-(4-thiomorpholino-4-oxobutyl)-1,2,3,4-tetrahydronaphthalene 124524-20-5 C27H33NO5S
1-(3,4-dimethoxy-6-methyl-2,5-benzoquinonyl)-2-(4-thiomorpholino-4-oxobutyl)-1,2,3,4-tetrahydronaphthalene
—— (3aS,3bR,6aS,7aR)-1,5,5,6a-Tetramethyl-hexahydro-[1,3]dioxolo[4',5':3,4]cyclopenta[1,2-c]isoxazole 136030-59-6 C11H19NO3
(3aS,3bR,6aS,7aR)-1,5,5,6a-Tetramethyl-hexahydro-[1,3]dioxolo[4',5':3,4]cyclopenta[1,2-c]isoxazole
—— cyclohexylammonium 6-(1',2'-dihydroxyethyl)-4,5-dihydroxy-4,5:1',2'-di-O-isopropylidene-D-manno-1,2λ<sup>5</sup>-oxaphosphorinan-2-one-2-oxide 126874-13-3 C6H13N*C6H13O7P
cyclohexylammonium 6-(1',2'-dihydroxyethyl)-4,5-dihydroxy-4,5:1',2'-di-O-isopropylidene-D-manno-1,2λ<sup>5</sup>-oxaphosphorinan-2-one-2-oxide
—— (S)-1-{(S)-2-[(S)-2-(2-methoxyethylamino)propionylamino]-3-methylbutyryl}-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid (2,6-difluorophenyl)amide 1595279-23-4 C25H31F2N5O4
(S)-1-{(S)-2-[(S)-2-(2-methoxyethylamino)propionylamino]-3-methylbutyryl}-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid (2,6-difluorophenyl)amide
—— (3R,4R)-3-Hydroxy-3,4-diphenyl-4,5,6,7,8,9-hexahydro-3H-benzo[b]oxepin-2-one 143618-70-6 C22H22O3
(3R,4R)-3-Hydroxy-3,4-diphenyl-4,5,6,7,8,9-hexahydro-3H-benzo[b]oxepin-2-one
—— (2S,4S)-5-Oxo-4-[(R)-phenyl-(toluene-4-sulfonylamino)-methyl]-pyrrolidine-1,2-dicarboxylic acid 2-benzyl ester 1-tert-butyl ester 135347-22-7 C31H34N2O7S
(2S,4S)-5-Oxo-4-[(R)-phenyl-(toluene-4-sulfonylamino)-methyl]-pyrrolidine-1,2-dicarboxylic acid 2-benzyl ester 1-tert-butyl ester
—— —— 1263422-35-0 C21H22BrN5O2
—— —— 1263422-16-7 C29H32N6O3
—— —— 1220902-62-4 C30H35Cl2N3O5
—— N-(trans-3-(2-cyclopropyl-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl)-1,7-naphthyridin-2-amine 1452551-09-5 C21H20N6
N-(trans-3-(2-cyclopropyl-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl)-1,7-naphthyridin-2-amine
—— tert-butyl (2S)-2-({4-[3-(6-fluoro-3-methyl-1H-indazol-1-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrrolidine-1-carboxylate 1415731-49-5 C25H33FN6O3
tert-butyl (2S)-2-({4-[3-(6-fluoro-3-methyl-1H-indazol-1-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrrolidine-1-carboxylate
—— —— 1332710-90-3 C23H26FN5O3S
—— —— 1404378-23-9 C30H42N2O5
—— —— 1072438-27-7 C47H71N3O5
—— 1-(3-Phenethyl-pyridin-2-yl)-ethanone 14578-26-8 C15H15NO
1-(3-Phenethyl-pyridin-2-yl)-ethanone
—— (S)-N-(3-(3-(cyclopropanecarboxamido)isoquinolin-7-yl)-4-methylphenyl)tetrahydrofuran-2-carboxamide 1382843-44-8 C25H25N3O3
(S)-N-(3-(3-(cyclopropanecarboxamido)isoquinolin-7-yl)-4-methylphenyl)tetrahydrofuran-2-carboxamide
—— 5-cyclopropyl-N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-1,3-oxazole-4-carboxamide 1416311-02-8 C27H37N5O3
5-cyclopropyl-N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-1,3-oxazole-4-carboxamide
—— (4-isopropoxy-3-methoxyphenyl)(4-isopropoxy-3-methoxyspiro[chroman-2,4'-piperidine]-1'-yl)methanone 1394030-58-0 C28H37NO6
(4-isopropoxy-3-methoxyphenyl)(4-isopropoxy-3-methoxyspiro[chroman-2,4'-piperidine]-1'-yl)methanone
—— (5R,8S)-N-{1-[(cyclopropylsulfonyl)carbamoyl]cyclobutyl}-7-[(2S)-2-{[(2S)-2-({[(2S)-1-isopropylpiperidin-2-yl]carbonyl}amino)-3,3-dimethylbutanoyl]amino}-3,3-dimethylbutanoyl]-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide 1247710-14-0 C41H68N6O7S
(5R,8S)-N-{1-[(cyclopropylsulfonyl)carbamoyl]cyclobutyl}-7-[(2S)-2-{[(2S)-2-({[(2S)-1-isopropylpiperidin-2-yl]carbonyl}amino)-3,3-dimethylbutanoyl]amino}-3,3-dimethylbutanoyl]-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide
—— (S)-5-{4-[3-(4-hydroxybenzylamino)piperidin-1-yl]-6-propylpyrimidin-2-ylamino}-2-methylbenzonitrile 1394804-77-3 C27H32N6O
(S)-5-{4-[3-(4-hydroxybenzylamino)piperidin-1-yl]-6-propylpyrimidin-2-ylamino}-2-methylbenzonitrile
—— N'-(2-tert-butylphenyl)-N-diphenylphosphanyl-4-methylbenzenecarboximidamide 1313508-28-9 C30H31N2P
N'-(2-tert-butylphenyl)-N-diphenylphosphanyl-4-methylbenzenecarboximidamide
—— methyl (2S)-3-[(3,5-dihydroxybenzoyl)amino]-2-[[5-[2-(3-hydroxyphenyl)ethylcarbamoyl]-3-methylthiophene-2-carbonyl]amino]propanoate 1400663-13-9 C26H27N3O8S
methyl (2S)-3-[(3,5-dihydroxybenzoyl)amino]-2-[[5-[2-(3-hydroxyphenyl)ethylcarbamoyl]-3-methylthiophene-2-carbonyl]amino]propanoate
—— (R)-2-((S)-4-tert-Butoxycarbonyl-4-{4-[(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-benzoylamino}-butyrylamino)-pentanedioic acid di-tert-butyl ester 145817-21-6 C42H55N5O9
(R)-2-((S)-4-tert-Butoxycarbonyl-4-{4-[(2-methyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-benzoylamino}-butyrylamino)-pentanedioic acid di-tert-butyl ester
—— [1-[7-(4-Morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-yl]piperidin-4-yl]methanamine 1415789-70-6 C23H28N6O
[1-[7-(4-Morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-yl]piperidin-4-yl]methanamine
—— 2-(2,4-dioxo-1-p-tolyl-1,3-diaza-spiro[4.5]dec-3-yl)-N-[1-(2-trifluoromethyl-phenyl)propyl]-acetamide 1240788-94-6 C27H30F3N3O3
2-(2,4-dioxo-1-p-tolyl-1,3-diaza-spiro[4.5]dec-3-yl)-N-[1-(2-trifluoromethyl-phenyl)propyl]-acetamide
—— N-(5-bicyclo[2.2.1]heptanylmethyl)-2-[3-[3-fluoro-4-(trifluoromethyl)phenyl]propylsulfanyl]pyridine-3-carboxylic acid amide 1242641-22-0 C24H26F4N2OS
N-(5-bicyclo[2.2.1]heptanylmethyl)-2-[3-[3-fluoro-4-(trifluoromethyl)phenyl]propylsulfanyl]pyridine-3-carboxylic acid amide
—— 5-(5-ethyl-1H-pyrazol-3-yl)-4-methyl-2-thiophen-2-yl-1,3-thiazole 1232031-17-2 C13H13N3S2
5-(5-ethyl-1H-pyrazol-3-yl)-4-methyl-2-thiophen-2-yl-1,3-thiazole
—— 3-[[4-[(1S,2R)-1-(4-chlorophenyl)-1-[2-chloro-4-(trifluoromethyl)phenoxy]pentan-2-yl]benzoyl]amino]propanoic acid 1242062-56-1 C28H26Cl2F3NO4
3-[[4-[(1S,2R)-1-(4-chlorophenyl)-1-[2-chloro-4-(trifluoromethyl)phenoxy]pentan-2-yl]benzoyl]amino]propanoic acid
—— 1-(1H-indazol-4-yl)-3-(2-(3-methoxypropyl)-4-(trifluoromethyl)benzyl)urea 1235487-49-6 C20H21F3N4O2
1-(1H-indazol-4-yl)-3-(2-(3-methoxypropyl)-4-(trifluoromethyl)benzyl)urea
—— N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-5-methyl-1,3,4-thiadiazole-2-carboxamide 1416311-10-8 C24H34N6O2S
N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-5-methyl-1,3,4-thiadiazole-2-carboxamide
—— (R)-6-cyclopropyl-2-(3-cyclopropyl-4-(3,3,3-trifluoropropanoyl)piperazin-1-yl)-5-(quinoxalin-5-yl)nicotinonitrile 1416140-82-3 C27H25F3N6O
(R)-6-cyclopropyl-2-(3-cyclopropyl-4-(3,3,3-trifluoropropanoyl)piperazin-1-yl)-5-(quinoxalin-5-yl)nicotinonitrile
—— [2'-(1-amino-ethyl)-5'-(3-fluoro-pyridin-4-ylcarbamoyl)-biphenyl-3-yloxy]-acetic acid propyl ester 1333399-81-7 C25H26FN3O4
[2'-(1-amino-ethyl)-5'-(3-fluoro-pyridin-4-ylcarbamoyl)-biphenyl-3-yloxy]-acetic acid propyl ester
—— 1-(4-fluorophenyl)-4-methyl-2-((2,3,6-trifluorobenzyl)thio)-1H-imidazole-5-carboxylic acid 1416267-09-8 C18H12F4N2O2S
1-(4-fluorophenyl)-4-methyl-2-((2,3,6-trifluorobenzyl)thio)-1H-imidazole-5-carboxylic acid
—— 2'-(1-amino-ethyl)-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carboxylic acid pentyl ester 1333398-56-3 C26H29N3O3
2'-(1-amino-ethyl)-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carboxylic acid pentyl ester
—— N-[6-amino-5-(2,5-dichlorophenyl)pyridin-2-yl]isoxazole-3-carboxamide 1079400-75-1 C15H10Cl2N4O2
N-[6-amino-5-(2,5-dichlorophenyl)pyridin-2-yl]isoxazole-3-carboxamide
—— N8-[3-(trifluoromethyl)benzyl][1,2,4]triazolo[4,3-a]pyrazine-3,8-diamine 1313187-11-9 C13H11F3N6
N8-[3-(trifluoromethyl)benzyl][1,2,4]triazolo[4,3-a]pyrazine-3,8-diamine
—— N-((R)-5-((1R,3aS,7aR,E)-4-(2-((3R,5R)-3,5-dihydroxycyclohexylidene)ethylidene)-7a-methyl-octahydro-7H-inden-1-yl)hexyl)-2-hydroxyethanesulfonamide 1188931-70-5 C26H45NO5S
N-((R)-5-((1R,3aS,7aR,E)-4-(2-((3R,5R)-3,5-dihydroxycyclohexylidene)ethylidene)-7a-methyl-octahydro-7H-inden-1-yl)hexyl)-2-hydroxyethanesulfonamide
—— 4-cyano-6-methyl-pyridine-2-carboxylic acid (1-methyl-1H-pyrazol-3-yl)-amide 1242967-75-4 C12H11N5O
4-cyano-6-methyl-pyridine-2-carboxylic acid (1-methyl-1H-pyrazol-3-yl)-amide
—— 1-[3-(6-methoxy-2,3-dihydro-indol-1-yl)-propyl]-1H-pyrazol-4-ylamine 1394162-26-5 C15H20N4O
1-[3-(6-methoxy-2,3-dihydro-indol-1-yl)-propyl]-1H-pyrazol-4-ylamine
—— N-(cyclopentylmethyl)-N-methyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.5]octane-8-sulfonamide 1384874-36-5 C19H28N6O2S
N-(cyclopentylmethyl)-N-methyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.5]octane-8-sulfonamide
—— 2-chloro-5-((4-fluoropyridin-2-yl)oxy)benzoic acid 1394348-53-8 C12H7ClFNO3
2-chloro-5-((4-fluoropyridin-2-yl)oxy)benzoic acid
—— 3-({(1H-benzotriazol-5-ylcarbonyl)[1-(4-fluorophenyl)ethyl]amino}methyl)benzoic acid 1398583-68-0 C23H19FN4O3
3-({(1H-benzotriazol-5-ylcarbonyl)[1-(4-fluorophenyl)ethyl]amino}methyl)benzoic acid
—— N-(1-{4-[2-(2-fluoro-4-methoxy-phenoxy)-thiazol-5-yloxy]-phenyl}-ethyl)-acetamide 1384191-89-2 C20H19FN2O4S
N-(1-{4-[2-(2-fluoro-4-methoxy-phenoxy)-thiazol-5-yloxy]-phenyl}-ethyl)-acetamide
—— 1-[2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carbonyl]-piperidine-2-carboxylic acid methyl ester 1333399-62-4 C27H28N4O4
1-[2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carbonyl]-piperidine-2-carboxylic acid methyl ester
—— (S)-N-(1-{2-[(3-chloro-4-hydroxyphenyl)amino]-6-propylpyrimidin-4-yl}pyrrolidin-3-yl)acetamide 1394317-12-4 C19H24ClN5O2
(S)-N-(1-{2-[(3-chloro-4-hydroxyphenyl)amino]-6-propylpyrimidin-4-yl}pyrrolidin-3-yl)acetamide
—— 2-((3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid 1228558-29-9 C21H19ClN2O6
2-((3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
—— 1-(2,2-dimethylpropyl)-3-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)carbonyl]piperidin-3-yl}-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1416309-54-0 C22H30N6O2
1-(2,2-dimethylpropyl)-3-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)carbonyl]piperidin-3-yl}-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— tert-butyl 4-{5-[4-(trifluoromethyl)phenyl]benzo[d]oxazol-2-yl}piperidine-1-carboxylate 1415991-39-7 C24H25F3N2O3
tert-butyl 4-{5-[4-(trifluoromethyl)phenyl]benzo[d]oxazol-2-yl}piperidine-1-carboxylate