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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid (2-{cyclopropyl-[2-cyclopropyl-5-(3-methoxy-phenyl)-thiazole-4-carbonyl]-amino}-ethyl)-amide 1117694-73-1 C26H27N5O3S2
6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid (2-{cyclopropyl-[2-cyclopropyl-5-(3-methoxy-phenyl)-thiazole-4-carbonyl]-amino}-ethyl)-amide
—— N-[2-hydroxy-1-(1H-indol-3-ylmethyl)-1-methyl-ethyl]-5-p-tolylethynyl-2-trifluoromethoxy-benzamide 1117834-18-0 C29H25F3N2O3
N-[2-hydroxy-1-(1H-indol-3-ylmethyl)-1-methyl-ethyl]-5-p-tolylethynyl-2-trifluoromethoxy-benzamide
—— (6aR,7S,10aS)-1,4-difluoro-7-methyl-7-(2-methylsulfonylethyl)-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6a,8,9,10-tetrahydro-6H-benzo[c]chromene 1100362-31-9 C24H25F5O5S2
(6aR,7S,10aS)-1,4-difluoro-7-methyl-7-(2-methylsulfonylethyl)-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6a,8,9,10-tetrahydro-6H-benzo[c]chromene
—— 4-methyl-2-[(E)-2-(3-methyl-5-pyridin-2-yl-3H-[1,2,3]triazol-4-yl)-vinyl]-thiazole-5-carboxylic acid (tetrahydro-pyran-4-yl)-amide 1374645-62-1 C20H22N6O2S
4-methyl-2-[(E)-2-(3-methyl-5-pyridin-2-yl-3H-[1,2,3]triazol-4-yl)-vinyl]-thiazole-5-carboxylic acid (tetrahydro-pyran-4-yl)-amide
—— (E)-2-Cyano-3-(3-fluoro-phenyl)-thioacrylamide 103868-11-7 C10H7FN2S
(E)-2-Cyano-3-(3-fluoro-phenyl)-thioacrylamide
—— N-(1-benzylpiperidine-4-yl)-2-(5,6-dichloropyridazine-4-ylamino)-N-methylacetamide 1080651-46-2 C19H23Cl2N5O
N-(1-benzylpiperidine-4-yl)-2-(5,6-dichloropyridazine-4-ylamino)-N-methylacetamide
—— 2-(3-amino-5-bromoindazol-1-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide 1023295-50-2 C21H20BrN7OS
2-(3-amino-5-bromoindazol-1-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
—— 3-(2,4,5-trifluoro-phenyl)-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole 1231908-35-2 C12H9F3N2O
3-(2,4,5-trifluoro-phenyl)-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole
—— (S)-4-[2-(3,5-bis-trifluoromethyl-phenyl)ethyl]-4,5-dihydrooxazol-2-ylamine 1043492-95-0 C13H12F6N2O
(S)-4-[2-(3,5-bis-trifluoromethyl-phenyl)ethyl]-4,5-dihydrooxazol-2-ylamine
—— (2S,4S)-1-(2-cyano-pyrimidin-4-yl)-4-(2-trifluoromethyl-benzenesulfonyl)-pyrrolidine-2-carboxylic acid 4-fluoro-benzylamide 1374674-85-7 C24H19F4N5O3S
(2S,4S)-1-(2-cyano-pyrimidin-4-yl)-4-(2-trifluoromethyl-benzenesulfonyl)-pyrrolidine-2-carboxylic acid 4-fluoro-benzylamide
—— 2-[5-(2-amino-pyrimidin-5-yl)-1-tert-butyl-1H-benzoimidazol-2-yl]-N-pyridin-3-yl-benzamide 1374150-25-0 C27H25N7O
2-[5-(2-amino-pyrimidin-5-yl)-1-tert-butyl-1H-benzoimidazol-2-yl]-N-pyridin-3-yl-benzamide
—— ethyl 5-(4-ethyl-phenyl)-1-oxy-6-phenyl-pyridine-2-carboxylate 1011467-32-5 C22H21NO3
ethyl 5-(4-ethyl-phenyl)-1-oxy-6-phenyl-pyridine-2-carboxylate
—— 4'-[(5-chloroquinoxalin-2-yl)oxy]-N-methylbiphenyl-3-sulfonamide 1225653-09-7 C21H16ClN3O3S
4'-[(5-chloroquinoxalin-2-yl)oxy]-N-methylbiphenyl-3-sulfonamide
—— (3R,4R)-3-[2-(4-fluorophenyl)ethylthio]-4-(4-hydroxyphenyl)-1-[4-(pyridin-3-yl)phenyl]azetidin-2-one 1056207-03-4 C28H23FN2O2S
(3R,4R)-3-[2-(4-fluorophenyl)ethylthio]-4-(4-hydroxyphenyl)-1-[4-(pyridin-3-yl)phenyl]azetidin-2-one
—— {4-[4-(4,4-difluoro-piperidine-1-sulfonyl)-phenoxy]-6-fluoro-3-methyl-naphthalen-2-yl}-acetic acid 1227384-49-7 C24H22F3NO5S
{4-[4-(4,4-difluoro-piperidine-1-sulfonyl)-phenoxy]-6-fluoro-3-methyl-naphthalen-2-yl}-acetic acid
—— (R)-1-[1-(acenaphthen-1-yl)piperidin-4-yl]-3-(2-methoxyethyl)-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1055322-85-4 C26H28N4O2
(R)-1-[1-(acenaphthen-1-yl)piperidin-4-yl]-3-(2-methoxyethyl)-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— ethyl 2-(8-(benzyloxy)quinolin-2-yl)-1-(3-butylureido)cyclopropanecarboxylate 1358916-64-9 C27H31N3O4
ethyl 2-(8-(benzyloxy)quinolin-2-yl)-1-(3-butylureido)cyclopropanecarboxylate
—— (+/-)-(8-chloro-3-hydroxyquinoxalin-2-yl)[2-(3-chlorobenzyl)pyrrolidin-1-yl]methanone 1374848-18-6 C20H17Cl2N3O2
(+/-)-(8-chloro-3-hydroxyquinoxalin-2-yl)[2-(3-chlorobenzyl)pyrrolidin-1-yl]methanone
—— 2-methyl-4-(4-methylpiperazinyl)-8-(trifluoromethyl)pyrazolo[3,4-c]quinoline 1217302-60-7 C17H18F3N5
2-methyl-4-(4-methylpiperazinyl)-8-(trifluoromethyl)pyrazolo[3,4-c]quinoline
—— 4-phenylbenzoyloxymethyl difluoromethanesulfonic acid sodium salt 1225186-03-7 C15H11F2O5S*Na
4-phenylbenzoyloxymethyl difluoromethanesulfonic acid sodium salt
—— {3-benzo[1,3]dioxol-5-yl-1-[1-(2-chloro-benzyl)-1H-tetrazol-5-yl]-2-methyl-propyl}-(1H-benzoimidazol-5-yl)-amine 1025368-12-0 C26H24ClN7O2
{3-benzo[1,3]dioxol-5-yl-1-[1-(2-chloro-benzyl)-1H-tetrazol-5-yl]-2-methyl-propyl}-(1H-benzoimidazol-5-yl)-amine
—— [6-fluoro-4-(4-methanesulfonyl-2-methyl-phenoxy)-3-methyl-naphthalen-2-yl]-acetic acid 1227384-03-3 C21H19FO5S
[6-fluoro-4-(4-methanesulfonyl-2-methyl-phenoxy)-3-methyl-naphthalen-2-yl]-acetic acid
—— 2-{3-[1-(3-bromoacenaphthen-1-yl)piperidin-4-yl]-2,3-dihydro-2-oxo-benzimidazol-1-yl}-N-methylacetamide 1055322-61-6 C27H27BrN4O2
2-{3-[1-(3-bromoacenaphthen-1-yl)piperidin-4-yl]-2,3-dihydro-2-oxo-benzimidazol-1-yl}-N-methylacetamide
—— (1H-benzoimidazol-5-yl)-{(3-fluoro-4-methoxy-phenyl)-[1-(tetrahydro-furan-2-ylmethyl)-1H-tetrazol-5-yl]-methyl}-amine 1025369-20-3 C21H22FN7O2
(1H-benzoimidazol-5-yl)-{(3-fluoro-4-methoxy-phenyl)-[1-(tetrahydro-furan-2-ylmethyl)-1H-tetrazol-5-yl]-methyl}-amine
—— N-(1-benzylpiperidine-4-yl)-2-(2-chloro-5-methylpyrimidine-4-ylamino)-N-methylacetamide 1080651-13-3 C20H26ClN5O
N-(1-benzylpiperidine-4-yl)-2-(2-chloro-5-methylpyrimidine-4-ylamino)-N-methylacetamide
—— (RS)-4-(5-chloro-2-trifluoromethylphenyl)-4,5-dihydrooxazol-2-ylamine 1043494-62-7 C10H8ClF3N2O
(RS)-4-(5-chloro-2-trifluoromethylphenyl)-4,5-dihydrooxazol-2-ylamine
—— (1H-benzoimidazol-5-yl)-{(3-bromo-4-methoxy-phenyl)-[1-(tetrahydro-furan-2-ylmethyl)-1H-tetrazol-5-yl]-methyl}-amine 1025368-04-0 C21H22BrN7O2
(1H-benzoimidazol-5-yl)-{(3-bromo-4-methoxy-phenyl)-[1-(tetrahydro-furan-2-ylmethyl)-1H-tetrazol-5-yl]-methyl}-amine
—— 8-Bromo-5-fluorochroman 1523009-39-3 C9H8BrFO
8-Bromo-5-fluorochroman
—— 1-(2-chloromethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-3-phenyl-propan-1-one-(2,4-dinitro-phenylhydrazone) 119640-90-3 C24H21ClN4O6
1-(2-chloromethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-3-phenyl-propan-1-one-(2,4-dinitro-phenylhydrazone)
—— 6,7-dimethyl-1'-[(2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)carbonyl]spiro[chromene-2,4'-piperidin]-4(3H)-one 1031415-04-9 C25H26N2O4
6,7-dimethyl-1'-[(2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)carbonyl]spiro[chromene-2,4'-piperidin]-4(3H)-one
—— tert-butyl N-[(2R,3S)-3-hydroxy-1-[methoxy(methyl)amino]-1-oxobutan-2-yl]carbamate 1301684-81-0 C11H22N2O5
tert-butyl N-[(2R,3S)-3-hydroxy-1-[methoxy(methyl)amino]-1-oxobutan-2-yl]carbamate
—— 7-[2-(6-Bromo-5-chloro-2-oxo-benzooxazol-3-yl)-acetylamino]-3-methyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 130970-61-5 C17H13BrClN3O6S
7-[2-(6-Bromo-5-chloro-2-oxo-benzooxazol-3-yl)-acetylamino]-3-methyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 2,1'-dinitro-[1,2']binaphthyl 112552-52-0 C20H12N2O4
2,1'-dinitro-[1,2']binaphthyl
—— Ethyl 2-(2,2,2-Trichloro-tert-butoxycarbonylamino)-2-hydroxy-3,3,3-trifluoropropionate 126535-85-1 C10H13Cl3F3NO5
Ethyl 2-(2,2,2-Trichloro-tert-butoxycarbonylamino)-2-hydroxy-3,3,3-trifluoropropionate
—— 2-(4-Bromomethyl-2,5-diphenyl-thiophen-3-ylmethylene)-malonic acid diethyl ester 162052-82-6 C25H23BrO4S
2-(4-Bromomethyl-2,5-diphenyl-thiophen-3-ylmethylene)-malonic acid diethyl ester
—— ethyl 2-(tert-butoxy)-2-[4-(isoquinolin-4-yl)-2,5-dimethylthiophen-3-yl]acetate 1402144-96-0 C23H27NO3S
ethyl 2-(tert-butoxy)-2-[4-(isoquinolin-4-yl)-2,5-dimethylthiophen-3-yl]acetate
—— ethyl 2-(tert-butoxy)-2-[4-(1H-inden-2-yl)-2,5-dimethylthiophen-3-yl]acetate 1402144-98-2 C23H28O3S
ethyl 2-(tert-butoxy)-2-[4-(1H-inden-2-yl)-2,5-dimethylthiophen-3-yl]acetate
—— Tert-butyl 4-[3-(2-methoxyethoxy)-6-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)pyridin-2-yl]piperazine-1-carboxylate 1312464-96-2 C31H45N3O4
Tert-butyl 4-[3-(2-methoxyethoxy)-6-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)pyridin-2-yl]piperazine-1-carboxylate
—— {4-[2-({3-[(dimethylamino)carbonyl]phenyl}sulfonyl)benzyl]-5-methyl-3-phenyl-1H-pyrazol-1-yl}acetic acid 1559061-53-8 C28H27N3O5S
{4-[2-({3-[(dimethylamino)carbonyl]phenyl}sulfonyl)benzyl]-5-methyl-3-phenyl-1H-pyrazol-1-yl}acetic acid
—— (S)-2-(3-(1,3-dimethyl-1H-pyrazol-5-yl)-1,4-dimethyl-1H-pyrazolo[3,4-b]pyridin-6-yloxy)-N-(1-p-tolylethyl)acetamide 1312946-58-9 C24H28N6O2
(S)-2-(3-(1,3-dimethyl-1H-pyrazol-5-yl)-1,4-dimethyl-1H-pyrazolo[3,4-b]pyridin-6-yloxy)-N-(1-p-tolylethyl)acetamide
—— N-tert-butoxycarbonyl-L-tryptophyl-γ-aminobutyryl-L-asparaginic acid α-amide 129280-49-5 C24H33N5O7
N-tert-butoxycarbonyl-L-tryptophyl-γ-aminobutyryl-L-asparaginic acid α-amide
—— (E)-N-(3-((4-hydroxybutyl)amino)-3-oxopropyl)-4-(2-(3-methoxybenzylidene)hydrazinecarbonyl)benzamide 1292823-96-1 C23H28N4O5
(E)-N-(3-((4-hydroxybutyl)amino)-3-oxopropyl)-4-(2-(3-methoxybenzylidene)hydrazinecarbonyl)benzamide
—— 11-Chloro-12-methoxy-6H-dibenzo[c,h]chromene-2,8-diol 1026709-73-8 C18H13ClO4
11-Chloro-12-methoxy-6H-dibenzo[c,h]chromene-2,8-diol
—— 1-[3-fluoro-4-(hydroxymethyl)phenyl]-3-[[2-(4-fluoro-3-methylphenyl)-5-(trifluoromethyl)-2H-pyrazol-3-yl]methyl]urea 1402582-79-9 C20H17F5N4O2
1-[3-fluoro-4-(hydroxymethyl)phenyl]-3-[[2-(4-fluoro-3-methylphenyl)-5-(trifluoromethyl)-2H-pyrazol-3-yl]methyl]urea
—— 1-((6-chloropyridin-3-yl)methyl)-8-nitro-1,2,3,4-tetrahydrothiazolo[3,4-a]pyrimidin-6-imine 1408310-73-5 C12H12ClN5O2S
1-((6-chloropyridin-3-yl)methyl)-8-nitro-1,2,3,4-tetrahydrothiazolo[3,4-a]pyrimidin-6-imine
—— ethyl (E)-3-(4-((E)-1-(4-cyano-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-5-yl)-2-cyclobutyl-2-phenylvinyl)phenyl)acrylate 1459254-59-1 C36H35N3O3
ethyl (E)-3-(4-((E)-1-(4-cyano-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-5-yl)-2-cyclobutyl-2-phenylvinyl)phenyl)acrylate
—— (R)-hexahydro-5-ethyl-2H-azepin-2-one 126694-36-8 C8H15NO
(R)-hexahydro-5-ethyl-2H-azepin-2-one
—— Tert-butyl 4-[5-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3,4-thiadiazol-2-yl]piperidine-1-carboxylate 1314087-83-6 C26H37N3O2S
Tert-butyl 4-[5-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3,4-thiadiazol-2-yl]piperidine-1-carboxylate
—— (E)-benzhydryl 5-((3aS,4R,5R,6aS)-5-hydroxy-4-((3S,E)-3-hydroxy-4-methyloct-1-en-6-yn-1-yl)hexahydropentalen-2(1H)-ylidene)pentanoate 1259542-03-4 C35H42O4
(E)-benzhydryl 5-((3aS,4R,5R,6aS)-5-hydroxy-4-((3S,E)-3-hydroxy-4-methyloct-1-en-6-yn-1-yl)hexahydropentalen-2(1H)-ylidene)pentanoate
—— Tert-butyl 8-bromo-4,10-dihydrotriazolo[5,1-c][1,4]benzodiazepine-5-carboxylate 1007309-53-6 C15H17BrN4O2
Tert-butyl 8-bromo-4,10-dihydrotriazolo[5,1-c][1,4]benzodiazepine-5-carboxylate