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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-6,6-difluoro-5-[2-fluoro-5-(tetrahydro-pyran-4-yl)-phenyl]-5,7,7-trimethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine 1401241-63-1 C19H25F3N2O2
(R)-6,6-difluoro-5-[2-fluoro-5-(tetrahydro-pyran-4-yl)-phenyl]-5,7,7-trimethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine
—— O2-{(3R)-1-[(cyclohexyloxy)carbonyl]pyrrolidin-3-yl}1-(N-tert-butylamino)diazen-1-ium-1,2-diolate 1398743-48-0 C15H28N4O4
O2-{(3R)-1-[(cyclohexyloxy)carbonyl]pyrrolidin-3-yl}1-(N-tert-butylamino)diazen-1-ium-1,2-diolate
—— 3-(4-(2-(4-(2-hydroxy-3-(prop-2-ynyloxy)propoxy)phenyl)propan-2-yl)phenoxy)propane-1,2-diol 1402419-05-9 C24H30O6
3-(4-(2-(4-(2-hydroxy-3-(prop-2-ynyloxy)propoxy)phenyl)propan-2-yl)phenoxy)propane-1,2-diol
—— S-[2-[[(2R,3R,4R,5R)-5-(2-amino-6-chloropurin-9-yl)-3,4-dihydroxy-4-methyloxolan-2-yl]methoxy-(propan-2-ylamino)phosphoryl]oxyethyl] 3-hydroxy-2,2-dimethylpropanethioate 1401314-27-9 C21H34ClN6O8PS
S-[2-[[(2R,3R,4R,5R)-5-(2-amino-6-chloropurin-9-yl)-3,4-dihydroxy-4-methyloxolan-2-yl]methoxy-(propan-2-ylamino)phosphoryl]oxyethyl] 3-hydroxy-2,2-dimethylpropanethioate
—— 1-[4-(2-cyanophenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid 1401320-84-0 C21H13N3O3
1-[4-(2-cyanophenoxy)phenyl]-1H-benzimidazole-6-carboxylic acid
—— 1-methanesulfonyl-3-[1-(6-morpholin-4-yl-pyridin-2-yl)-methylidene]-5-phenyl-piperidine-2,4-dione 1096166-41-4 C22H23N3O5S
1-methanesulfonyl-3-[1-(6-morpholin-4-yl-pyridin-2-yl)-methylidene]-5-phenyl-piperidine-2,4-dione
—— 3-fluoro-N6-((1S)-1-(5-fluoropyrimidin-2-yl)ethyl)-N2-(5-isopropoxy-1H-pyrazol-3-yl)-5-nitropyridine-2,6-diamine 1073149-14-0 C17H18F2N8O3
3-fluoro-N6-((1S)-1-(5-fluoropyrimidin-2-yl)ethyl)-N2-(5-isopropoxy-1H-pyrazol-3-yl)-5-nitropyridine-2,6-diamine
—— [(S)-1-(3-amino-1H-indazol-6-ylcarbamoyl)-2-phenylethyl]carbamic acid tert-butyl ester 1094106-97-4 C21H25N5O3
[(S)-1-(3-amino-1H-indazol-6-ylcarbamoyl)-2-phenylethyl]carbamic acid tert-butyl ester
—— dimethyl 2-(3-(2-(tert-butoxycarbonyl(methyl)amino)ethyl)phenyl)malonate 1093938-88-5 C19H27NO6
dimethyl 2-(3-(2-(tert-butoxycarbonyl(methyl)amino)ethyl)phenyl)malonate
—— 2-[(5-phenoxy-2-phenyl-1H-indole-7-yl)amino]-acetic acid 1120333-51-8 C22H18N2O3
2-[(5-phenoxy-2-phenyl-1H-indole-7-yl)amino]-acetic acid
—— N-(3-oxo-2-quinolin-6-yl-1H-isoindol-5-yl)propanamide 1402890-38-3 C20H17N3O2
N-(3-oxo-2-quinolin-6-yl-1H-isoindol-5-yl)propanamide
—— [5-amino-1-(2-methyl-1H-benzimidazol-5-yl)-1H-pyrazol-4-yl]-(5-fluoro-1H-indol-2-yl)-methanone 1265230-84-9 C20H15FN6O
[5-amino-1-(2-methyl-1H-benzimidazol-5-yl)-1H-pyrazol-4-yl]-(5-fluoro-1H-indol-2-yl)-methanone
—— (3-{[(5-{3-fluoro-4-[3-(2-methylphenyl)propyl]phenyl}quinolin-8-yl)methyl]amino}propyl)phosphonic acid 1403379-67-8 C29H32FN2O3P
(3-{[(5-{3-fluoro-4-[3-(2-methylphenyl)propyl]phenyl}quinolin-8-yl)methyl]amino}propyl)phosphonic acid
—— diethyl 4-(3'-cyanobiphenyl-2-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate 1099641-01-6 C26H26N2O4
diethyl 4-(3'-cyanobiphenyl-2-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate
—— 1-(4-fluoro-benzyl)-3,3-dimethyl-5-[1-(6-morpholin-4-yl-pyridin-2-yl)-methylidene]-piperidin-4-one 1096165-90-0 C24H28FN3O2
1-(4-fluoro-benzyl)-3,3-dimethyl-5-[1-(6-morpholin-4-yl-pyridin-2-yl)-methylidene]-piperidin-4-one
—— 1-cyclopropyl-3,3-dimethyl-5-[1-pyridin-2-yl-methylidene]-piperidin-4-one 1096165-65-9 C16H20N2O
1-cyclopropyl-3,3-dimethyl-5-[1-pyridin-2-yl-methylidene]-piperidin-4-one
—— Ethyl (4RS,5SR)-5-Isopropyl-2-oxooxazolidine-4-carboxylate 135524-14-0 C9H15NO4
Ethyl (4RS,5SR)-5-Isopropyl-2-oxooxazolidine-4-carboxylate
—— 5-fluoromethoxy-pyridine-2-carboxylic acid [3-((4R,5R)-2-amino-5-fluoro-4-methyl-5,6-dihydro-4H-[1,3]oxazin-4-yl)-4-fluoro-phenyl]-amide 1402412-34-3 C18H17F3N4O3
5-fluoromethoxy-pyridine-2-carboxylic acid [3-((4R,5R)-2-amino-5-fluoro-4-methyl-5,6-dihydro-4H-[1,3]oxazin-4-yl)-4-fluoro-phenyl]-amide
—— N2-[2-(7-methoxy-1H-indol-3-yl)ethyl]-N4-(2-methyl-1H-indol-5-yl)pyrimidine-2,4-diamine 1400890-23-4 C24H24N6O
N2-[2-(7-methoxy-1H-indol-3-yl)ethyl]-N4-(2-methyl-1H-indol-5-yl)pyrimidine-2,4-diamine
—— 2-{3-[2-(tetrahydropyran-4-ylamino)pyrimidin-4-yl]imidazo[1,2-a]pyrazin-8-ylamino}ethanol 1400669-77-3 C17H21N7O2
2-{3-[2-(tetrahydropyran-4-ylamino)pyrimidin-4-yl]imidazo[1,2-a]pyrazin-8-ylamino}ethanol
—— N-(5-{3-[(1-{[4-(methyloxy)phenyl]sulfonyl}-4-piperidinyl)amino]-6-quinoxalinyl}-3-pyridinyl)benzenesulfonamide 1083322-24-0 C31H30N6O5S2
N-(5-{3-[(1-{[4-(methyloxy)phenyl]sulfonyl}-4-piperidinyl)amino]-6-quinoxalinyl}-3-pyridinyl)benzenesulfonamide
—— 5-hydroxy-2,6-dimethyl-4-[5-methyl-3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl]-3(2H)-pyridazinone 1164164-04-8 C17H15F3N4O2
5-hydroxy-2,6-dimethyl-4-[5-methyl-3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl]-3(2H)-pyridazinone
—— [3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 4-ethoxybenzoate 1403240-48-1 C28H28N4O4
[3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 4-ethoxybenzoate
—— (3-chloro-4-(2-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridin-6-ylamino)phenyl)(3-methoxyazetidin-1-yl)methanone 1400286-03-4 C22H21ClN6O2
(3-chloro-4-(2-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridin-6-ylamino)phenyl)(3-methoxyazetidin-1-yl)methanone
—— 4-[3-(4-bromophenyl)-5-methyl-1H-pyrazol-1-yl]-5-methoxy-2-(tetrahydro-2H-pyran-2-yl)-3(2H)-pyridazinone 1164166-20-4 C20H21BrN4O3
4-[3-(4-bromophenyl)-5-methyl-1H-pyrazol-1-yl]-5-methoxy-2-(tetrahydro-2H-pyran-2-yl)-3(2H)-pyridazinone
—— N-{1-[(1-ethyl-piperidin-4-ylmethyl)-carbamoyl]-1-methyl-ethyl}-4-(2-phenoxy-phenylsulfamoyl)-benzamide 1021523-60-3 C31H38N4O5S
N-{1-[(1-ethyl-piperidin-4-ylmethyl)-carbamoyl]-1-methyl-ethyl}-4-(2-phenoxy-phenylsulfamoyl)-benzamide
—— 1-{4-[(3S)-2,3-dihydro[1,4]dioxino[2,3-b]pyridin-3-yl]benzyl}-N-(2-hydroxyethyl)piperidine-4-carboxamide 1400795-67-6 C22H27N3O4
1-{4-[(3S)-2,3-dihydro[1,4]dioxino[2,3-b]pyridin-3-yl]benzyl}-N-(2-hydroxyethyl)piperidine-4-carboxamide
—— 2-fluoro-5-{[6-oxo-4-(trifluoromethyl)-1,6-dihydropyridazin-3-yl]methyl}-benzoic acid 1154868-51-5 C13H8F4N2O3
2-fluoro-5-{[6-oxo-4-(trifluoromethyl)-1,6-dihydropyridazin-3-yl]methyl}-benzoic acid
—— [1-methyl-6-(4-methyl-5-methylaminopyridin-2-yloxy)-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone 1150460-61-9 C30H32F3N5O3
[1-methyl-6-(4-methyl-5-methylaminopyridin-2-yloxy)-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone
—— N-{2-[4'-(2-butyl-4-chloro-5-hydroxymethylimidazol-1-ylmethyl)biphenyl-2-sulfonylamino]-2-oxoethyl}-2-mercaptomethyl-3-methylbutyramide 1192346-23-8 C29H37ClN4O5S2
N-{2-[4'-(2-butyl-4-chloro-5-hydroxymethylimidazol-1-ylmethyl)biphenyl-2-sulfonylamino]-2-oxoethyl}-2-mercaptomethyl-3-methylbutyramide
—— (4-iodophenyl) (4S)-4-cyano-4-[3-methoxy-2-(methoxymethoxy)phenyl]-5-oxohexanoate 1334171-11-7 C22H22INO6
(4-iodophenyl) (4S)-4-cyano-4-[3-methoxy-2-(methoxymethoxy)phenyl]-5-oxohexanoate
—— 4-{[[(2,2-dimethyl-2,3-dihydro-1H-inden-5-yl)methyl](4-methylisoquinolin-3-yl)amino]sulfonyl}benzoic acid 1400699-16-2 C29H28N2O4S
4-{[[(2,2-dimethyl-2,3-dihydro-1H-inden-5-yl)methyl](4-methylisoquinolin-3-yl)amino]sulfonyl}benzoic acid
—— (4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-4a,6a-dimethyl-2-oxo-8-(2-phenoxy-ethyl)-2,4a,4b,5,6,6a,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-aza-pentaleno[2,1-a]phenanthrene-6b-carbothioic acid S-fluoromethyl ester 1400571-70-1 C30H34F3NO5S
(4aS,4bR,5S,6aS,6bR,9aS,10aS,10bS,12S)-4b,12-difluoro-5-hydroxy-4a,6a-dimethyl-2-oxo-8-(2-phenoxy-ethyl)-2,4a,4b,5,6,6a,8,9,9a,10,10a,10b,11,12-tetradecahydro-7-oxa-8-aza-pentaleno[2,1-a]phenanthrene-6b-carbothioic acid S-fluoromethyl ester
—— 2-[2-fluoro-4-[2-[(1S,2R)-2-[1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-1-[2-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl]ethanone 1402553-80-3 C29H35F4N7O3
2-[2-fluoro-4-[2-[(1S,2R)-2-[1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-1-[2-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl]ethanone
—— 1-(4-(4-(2-(1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridin-6-ylamino)phenyl)piperazin-1-yl)ethanone 1400286-30-7 C22H23N7O
1-(4-(4-(2-(1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridin-6-ylamino)phenyl)piperazin-1-yl)ethanone
—— [(3S,5R,8R,9S,10S,13R,14S,17R)-14-hydroxy-10,13-dimethyl-17-(6-oxopyran-3-yl)-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta[a]phenanthren-3-yl] imidazolidine-1-carboxylate 1385012-00-9 C28H40N2O5
[(3S,5R,8R,9S,10S,13R,14S,17R)-14-hydroxy-10,13-dimethyl-17-(6-oxopyran-3-yl)-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta[a]phenanthren-3-yl] imidazolidine-1-carboxylate
—— [(3R)-1-{4-[(2S)-2,3-dihydro-1,4-benzodioxin-2-yl]benzyl}piperidin-3-yl]acetic acid 1400796-21-5 C22H25NO4
[(3R)-1-{4-[(2S)-2,3-dihydro-1,4-benzodioxin-2-yl]benzyl}piperidin-3-yl]acetic acid
—— {methyl-[4-(2-phenoxy-phenylsulfamoyl)-benzoyl]-amino}-acetic acid 1021522-83-7 C22H20N2O6S
{methyl-[4-(2-phenoxy-phenylsulfamoyl)-benzoyl]-amino}-acetic acid
—— ethyl 3-[4-(6-methoxycarbonylmethyl-10H-9-oxa-3-thiabenzo[f]azulen-4-ylidene)piperidin-1-yl]propionate hydrochloride 1176738-82-1 C25H29NO5S*ClH
ethyl 3-[4-(6-methoxycarbonylmethyl-10H-9-oxa-3-thiabenzo[f]azulen-4-ylidene)piperidin-1-yl]propionate hydrochloride
—— (S)-3-{2-ethyl-4-[5-(2-isobutylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-6-methyl-phenoxy}-propane-1,2-diol 1150645-91-2 C23H31N5O4
(S)-3-{2-ethyl-4-[5-(2-isobutylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-6-methyl-phenoxy}-propane-1,2-diol
—— N-{4-[3-(4-chloro-phenyl)-5-trifluoromethyl-4,5-dihydro-isoxazol-5-yl]-2,6-dimethyl-phenyl}-4-cyano-3-(4-fluoro-benzoylamino)-benzamide 1146469-33-1 C33H23ClF4N4O3
N-{4-[3-(4-chloro-phenyl)-5-trifluoromethyl-4,5-dihydro-isoxazol-5-yl]-2,6-dimethyl-phenyl}-4-cyano-3-(4-fluoro-benzoylamino)-benzamide
—— 3-(7-(2-(trifluoromethyl)phenyl-sulfonamido)-1H-indol-1-yl)propionic acid 1239711-42-2 C18H15F3N2O4S
3-(7-(2-(trifluoromethyl)phenyl-sulfonamido)-1H-indol-1-yl)propionic acid
—— [5-(5-aminopyridin-2-yloxy)-1-methyl-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone 1150743-51-3 C28H28F3N5O3
[5-(5-aminopyridin-2-yloxy)-1-methyl-1H-indol-2-yl]{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazin-1-yl}methanone
—— 4-{1-methyl-6-[5-(4-trifluoromethoxybenzoylamino)pyridin-2-yloxy]-1H-indole-2-carbonyl}piperazine-1-carboxylic acid tert-butyl ester 1150745-13-3 C32H32F3N5O6
4-{1-methyl-6-[5-(4-trifluoromethoxybenzoylamino)pyridin-2-yloxy]-1H-indole-2-carbonyl}piperazine-1-carboxylic acid tert-butyl ester
—— 2-(4-Fluorophenyl)-5-[2-(methylamino)-4-thiazolyl]-3-[4-(methylsulfonyl)phenyl]thiophene 140403-85-6 C21H17FN2O2S3
2-(4-Fluorophenyl)-5-[2-(methylamino)-4-thiazolyl]-3-[4-(methylsulfonyl)phenyl]thiophene
—— N-(2-chloro-4-fluorophenyl)-5-fluoro-4-imino-3-methyl-2-oxopyrimidine-1-carboxamide 1616685-23-4 C12H9ClF2N4O2
N-(2-chloro-4-fluorophenyl)-5-fluoro-4-imino-3-methyl-2-oxopyrimidine-1-carboxamide
—— 2-[2-(5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl]-6-fluoro-8-methylquinoline 1445746-00-8 C19H18FN5
2-[2-(5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl]-6-fluoro-8-methylquinoline
—— —— 1622254-25-4 C19H20O
—— 4-[(1R,3S)-3-bromomethyl-2,2-dimethylcyclopropyl]butan-2-one 1422560-69-7 C10H17BrO
4-[(1R,3S)-3-bromomethyl-2,2-dimethylcyclopropyl]butan-2-one
—— N,N-dimethyl-9H-pyrido[3,4-b]indole-9-carboxamide 1613335-90-2 C14H13N3O
N,N-dimethyl-9H-pyrido[3,4-b]indole-9-carboxamide