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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-{(1RS,2RS)-2-(4-Chlorophenyl)-3-(4-fluorophenyl)-1-methylpropyl}carbamoylmethylsuccinic acid 162036-88-6 C22H23ClFNO5
N-{(1RS,2RS)-2-(4-Chlorophenyl)-3-(4-fluorophenyl)-1-methylpropyl}carbamoylmethylsuccinic acid
—— 3-methyl-1-phenyl-6-(1-(piperidine-4-carbonyl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one hydrochloride 1345405-07-3 C23H28N6O2*ClH
3-methyl-1-phenyl-6-(1-(piperidine-4-carbonyl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one hydrochloride
—— 8-(4-cyanophenyl)-2-cyclopropylcarbonylamino-7-hydroxy-6-[2-methyl-5-N-(3-trifluoromethylphenyl)carbamoylphenyl]quinazoline 1191931-53-9 C34H24F3N5O3
8-(4-cyanophenyl)-2-cyclopropylcarbonylamino-7-hydroxy-6-[2-methyl-5-N-(3-trifluoromethylphenyl)carbamoylphenyl]quinazoline
—— tert-butyl 4-((6-(4-((2,2-dioxido-1,3,2-dioxathiolan-4-yl)methyl)phenoxy)-5-methylpyrimidin-4-yl)oxy)piperidine-1-carboxylate 1258604-11-3 C24H31N3O8S
tert-butyl 4-((6-(4-((2,2-dioxido-1,3,2-dioxathiolan-4-yl)methyl)phenoxy)-5-methylpyrimidin-4-yl)oxy)piperidine-1-carboxylate
—— (S)-(4Z,17Z)-4-hydroxymethyl-1-trimethylsilyl-3-triethylsilyloxy-4,17-docosadien-1-yne 1256266-68-8 C32H62O2Si2
(S)-(4Z,17Z)-4-hydroxymethyl-1-trimethylsilyl-3-triethylsilyloxy-4,17-docosadien-1-yne
—— 2-chloro-N,6-dimethyl-N-[[7-(3-pyridin-4-yl-3,9-diazaspiro[5.5]undecane-9-carbonyl)-1H-benzoimidazol-2-yl]-methyl]-benzenesulfonic acid amide 1258069-52-1 C31H35ClN6O3S
2-chloro-N,6-dimethyl-N-[[7-(3-pyridin-4-yl-3,9-diazaspiro[5.5]undecane-9-carbonyl)-1H-benzoimidazol-2-yl]-methyl]-benzenesulfonic acid amide
—— N-(2-((5-chloro-2-((1-(cyclopropylmethyl)-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)methanesulfonamide 1258944-30-7 C19H22ClN7O3S
N-(2-((5-chloro-2-((1-(cyclopropylmethyl)-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)methanesulfonamide
—— 2-[4-[{4-butyl-2-methyl-6-oxo-1-(pyridin-2-yl)-1,6-dihydropyrimidin-5-yl}methyl]-2,6-dipropylphenoxy]-2-(2-chlorophenyl)acetic acid 1256779-59-5 C35H40ClN3O4
2-[4-[{4-butyl-2-methyl-6-oxo-1-(pyridin-2-yl)-1,6-dihydropyrimidin-5-yl}methyl]-2,6-dipropylphenoxy]-2-(2-chlorophenyl)acetic acid
—— 5,7-dichloro-4-[1-(3-hydroxymethylphenylcarbamoyl)-ethoxy]-naphthalene-2-carboxylic acid 1257342-45-2 C21H17Cl2NO5
5,7-dichloro-4-[1-(3-hydroxymethylphenylcarbamoyl)-ethoxy]-naphthalene-2-carboxylic acid
—— N-(2-((5-chloro-2-((1-propyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)methanesulfonamide 1258946-56-3 C18H22ClN7O3S
N-(2-((5-chloro-2-((1-propyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)methanesulfonamide
—— 5-(3-chlorophenyl)-2,7-dioxo-N-(pyridin-2-yl)-1,2,4,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 1257440-19-9 C18H12ClN5O3
5-(3-chlorophenyl)-2,7-dioxo-N-(pyridin-2-yl)-1,2,4,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 2-(1-azetidin-3-yl-1H-pyrazol-4-yl)-8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxaline 1092500-10-1 C25H24F2N6O
2-(1-azetidin-3-yl-1H-pyrazol-4-yl)-8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxaline
—— 2-(2-chloropyridin-4-yl)-N-(3-ethylphenyl)-4-(2-methylphenyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide 1095716-54-3 C28H26ClN5O
2-(2-chloropyridin-4-yl)-N-(3-ethylphenyl)-4-(2-methylphenyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide
—— Methyl 4-[2-[3,5-dichloro-2-[(3,5-dimethoxyphenoxy)methyl]-6-oxopyridin-1-yl]ethyl]benzoate 1091595-93-5 C24H23Cl2NO6
Methyl 4-[2-[3,5-dichloro-2-[(3,5-dimethoxyphenoxy)methyl]-6-oxopyridin-1-yl]ethyl]benzoate
—— (S,E)-methyl 2-(2-(3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)-[1,2,4]triazolo[1,5-a]pyridine-7-carboxylate 1094104-07-0 C27H22ClN9O4
(S,E)-methyl 2-(2-(3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)-[1,2,4]triazolo[1,5-a]pyridine-7-carboxylate
—— 3-(2,5-difluorophenyl)-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile 1056890-75-5 C21H18F2N2O
3-(2,5-difluorophenyl)-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile
—— 1-(3-benzothienyl)-3-(tetrahydro-2H-pyran-2-yloxy)-1-propyne 1093173-48-8 C16H16O2S
1-(3-benzothienyl)-3-(tetrahydro-2H-pyran-2-yloxy)-1-propyne
—— methanesulfonic acid 6-(4-fluoro-2-methyl-1H-indol-5-yloxy)-pyrimidin-4-ylmethyl ester 1229448-52-5 C15H14FN3O4S
methanesulfonic acid 6-(4-fluoro-2-methyl-1H-indol-5-yloxy)-pyrimidin-4-ylmethyl ester
—— (S,E)-3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-N-(1-oxo-3-phenyl-1-(3-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-8-ylamino)propan-2-yl)acrylamide 1094104-68-3 C26H19ClF3N9O2
(S,E)-3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-N-(1-oxo-3-phenyl-1-(3-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-8-ylamino)propan-2-yl)acrylamide
—— (S)-N-hydroxy-3-[4-(2-methylquinolin-4-ylmethoxy)benzenesulfonylamino]-2-[4-(propane-2-sulfonyl)piperazin-1-yl]propionamide 1260171-77-4 C27H35N5O7S2
(S)-N-hydroxy-3-[4-(2-methylquinolin-4-ylmethoxy)benzenesulfonylamino]-2-[4-(propane-2-sulfonyl)piperazin-1-yl]propionamide
—— N-(2-(5-chloro-2-(1,3,5-trimethyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide 1258943-84-8 C18H22ClN7O3S
N-(2-(5-chloro-2-(1,3,5-trimethyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide
—— 1-{[7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}-4-phenylpiperidin-4-ol 1257320-28-7 C29H30N4O3
1-{[7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}-4-phenylpiperidin-4-ol
—— (S)-6-(6-(3-ethylureido)-4-(4-phenylthiazol-2-yl)pyridin-3-yl)-1-(1-(2-morpholinoethyl)piperidin-3-yl)-4-oxo-1,4-dihydro-1,7-naphthyridine-3-carboxylic acid 1256912-56-7 C37H40N8O5S
(S)-6-(6-(3-ethylureido)-4-(4-phenylthiazol-2-yl)pyridin-3-yl)-1-(1-(2-morpholinoethyl)piperidin-3-yl)-4-oxo-1,4-dihydro-1,7-naphthyridine-3-carboxylic acid
—— 4-(5-methyl-pyridin-2-yl)-1-phenyl-1H-indazole-6-carboxylic acid (5-methyl-pyrazin-2-ylmethyl)-amide 1258940-41-8 C26H22N6O
4-(5-methyl-pyridin-2-yl)-1-phenyl-1H-indazole-6-carboxylic acid (5-methyl-pyrazin-2-ylmethyl)-amide
—— 3-(4-isopropylthiazol-2-yl)-5-thioxo-1H-(1,2,4-triazol-4(5H)-yl) 4-methylbenzamide 1257424-36-4 C16H17N5OS2
3-(4-isopropylthiazol-2-yl)-5-thioxo-1H-(1,2,4-triazol-4(5H)-yl) 4-methylbenzamide
—— 4-((2R)-1-(3-(4-fluorophenyl)pyrrolidin-1-yl)-1-oxobutan-2-yl)-4,5-dihydropyrrolo[4,3,2-de][2,6]naphthyridin-3(1H)-one 1258065-85-8 C23H23FN4O2
4-((2R)-1-(3-(4-fluorophenyl)pyrrolidin-1-yl)-1-oxobutan-2-yl)-4,5-dihydropyrrolo[4,3,2-de][2,6]naphthyridin-3(1H)-one
—— N-((S)-1-((R)-4-(4-fluorophenyl)-1-oxo-2,8-diazaspiro[4.5]decan-8-yl)propan-2-yl)-1H-indole-2-carboxamide 2,2,2-trifluoroacetate 1262536-71-9 C2HF3O2*C26H29FN4O2
N-((S)-1-((R)-4-(4-fluorophenyl)-1-oxo-2,8-diazaspiro[4.5]decan-8-yl)propan-2-yl)-1H-indole-2-carboxamide 2,2,2-trifluoroacetate
—— 4-hydroxy-5,6-dimethoxy-3-(5-methoxy-2-methylpentanoyl)pyridin-2(1H)-one 1231945-01-9 C14H21NO6
4-hydroxy-5,6-dimethoxy-3-(5-methoxy-2-methylpentanoyl)pyridin-2(1H)-one
—— N-({(5S)-3-[4-(3-allyl-2-oxopyridin-1(2H)-yl)-2-fluorophenyl]-2-oxo-1,3-oxazolidin-5-yl}methyl)-5-chlorothiophene-2-carboxamide 1093629-15-2 C23H19ClFN3O4S
N-({(5S)-3-[4-(3-allyl-2-oxopyridin-1(2H)-yl)-2-fluorophenyl]-2-oxo-1,3-oxazolidin-5-yl}methyl)-5-chlorothiophene-2-carboxamide
—— N-(2-(5-chloro-2-(1-methyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide 1258943-77-9 C16H18ClN7O3S
N-(2-(5-chloro-2-(1-methyl-1H-pyrazol-4-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide
—— chlorogold;diphenylphosphinothioylmethyl-diphenyl-sulfanylidene-λ5-phosphane 192765-62-1 C25H22Au2Cl2P2S2
chlorogold;diphenylphosphinothioylmethyl-diphenyl-sulfanylidene-λ5-phosphane
—— N-(5-ethylpyridin-3-yl)-4-(2-methylphenyl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide 1095716-29-2 C27H26N6O
N-(5-ethylpyridin-3-yl)-4-(2-methylphenyl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide
—— (Z)-3-((4-acetyl-5-methyl-3-(3-(4-methylpiperazin-1-yl)-3-oxopropyl)-1H-pyrrol-2-yl)methylene)-5-fluoroindolin-2-one 1235459-41-2 C24H27FN4O3
(Z)-3-((4-acetyl-5-methyl-3-(3-(4-methylpiperazin-1-yl)-3-oxopropyl)-1H-pyrrol-2-yl)methylene)-5-fluoroindolin-2-one
—— 2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-quinoxalin-6-ylpropanenitrile 1056889-39-4 C23H20N4O
2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-quinoxalin-6-ylpropanenitrile
—— 3-[3-(3-cyanopropoxy)phenyl]-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile 1056888-20-0 C25H25N3O2
3-[3-(3-cyanopropoxy)phenyl]-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile
—— N-(2-(4-(4-cyano-1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)-2-(trifluoromethyl)-phenoxy)ethyl)-2-((2-methoxyethyl)(methyl)amino)-N-methylacetamide 1235841-37-8 C24H27F3N6O3
N-(2-(4-(4-cyano-1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)-2-(trifluoromethyl)-phenoxy)ethyl)-2-((2-methoxyethyl)(methyl)amino)-N-methylacetamide
—— (2R,3S)-4-(((4S)-6-ethyl-3,4-dihydrospiro[chromene-2,1'-cyclobutan]-4-yl)amino)-3-((2-fluorophenyl)amino)-4-phenyl-2-butanol 1154096-56-6 C30H35FN2O2
(2R,3S)-4-(((4S)-6-ethyl-3,4-dihydrospiro[chromene-2,1'-cyclobutan]-4-yl)amino)-3-((2-fluorophenyl)amino)-4-phenyl-2-butanol
—— 5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid (5-tert-butyl-4-methoxymethyl-isoxazol-3-yl)-amide 1229452-99-6 C24H26N6O4
5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid (5-tert-butyl-4-methoxymethyl-isoxazol-3-yl)-amide
—— N-[3-(1,3-dimethyl-2-oxobenzimidazol-5-yl)-5-ethylphenyl]-4-(2-methylphenyl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide 1095716-81-6 C37H35N7O2
N-[3-(1,3-dimethyl-2-oxobenzimidazol-5-yl)-5-ethylphenyl]-4-(2-methylphenyl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide
—— 5-(6-pyrazol-1-ylmethyl-pyrimidin-4-yloxy)-indole-1-carboxylic acid (2-fluoro-5-trifluoromethyl-phenyl)-amide 1229449-29-9 C24H16F4N6O2
5-(6-pyrazol-1-ylmethyl-pyrimidin-4-yloxy)-indole-1-carboxylic acid (2-fluoro-5-trifluoromethyl-phenyl)-amide
—— [9-(2,6-Diethyl-4-methylphenyl)-10-oxo-3-oxaspiro[5.5]undec-8-en-8-yl] 2-methoxyacetate 1058730-41-8 C24H32O5
[9-(2,6-Diethyl-4-methylphenyl)-10-oxo-3-oxaspiro[5.5]undec-8-en-8-yl] 2-methoxyacetate
—— (S,E)-methyl 3-(2-(3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)benzo[d]isoxazol-7-ylcarbamate 1094104-69-4 C28H23ClN8O5
(S,E)-methyl 3-(2-(3-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)acrylamido)-3-phenylpropanamido)benzo[d]isoxazol-7-ylcarbamate
—— 2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-ethoxypiperidin-1-yl]-4-{5-[4-(2-hydroxyethyl)piperazin-1-yl]pyrazin-2-yl}-1,3-thiazole-5-carboxylic acid 1229572-25-1 C27H34Cl2N8O5S
2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-ethoxypiperidin-1-yl]-4-{5-[4-(2-hydroxyethyl)piperazin-1-yl]pyrazin-2-yl}-1,3-thiazole-5-carboxylic acid
—— thiazole-4-carboxylic acid [5-(2-methoxy-1-methylethylcarbamoyl)-4'-methylbiphenyl-3-yl]amide 1258858-41-1 C22H23N3O3S
thiazole-4-carboxylic acid [5-(2-methoxy-1-methylethylcarbamoyl)-4'-methylbiphenyl-3-yl]amide
—— 1-(5-chloro-thiophene-2-sulfonyl)-4,4-difluoro-pyrrolidine-2S-carboxylic acid [2-(4-isobutyl-piperazin-1-yl)-6-(4-trifluoromethyl-phenyl)-pyrimidin-4-ylmethyl]-amide 1257433-41-2 C29H32ClF5N6O3S2
1-(5-chloro-thiophene-2-sulfonyl)-4,4-difluoro-pyrrolidine-2S-carboxylic acid [2-(4-isobutyl-piperazin-1-yl)-6-(4-trifluoromethyl-phenyl)-pyrimidin-4-ylmethyl]-amide
—— 4-(5-benzyl-1,5-diazocan-1-yl)pyrimidin-2-amine 1259940-17-4 C17H23N5
4-(5-benzyl-1,5-diazocan-1-yl)pyrimidin-2-amine
—— (3-dimethylamino-pyrrolidine-1-yl)-{(S)-1-[3-(1-methyl-1H-benzoimidazole-2-yl)-phenyl]-piperidin-3-yl}-methanone 1258279-13-8 C26H33N5O
(3-dimethylamino-pyrrolidine-1-yl)-{(S)-1-[3-(1-methyl-1H-benzoimidazole-2-yl)-phenyl]-piperidin-3-yl}-methanone
—— 4-[(5-Chloropyridin-2-yl)methoxy]-1-[6-(3-pyridin-4-ylpyrrolidin-1-yl)pyridin-3-yl]pyridin-2-one 1257315-28-8 C25H22ClN5O2
4-[(5-Chloropyridin-2-yl)methoxy]-1-[6-(3-pyridin-4-ylpyrrolidin-1-yl)pyridin-3-yl]pyridin-2-one
—— tert-butyl 4-(4-((4-(2,2-dioxido-1,3,2-dioxathian-5-yl)phenoxy)methyl)phenoxy)piperidine-1-carboxylate 1258604-08-8 C26H33NO8S
tert-butyl 4-(4-((4-(2,2-dioxido-1,3,2-dioxathian-5-yl)phenoxy)methyl)phenoxy)piperidine-1-carboxylate
—— 2-methyl-N-(thietan-3-yl)-4-[(E)-4,4,4-trifluoro-3-(3,4,5-trichlorophenyl)but-1-enyl]benzamide 1416976-94-7 C21H17Cl3F3NOS
2-methyl-N-(thietan-3-yl)-4-[(E)-4,4,4-trifluoro-3-(3,4,5-trichlorophenyl)but-1-enyl]benzamide