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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide 1254783-04-4 C24H26N6O2
N-[3-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide
—— 1-(2,4-Difluorophenyl)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]urea 1227091-42-0 C17H18F2N4O
1-(2,4-Difluorophenyl)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]urea
—— US8653087, III-203 1213244-88-2 C22H28N8O
US8653087, III-203
—— N-phenethyl-1H-indole-4-carboxamide 1153854-13-7 C17H16N2O
N-phenethyl-1H-indole-4-carboxamide
—— N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3-[[6-[methyl(oxan-2-ylmethyl)amino]pyrimido[5,4-d]pyrimidin-4-yl]amino]benzamide 1213247-62-1 C29H30F3N7O3
N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3-[[6-[methyl(oxan-2-ylmethyl)amino]pyrimido[5,4-d]pyrimidin-4-yl]amino]benzamide
—— US8653087, III-231 1213245-17-0 C26H26F4N8O
US8653087, III-231
—— US8653087, III-202 1213244-87-1 C25H28N8O
US8653087, III-202
—— 2-[1-[(1-Acetylpiperidin-4-yl)methyl]-2-tert-butylbenzimidazol-5-yl]sulfonylpropanenitrile 1067154-03-3 C22H30N4O3S
2-[1-[(1-Acetylpiperidin-4-yl)methyl]-2-tert-butylbenzimidazol-5-yl]sulfonylpropanenitrile
—— 5(4)-amino-N-cyclopropyl-1H-imidazole-4(5)-sulfonamide 1383939-24-9 C6H10N4O2S
5(4)-amino-N-cyclopropyl-1H-imidazole-4(5)-sulfonamide
—— 3-(1,3-Benzothiazol-6-ylamino)-6-ethyl-5-[(4-pyrrolidin-1-ylcyclohexyl)amino]pyrazine-2-carboxamide 1254050-99-1 C24H31N7OS
3-(1,3-Benzothiazol-6-ylamino)-6-ethyl-5-[(4-pyrrolidin-1-ylcyclohexyl)amino]pyrazine-2-carboxamide
—— 2-Butyl-4-hydroxy-3-phenyl-4-(3-phenyl-prop-1-ynyl)-cyclobut-2-enone 144790-94-3 C23H22O2
2-Butyl-4-hydroxy-3-phenyl-4-(3-phenyl-prop-1-ynyl)-cyclobut-2-enone
—— 1-methyl-1'-(2-(2-(trifluoromethyl)phenyl)acetyl)spiro[indoline-3,4'-piperidin]-2-one 1185754-23-7 C22H21F3N2O2
1-methyl-1'-(2-(2-(trifluoromethyl)phenyl)acetyl)spiro[indoline-3,4'-piperidin]-2-one
—— 1-(4-bromophenyl)-3-((4-chlorophenyl)amino)-3-(p-tolyl)propan-1-one 1612152-87-0 C22H19BrClNO
1-(4-bromophenyl)-3-((4-chlorophenyl)amino)-3-(p-tolyl)propan-1-one
—— 2-sec-butylsulfanyl-2-methyl-propionic acid ethyl ester 1017539-66-0 C10H20O2S
2-sec-butylsulfanyl-2-methyl-propionic acid ethyl ester
—— 6-[(3S,4S)-3-[(5S)-4-acetyl-5-(4-chlorophenyl)-1,4-diazocane-1-carbonyl]-4-(5-chloropyridin-2-yl)pyrrolidin-1-yl]-2-methylpyridazin-3-one 1207511-41-8 C29H32Cl2N6O3
6-[(3S,4S)-3-[(5S)-4-acetyl-5-(4-chlorophenyl)-1,4-diazocane-1-carbonyl]-4-(5-chloropyridin-2-yl)pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— diethyl (4-{[4-{[7-(3-hydroxyazetidin-1-yl)-2-methyl-3-oxo-2,3-dihydro-1H-isoindol-4-yl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzyl)phosphonate 1257995-45-1 C28H32F3N6O5P
diethyl (4-{[4-{[7-(3-hydroxyazetidin-1-yl)-2-methyl-3-oxo-2,3-dihydro-1H-isoindol-4-yl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzyl)phosphonate
—— 9-phenyl-N-(5-(1-piperazinyl)-2-pyridinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine 1169692-08-3 C24H22N8
9-phenyl-N-(5-(1-piperazinyl)-2-pyridinyl)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-2-amine
—— (4-dimethylaminobenzyl)-[5-(6-methoxypyridin-3-yl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]amine 1206203-96-4 C19H20N6OS
(4-dimethylaminobenzyl)-[5-(6-methoxypyridin-3-yl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]amine
—— 4-[2-(4-fluorobenzylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]-N-(2-hydroxyethyl)benzamide 1206205-05-1 C20H18FN5O2S
4-[2-(4-fluorobenzylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]-N-(2-hydroxyethyl)benzamide
—— (S)-4-((6-ethynyl-4-(1,1,1-trifluoropropan-2-ylamino)pyrido[3,2-d]pyrimidin-2-ylamino)methyl)benzenesulfonamide 1203654-88-9 C19H17F3N6O2S
(S)-4-((6-ethynyl-4-(1,1,1-trifluoropropan-2-ylamino)pyrido[3,2-d]pyrimidin-2-ylamino)methyl)benzenesulfonamide
—— diethyl [4-({4-[(2-methyl-1-oxo-1,2-dihydroisoquinolin-8-yl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzyl]phosphonate 1257994-48-1 C26H27F3N5O4P
diethyl [4-({4-[(2-methyl-1-oxo-1,2-dihydroisoquinolin-8-yl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzyl]phosphonate
—— [5-[1-(6-chloro-1,3-benzothiazol-2-yl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-5-oxo-2H-pyrrol-2-yl]furan-2-yl]methyl acetate 1071951-43-3 C24H17ClN2O7S
[5-[1-(6-chloro-1,3-benzothiazol-2-yl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-5-oxo-2H-pyrrol-2-yl]furan-2-yl]methyl acetate
—— (2S)-1-[(2R,3'S)-3'-(2-aminoethyl)-5-(2,5-difluorophenyl)-6',8'-difluorospiro[1,3,4-thiadiazole-2,4'-2,3-dihydrochromene]-3-yl]-2-methoxypropan-1-one 1146210-16-3 C22H21F4N3O3S
(2S)-1-[(2R,3'S)-3'-(2-aminoethyl)-5-(2,5-difluorophenyl)-6',8'-difluorospiro[1,3,4-thiadiazole-2,4'-2,3-dihydrochromene]-3-yl]-2-methoxypropan-1-one
—— 4-((6-(4-(difluoromethoxy)-3-(methylsulfonyl)phenyl)-4-(2,2,2-trifluoroethylamino)pyrido[3,2-d]pyrimidin-2-ylamino)methyl)benzenesulfonamide 1203653-49-9 C24H21F5N6O5S2
4-((6-(4-(difluoromethoxy)-3-(methylsulfonyl)phenyl)-4-(2,2,2-trifluoroethylamino)pyrido[3,2-d]pyrimidin-2-ylamino)methyl)benzenesulfonamide
—— US8653087, III-449 1213247-36-9 C28H30F3N9O
US8653087, III-449
—— 3-[(2-iodo-phenylmethanesulfonyl)-(2,2-difluoro-ethyl)-amino]-pyrazine-2-carboxylic acid methyl ester 1154617-04-5 C15H14F2IN3O4S
3-[(2-iodo-phenylmethanesulfonyl)-(2,2-difluoro-ethyl)-amino]-pyrazine-2-carboxylic acid methyl ester
—— N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-3,5-dimethyl-N-(2-(methylsulfonamido)ethyl)isoxazole-4-carboxamide 1108707-56-7 C21H25FN6O5S2
N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-3,5-dimethyl-N-(2-(methylsulfonamido)ethyl)isoxazole-4-carboxamide
—— N2-(4-(1H-1,2,4-triazol-1-yl)benzyl)-6-(6-aminopyridin-3-yl)-N4-(1-(trifluoromethyl)cyclopropyl)pyrido[3,2-d]pyrimidine-2,4-diamine 1203653-09-1 C25H21F3N10
N2-(4-(1H-1,2,4-triazol-1-yl)benzyl)-6-(6-aminopyridin-3-yl)-N4-(1-(trifluoromethyl)cyclopropyl)pyrido[3,2-d]pyrimidine-2,4-diamine
—— 3-[1-(2,4-dichlorobenzyl)-2,3-dihydro-1H-pyrrolo[2,3-b]pyridin-6-yl]-N-(3-hydroxypropyl)benzamide 1202500-72-8 C24H23Cl2N3O2
3-[1-(2,4-dichlorobenzyl)-2,3-dihydro-1H-pyrrolo[2,3-b]pyridin-6-yl]-N-(3-hydroxypropyl)benzamide
—— N-cyclopropyl-5-(5-fluorobenzimidazol-1-yl)thiophene-2-carboxamide 1195774-59-4 C15H12FN3OS
N-cyclopropyl-5-(5-fluorobenzimidazol-1-yl)thiophene-2-carboxamide
—— sodium 3-((4-((12-(methacryloyloxy)dodecyloxy)carbonyl)phenoxy)sulfonyl)-1,1,2,2,3,3-hexafluoropropane-1-sulfonate 1134354-57-6 C26H33F6O10S2*Na
sodium 3-((4-((12-(methacryloyloxy)dodecyloxy)carbonyl)phenoxy)sulfonyl)-1,1,2,2,3,3-hexafluoropropane-1-sulfonate
—— [1-15N]-2'-deoxyguanosine 130434-96-7 C10H13N5O4
[1-15N]-2'-deoxyguanosine
—— 5-(3-chlorophenyl)-1-(3-cyano-4-fluorophenyl)-1H-pyrazole-3-carboxylic acid 1187919-09-0 C17H9ClFN3O2
5-(3-chlorophenyl)-1-(3-cyano-4-fluorophenyl)-1H-pyrazole-3-carboxylic acid
—— 3-(4-chloro-3-{[(2S,3R)-2-(4-chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}-2-methyl-phenyl)-2-methylpropanoic acid 1297548-09-4 C22H22Cl2F3NO3
3-(4-chloro-3-{[(2S,3R)-2-(4-chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}-2-methyl-phenyl)-2-methylpropanoic acid
—— 4-{2-[2-(4-cyclopropane-sulfonyl-phenyl)-2-(3-trifluoromethyl-phenoxy)acetyl-amino]thiazol-5-yloxy}benzoic acid 1328986-54-4 C28H21F3N2O7S2
4-{2-[2-(4-cyclopropane-sulfonyl-phenyl)-2-(3-trifluoromethyl-phenoxy)acetyl-amino]thiazol-5-yloxy}benzoic acid
—— [5-(2-dimethylaminophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]isobutylamine 1206203-24-8 C16H21N5S
[5-(2-dimethylaminophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]isobutylamine
—— 4-(1-benzyl-1,7-diazaspiro[4.4]nonan-7-yl)-7H-pyrrolo[2,3-d]pyrimidine 1263773-64-3 C20H23N5
4-(1-benzyl-1,7-diazaspiro[4.4]nonan-7-yl)-7H-pyrrolo[2,3-d]pyrimidine
—— 1-(4-chloro-1,3-benzothiazol-2-yl)-2-(2,4-difluorophenyl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-2H-pyrrol-5-one 1071948-89-4 C23H13ClF2N2O4S
1-(4-chloro-1,3-benzothiazol-2-yl)-2-(2,4-difluorophenyl)-4-hydroxy-3-(5-methylfuran-2-carbonyl)-2H-pyrrol-5-one
—— 1-[(2R,3'S)-3'-(2-aminoethyl)-5-(3,5-difluorophenyl)-6'-fluorospiro[1,3,4-thiadiazole-2,4'-2,3-dihydrochromene]-3-yl]ethanone 1146210-07-2 C20H18F3N3O2S
1-[(2R,3'S)-3'-(2-aminoethyl)-5-(3,5-difluorophenyl)-6'-fluorospiro[1,3,4-thiadiazole-2,4'-2,3-dihydrochromene]-3-yl]ethanone
—— benzyl N-[4-[3-ethynyl-5-(trifluoromethoxy)phenyl]butyl]carbamate 1292220-55-3 C21H20F3NO3
benzyl N-[4-[3-ethynyl-5-(trifluoromethoxy)phenyl]butyl]carbamate
—— 4-[[4-[2-[2-(2-benzamidoethoxy)ethoxy]ethylamino]-6-(4-hydroxyanilino)-1,3,5-triazin-2-yl]amino]-N-(2-phenylpropan-2-yl)benzamide 1282037-77-7 C38H42N8O5
4-[[4-[2-[2-(2-benzamidoethoxy)ethoxy]ethylamino]-6-(4-hydroxyanilino)-1,3,5-triazin-2-yl]amino]-N-(2-phenylpropan-2-yl)benzamide
—— US8653087, III-111 1213243-96-9 C29H29F3N8O
US8653087, III-111
—— (+)-3-(4-chloro-3-{[(2S,3R)-4,4,4-trifluoro-3-methyl-2-(4-vinylphenyl)butanoyl]amino}phenyl)-propanoic acid 1297546-86-1 C22H21ClF3NO3
(+)-3-(4-chloro-3-{[(2S,3R)-4,4,4-trifluoro-3-methyl-2-(4-vinylphenyl)butanoyl]amino}phenyl)-propanoic acid
—— cyclohexyl-[5-(5-methoxypyridin-3-yl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-amine 1137143-98-6 C16H19N5OS
cyclohexyl-[5-(5-methoxypyridin-3-yl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-amine
—— tert-butyl 2-(2-amino-5-fluorophenyl)acetate 1646556-41-3 C12H16FNO2
tert-butyl 2-(2-amino-5-fluorophenyl)acetate
—— —— 1315459-02-9 C26H27N5O4
—— (5-cyclopropylidenepent-1-yn-1-yl)benzene 1590431-65-4 C14H14
(5-cyclopropylidenepent-1-yn-1-yl)benzene
—— 7-methyl-2-(2-(methylthio)ethyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one 1146966-71-3 C9H11N3OS2
7-methyl-2-(2-(methylthio)ethyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— (2S,3R)-2-[3,4,5-tris[[tert-butyl(dimethyl)silyl]oxy]phenyl]-3,4-dihydro-2H-chromen-3-ol 1131849-82-5 C33H56O5Si3
(2S,3R)-2-[3,4,5-tris[[tert-butyl(dimethyl)silyl]oxy]phenyl]-3,4-dihydro-2H-chromen-3-ol
—— (1R)-2,2-dimethyl-1-[(4S)-4-propan-2-yl-4,5-dihydro-1,3-thiazol-2-yl]propan-1-ol 1133443-22-7 C11H21NOS
(1R)-2,2-dimethyl-1-[(4S)-4-propan-2-yl-4,5-dihydro-1,3-thiazol-2-yl]propan-1-ol