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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-cyclopropyl-N-((S)-1-methyl-3-phenyl-piperidin-3-yl)-4-trifluoromethyl-benzamide hydrochloride 1236303-94-8 C23H25F3N2O*ClH
2-cyclopropyl-N-((S)-1-methyl-3-phenyl-piperidin-3-yl)-4-trifluoromethyl-benzamide hydrochloride
—— N-Benzyl-N-(2,6-dimethyl-phenyl)-3-methyl-isonicotinamide 951028-78-7 C22H22N2O
N-Benzyl-N-(2,6-dimethyl-phenyl)-3-methyl-isonicotinamide
—— 5-acetyl-4-amino-6-benzofuran-2-yl-2-ethyl-2H-pyridazin-3-one 720718-70-7 C16H15N3O3
5-acetyl-4-amino-6-benzofuran-2-yl-2-ethyl-2H-pyridazin-3-one
—— [4-(2-hydroxy-2-methyl-propoxy)-3-methyl-phenyl]-[10-(methoxymethyl)-8-pyrimidin-2-yl-11-oxa-3,8-diazaspiro[5.5]undecan-3-yl]methanone 1400641-67-9 C26H36N4O5
[4-(2-hydroxy-2-methyl-propoxy)-3-methyl-phenyl]-[10-(methoxymethyl)-8-pyrimidin-2-yl-11-oxa-3,8-diazaspiro[5.5]undecan-3-yl]methanone
—— N-ethyl-2-methyl-4-{6-(pyridin-4-yl)-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide 1402594-23-3 C25H24F3N5O
N-ethyl-2-methyl-4-{6-(pyridin-4-yl)-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyridin-3-yl}benzamide
—— 1-tert-butyl-5-[2-(dimethylamino)pyrimidin-4-yl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide 1403332-77-3 C17H26N6O
1-tert-butyl-5-[2-(dimethylamino)pyrimidin-4-yl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
—— 1-[3-(4-Amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)phenyl]-3-(2-methylpropyl)urea 1401530-68-4 C21H21N5OS
1-[3-(4-Amino-[1]benzothiolo[3,2-d]pyrimidin-7-yl)phenyl]-3-(2-methylpropyl)urea
—— 2-[2,6-difluoro-4-[2-[(1S,2R)-2-[1-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-1-morpholin-4-ylethanone 1402553-93-8 C26H34F2N4O5
2-[2,6-difluoro-4-[2-[(1S,2R)-2-[1-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]piperidin-4-yl]cyclopropyl]ethoxy]phenyl]-1-morpholin-4-ylethanone
—— Fmoc-Val-N(Me)Val-OIle-OH 1393736-44-1 C32H42N2O7
Fmoc-Val-N(Me)Val-OIle-OH
—— N-biphenyl-2-yl-N-isobutyl-3-methyl-isonicotinamide 951029-52-0 C23H24N2O
N-biphenyl-2-yl-N-isobutyl-3-methyl-isonicotinamide
—— N-(3-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)-1-(p-tolyl)-1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1401219-15-5 C22H22N6O3S
N-(3-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)-1-(p-tolyl)-1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 4-[2-(2-{4-[2-(2,4-dichloro-phenoxy)-phenylsulfamoyl]-benzoylamino}-acetylamino)-ethyl]-piperidine-1-carboxylic acid tert-butyl ester 1021522-96-2 C33H38Cl2N4O7S
4-[2-(2-{4-[2-(2,4-dichloro-phenoxy)-phenylsulfamoyl]-benzoylamino}-acetylamino)-ethyl]-piperidine-1-carboxylic acid tert-butyl ester
—— N-{[2-chloro-4-(4-methyl-1H-benzimidazol-5-yl)phenyl]methyl}-2-cyclohexylethanamine hydrochloride 1008359-39-4 C23H28ClN3*ClH
N-{[2-chloro-4-(4-methyl-1H-benzimidazol-5-yl)phenyl]methyl}-2-cyclohexylethanamine hydrochloride
—— (1S,3R)-1-trimethylsilyl-1,3-butanediol 1017293-84-3 C7H18O2Si
(1S,3R)-1-trimethylsilyl-1,3-butanediol
—— 4-(2-biphenyl-4-yl-5-methyl-pyrrol-1-yl)-benzenesulfonamide 1000280-19-2 C23H20N2O2S
4-(2-biphenyl-4-yl-5-methyl-pyrrol-1-yl)-benzenesulfonamide
—— N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-1,3-thiazole-2-carboxamide 1141877-13-5 C14H9ClF3N3O3S
N-{[6-chloro-2-oxo-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}-1,3-thiazole-2-carboxamide
—— 4-methylthiomethyl-1,4H-3,1-benzoxazin-2-one 123197-58-0 C10H11NO2S
4-methylthiomethyl-1,4H-3,1-benzoxazin-2-one
—— N-[(4,4-difluoropiperidin-3-yl)methyl]-7-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-amine 1400587-45-2 C17H19F2N7
N-[(4,4-difluoropiperidin-3-yl)methyl]-7-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-amine
—— N-[2-(cyclopentylamino)-1-(3,4-difluorophenyl)-2-oxoethyl]-N-[3-methyl-4-(tetrazol-1-yl)phenyl]prop-2-ynamide 1401089-12-0 C24H22F2N6O2
N-[2-(cyclopentylamino)-1-(3,4-difluorophenyl)-2-oxoethyl]-N-[3-methyl-4-(tetrazol-1-yl)phenyl]prop-2-ynamide
—— 1-[4-(9-Amino-7,10,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-7-yl)phenyl]-3-[4-methoxy-3-(trifluoromethyl)phenyl]urea 1402558-93-3 C24H21F3N6O2
1-[4-(9-Amino-7,10,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-7-yl)phenyl]-3-[4-methoxy-3-(trifluoromethyl)phenyl]urea
—— 4-((3S,4S)-4-methyl-1-(methylsulfonyl)pyrrolidin-3-ylamino)-6-(6-(methylcarbamoyl)pyridin-3-yl)pyrrolo[1,2-b]pyridazine-3-carboxamide 1400578-79-1 C21H25N7O4S
4-((3S,4S)-4-methyl-1-(methylsulfonyl)pyrrolidin-3-ylamino)-6-(6-(methylcarbamoyl)pyridin-3-yl)pyrrolo[1,2-b]pyridazine-3-carboxamide
—— ethyl 2-amino-5-(4-benzyloxybutyl)-thiophene-3-carboxylate 1186474-58-7 C18H23NO3S
ethyl 2-amino-5-(4-benzyloxybutyl)-thiophene-3-carboxylate
—— 7-(trifluoromethyl)isoxazolo[5,4-c]pyridin-3-amine 1242515-53-2 C7H4F3N3O
7-(trifluoromethyl)isoxazolo[5,4-c]pyridin-3-amine
—— 1-(1H-indazol-4-yl)-3-{(3S)-3-[4-(methylsulfanyl)phenyl]cyclopentyl}urea 1401074-91-6 C20H22N4OS
1-(1H-indazol-4-yl)-3-{(3S)-3-[4-(methylsulfanyl)phenyl]cyclopentyl}urea
—— N-(4-((1R,3R,4R,5S)-3-amino-4-hydroxy-4,5-dimethylcyclohexyl)pyridin-3-yl)-6-(2,6-difluoro-3-(2-hydroxyethoxy)phenyl)-5-fluoropicolinamide 1395276-12-6 C27H29F3N4O4
N-(4-((1R,3R,4R,5S)-3-amino-4-hydroxy-4,5-dimethylcyclohexyl)pyridin-3-yl)-6-(2,6-difluoro-3-(2-hydroxyethoxy)phenyl)-5-fluoropicolinamide
—— 5-(4-((1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)sulfonyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)thiophene-2-carbonitrile 1401774-41-1 C22H18N4O4S2
5-(4-((1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)sulfonyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)thiophene-2-carbonitrile
—— N-cyclopropyl-2-methyl-4-{6-[4-(morpholin-4-yl)phenoxy]-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}benzamide 1401450-44-9 C31H32F3N5O3
N-cyclopropyl-2-methyl-4-{6-[4-(morpholin-4-yl)phenoxy]-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}benzamide
—— N-octyl-N-hydroxy-2-(4-hydroxy-3-methoxyphenyl)acetamide 1400943-52-3 C17H27NO4
N-octyl-N-hydroxy-2-(4-hydroxy-3-methoxyphenyl)acetamide
—— N-[(2S)-morpholin-2-ylmethyl]-7-(1-propyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-amine 1400587-29-2 C18H23N7O
N-[(2S)-morpholin-2-ylmethyl]-7-(1-propyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-amine
—— (3S,4S)-4-(2-methoxy-ethoxy)-4-[4-(2-methoxy-ethoxymethyl)-phenyl]-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-piperidine-1-carboxylic acid tert-butyl ester 1146169-35-8 C36H54N2O9
(3S,4S)-4-(2-methoxy-ethoxy)-4-[4-(2-methoxy-ethoxymethyl)-phenyl]-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-piperidine-1-carboxylic acid tert-butyl ester
—— N-cyclopropyl-N-[(4-oxo4,5-dihydropyrrolo[1,2-a]quinoxalin-7-yl)methyl]methanesulfonamide 1036726-61-0 C16H17N3O3S
N-cyclopropyl-N-[(4-oxo4,5-dihydropyrrolo[1,2-a]quinoxalin-7-yl)methyl]methanesulfonamide
—— 5-[4-(2-trifluoromethyl-phenyl)-oxazol-2-yl]-pentanoic acid 847266-84-6 C15H14F3NO3
5-[4-(2-trifluoromethyl-phenyl)-oxazol-2-yl]-pentanoic acid
—— 1-[[4-Fluoro-3-[4-[(2-methylpropan-2-yl)oxy]piperidine-1-carbonyl]phenyl]methyl]quinazoline-2,4-dione 1399119-29-9 C25H28FN3O4
1-[[4-Fluoro-3-[4-[(2-methylpropan-2-yl)oxy]piperidine-1-carbonyl]phenyl]methyl]quinazoline-2,4-dione
—— 2-{8-(3,3-dimethyl-2-oxo-butyl)-7-oxo-7,8-dihydro-2-trifluoromethyl-[1,8]-naphthyridine-3-carbonyl}-cyclohexane-1,3-dione 1188432-39-4 C22H21F3N2O5
2-{8-(3,3-dimethyl-2-oxo-butyl)-7-oxo-7,8-dihydro-2-trifluoromethyl-[1,8]-naphthyridine-3-carbonyl}-cyclohexane-1,3-dione
—— 3-(2-methoxyethyl)-8-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-3,8-dihydro[1,2,3]triazino[4,5-g]quinazoline-4,9-dione 1134100-71-2 C16H17N9O3
3-(2-methoxyethyl)-8-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-3,8-dihydro[1,2,3]triazino[4,5-g]quinazoline-4,9-dione
—— N-cyclopentyl-2-cyclopropylamino-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide 1138321-84-2 C27H30N6O2
N-cyclopentyl-2-cyclopropylamino-6-[4-(3-pyridin-3-ylmethyl-ureido)-phenyl]-nicotinamide
—— 1-(2-chlorophenyl)-2-(5H-imidazo[5,1-α]isoindol-5-yl)ethanol 1402836-69-4 C18H15ClN2O
1-(2-chlorophenyl)-2-(5H-imidazo[5,1-α]isoindol-5-yl)ethanol
—— (3S)-3-({[7-(1,3-dimethyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-yl]oxy}methyl)piperidine hydrochloride 1400587-04-3 C18H22N6O*ClH
(3S)-3-({[7-(1,3-dimethyl-1H-pyrazol-4-yl)pyrido[3,4-b]pyrazin-5-yl]oxy}methyl)piperidine hydrochloride
—— 2-[(4-methoxybenzyl)oxy]-1-nitro-3-{2-[4-(4-phenylbutoxy)phenyl]vinyl}benzene 847657-78-7 C32H31NO5
2-[(4-methoxybenzyl)oxy]-1-nitro-3-{2-[4-(4-phenylbutoxy)phenyl]vinyl}benzene
—— 4-[3-(2-tert-butylphenoxy)azetidin-1-yl]-4-oxo-N-(pentylsulfonyl)butanamide 1146958-11-3 C22H34N2O5S
4-[3-(2-tert-butylphenoxy)azetidin-1-yl]-4-oxo-N-(pentylsulfonyl)butanamide
—— 3-[1-(3',5'-dimethoxybiphenyl-3-yl)-1H-benzimidazol-6-yl]-1,2,4-oxadiazol-5(2H)-one 1401321-39-8 C23H18N4O4
3-[1-(3',5'-dimethoxybiphenyl-3-yl)-1H-benzimidazol-6-yl]-1,2,4-oxadiazol-5(2H)-one
—— 6-[5-(acetylmethylamino)pyridin-2-yloxy]indole-1,2-dicarboxylic acid 1-tert-butyl ester 2-ethyl ester 1150745-86-0 C24H27N3O6
6-[5-(acetylmethylamino)pyridin-2-yloxy]indole-1,2-dicarboxylic acid 1-tert-butyl ester 2-ethyl ester
—— 5-amino-2-chloro-N-cyclopentyl-4-methylaminobenzamide 1242268-53-6 C13H18ClN3O
5-amino-2-chloro-N-cyclopentyl-4-methylaminobenzamide
—— 1-[4-(9-Amino-7,10,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-7-yl)phenyl]-3-[4-chloro-3-(trifluoromethyl)phenyl]urea 1402558-97-7 C23H18ClF3N6O
1-[4-(9-Amino-7,10,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-7-yl)phenyl]-3-[4-chloro-3-(trifluoromethyl)phenyl]urea
—— 3-(1-{[3-chloro-6-(3-furanyl)-8-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-3-hydroxy-4-piperidinyl)-1,3-oxazolidin-2-one 1237842-01-1 C21H18ClF3N4O5
3-(1-{[3-chloro-6-(3-furanyl)-8-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-3-hydroxy-4-piperidinyl)-1,3-oxazolidin-2-one
—— [3-cyclohexyl-2-[2-({[2-(dimethylamino)ethyl]amino}methyl)phenyl]-6-(methoxycarbonyl)-1H-indol-1-yl]acetic acid 886041-24-3 C29H37N3O4
[3-cyclohexyl-2-[2-({[2-(dimethylamino)ethyl]amino}methyl)phenyl]-6-(methoxycarbonyl)-1H-indol-1-yl]acetic acid
—— 3-(2-methyl-5-(3-trifluoromethyl-phenyl)-pyrrol-1-yl)-benzenesulfonamide 1000280-15-8 C18H15F3N2O2S
3-(2-methyl-5-(3-trifluoromethyl-phenyl)-pyrrol-1-yl)-benzenesulfonamide
—— {[4-(1H-benzimidazol-5-yl)phenyl]methyl}cyclohexylamine trifluoroacetate 1008358-12-0 C2HF3O2*C20H23N3
{[4-(1H-benzimidazol-5-yl)phenyl]methyl}cyclohexylamine trifluoroacetate
—— [3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 2-methoxybenzoate 1403240-49-2 C27H26N4O4
[3-[4-[(4-oxo-3H-quinazolin-2-yl)methyl]piperazin-1-yl]phenyl] 2-methoxybenzoate
—— 4-{6-(2,3-difluorophenoxy)-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}-N-ethyl-2-methylbenzamide 1401450-50-7 C26H23F5N4O2
4-{6-(2,3-difluorophenoxy)-4-[(3,3,3-trifluoropropyl)amino]-1H-benzimidazol-1-yl}-N-ethyl-2-methylbenzamide