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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[6-(4-Methoxy-phenoxy)-hexyl]-1,5-dimethyl-2-oxo-1,2,3,5-tetrahydro-2λ<sup>4</sup>-imidazo[4,5-c][1,2,6]thiadiazin-4-one 117835-58-2 C19H26N4O4S
3-[6-(4-Methoxy-phenoxy)-hexyl]-1,5-dimethyl-2-oxo-1,2,3,5-tetrahydro-2λ<sup>4</sup>-imidazo[4,5-c][1,2,6]thiadiazin-4-one
—— 2-[(2-amino-2-oxoethyl)(3,4-dichlorophenyl)amino]-N-methyl-N-[1-{3'-[(methylsulfonyl)amino]-4-biphenylyl}-2-(4-morpholinyl)ethyl]acetamide 1003876-00-3 C30H35Cl2N5O5S
2-[(2-amino-2-oxoethyl)(3,4-dichlorophenyl)amino]-N-methyl-N-[1-{3'-[(methylsulfonyl)amino]-4-biphenylyl}-2-(4-morpholinyl)ethyl]acetamide
—— N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-4-chloro-3-[2-(4-methyl-[1,4]diazepan-1-ylmethyl)-pyrimidin-4-yloxy]-benzamide 1215029-69-8 C30H39ClN6O5S
N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-4-chloro-3-[2-(4-methyl-[1,4]diazepan-1-ylmethyl)-pyrimidin-4-yloxy]-benzamide
—— butyl 2-[4-(3'-methoxy-1,1'-biphenyl-4-yl)-1H-imidazol-2-yl]ethylcarbamate 717914-96-0 C23H27N3O3
butyl 2-[4-(3'-methoxy-1,1'-biphenyl-4-yl)-1H-imidazol-2-yl]ethylcarbamate
—— N-(2-{2-[4-(phenylsulphonyl-methyl-amino)-phenylamino]-5-trifluoromethyl-pyrimidin-4-ylamino}-ethyl)-acetamide 514841-63-5 C22H23F3N6O3S
N-(2-{2-[4-(phenylsulphonyl-methyl-amino)-phenylamino]-5-trifluoromethyl-pyrimidin-4-ylamino}-ethyl)-acetamide
—— methyl 2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoate 1228781-68-7 C35H38ClN3O3
methyl 2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoate
—— N-(3-fluoro-4-(3-(piperidin-4-yloxy)-1H-pyrazolo[3,4-b]pyridin-4-yloxy)phenyl)-2-methyl-3-oxo-2,3-dihydropyridazine-4-carboxamide 1129457-62-0 C23H22FN7O4
N-(3-fluoro-4-(3-(piperidin-4-yloxy)-1H-pyrazolo[3,4-b]pyridin-4-yloxy)phenyl)-2-methyl-3-oxo-2,3-dihydropyridazine-4-carboxamide
—— acetic acid (R,R)-2-(5-[4-(benzothiazol-2-yloxy)-benzyl]-2,5-diaza-bicyclo[2.2.1]hept-2-yl)-2-oxo-ethyl ester 1146691-94-2 C23H23N3O4S
acetic acid (R,R)-2-(5-[4-(benzothiazol-2-yloxy)-benzyl]-2,5-diaza-bicyclo[2.2.1]hept-2-yl)-2-oxo-ethyl ester
—— 4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(3-fluorophenoxy)-N-({4-[(1-methylpiperidin-4-yl)amino]-3-nitrophenyl}sulfonyl)benzamide 1228939-03-4 C44H50ClFN6O6S
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(3-fluorophenoxy)-N-({4-[(1-methylpiperidin-4-yl)amino]-3-nitrophenyl}sulfonyl)benzamide
—— (R)-1-amino-3-(2-bromo-4-fluorophenoxy)propan-2-ol 1008451-15-7 C9H11BrFNO2
(R)-1-amino-3-(2-bromo-4-fluorophenoxy)propan-2-ol
—— 6-allyl-7-methoxy-5-methylimidazo<1,2-a>pyrimidine-2-carbohydrazide 106073-10-3 C12H15N5O2
6-allyl-7-methoxy-5-methylimidazo<1,2-a>pyrimidine-2-carbohydrazide
—— 1-(7,8-Dichloro-2-hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-ethanone 103829-73-8 C11H10Cl2O4
1-(7,8-Dichloro-2-hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-ethanone
—— N-4-tert-butylbenzyl-N-ethyl-1-naphthalenemethylamine 101828-38-0 C24H29N
N-4-tert-butylbenzyl-N-ethyl-1-naphthalenemethylamine
—— 2,2-difluoro-8-[(1S)-1-hydroxyethyl]-4-(1H-indazol-4-ylmethyl)-2H-1,4-benzoxazin-3(4H)-one 1263412-83-4 C18H15F2N3O3
2,2-difluoro-8-[(1S)-1-hydroxyethyl]-4-(1H-indazol-4-ylmethyl)-2H-1,4-benzoxazin-3(4H)-one
—— 4-Amino-6-methylmercapto-5-cyan-3-methyl-3H-pyrrolo<2,3-d>pyrimidin 16754-94-2 C9H9N5S
4-Amino-6-methylmercapto-5-cyan-3-methyl-3H-pyrrolo<2,3-d>pyrimidin
—— 8-Amino-6-hydrazino-tetrazolo<1,5-b>pyridazin 1589-08-8 C4H6N8
8-Amino-6-hydrazino-tetrazolo<1,5-b>pyridazin
—— 1-methyl-3-[3-(1-benzyl-4-piperidyl)propionyl]indazole oxalate 155868-77-2 C2H2O4*C23H27N3O
1-methyl-3-[3-(1-benzyl-4-piperidyl)propionyl]indazole oxalate
—— (2-{4-[2-(2-fluoro-5-trifluoromethyl-phenylamino)-1-methyl-1H-benzoimidazol-5-yloxy]-pyridin-2-yl}-5-trifluoromethyl-1H-imidazol-4-yl)-methanol 927881-05-8 C25H17F7N6O2
(2-{4-[2-(2-fluoro-5-trifluoromethyl-phenylamino)-1-methyl-1H-benzoimidazol-5-yloxy]-pyridin-2-yl}-5-trifluoromethyl-1H-imidazol-4-yl)-methanol
—— 4,5-diphenyl-1-(phenylthio)imidazo[1,5-a]quinoline 1428368-46-0 C29H20N2S
4,5-diphenyl-1-(phenylthio)imidazo[1,5-a]quinoline
—— —— 864058-33-3 C32H40O3Si
—— 2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)cyclohept-1-enyl)methyl)piperazin-1-yl)benzoic acid 1228783-73-0 C33H34ClN3O3
2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)cyclohept-1-enyl)methyl)piperazin-1-yl)benzoic acid
—— N-[5-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-2-methyl-benzenesulfonamide 1080826-91-0 C24H25N5O4S
N-[5-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-2-methyl-benzenesulfonamide
—— [4-(3,5-di-tert-butylphenyl)-1,3-thiazol-2-yl]methylamine 717915-76-9 C18H26N2S
[4-(3,5-di-tert-butylphenyl)-1,3-thiazol-2-yl]methylamine
—— 2,5-dimethyl-(N-dichlorofluoromethylsulphenyl-N-methyl)-benzenesulphonamide 107879-09-4 C10H12Cl2FNO2S2
2,5-dimethyl-(N-dichlorofluoromethylsulphenyl-N-methyl)-benzenesulphonamide
—— 1-[N-5-(4-trifluoromethylthiophenoxy)-pentyl-N-propyl-carbamoyl]-imidazole 102793-39-5 C19H24F3N3O2S
1-[N-5-(4-trifluoromethylthiophenoxy)-pentyl-N-propyl-carbamoyl]-imidazole
—— 3,6-Heptanooxepin-4,5-dimethanol 102652-09-5 C15H22O3
3,6-Heptanooxepin-4,5-dimethanol
—— benzo[b]thiophen-3-yl-[7-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-4,7-diaza-spiro[2.5]oct-4-yl]-methanone 1261356-47-1 C21H19N5OS
benzo[b]thiophen-3-yl-[7-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-4,7-diaza-spiro[2.5]oct-4-yl]-methanone
—— 7-(benzylsulfanyl)[1,2,4]triazolo[1,5-a]pyridine 1431878-03-3 C13H11N3S
7-(benzylsulfanyl)[1,2,4]triazolo[1,5-a]pyridine
—— 3-[5-(5-{[(5-fluoropyridin-2-yl)oxy]methyl}-1-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-N-[2-(methylamino)ethyl]benzenesulfonamide 1359029-04-1 C21H22FN7O4S
3-[5-(5-{[(5-fluoropyridin-2-yl)oxy]methyl}-1-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-N-[2-(methylamino)ethyl]benzenesulfonamide
—— 6-[9-(4-chloro-3-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-3,3-dimethyl-6-oxohexanoic acid 1354803-29-4 C25H27ClFN3O3
6-[9-(4-chloro-3-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-3,3-dimethyl-6-oxohexanoic acid
—— N-(adamantan-1-ylmethyl)-2-{2-[ethyl(methyl)amino]-2-oxoethyl}imidazo[1,2-a]pyridine-5-carboxamide 1031831-32-9 C24H32N4O2
N-(adamantan-1-ylmethyl)-2-{2-[ethyl(methyl)amino]-2-oxoethyl}imidazo[1,2-a]pyridine-5-carboxamide
—— 1,6-Dioxo-5,6-dihydro-1H-pyrido[1,2-a]quinazoline-2,4-dicarboxylic acid diethyl ester 121583-02-6 C18H16N2O6
1,6-Dioxo-5,6-dihydro-1H-pyrido[1,2-a]quinazoline-2,4-dicarboxylic acid diethyl ester
—— 4-(4-(4-(1-butylazetidin-3-yloxy)phenyl)-3-(2-chlorophenyl)isoxazol-5-yl)-phenol hydrochloride 1383928-82-2 C28H27ClN2O3*ClH
4-(4-(4-(1-butylazetidin-3-yloxy)phenyl)-3-(2-chlorophenyl)isoxazol-5-yl)-phenol hydrochloride
—— 4-(1,1-dioxo-2-phenyl-1<i>H</i>-1λ<sup>6</sup>-benzo[<i>b</i>]thiophen-3-yl)-morpholine 55118-74-6 C18H17NO3S
4-(1,1-dioxo-2-phenyl-1<i>H</i>-1λ<sup>6</sup>-benzo[<i>b</i>]thiophen-3-yl)-morpholine
—— 5-[5-(3-chlorophenyl)-1H-imidazol-2-yl]-3-phenyl-1H-pyrazol-4-ol 1197337-76-0 C18H13ClN4O
5-[5-(3-chlorophenyl)-1H-imidazol-2-yl]-3-phenyl-1H-pyrazol-4-ol
—— 2-amino-7-hydroxy-6-[2-methyl-5-N-(-4-trifluoromethylpyrimidin-6-yl)carbamoylphenyl]-8-(pyridin-2-yl)quinazoline 1191932-12-3 C26H18F3N7O2
2-amino-7-hydroxy-6-[2-methyl-5-N-(-4-trifluoromethylpyrimidin-6-yl)carbamoylphenyl]-8-(pyridin-2-yl)quinazoline
—— 3-nitro-5,6,7,8-tetrahydro-5,8-methanoisoquinoline-6-(exo)-ol nitrate N-oxide 106203-61-6 C10H9N3O6
3-nitro-5,6,7,8-tetrahydro-5,8-methanoisoquinoline-6-(exo)-ol nitrate N-oxide
—— 3-phenyl-5-(4-ethoxyphenyl)-isoxazole 79182-03-9 C17H15NO2
3-phenyl-5-(4-ethoxyphenyl)-isoxazole
—— 2,4,6-Triamino-5-<3-(N-acetyl-4-aethoxycarbonyl-anilino)-propionylamino>-pyrimidin 17415-04-2 C18H23N7O4
2,4,6-Triamino-5-<3-(N-acetyl-4-aethoxycarbonyl-anilino)-propionylamino>-pyrimidin
—— 6-chloro-3-(2-cyclopropyl-6-methylphenoxy)-4-pyridazinyl 1-propanesulfonate 499230-85-2 C17H19ClN2O4S
6-chloro-3-(2-cyclopropyl-6-methylphenoxy)-4-pyridazinyl 1-propanesulfonate
—— 6-chloro-3-(2-cyclopropyl-6-methylphenoxy)-4-pyridazinyl 5-acetyl-2-thiophenecarboxylate 499233-60-2 C21H17ClN2O4S
6-chloro-3-(2-cyclopropyl-6-methylphenoxy)-4-pyridazinyl 5-acetyl-2-thiophenecarboxylate
—— 2-(2-aminocyclohexylamino)-6-(3-carboxy-4-chloroanilino)-8-azapurine 663889-20-1 C17H19ClN8O2
2-(2-aminocyclohexylamino)-6-(3-carboxy-4-chloroanilino)-8-azapurine
—— (E)-N-[4-(4-methoxyphenyl)thiazol-2-yl]-3-(3-methoxy-4-(2,2-difluoroethoxy)-phenyl)acrylamide 1070794-59-0 C22H20F2N2O4S
(E)-N-[4-(4-methoxyphenyl)thiazol-2-yl]-3-(3-methoxy-4-(2,2-difluoroethoxy)-phenyl)acrylamide
—— ethyl 2-(4-(hydroxymethyl)phenylamino)-6-(2-methoxyphenylamino)-5-nitropyrimidine-4-carboxylate 1022158-05-9 C21H21N5O6
ethyl 2-(4-(hydroxymethyl)phenylamino)-6-(2-methoxyphenylamino)-5-nitropyrimidine-4-carboxylate
—— 2-(6-isopropoxy-indol-3-yl)-ethylamine 131762-50-0 C13H18N2O
2-(6-isopropoxy-indol-3-yl)-ethylamine
—— 3-{2-[9-(4-chloro-2-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-2-oxoethoxy}-2,2-dimethylpropanoic acid 1354803-44-3 C24H25ClFN3O4
3-{2-[9-(4-chloro-2-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]-2-oxoethoxy}-2,2-dimethylpropanoic acid
—— 2-adamantan-1-yl-N-(2-{[4-(trifluoromethyl)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridin-5-yl)acetamide 1031833-71-2 C26H31F3N4O2
2-adamantan-1-yl-N-(2-{[4-(trifluoromethyl)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridin-5-yl)acetamide
—— 1-{2-tert-butyl-4-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-5-yl}-3-[4-(6,7-dimethoxyquinolin-4-yloxy)phenyl]urea 1355347-05-5 C31H34N8O4
1-{2-tert-butyl-4-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-5-yl}-3-[4-(6,7-dimethoxyquinolin-4-yloxy)phenyl]urea
—— N-(3-((2-((4-(2-methoxyethoxy)phenyl)amino)thieno[3,2-d]pyrimidin-4-yl)oxy)phenyl)acrylamide 1353550-74-9 C24H22N4O4S
N-(3-((2-((4-(2-methoxyethoxy)phenyl)amino)thieno[3,2-d]pyrimidin-4-yl)oxy)phenyl)acrylamide
—— tert-butyl 4-(3-(1-(cyclohexyl(methyl)carbamoyl)-1H-imidazol-4-yl)benzamido)piperidine-1-carboxylate 1356960-68-3 C28H39N5O4
tert-butyl 4-(3-(1-(cyclohexyl(methyl)carbamoyl)-1H-imidazol-4-yl)benzamido)piperidine-1-carboxylate