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—— methyl (3aR,6aR)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C20H16ClN3O5
methyl (3aR,6aR)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— Methyl 2-[[4-(difluoromethoxy)benzoyl]amino]-5-phenylthiophene-3-carboxylate —— C20H15F2NO4S
Methyl 2-[[4-(difluoromethoxy)benzoyl]amino]-5-phenylthiophene-3-carboxylate
—— methyl (3aS,6aR)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C20H16ClN3O5
methyl (3aS,6aR)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl 4-[(2S)-3-acetyl-1-(3-bromo-4-methylphenyl)-4-hydroxy-5-oxo-2H-pyrrol-2-yl]benzoate —— C21H18BrNO5
methyl 4-[(2S)-3-acetyl-1-(3-bromo-4-methylphenyl)-4-hydroxy-5-oxo-2H-pyrrol-2-yl]benzoate
—— methyl (3aS,6aS)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C20H16ClN3O5
methyl (3aS,6aS)-5-(4-chlorophenyl)-1-(2-methoxyphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl (7R)-6-benzoyl-7-(3-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate —— C19H14FN5O3
methyl (7R)-6-benzoyl-7-(3-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate
—— methyl (1R,1aR,7bR)-6-bromo-1-ethyl-1-(4-methylbenzoyl)-2-oxo-7bH-cyclopropa[c]chromene-1a-carboxylate —— C22H19BrO5
methyl (1R,1aR,7bR)-6-bromo-1-ethyl-1-(4-methylbenzoyl)-2-oxo-7bH-cyclopropa[c]chromene-1a-carboxylate
—— methyl 5-hydroxy-2-methyl-1-{2-[5-methyl-2-(propan-2-yl)phenoxy]ethyl}-1H-indole-3-carboxylate —— C23H27NO4
methyl 5-hydroxy-2-methyl-1-{2-[5-methyl-2-(propan-2-yl)phenoxy]ethyl}-1H-indole-3-carboxylate
—— Methyl 2-[2-(2-bromo-4-chlorophenoxy)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C18H17BrClNO4S
Methyl 2-[2-(2-bromo-4-chlorophenoxy)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl (7R)-6-(4-chlorobenzoyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate —— C19H14ClN5O3
methyl (7R)-6-(4-chlorobenzoyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate
—— Methyl 2-[2-(3,4-diethoxyphenyl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H27NO5S
Methyl 2-[2-(3,4-diethoxyphenyl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 4-[(4S)-6-amino-5-cyano-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate —— C21H15FN4O3
methyl 4-[(4S)-6-amino-5-cyano-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate
—— methyl 2-[(4S)-6-amino-5-cyano-3-(4-methoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C24H19N5O5
methyl 2-[(4S)-6-amino-5-cyano-3-(4-methoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(4R)-6-amino-3-(5-chlorothiophen-2-yl)-5-cyano-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate —— C19H13ClN4O3S
methyl 4-[(4R)-6-amino-3-(5-chlorothiophen-2-yl)-5-cyano-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate
—— methyl 4-[(4S)-6-amino-3-(5-chlorothiophen-2-yl)-5-cyano-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate —— C19H13ClN4O3S
methyl 4-[(4S)-6-amino-3-(5-chlorothiophen-2-yl)-5-cyano-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate
—— Methyl 2-[[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-4,5-dimethoxybenzoate —— C21H19ClN2O6
Methyl 2-[[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-4,5-dimethoxybenzoate
—— methyl (7S)-6-acetyl-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate —— C14H12BrN5O3
methyl (7S)-6-acetyl-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylate
—— methyl 4-[(6S,9S)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C29H26N2O4
methyl 4-[(6S,9S)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9R)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C29H26N2O4
methyl 4-[(6R,9R)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9R)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H30N2O4
methyl 4-[(6R,9R)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(4S)-6-amino-5-cyano-3-(3,4-dichlorophenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C23H15Cl2N5O4
methyl 2-[(4S)-6-amino-5-cyano-3-(3,4-dichlorophenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 2-[(4S)-6-amino-5-cyano-3-(4-ethoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C25H21N5O5
methyl 2-[(4S)-6-amino-5-cyano-3-(4-ethoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 2-[(3R)-6'-amino-1'-(3-chlorophenyl)-5'-cyano-3'-methyl-2-oxospiro[indole-3,4'-pyrano[2,3-c]pyrazole]-1-yl]acetate —— C24H18ClN5O4
methyl 2-[(3R)-6'-amino-1'-(3-chlorophenyl)-5'-cyano-3'-methyl-2-oxospiro[indole-3,4'-pyrano[2,3-c]pyrazole]-1-yl]acetate
—— methyl 2-[(4S,7R)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate —— C24H19N3O6
methyl 2-[(4S,7R)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate
—— methyl 5-hydroxy-2-methyl-1-[2-(2,4,6-trimethylphenoxy)ethyl]-1H-indole-3-carboxylate —— C22H25NO4
methyl 5-hydroxy-2-methyl-1-[2-(2,4,6-trimethylphenoxy)ethyl]-1H-indole-3-carboxylate
—— methyl 4-[(4R)-6-amino-5-cyano-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate —— C21H15FN4O3
methyl 4-[(4R)-6-amino-5-cyano-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]benzoate
—— methyl 4-[(6R,9S)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H32N2O4
methyl 4-[(6R,9S)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(4R)-6-amino-5-cyano-3-(4-methoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C24H19N5O5
methyl 2-[(4R)-6-amino-5-cyano-3-(4-methoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(6R,9R)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H32N2O4
methyl 4-[(6R,9R)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(3S)-6'-amino-1'-(3-chlorophenyl)-5'-cyano-3'-methyl-2-oxospiro[indole-3,4'-pyrano[2,3-c]pyrazole]-1-yl]acetate —— C24H18ClN5O4
methyl 2-[(3S)-6'-amino-1'-(3-chlorophenyl)-5'-cyano-3'-methyl-2-oxospiro[indole-3,4'-pyrano[2,3-c]pyrazole]-1-yl]acetate
—— methyl 2-[(4R)-6-amino-5-cyano-2'-oxo-3-propan-2-ylspiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C20H19N5O4
methyl 2-[(4R)-6-amino-5-cyano-2'-oxo-3-propan-2-ylspiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 2-[(4S)-6-amino-5-cyano-3-(4-methylphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C24H19N5O4
methyl 2-[(4S)-6-amino-5-cyano-3-(4-methylphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 2-[(4R)-6-amino-5-cyano-3-(3,4-dichlorophenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C23H15Cl2N5O4
methyl 2-[(4R)-6-amino-5-cyano-3-(3,4-dichlorophenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(6S,9R)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H30N2O4
methyl 4-[(6S,9R)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6S,9R)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C31H28N2O4
methyl 4-[(6S,9R)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6S,9S)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H32N2O4
methyl 4-[(6S,9S)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-({2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethyl}carbamoyl)benzoate —— C21H19F3N2O4
methyl 4-({2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethyl}carbamoyl)benzoate
—— methyl 4-[(6S,9S)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C31H28N2O4
methyl 4-[(6S,9S)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(4R)-6-amino-5-cyano-3-(4-methylphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C24H19N5O4
methyl 2-[(4R)-6-amino-5-cyano-3-(4-methylphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 2-[(4S,7S)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate —— C24H19N3O6
methyl 2-[(4S,7S)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(6S,9R)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H32N2O4
methyl 4-[(6S,9R)-5-(3-methylbutanoyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(4R,7R)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate —— C24H19N3O6
methyl 2-[(4R,7R)-2-amino-3-cyano-7-(furan-2-yl)-2',5-dioxospiro[7,8-dihydro-6H-chromene-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(6R,9R)-7-oxo-5-propanoyl-9-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C28H26N2O4S
methyl 4-[(6R,9R)-7-oxo-5-propanoyl-9-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9R)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C31H28N2O4
methyl 4-[(6R,9R)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9S)-7-oxo-5-propanoyl-9-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C28H26N2O4S
methyl 4-[(6R,9S)-7-oxo-5-propanoyl-9-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9S)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C29H26N2O4
methyl 4-[(6R,9S)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6S,9R)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C29H26N2O4
methyl 4-[(6S,9R)-5-acetyl-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 4-[(6R,9S)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C31H28N2O4
methyl 4-[(6R,9S)-5-(cyclopropanecarbonyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate
—— methyl 2-[(4R)-6-amino-5-cyano-3-(4-ethoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate —— C25H21N5O5
methyl 2-[(4R)-6-amino-5-cyano-3-(4-ethoxyphenyl)-2'-oxospiro[2H-pyrano[2,3-c]pyrazole-4,3'-indole]-1'-yl]acetate
—— methyl 4-[(6S,9S)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate —— C32H30N2O4
methyl 4-[(6S,9S)-5-(cyclopropanecarbonyl)-9-(4-methylphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-6-yl]benzoate