| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 5,8-dimethyl-2-[2-(1-methyl-4-thiazol-4-yl-1H-imidazol-2-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312160-46-5 | C16H17N7S |
| —— | (R,R)-N-benzyl-N-(α-methylbenzyl)-1-(2',4',5'-trifluorophenyl)-4-oxo-4-{3''-(trifluoromethyl)-5'',6''-dihydro-1'',2'',4''-triazolo[4,3-α]pyrazin-7''(8''H)-yl}butan-2-amine | 1380521-88-9 | C31H29F6N5O |
| —— | (R)-2-(4-chlorophenyl)-4-(8-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)thiazole hydrochloride | 1338376-14-9 | C15H14ClN5S*ClH |
| —— | (S)-3-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-ylamino]-pyrrolidine-1-carboxylic acid tert-butyl ester | 1215210-20-0 | C24H31F3N8O2S |
| —— | 2-[6-isopropyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-ylamino]-ethanol | 1215214-00-8 | C17H20F3N7OS |
| —— | 2-methanesulfonyl-N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-acetamide | 1215221-83-2 | C20H24F3N7O4S2 |
| —— | 2-(chloromethyl)-5,8-dimethyl-[1,2,4]triazolo[1,5-c]pyrimidine | 1351515-93-9 | C8H9ClN4 |
| —— | {1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-piperidin-2-yl}-methanol | 1215167-57-9 | C21H26F3N7OS |
| —— | 2-oxiranylmethyl-3-oxo-2,5,6,8-tetrahydro-3H-[1,2,4]triazolo[4,3-a]pyrazine-7-carboxylic acid tert-butyl ester | 1182359-43-8 | C13H20N4O4 |
| —— | 7-[2-(5,6-dihydro-8H-imidazo[1,2-a]pyrazin-7-yl)-6-propyl-thieno[2,3-d]pyrimidin-4-yl]-3-trifluoromethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine | 1215205-34-7 | C21H22F3N9S |
| —— | 2-{(2-hydroxy-ethyl)-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-amino}-ethanol | 1215167-64-8 | C19H24F3N7O2S |
| —— | azetidin-3-yl-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-amine | 1215205-52-9 | C18H21F3N8S |
| —— | (R)-1-[6-isobutyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidin-3-ol | 1215214-20-2 | C20H24F3N7OS |
| —— | 7-[6-propyl-2-(tetrahydro-furan-2-ylmethoxy)-thieno[2,3-d]pyrimidin-4-yl]-3-trifluoromethyl-5.6.7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine | 1215214-43-9 | C20H23F3N6O2S |
| —— | (R)-N-benzyl-1-(2',4',5'-trifluorophenyl)-4-oxo-4-{3''-(trifluoromethyl)-5'',6''-dihydro-1'',2'',4''-triazolo[4,3-α]pyrazin-7''(8''H)-yl}butan-2-amine | 1393363-87-5 | C32H31F6N5O2 |
| —— | (1-benzyl-pyrrolidin-3-ylmethyl)-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-amine | 1215167-38-6 | C27H31F3N8S |
| —— | 7-[2-(2-methoxy-ethoxy)-6-propyl-thieno[2,3-d]pyrimidin-4-yl]-3-trifluoromethyl-5.6.7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine | 1215214-40-6 | C18H21F3N6O2S |
| —— | pyridine-2-carboxylic acid {2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-amide | 1215221-87-6 | C23H23F3N8O2S |
| —— | (S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-piperidin-3-ylamine | 1215210-19-7 | C20H25F3N8S |
| —— | cyclopentyl-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-amine | 1215167-60-4 | C20H24F3N7S |
| —— | N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-methanesulfonamide | 1215221-80-9 | C18H22F3N7O3S2 |
| —— | 2-cyano-N-{(S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidin-3-yl}-acetamide | 1215209-93-0 | C22H24F3N9OS |
| —— | (S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidine-3-carboxylic acid 2,2-dimethyl-propionyloxymethyl ester | 1215205-08-5 | C26H32F3N7O4S |
| —— | {(R)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidin-3-yl}-carbamic acid tert-butyl ester | 1215167-40-0 | C24H31F3N8O2S |
| —— | [6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-acetic acid | 1215214-49-5 | C17H17F3N6O3S |
| —— | 2-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-thiazol-4-yl}-ethanol | 1215226-35-9 | C20H20F3N7OS2 |
| —— | 2-(1H-imidazol-4-yl)-N-{(S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidin-3-yl}-acetamide | 1215210-13-1 | C24H27F3N10OS |
| —— | 1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-piperidine-3-carboxylic acid dimethylamide | 1215205-69-8 | C23H29F3N8OS |
| —— | (S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidine-3-carboxylic acid dimethylamide | 1215205-60-9 | C22H27F3N8OS |
| —— | 2-[[6-ethyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-(2-hydroxy-ethyl)-amino]-ethanol | 1215210-42-6 | C18H22F3N7O2S |
| —— | {2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxymethyl]-oxazol-4-yl}-acetic acid ethyl ester | 1215214-73-5 | C23H24F3N7O4S |
| —— | 2-[2-(5,8-Dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethenyl]-5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazine | 1384868-06-7 | C16H16N8 |
| —— | 2-[6-butyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-ylamino]-ethanol | 1215214-11-1 | C18H22F3N7OS |
| —— | (R)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)thieno[2,3-d]pyrimidin-2-ylmethyl]pyrrolidin-3-ol | 1215222-14-2 | C20H24F3N7OS |
| —— | (S)-1-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yl]-pyrrolidine-3-carboxylic acid | 1215205-06-3 | C20H22F3N7O2S |
| —— | 8-N-benzyl-[1,2,4]triazolo[1,5-a]pyrazine-2,8-diamine | 1360612-79-8 | C12H12N6 |
| —— | 5,8-dimethyl-2-[2-(2-methyl-5-thiazol-5-yl-2H-[1,2,4]triazol-3-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-54-4 | C15H16N8S |
| —— | 6-(2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl)-3-ethyl-4-methyl-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine | 1612163-58-2 | C19H24N6O |
| —— | 2-[2-(2-furan-3-yl-1H-imidazol-4-yl)-ethyl]-5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazine | 1312325-55-5 | C16H16N6O |
| —— | 2-[2-(5-furan-2-yl-1-methyl-1H-[1,2,4]triazol-3-yl)-ethyl]-5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-45-3 | C16H17N7O |
| —— | 2-[2-(2-furan-2-yl-1H-imidazol-4-yl)-ethyl]-5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazine | 1312325-57-7 | C16H16N6O |
| —— | (6-chloro-pyrazolo[1,5-a]pyrimidin-2-yl)-(8-methyl-3-thiophen-2-yl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-methanone | 1174647-51-8 | C17H14ClN7OS |
| —— | 5,8-dimethyl-2-{2-[2-methyl-5-(5-methyl-thiazol-2-yl)-2H-[1,2,4]triazol-3-yl]-ethyl}-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-48-6 | C16H18N8S |
| —— | 5,8-dimethyl-2-[2-(2-methyl-5-thiazol-2-yl-2H-[1,2,4]triazol-3-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-55-5 | C15H16N8S |
| —— | (6-chloro-pyrazolo[1,5-a]pyrimidin-2-yl)-(3-furan-3-yl-8-methyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-methanone | 1174647-78-9 | C17H14ClN7O2 |
| —— | (6-bromo-pyrazolo[1,5-a]pyrimidin-2-yl)-(1-methyl-6-thiophen-3-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl)-methanone | 1174646-89-9 | C19H16BrN5OS |
| —— | 5,8-dimethyl-2-[2-(2-methyl-5-oxazol-2-yl-2H-[1,2,4]triazol-3-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-50-0 | C15H16N8O |
| —— | 5,8-dimethyl-2-[2-(2-thiazol-2-yl-1H-imidazol-4-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312325-54-4 | C15H15N7S |
| —— | 5,8-dimethyl-2-[2-(2-methyl-5-thiophen-2-yl-2H-[1,2,4]triazol-3-yl)-ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | 1312301-51-1 | C16H17N7S |
| —— | 6-(2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl)-3,4-dimethyl-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine | 1612163-50-4 | C18H22N6O |