| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 1-[3-[(2R)-1-acetylpiperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C14H21N5O2 |
| —— | 3-(2-methylphenoxy)-1-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]propan-1-one | —— | C19H25N5O2 |
| —— | (3-methyl-1-benzofuran-2-yl)-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone | —— | C19H21N5O2 |
| —— | 3-cyclopentyl-1-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]propan-1-one | —— | C19H31N5O |
| —— | 7-(4,6-dimethylpyrimidin-2-yl)-3-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C16H23N7 |
| —— | 3-[(2S)-1-[(4-fluorophenyl)methylsulfonyl]piperidin-2-yl]-7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C18H24FN5O2S |
| —— | 3-(2-methylphenoxy)-1-[3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]propan-1-one | —— | C19H25N5O2 |
| —— | 3-[(2R)-1-[(4-fluorophenyl)methylsulfonyl]piperidin-2-yl]-7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C18H24FN5O2S |
| —— | 7-methyl-3-[(2R)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C19H27N5O2S |
| —— | 3-[(2S)-1-[(3-fluorophenyl)methylsulfonyl]piperidin-2-yl]-7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C18H24FN5O2S |
| —— | 1-[3-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C15H19N7O |
| —— | 1-[3-[(2S)-1-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C21H27N5O3 |
| —— | [(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone | —— | C16H22N6OS |
| —— | 7-methyl-3-[(2R)-1-(2-phenylethylsulfonyl)piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C19H27N5O2S |
| —— | 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C21H29N5O |
| —— | [3-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C20H27N5O2 |
| —— | [3-[(2R)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C20H27N5O2 |
| —— | 3-(4-methoxyphenyl)-1-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H27N5O2 |
| —— | 2-(2,4-difluorophenoxy)-1-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]ethanone | —— | C18H21F2N5O2 |
| —— | 1-[3-[(2R)-1-[[4-ethoxy-3-(hydroxymethyl)phenyl]methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C21H29N5O3 |
| —— | 1-[3-[(2R)-1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | (3-methoxyphenyl)-[3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone | —— | C17H21N5O2 |
| —— | 3-(4-methoxyphenyl)-1-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H27N5O2 |
| —— | 7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C18H25N5O |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H28N6O2 |
| —— | 1-[3-[(2S)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | 1-[3-[(2R)-1-(3-methoxybenzoyl)pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C19H23N5O3 |
| —— | 1-[3-[(2R)-1-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C21H27N5O3 |
| —— | 3-[(2R)-1-methylpyrrolidin-2-yl]-7-pyrimidin-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C14H19N7 |
| —— | 3-(4-methoxyphenyl)-1-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]propan-1-one | —— | C19H25N5O2 |
| —— | 1-[3-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C15H19N7O |
| —— | 1-[(2S)-2-(7-acetyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one | —— | C21H27N5O3 |
| —— | [4-(ethoxymethyl)phenyl]-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone | —— | C19H25N5O2 |
| —— | 1-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]-2-phenoxyethanone | —— | C18H23N5O2 |
| —— | 2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H27N5O3 |
| —— | 2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H27N5O3 |
| —— | [4-(ethoxymethyl)phenyl]-[3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone | —— | C19H25N5O2 |
| —— | 1-[3-[(2S)-1-(3-methoxybenzoyl)pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C19H23N5O3 |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H28N6O2 |
| —— | 1-[3-[(2R)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | (2R)-N,N-diethyl-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidine-1-sulfonamide | —— | C14H26N6O2S |
| —— | 1-[3-[(2S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C22H29N5O2 |
| —— | 1-[3-[(2S)-1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | 1-[3-[(2R)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C22H29N5O2 |
| —— | (3,5-dimethyl-1,2-oxazol-4-yl)-[3-(hydroxymethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone | —— | C12H15N5O3 |
| —— | 1-[(2R)-2-(7-acetyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one | —— | C21H27N5O3 |
| —— | 7-methyl-3-[(2S)-1-propan-2-ylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine | —— | C13H23N5 |
| —— | [3-(hydroxymethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(5-propylfuran-2-yl)methanone | —— | C14H18N4O3 |
| —— | 1-[3-[(2R)-1-(3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C21H23N5O3 |
| —— | 1-[3-[(2S)-1-[4-(ethoxymethyl)benzoyl]pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]ethanone | —— | C21H27N5O3 |