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吡啶二氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-3-ylmethanone —— C18H24N4OS
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-3-ylmethanone
—— 1-methyl-4-pyridin-2-yl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H16N4
1-methyl-4-pyridin-2-yl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1-methylpyrrol-2-yl)methanone —— C18H22N4O
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1-methylpyrrol-2-yl)methanone
—— N,N-dimethyl-2-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanamine —— C18H28N6
N,N-dimethyl-2-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanamine
—— [(2S)-oxolan-2-yl]-[1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C19H22N4O2
[(2S)-oxolan-2-yl]-[1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]-N,N-dimethylethanamine —— C18H27N5O
2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]-N,N-dimethylethanamine
—— 4-(cyclopropylmethyl)-8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C18H25N5
4-(cyclopropylmethyl)-8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-(1-prop-2-enyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carbonyl)benzonitrile —— C19H18N4O
4-(1-prop-2-enyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carbonyl)benzonitrile
—— 8-methyl-4-(oxan-4-yl)-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C20H26N4O
8-methyl-4-(oxan-4-yl)-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-morpholin-4-ylmethanone —— C18H29N5O2
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-morpholin-4-ylmethanone
—— 1,8-dimethyl-4-[(1-methylpyrazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C15H21N5
1,8-dimethyl-4-[(1-methylpyrazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-2-pyridin-2-ylethanone —— C16H18N4O
1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-2-pyridin-2-ylethanone
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(furan-2-yl)methanone —— C18H24N4O2
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(furan-2-yl)methanone
—— 1-(2-methoxyethyl)-4-(6-methoxypyrimidin-4-yl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H23N5O2
1-(2-methoxyethyl)-4-(6-methoxypyrimidin-4-yl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrrolidin-1-ylmethanone —— C17H26N4O2
[1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrrolidin-1-ylmethanone
—— cyclopent-3-en-1-yl-[1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C17H23N3O2
cyclopent-3-en-1-yl-[1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 1-(2-methoxyethyl)-8-methyl-4-(6-methylpyridin-2-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C18H24N4O
1-(2-methoxyethyl)-8-methyl-4-(6-methylpyridin-2-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-methyl-4-(5-methylpyrimidin-2-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H17N5
1-methyl-4-(5-methylpyrimidin-2-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-(benzenesulfonyl)-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H21N3O3S
4-(benzenesulfonyl)-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— cyclopent-3-en-1-yl-[8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C21H24N4O
cyclopent-3-en-1-yl-[8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 4-ethylsulfonyl-8-methyl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H22N4O2S
4-ethylsulfonyl-8-methyl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(furan-3-yl)methanone —— C18H24N4O2
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(furan-3-yl)methanone
—— 3,5-dimethyl-4-[[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methyl]-1,2-oxazole —— C20H23N5O
3,5-dimethyl-4-[[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methyl]-1,2-oxazole
—— pyridazin-4-yl-[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C19H18N6O
pyridazin-4-yl-[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 3-[(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)methyl]benzonitrile —— C17H18N4
3-[(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)methyl]benzonitrile
—— pyridin-4-yl-[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C20H19N5O
pyridin-4-yl-[1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— N-propan-2-yl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C17H24N6O
N-propan-2-yl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 4-cyclopropylsulfonyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C12H17N3O2S
4-cyclopropylsulfonyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyridin-3-ylmethanone —— C18H20N4O
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyridin-3-ylmethanone
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-2-ylmethanone —— C17H19N3OS
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-2-ylmethanone
—— 1-[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-2-methoxyethanone —— C15H21N3O2
1-[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-2-methoxyethanone
—— 1-prop-2-enyl-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H19N3S
1-prop-2-enyl-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— (1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-(1-methylpyrrol-2-yl)methanone —— C15H18N4O
(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-(1-methylpyrrol-2-yl)methanone
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(oxan-4-yl)methanone —— C18H25N3O2
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(oxan-4-yl)methanone
—— N,N,1-trimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C12H18N4O
N,N,1-trimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 1-(2-methoxyethyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C12H19N3O3S
1-(2-methoxyethyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-(cyclopropylmethyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C13H19N3O2S
1-(cyclopropylmethyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrrolidin-1-ylmethanone —— C17H24N4O
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrrolidin-1-ylmethanone
—— 4-ethylsulfonyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C11H17N3O2S
4-ethylsulfonyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-cyclopropylsulfonyl-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H21N3O3S
4-cyclopropylsulfonyl-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-[(4-fluorophenyl)methyl]-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H18FN3
4-[(4-fluorophenyl)methyl]-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-methyl-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C10H15N3O2S
1-methyl-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-ethylsulfonyl-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C13H21N3O3S
4-ethylsulfonyl-1-(2-methoxyethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— (1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-pyrrolidin-1-ylmethanone —— C14H20N4O
(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-pyrrolidin-1-ylmethanone
—— 2-methoxy-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)ethanone —— C12H17N3O2
2-methoxy-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)ethanone
—— 1-methyl-4-(6-methylpyridazin-3-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H17N5
1-methyl-4-(6-methylpyridazin-3-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-(cyclopropylmethyl)-4-ethylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H21N3O2S
1-(cyclopropylmethyl)-4-ethylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 9-(2-Chlorophenyl)-6,13-dimethyl-2,4,5,8,12-pentazatricyclo[8.4.0.03,7]tetradeca-1(10),3,6,8,11,13-hexaene —— C17H14ClN5
9-(2-Chlorophenyl)-6,13-dimethyl-2,4,5,8,12-pentazatricyclo[8.4.0.03,7]tetradeca-1(10),3,6,8,11,13-hexaene
—— 9-methoxy-10-[(5R)-2-oxa-9-azaspiro[4.5]decane-9-carbonyl]-2,3,4,5-tetrahydro-1H-pyrido[1,2-d][1,4]diazepin-7-one —— C19H27N3O4
9-methoxy-10-[(5R)-2-oxa-9-azaspiro[4.5]decane-9-carbonyl]-2,3,4,5-tetrahydro-1H-pyrido[1,2-d][1,4]diazepin-7-one
—— 9-methoxy-10-[(5S)-2-oxa-9-azaspiro[4.5]decane-9-carbonyl]-2,3,4,5-tetrahydro-1H-pyrido[1,2-d][1,4]diazepin-7-one —— C19H27N3O4
9-methoxy-10-[(5S)-2-oxa-9-azaspiro[4.5]decane-9-carbonyl]-2,3,4,5-tetrahydro-1H-pyrido[1,2-d][1,4]diazepin-7-one