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吡啶二氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Isobutyl-4,5-dihydro-1H-pyrido[2,3-b][1,4]diazepin-2(3H)-one —— C12H17N3O
5-Isobutyl-4,5-dihydro-1H-pyrido[2,3-b][1,4]diazepin-2(3H)-one
—— 5-Cyclopropylmethyl-2,3,4,5-tetrahydro-1H-pyrido[3,4-b][1,4]diazepine —— C12H17N3
5-Cyclopropylmethyl-2,3,4,5-tetrahydro-1H-pyrido[3,4-b][1,4]diazepine
—— 1-Isobutyl-2,3-dihydro-1H-pyrido[3,4-b][1,4]diazepin-4(5H)-one —— C12H17N3O
1-Isobutyl-2,3-dihydro-1H-pyrido[3,4-b][1,4]diazepin-4(5H)-one
—— 8-methyl-N-propan-2-yl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C18H26N6O
8-methyl-N-propan-2-yl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— N-cyclopropyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C13H18N4O
N-cyclopropyl-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 4-[(5-ethylfuran-2-yl)methyl]-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H21N3O
4-[(5-ethylfuran-2-yl)methyl]-1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-[[4-(furan-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]methyl]-2-methyl-1,3-thiazole —— C18H20N4OS
4-[[4-(furan-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]methyl]-2-methyl-1,3-thiazole
—— 1-(cyclopropylmethyl)-4-(furan-2-ylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C18H23N3O
1-(cyclopropylmethyl)-4-(furan-2-ylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 2-ethyl-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)butan-1-one —— C15H23N3O
2-ethyl-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)butan-1-one
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-2-ylmethanone —— C18H24N4OS
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-thiophen-2-ylmethanone
—— 8-methyl-4-methylsulfonyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H20N4O2S
8-methyl-4-methylsulfonyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— N-cyclopropyl-1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C17H24N4O
N-cyclopropyl-1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 1-[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]butan-1-one —— C17H28N4O
1-[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]butan-1-one
—— 1-(cyclopropylmethyl)-4-cyclopropylsulfonyl-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H23N3O2S
1-(cyclopropylmethyl)-4-cyclopropylsulfonyl-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— (1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-thiophen-3-ylmethanone —— C15H17N3OS
(1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)-thiophen-3-ylmethanone
—— 8-methyl-4-(oxan-4-yl)-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C19H27N5O
8-methyl-4-(oxan-4-yl)-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 8-methyl-4-(pyridin-2-ylmethyl)-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C21H23N5
8-methyl-4-(pyridin-2-ylmethyl)-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— cyclopropyl-(1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)methanone —— C14H19N3O
cyclopropyl-(1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)methanone
—— 4-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H22N4O
4-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— N-propan-2-yl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C18H23N5O
N-propan-2-yl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 4-ethylsulfonyl-8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H23N5O2S
4-ethylsulfonyl-8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 2-cyclopropyl-1-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone —— C19H25N5O
2-cyclopropyl-1-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone
—— cyclobutyl-[8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C20H24N4O
cyclobutyl-[8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 1-[1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-3-methoxypropan-1-one —— C17H25N3O2
1-[1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-3-methoxypropan-1-one
—— 2-(3-fluorophenyl)-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)ethanone —— C17H18FN3O
2-(3-fluorophenyl)-1-(1-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl)ethanone
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1,3-thiazol-4-yl)methanone —— C17H23N5OS
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1,3-thiazol-4-yl)methanone
—— 1-(2-methoxyethyl)-8-methyl-4-propylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C15H25N3O3S
1-(2-methoxyethyl)-8-methyl-4-propylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— N-cyclopropyl-1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C14H20N4O
N-cyclopropyl-1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 2-methoxy-1-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone —— C17H23N5O2
2-methoxy-1-[8-methyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone
—— [1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1H-pyrrol-2-yl)methanone —— C18H25N5O
[1-[2-(dimethylamino)ethyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(1H-pyrrol-2-yl)methanone
—— 4-ethylsulfonyl-8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H22N4O2S
4-ethylsulfonyl-8-methyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— N-cyclopropyl-1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C16H24N4O2
N-cyclopropyl-1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— [1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrazin-2-ylmethanone —— C17H19N5O
[1-(cyclopropylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-pyrazin-2-ylmethanone
—— 8-methyl-4-methylsulfonyl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C16H20N4O2S
8-methyl-4-methylsulfonyl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 8-methyl-4-[(1-methylpyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C20H24N6
8-methyl-4-[(1-methylpyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— [1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(3-fluoropyridin-4-yl)methanone —— C19H21FN4O
[1-(cyclopropylmethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-(3-fluoropyridin-4-yl)methanone
—— 1-(2-methoxyethyl)-8-methyl-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C13H21N3O3S
1-(2-methoxyethyl)-8-methyl-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 4-[[1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methyl]-3,5-dimethyl-1,2-oxazole —— C18H26N4O2
4-[[1-(2-methoxyethyl)-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methyl]-3,5-dimethyl-1,2-oxazole
—— 3-methoxy-1-[8-methyl-1-(2-methylpropyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]propan-1-one —— C17H27N3O2
3-methoxy-1-[8-methyl-1-(2-methylpropyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]propan-1-one
—— 4-(furan-2-ylmethyl)-1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C15H19N3O
4-(furan-2-ylmethyl)-1,8-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 8-methyl-4-methylsulfonyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C15H21N5O2S
8-methyl-4-methylsulfonyl-1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-[8-methyl-1-(2-methylpropyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-2-pyridin-2-ylethanone —— C20H26N4O
1-[8-methyl-1-(2-methylpropyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]-2-pyridin-2-ylethanone
—— 2-cyclopropyl-1-[1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone —— C19H22N4O
2-cyclopropyl-1-[1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]ethanone
—— 2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]-N,N-dimethylethanamine —— C19H29N5O
2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-8-methyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-1-yl]-N,N-dimethylethanamine
—— [(2R)-oxolan-2-yl]-[1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone —— C18H23N5O2
[(2R)-oxolan-2-yl]-[1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]methanone
—— 1,8-dimethyl-N-propan-2-yl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide —— C14H22N4O
1,8-dimethyl-N-propan-2-yl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
—— 1-[1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]propan-1-one —— C16H21N5O
1-[1-(2-pyrazol-1-ylethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepin-4-yl]propan-1-one
—— 1-(2-methoxyethyl)-8-methyl-4-(6-methylpyridazin-3-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C17H23N5O
1-(2-methoxyethyl)-8-methyl-4-(6-methylpyridazin-3-yl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 8-methyl-1-(2-methylpropyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C14H23N3O2S
8-methyl-1-(2-methylpropyl)-4-methylsulfonyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine
—— 1-(cyclopropylmethyl)-8-methyl-4-[(1-methylpyrazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine —— C18H25N5
1-(cyclopropylmethyl)-8-methyl-4-[(1-methylpyrazol-4-yl)methyl]-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine