| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | [D-Ala17]orexin-B | —— | C123H212N44O35S |
| —— | [Trp11]orexin-B | —— | C128H211N45O35S |
| —— | [D-Ala22]orexin-B | —— | C123H212N44O35S |
| —— | (2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-4-[(1S,2R)-2-aminocyclopropyl]-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-hydroxybutanoyl]amino]butanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acid | —— | C95H172N36O28 |
| —— | [D-Leu11]orexin-B | —— | C123H212N44O35S |
| —— | [D-Ala6]orexin-B | —— | C124H214N44O35S |
| —— | [Ala2]orexin-B | —— | C123H212N44O34S |
| —— | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(3S,6R,9S,14S,17R,20S,23R,26S,29R,32S,35R)-3-(2-amino-2-oxoethyl)-29-[(2S)-butan-2-yl]-23,32-bis(3-carbamimidamidopropyl)-6,26-bis(carboxymethyl)-17-[(4-hydroxyphenyl)methyl]-20-(1H-indol-3-ylmethyl)-9-[[(2S)-4-methyl-2-[[(2S)-2-(quinoline-2-carbonylamino)propanoyl]amino]pentanoyl]amino]-2,5,8,16,19,22,25,28,31,34-decaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33-decazabicyclo[33.3.0]octatriacontane-14-carbonyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]-5-[(2-amino-2-oxoethyl)amino]-5-oxopentanoic acid | —— | C106H145N29O28S2 |
| —— | [Ala15]orexin-B | —— | C120H206N44O35S |
| —— | F-G-G-F-T-G-A-R-K-S-A-R-K-L-Aib-N-Q-CONH2 | —— | C80H132N28O21 |
| —— | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-carboxypropanoyl]amino]propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]-5-[[(2S)-1-[[(3S,6S,9S,12S,15S,18R,23R,26S,29S)-23-[[(2R,3R)-1-[[(2R)-1-[[(2R)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-12-[(4-hydroxyphenyl)methyl]-15,26-bis(1H-imidazol-5-ylmethyl)-3-(2-methylpropyl)-2,5,8,11,14,17,25,28-octaoxo-6-[4-[[2-[2-oxo-2-[4-[3-oxo-3-(2-oxoazetidin-1-yl)propyl]anilino]ethoxy]acetyl]amino]butyl]-20,21-dithia-1,4,7,10,13,16,24,27-octazabicyclo[27.3.0]dotriacontan-18-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-oxopentanoic acid | —— | C116H161N29O31S2 |
| —— | [Ala16]orexin-B | —— | C121H209N43O34S |
| —— | Glu-Ser-OctSer-phe-Leu-Ser-Pro-Glu-Arg-Val_Gln-Gln-Arg-Lys-Glu Ser-Lys-Lys-Pro-Pro-Pro-Ala-Lya-Leu-Gln-Pro-Arg | —— | C154H256N48O43 |
| —— | [Ala9]orexin-B | —— | C124H214N44O35S |
| —— | [D-Gln12]orexin-B | —— | C123H212N44O35S |
| —— | (4S)-5-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[2-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-1-oxohexan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-carboxy-1-oxobutan-2-yl]amino]-4-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[2-[[(2S)-2-[[(2S)-1-[2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-hydroxypropanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]acetyl]amino]-3-hydroxybutanoyl]amino]-4-methylpentanoyl]amino]propanoyl]amino]-5-oxopentanoic acid | —— | C126H195N37O37 |
| —— | (4S)-5-[[(2S)-1-[[(2S)-1-[[(2S)-4-amino-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-6-amino-1-[[2-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[di(piperidin-1-yl)amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1,4-dioxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-carboxy-1-oxobutan-2-yl]amino]-4-[[(2S)-2-[[(2S)-2-[[(2S)-4-amino-2-[[2-[[(2S)-2-[[(2S)-1-[2-[[(2S)-2-[[(2S,3R)-2-amino-3-hydroxybutanoyl]amino]-3-hydroxypropanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]acetyl]amino]-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]propanoyl]amino]-5-oxopentanoic acid | —— | C137H213N39O37 |
| —— | N-[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-acetamido-4-methylpentanoyl]amino]-3-hydroxybutanoyl]amino]-3-phenylpropanoyl]amino]-6-(2-methylprop-2-enoylamino)hexanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-6-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]-2-(4-methoxyphenyl)tetrazole-5-carboxamide | —— | C91H127N25O20 |
| —— | [Ala5]orexin-B | —— | C122H211N45O36S |
| —— | [Ala12]orexin-B | —— | C121H209N43O34S |
| —— | [D-Ala9]orexin-B | —— | C124H214N44O35S |
| —— | F-G-G-F-T-G-MeA-R-K-S-A-R-K-L-A-N-Q-CONH2 | —— | C80H132N28O21 |
| —— | SALRHYINLITRQRY | 718628-68-3 | C85H138N28O22 |
| —— | [Ala25]orexin-B | —— | C120H206N44O35S |
| —— | [Gly17]orexin-B | —— | C122H210N44O35S |
| —— | F-G-G-F-T-G-Aib-R-K-S-A-R-K-L-A-N-Q-COOH | —— | C80H131N27O22 |
| —— | [Ala26]orexin-B | —— | C120H206N44O35S |
| —— | [Ala14]orexin-B | —— | C120H206N44O35S |
| —— | DOTA-ReCCEHdFRWCKPVD-OH | —— | C79H112N25O25ReS3-5 |
| —— | [D-Ser2]orexin-B | —— | C123H212N44O35S |
| —— | 3-[(3S,6R,9S,14S,17R,20S,23R,26S,29R,32S,35R)-14-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[(2-amino-2-oxoethyl)amino]-4-carboxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1,5-dioxopentan-2-yl]carbamoyl]-3-(2-amino-2-oxoethyl)-29-[(2S)-butan-2-yl]-23-(3-carbamimidamidopropyl)-6,26-bis(carboxymethyl)-17-[(4-hydroxyphenyl)methyl]-20-(1H-indol-3-ylmethyl)-9-[[(2S)-4-methyl-2-[[(2S)-2-[[5-(2-nitrophenyl)furan-2-carbonyl]amino]propanoyl]amino]pentanoyl]amino]-2,5,8,16,19,22,25,28,31,34-decaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33-decazabicyclo[33.3.0]octatriacontan-32-yl]propyl-[amino(azaniumylidene)methyl]azanide | —— | C107H145N29O31S2 |
| —— | 5-[[1-[[(2S)-1-[[5-carbamimidamido-1-[[1-[[2-[[5-carbamimidamido-1-[2-[(1-carboxy-2-methylpropyl)carbamoyl]pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-2-oxo-1-sulfanylethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-5-oxo-4-[[2-sulfanyl-2-[[2-sulfanyl-2-[[2-[4,7,10-tris(carboxymethyl)-1,4,7,10-tetrazacyclododec-1-yl]acetyl]amino]acetyl]amino]acetyl]amino]pentanoic acid | —— | C75H110N24O21S3 |
| —— | [Gly23]orexin-B | —— | C122H210N44O35S |
| —— | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(3S,6R,9S,14S,17R,20S,23R,26S,29R,32S,35R)-3-(2-amino-2-oxoethyl)-29-[(2S)-butan-2-yl]-23,32-bis(3-carbamimidamidopropyl)-6,26-bis(carboxymethyl)-17-[(4-hydroxyphenyl)methyl]-20-(1H-indol-3-ylmethyl)-9-[[(2S)-4-methyl-2-[[(2S)-2-[(4-phenylbenzoyl)amino]propanoyl]amino]pentanoyl]amino]-2,5,8,16,19,22,25,28,31,34-decaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33-decazabicyclo[33.3.0]octatriacontane-14-carbonyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]-5-[(2-amino-2-oxoethyl)amino]-5-oxopentanoic acid | —— | C109H148N28O28S2 |
| —— | 2-[(3R,6S,9R,14S,17R,20S,23R,26S,29R,32S,38S)-14-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-9-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-3-benzyl-20-[(2S)-butan-2-yl]-23,32-bis(3-carbamimidamidopropyl)-17-(hydroxymethyl)-6-(1H-imidazol-5-ylmethyl)-29-(2-methylsulfanylethyl)-2,5,8,16,19,22,25,28,31,34,37-undecaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33,36-undecazabicyclo[36.3.0]hentetracontan-26-yl]acetic acid | —— | C78H121N27O19S4 |
| —— | [D-Arg13]orexin-B | —— | C123H212N44O35S |
| —— | 2-[(4S,7R,10S,13R,16S,19R,22S,28S,31R,34R)-4-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-34-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-28-benzyl-10-[(2S)-butan-2-yl]-13,22-bis(3-carbamimidamidopropyl)-7-(hydroxymethyl)-31-(1H-imidazol-5-ylmethyl)-19-(2-methylsulfanylethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-16-yl]acetic acid | —— | C73H114N26O18S4 |
| —— | 2-[(4S,7R,10S,13R,16S,19R,22S,31R,34S,37R)-4-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-37-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-31-benzyl-10-[(2S)-butan-2-yl]-13,22-bis(3-carbamimidamidopropyl)-7-(hydroxymethyl)-34-(1H-imidazol-5-ylmethyl)-19-(2-methylsulfanylethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacont-16-yl]acetic acid | —— | C75H117N27O19S4 |
| —— | F-G-G-F-T-G-Aib-R-K-S-A-R-K-L-A-N-Q-CONH2 | —— | C80H132N28O21 |
| —— | (alpha-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | —— | C77H99N19O19S2 |
| —— | 2-[(4S,7R,10S,13R,16S,19R,22S,31R,34S,37R)-4-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-37-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-31-benzyl-10-[(2S)-butan-2-yl]-13,22-bis(3-carbamimidamidopropyl)-7-(hydroxymethyl)-34-(1H-imidazol-5-ylmethyl)-19-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacont-16-yl]acetic acid | —— | C73H113N27O19S3 |
| —— | F-G-G-F-T-G-A-R-K-S-A-R-K-L-MeA-N-Q-CONH2 | —— | C80H132N28O21 |
| —— | 2-[(3R,12R,15S,18R,23R,26S,29R,32S,35R,38S)-23-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-18-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-12-benzyl-29-[(2S)-butan-2-yl]-3,32-bis(3-carbamimidamidopropyl)-26-(hydroxymethyl)-15-(1H-imidazol-5-ylmethyl)-2,5,8,11,14,17,25,28,31,34,37-undecaoxo-20,21-dithia-1,4,7,10,13,16,24,27,30,33,36-undecazabicyclo[36.3.0]hentetracontan-35-yl]acetic acid | —— | C75H115N27O19S3 |
| —— | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(3S,6R,9S,14S,17R,20S,23R,26S,29R,32S,35R)-3-(2-amino-2-oxoethyl)-29-[(2S)-butan-2-yl]-23,32-bis(3-carbamimidamidopropyl)-6,26-bis(carboxymethyl)-17-[(4-hydroxyphenyl)methyl]-20-(1H-indol-3-ylmethyl)-9-[[(2S)-4-methyl-2-[[(2S)-2-[(3-methylphenyl)carbamoylamino]propanoyl]amino]pentanoyl]amino]-2,5,8,16,19,22,25,28,31,34-decaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33-decazabicyclo[33.3.0]octatriacontane-14-carbonyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]-5-[(2-amino-2-oxoethyl)amino]-5-oxopentanoic acid | —— | C104H147N29O28S2 |
| —— | [Pro7]mintANP | —— | C74H112N24O19S4 |
| —— | [Ala13]orexin-B | —— | C120H205N41O35S |
| —— | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(3S,6R,9S,14S,17R,20S,23R,26S,29R,32S,35R)-3-(2-amino-2-oxoethyl)-29-[(2S)-butan-2-yl]-23,32-bis(3-carbamimidamidopropyl)-6,26-bis(carboxymethyl)-17-[(4-hydroxyphenyl)methyl]-20-(1H-indol-3-ylmethyl)-9-[[(2S)-4-methyl-2-[[(2S)-2-(quinoline-3-carbonylamino)propanoyl]amino]pentanoyl]amino]-2,5,8,16,19,22,25,28,31,34-decaoxo-11,12-dithia-1,4,7,15,18,21,24,27,30,33-decazabicyclo[33.3.0]octatriacontane-14-carbonyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]-5-[(2-amino-2-oxoethyl)amino]-5-oxopentanoic acid | —— | C106H145N29O28S2 |
| —— | 2-[(6R,9S,12R,17S,20R,23S,26R,29S,32R,35S,38R)-17-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-12-[[(2S)-2-amino-4-methylsulfanylbutanoyl]amino]-6-benzyl-23-[(2S)-butan-2-yl]-26,35-bis(3-carbamimidamidopropyl)-20-(hydroxymethyl)-9-(1H-imidazol-5-ylmethyl)-32-(2-methylsulfanylethyl)-2,5,8,11,19,22,25,28,31,34,37-undecaoxo-14,15-dithia-1,4,7,10,18,21,24,27,30,33,36-undecazabicyclo[36.3.0]hentetracontan-29-yl]acetic acid | —— | C78H121N27O19S4 |
| —— | [D-Pro4]orexin-B | —— | C123H212N44O35S |
| —— | F-G-G-F-T-G-A-R-K-S-MeA-R-K-L-A-N-Q-COOH | —— | C80H131N27O22 |