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三唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H29N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O4
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O4
(7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O3
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3S
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H26ClN5O3S
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O4
(7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O3S
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H19ClF3N5O3
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— methyl (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H22N4O5
methyl (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H29N5O5
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O4
(7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O3S
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O4
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 1-[(7S)-2-benzyl-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C24H24N4O3
1-[(7S)-2-benzyl-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— (7R)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7R)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H22F3N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H19ClF3N5O3
(7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O4
(7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4S
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O3
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3S
(7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O3
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O3
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O5
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O5
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— methyl (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H22N4O4S
methyl (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4S
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(furan-2-yl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(furan-2-yl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24ClN5O3
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide