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三唑并嘧啶类

中文名称 英文名称 CAS号 化学式
—— N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]propanamide —— C19H23F3N6OS
—— N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]propanamide —— C19H23F3N6OS
—— 2-(5,7-dimethyl-2-methylsulfanyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]acetamide —— C20H24N8OS2
—— 2-(5,7-dimethyl-2-methylsulfanyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]acetamide —— C20H24N8OS2
—— N-[(1R)-1-(4-chlorophenyl)ethyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C18H20ClN5O
—— N-[(1S)-1-(2,4-difluorophenyl)ethyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C18H19F2N5O
—— N-[(2,4-dichlorophenyl)methyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-methylpropanamide —— C18H19Cl2N5O
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[(1S)-1-(4-methylphenyl)propyl]propanamide —— C20H25N5O
—— N-[(1S)-1-(3,4-diethoxyphenyl)ethyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C22H29N5O3
—— N-(3,4-difluorophenyl)-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C16H15F2N5O
—— (2R)-N'-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoyl]-2-(4-fluorophenoxy)propanehydrazide —— C19H21FN6O3
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]propanamide —— C22H29N5O
—— N-[(1R)-1-(2,4-dichloro-5-fluorophenyl)ethyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C18H18Cl2FN5O
—— N-(3-cyanophenyl)-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C17H16N6O
—— N-[4-(difluoromethoxy)phenyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C17H17F2N5O2
—— N'-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoyl]-4-ethoxybenzohydrazide —— C19H22N6O3
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[(2S)-2-phenylpropyl]propanamide —— C19H23N5O
—— N-[(5-chlorothiophen-2-yl)methyl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-prop-2-enylpropanamide —— C18H20ClN5OS
—— N'-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoyl]-2,5-dimethylfuran-3-carbohydrazide —— C17H20N6O3
—— 1-[3-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoylamino]-3-(4-fluorophenyl)thiourea —— C17H18FN7OS
—— 1-Tert-butyl-3-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoylamino]thiourea —— C15H23N7OS
—— N'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)acetohydrazide —— C16H20N8O2
—— 3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]propan-1-one —— C20H20F3N5O
—— 3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]propan-1-one —— C20H20F3N5O
—— 3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[(1R)-1-(4-methoxyphenyl)-2-methylpropyl]propanamide —— C22H26F3N5O2
—— [(2S)-1-[(1-cyanocyclohexyl)amino]-1-oxopropan-2-yl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H22N6O3
—— [2-(5-Bromothiophen-2-yl)-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C14H11BrN4O3S
—— [(2R)-1-(3,5-dichloroanilino)-1-oxopropan-2-yl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C17H15Cl2N5O3
—— (2-Morpholin-4-yl-2-oxoethyl) 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C14H17N5O4
—— [(2S)-1-(1H-indol-3-yl)-1-oxopropan-2-yl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C19H17N5O3
—— [2-[[(1S)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C16H18N6O3
—— [2-[[(2R)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C16H20N6O3
—— [2-(4-Ethoxycarbonylpiperidin-1-yl)-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H23N5O5
—— [(1R)-1-cyanoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C11H11N5O2
—— [2-(2,6-Difluoroanilino)-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C16H13F2N5O3
—— [2-[[(1S)-1-(2,4-difluorophenyl)ethyl]amino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H17F2N5O3
—— [2-(2,5-Dimethyl-1-propan-2-ylpyrrol-3-yl)-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C19H23N5O3
—— [(2S)-1-[benzyl(methyl)amino]-1-oxopropan-2-yl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C19H21N5O3
—— [(2R)-1-(3-methoxyanilino)-1-oxopropan-2-yl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H19N5O4
—— [2-[(2-Methoxyphenyl)methylamino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H19N5O4
—— [2-[[(1S)-1-(1-adamantyl)ethyl]amino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C22H29N5O3
—— [2-[[(1R)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C16H18N6O3
—— N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)acetamide —— C19H20ClN5O3
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-(5-fluoro-2-methylphenyl)propanamide —— C17H18FN5O
—— N-(4-chloro-2-fluorophenyl)-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C16H15ClFN5O
—— 3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[2-(4-fluorophenyl)ethyl]propanamide —— C19H19F4N5O
—— N-[(2-chlorophenyl)methyl]-3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]propanamide —— C18H17ClF3N5O
—— 2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]acetamide —— C21H25N5O3
—— 3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-N-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]propanamide —— C22H27N5O3
—— N-[4-(3,4-dimethylphenyl)-1,3-thiazol-2-yl]-3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanamide —— C21H22N6OS