| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | N-[2-(diaminomethylideneamino)oxyethyl]-2-[(3S)-3-[[4-(4-methylphenyl)phenyl]sulfonylamino]-2-oxopiperidin-1-yl]acetamide | —— | C23H30N6O5S |
| —— | Bis(2-cyanoethyl) [(3,5-difluorophenoxy)-(10-methylacridin-9-ylidene)methyl] phosphate | —— | C27H22F2N3O5P |
| —— | 4-chloro-N-{[5-({4-[(2E)-3-phenylprop-2-enoyl]piperazin-1-yl}sulfonyl)thien-2-yl]methyl}benzamide | —— | C25H24ClN3O4S2 |
| —— | (3R)-N-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-1,1-dioxo-N-propylthiolan-3-amine | —— | C17H21FN2O3S |
| —— | (2S,5S)-4-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-2,5-dimethylmorpholine | —— | C16H20FN3O3 |
| —— | (3S)-3-[[4-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]oxolane-2,5-dione | —— | C17H22N2O3 |
| —— | (2S)-1-[(2R,5S)-2,5-dimethylmorpholin-4-yl]-3-(4-ethoxyphenoxy)propan-2-ol | —— | C17H27NO4 |
| —— | (3R)-3-(pyridin-4-ylmethyl)oxolane-2,5-dione | —— | C10H9NO3 |
| —— | [(1R,2S,10R,12R,13S,15R)-12-cyano-8-methoxy-16-methyl-15-(methylsulfonyloxymethyl)-11,16-diazatetracyclo[11.2.1.02,11.04,9]hexadeca-4(9),5,7-trien-10-yl]methyl benzoate | —— | C27H31N3O6S |
| —— | 5-benzyloxy-2-(4-flouro-phenyl)-3-methyl-1-[4-(2-piperidin-1-yl-ethoxy)-benzyl]-1H-indole | —— | C36H37FN2O2 |
| —— | 3-O-[3-(4-hydroxyphenyl)-4-oxochromen-7-yl] 1-O-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl] propanedioate | —— | C24H22O12 |
| —— | (2S,6S)-N,2,6-trimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]morpholine-4-sulfonamide | —— | C12H21N3O4S |
| —— | 3-(2-chloro-4-(1-propoxy)benzyl)-2,7-dimethyl-5-[(4-methylbenzene)sulfonylcarbamoyl]-3H-imidazo[4,5-b]pyridine | 275380-76-2 | C26H27ClN4O4S |
| —— | (2R,5R)-2,5-dimethyl-4-(3-methylquinolin-8-yl)sulfonylmorpholine | —— | C16H20N2O3S |
| —— | (2R)-4-[2-[(2R,5S)-2,5-dimethylmorpholin-4-yl]acetyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide | —— | C17H23N3O4 |
| —— | (2R,5S)-4-[[2-(2,4-dimethoxyphenyl)-1,3-thiazol-4-yl]methyl]-2,5-dimethylmorpholine | —— | C18H24N2O3S |
| —— | (NE)-N-[(4E,8R)-8-(1,3-benzothiazol-2-ylsulfanyl)cyclooct-4-en-1-ylidene]hydroxylamine | —— | C15H16N2OS2 |
| —— | 3-(2-Methylpropoxycarbonylamino)-3-[3-[[3-(propylcarbamoylamino)phenyl]sulfonylamino]phenyl]propanoic acid | —— | C24H32N4O7S |
| —— | 2-[[2-[4-[4-[2-(4-Acetamidophenyl)ethoxy]phenoxy]phenyl]acetyl]amino]benzoic acid | —— | C31H28N2O6 |
| —— | 1-[(2S)-2-(4,4,5,5,5-pentafluoropentylsulfanylmethyl)pyrrolidin-1-yl]-2-(3,4,5-trimethoxyphenyl)ethane-1,2-dione | —— | C21H26F5NO5S |
| —— | (3S)-3-(thiophen-2-ylmethyl)oxolane-2,5-dione | —— | C9H8O3S |
| —— | thien-3-ylcarbonyl-Trp-piperazine-4-nitrophenyl | —— | C26H25N5O4S |
| —— | 2-methyl-1-[4-[(3S)-1-(4-methylbenzoyl)piperidine-3-carbonyl]piperazin-1-yl]-2-phenylpropan-1-one | —— | C28H35N3O3 |
| —— | 2-[(3R)-3-methyl-4-[2-(4-methylsulfanylanilino)-2-oxoethyl]piperazin-1-yl]-N-(4-methylsulfanylphenyl)acetamide | —— | C23H30N4O2S2 |
| —— | ethyl (2Z,5S)-2-[(5-bromofuran-2-yl)methylidene]-7-methyl-3-oxo-5-(2-propan-2-yloxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate | —— | C24H23BrN2O5S |
| —— | (1-hydroxy-5H-pyrido[3,2-c][1,5]benzodiazepin-6-yl)-[2-(trifluoromethyl)-4-[3-(trifluoromethyl)pyrazol-1-yl]phenyl]methanone | —— | C24H15F6N5O2 |
| —— | 4-[3-(5-Bromo-2-phenylmethoxyphenyl)thiophen-2-yl]-2-methylbenzoic acid | —— | C25H19BrO3S |
| —— | 1H-indole-5-carboxylic acid-{(R)-1-(cyanomethyl-carbamoyl)-2-[2-(1,1-difluoro-methoxy)-phenylmethanesulfonyl]-ethyl}-amide | 330475-23-5 | C22H20F2N4O5S |
| —— | 3,7-dimethyl-1-[11-[[(E)-tridec-9-enyl]amino]undecyl]purine-2,6-dione | —— | C31H55N5O2 |
| —— | N-[2-(dimethylamino)ethyl]-N-[1-[3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]ethyl]-7-methyloctanamide | —— | C29H39FN4O2 |
| —— | N-[[7-chloro-1-(2,4-dichlorophenyl)-4,4-dioxo-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]piperidin-1-amine | —— | C22H21Cl3N4O2S |
| —— | (2R)-1-[(2R,5S)-2,5-dimethylmorpholin-4-yl]-3-(4-fluorophenoxy)propan-2-ol | —— | C15H22FNO3 |
| —— | N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-4-(2-methylpropyl)benzenesulfonamide | —— | C21H30N2O4S |
| —— | 1-[(1R,4R)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]methanesulfonamide | —— | C16H27NO4S |
| —— | 5-chloro-2-[(4-chlorophenyl)sulfonylamino]-N-(2-methoxy-4-nitrophenyl)benzamide | —— | C20H15Cl2N3O6S |
| —— | 3-[3-(4-chloro-3-ethylphenoxy)-N-[[4-fluoro-2-(trifluoromethyl)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-ol | —— | C25H21ClF7NO2 |
| —— | 2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5-[3-(2-methylpropyl)-1,2,4-triaza-3-boranuidacyclopenta-3,5-dien-5-yl]-4-(trifluoromethylsulfanyl)-1H-pyrazol-2-ium-3-amine | —— | C16H15BCl2F6N6S |
| —— | 3-(3,4-dimethoxyphenoxy)-N-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]propanamide | —— | C27H28N4O6 |
| —— | ethyl 5-[[(3S)-3-benzamidobutanoyl]amino]-1-benzothiophene-2-carboxylate | —— | C22H22N2O4S |
| —— | US8530490, Comparative 2 | —— | C21H22N4O7S |
| —— | 3,5-dimethyl-4-[(2R)-4-methyl-2-phenylpiperazin-1-yl]sulfonyl-1,2-oxazole | —— | C16H21N3O3S |
| —— | 1-Bicyclo[2.2.1]hept-2-yl-7-{4-[4-(3-morpholin-4-ylpropyl)piperidin-1-yl]phenylamino}pyrimido[4,5-d]pyrimidin-2(1H)-one | —— | C31H41N7O2 |
| —— | (2S)-1-(6-phenyl-2-pyridin-3-ylthieno[2,3-d]pyrimidin-4-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-2-carboxamide | —— | C24H20F3N5OS |
| —— | (2S)-4-[4-(4-bromophenyl)phenyl]-2-[2-(1,3-dioxoisoindol-2-yl)ethyl]-4-oxobutanoic acid | —— | C26H20BrNO5 |
| —— | 2-[(1S)-1-[[butyl(methyl)sulfamoyl]amino]ethyl]-7-ethoxy-1-benzofuran | —— | C17H26N2O4S |
| —— | [10R,4bR-(4bβ,9aβ)]-7-[(N-(4-trifluoromethyl)phenylmethyl-N-isopropyl)aminocarbonyl]-4b,5,9,9a,10,11-hexahydro-9a-hydroxy-(6H)-8-methyl-10,4b-(iminoethano)-phenanthro[3,2-b]pyrrole | 302900-30-7 | C31H34F3N3O2 |
| —— | (2S,5S)-2,5-dimethyl-4-[[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl]morpholine | —— | C13H23N3O2 |
| —— | 1-(5-chloro-2-methoxybenzoyl)-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]piperidine-4-carboxamide | —— | C24H33ClN2O3 |
| —— | benzyl N-[(2R)-1-[4-methoxy-3-(2-methoxyethoxy)anilino]-1-oxo-3-phenylpropan-2-yl]carbamate | —— | C27H30N2O6 |
| —— | N-[(2S)-1-[4-methoxy-3-(2-methoxyethoxy)anilino]-4-methylsulfanyl-1-oxobutan-2-yl]-3-methylbenzamide | —— | C23H30N2O5S |