| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 2-hydroxy-1-[4-[2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]oxy-1,3-benzothiazol-6-yl]-3,6-dihydro-2H-pyridin-1-yl]ethanone | 1346624-92-7 | C26H31N5O3S |
| —— | 3-[3-acetyl-1-(4-chlorophenyl)-1H-pyrazole-4-carbonyl]-1,5-diphenyl-1H-pyrazole-4-carbonitrile | 1261418-33-0 | C28H18ClN5O2 |
| —— | methyl 3-{[(2-hydroxy-3-methylquinolin-6-yl)amino]sulfonyl}benzoate | 1425927-19-0 | C18H16N2O5S |
| —— | Cyclobutylmethyl 4-[[6-[4-(4-hydroxy-4-methylpentyl)sulfonylpiperazin-1-yl]-1,3-benzothiazol-2-yl]oxy]piperidine-1-carboxylate | 1346625-74-8 | C28H42N4O6S2 |
| —— | 1-[4-[2-[[2-Cyano-4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]phenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylic acid | 1423067-78-0 | C29H32N4O5S2 |
| —— | 5-ethyl-6-[2-fluoro-4-(piperidin-1-yl)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426660-11-8 | C19H21FN2O3 |
| —— | 4-[4-(4-diethylaminomethyl-2-fluoro-phenyl)-[1,2,3]triazol-1-ylmethyl]-N-hydroxy-benzamide | 1267502-39-5 | C21H24FN5O2 |
| —— | 6-(4-{3-[1-(dimethylamino)cyclopropyl]pyrrolidin-1-yl}phenyl)-5-ethyl-4-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426666-72-9 | C23H29N3O4 |
| —— | 1-cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(pyrrolidin-1-yl)-1H-indole-4-carboxamide | 1346574-90-0 | C26H32N4O2 |
| —— | 1-[6-(3-bromo-phenyl)-pyrimidine-4-carbonyl]-pyrrolidine-3-carboxylic acid | 1426411-92-8 | C16H14BrN3O3 |
| —— | 2-amino-4-[[(1S)-1-[2-cyclopropyl-8-(6-methoxypyridin-3-yl)-1-oxoisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile | 1425042-53-0 | C25H23N7O2 |
| —— | 2-amino-4-[[(1S)-1-[8-chloro-2-(2,3-difluorophenyl)-1-oxoisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile | 1425043-44-2 | C22H15ClF2N6O |
| —— | 1-cyclopentyl-2-(4-((1-ethylpiperidin-4-ylidene)methyl)phenyl)ethanol | 1425972-10-6 | C21H31NO |
| —— | (18S)-26-methoxy-23-methyl-5,7,14,20,23,31-hexazapentacyclo[23.3.1.12,6.18,12.014,18]hentriaconta-1(29),2(31),3,5,8,10,12(30),25,27-nonaen-19-one | 1187659-83-1 | C27H32N6O2 |
| —— | 6-(benzofuran-5-yl)-5-ethyl-4-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426527-33-4 | C16H13NO5 |
| —— | 4-hydroxy-5-methoxy-6-(1-methyl-1H-indol-5-yl)-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426527-45-8 | C16H14N2O5 |
| —— | 1-[4-[2-[[2-Cyano-4-[[methyl(oxan-4-ylmethyl)amino]methyl]phenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylic acid | 1423067-71-3 | C32H38N4O4S |
| —— | 1-[2-(2-methoxypyridin-4-yl)ethyl]-4-[3-(tetrahydropyran-4-yl)-[1,2,4]thiadiazol-5-yl]piperazine | 1423042-38-9 | C19H27N5O2S |
| —— | (5-methyl-6-(2-morpholinoethyl)-6H-thieno[2,3-b]pyrrol-2-yl)(6-methylpyridin-3-yl)methanone | 1261150-93-9 | C20H23N3O2S |
| —— | 4-methoxy-N-[1-(4-methoxyphenyl)-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl]benzamide | 1266083-91-3 | C22H20BNO4 |
| —— | Ethyl 1-[4-(5-chloro-2-hydroxyphenyl)-1,3-thiazol-2-yl]-3-(trifluoromethyl)piperidine-4-carboxylate | 1423070-78-3 | C18H18ClF3N2O3S |
| —— | 6-{4-[(3R,4S)-3,4-dihydroxypyrrolidin-1-yl]phenyl}-5-ethyl-4-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426668-70-3 | C18H20N2O6 |
| —— | 6-[5-(dimethylamino)thiophen-2-yl]-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426668-72-5 | C14H16N2O3S |
| —— | 5-fluoro-N-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-6-{[(1S,2S)-2-(1,5-naphthyridin-2-yl)cyclopropyl]methoxy}pyrimidine-2,4-diamine | 1424374-01-5 | C20H19FN8OS |
| —— | (4aR,6R,8aS)-6-[(benzyloxy)methyl]-8a-(2,4-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-amine | 1425947-71-2 | C21H22F2N2O2S |
| —— | 6-(6-chloro-1-methyl-2-(morpholinomethyl)-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid | 1426524-63-1 | C22H24ClN3O4 |
| —— | 2-[(2-hydroxy-3-hexadecyloxypropyl)(15-(4-iodophenyl)pentadecanoyl)amino]ethyl 2-acetamido-2-deoxy-β-D-glucopyranosyl-(1→2)-α-D-mannopyranosyl-(1→6)-β-D-glucopyranoside | 1499188-77-0 | C62H109IN2O19 |
| —— | (R)-(3-aminopiperidin-1-yl)(2-(1-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-1-methyl-7-(trifluoromethoxy)-1H-benzo[d]imidazol-5-yl)methanone | 1549811-09-7 | C24H25F3N6O2 |
| —— | 3,4-bis(benzyloxy)-6-(3,6-dihydro-2H-pyran-4-yl)pyridazine | 1616378-89-2 | C23H22N2O3 |
| —— | N-(1-(3-((ethylamino)methyl)benzyl)-1H-pyrazol-4-yl)-1H-indazole-3-carboxamide | 1422980-59-3 | C21H22N6O |
| —— | N-[(2-fluorophenyl)methylideneamino]-1,2-benzothiazole-3-carboxamide | 902772-45-6 | C15H10FN3OS |
| —— | US10138229, Example 67 | 1558036-98-8 | C25H26N4O4 |
| —— | (2R,3R,4S)-4-amino-2-tetradecylpyrrolidin-3-ol | 1254942-89-6 | C18H38N2O |
| —— | 4-(4-bromobenzylidene)-1-(3-{[tert-butyl(dimethyl)silyl]oxy}cyclobutyl)piperidine | 1425972-22-0 | C22H34BrNOSi |
| —— | N-(1-(3-((2-(dimethylamino)ethylamino)methyl)benzyl)-1H-pyrazol-4-yl)-1H-indazole-3-carboxamide | 1422980-62-8 | C23H27N7O |
| —— | 3-methyl-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzene-sulfonamide | 1425926-90-4 | C16H17N3O3S |
| —— | 5-amino-2-(2,6-difluorophenyl)-N-(5-((4-hydroxy-4-methylpentyl)oxy)isothiazol-4-yl)thiazole-4-carboxamide | 1422395-14-9 | C19H20F2N4O3S2 |
| —— | 6-(1-methylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2-[(3S)-1-(5-propylpyrimidin-2-yl)pyrrolidin-3-yl]oxy-1,3-benzothiazole | 1346624-87-0 | C24H29N5O3S2 |
| —— | 2-amino-4-[[(1S)-1-[5-(1-methylpyrazol-4-yl)-4-oxo-3-phenylquinazolin-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | 1425042-27-8 | C25H21N9O |
| —— | tert-Butyl 3'-bromo-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[1,2-a]imidazole]-1-carboxylate | 1251000-16-4 | C15H22BrN3O2 |
| —— | 5-(4-chlorophenyl)-N-(5-(morpholinomethyl)-2-oxooxazolidin-3-yl)-6-(2,2,2-trifluoroethoxy)-3-pyridinecarboxamide | 1427064-17-2 | C22H22ClF3N4O5 |
| —— | 2-{[(2-Ethoxy-phenylcarbamoyl)-methyl]-amino}-benzoic acid methyl ester | 57037-26-0 | C18H20N2O4 |
| —— | (1R,2S)-N-[5-methyl-8-(6-trifluoromethyl-1H-indol-3-yl)-pyrido[4,3-d]pyrimidin-2-yl]-cyclohexane-1,2-diamine | 1562987-55-6 | C23H23F3N6 |
| —— | (2S,3S,4R)-4-amino-2-tetradecylpyrrolidin-3-ol | 1254942-82-9 | C18H38N2O |
| —— | (S)-1-benzyl-2-methyl-7-morpholin-4-yl-2-trifluoromethyl-2,3-dihydro-1H-imidazo[1,2-a]pyrimidin-5-one | 1260983-15-0 | C19H21F3N4O2 |
| —— | US10138229, Example 82 | 1558037-13-0 | C27H29N5O3 |
| —— | N-ethyl-6-(N-methylcyclohexanecarboxamido)-2-(pyrazine-2-carboxamido)-1H-indole-3-carboxamide | 1562185-23-2 | C24H28N6O3 |
| —— | 3-[(2S,8S,9S)-11-[(2R)-1-hydroxypropan-2-yl]-2,9-dimethyl-8-{[N-methyl(4-fluorobenzene)sulfonamido]methyl}-12-oxo-2,3,4,5,6,8,9,10,11,12-decahydro-1,7,11-benzodioxazacyclotetradecin-14-yl]-1-phenylurea | 1255392-37-0 | C35H45FN4O7S |
| —— | Tert-butyl 4-[2-fluoro-4-(oxetan-3-yloxy)phenyl]piperazine-1-carboxylate | 929884-54-8 | C18H25FN2O4 |
| —— | 2-Anilino-7-methyl-1-phenyl-5-piperidin-1-yl-1,6-naphthyridin-4-one | 503437-02-3 | C26H26N4O |