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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1235867-27-2 C43H52N6O3
—— tert-butyl (((2R,3S)-5-((S)-1-((4-methoxybenzyl)oxy)propan-2-yl)-3-methyl-8-nitro-6-oxo-3,4,5,6-tetrahydro-2H-benzo[b][1,5]oxazocin-2-yl)methyl)(methyl)carbamate 1255212-97-5 C29H39N3O8
tert-butyl (((2R,3S)-5-((S)-1-((4-methoxybenzyl)oxy)propan-2-yl)-3-methyl-8-nitro-6-oxo-3,4,5,6-tetrahydro-2H-benzo[b][1,5]oxazocin-2-yl)methyl)(methyl)carbamate
—— methyl 5-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino-2-furancarboxylate 383667-79-6 C32H35ClN2O10
methyl 5-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino-2-furancarboxylate
—— methyl 5-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-7-ethoxy-1-benzofuran-2-carboxylate 383673-59-4 C38H41ClN2O11
methyl 5-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-7-ethoxy-1-benzofuran-2-carboxylate
—— 4-furan-2-yl-4,5-dihydro-benzo[<i>d</i>][1,3]oxazepine 68028-87-5 C13H11NO2
4-furan-2-yl-4,5-dihydro-benzo[<i>d</i>][1,3]oxazepine
—— 4,4-dibenzyl-2,3,4,4a-tetrahydronaphtho[2,3-e]pyrido[2,1-b][1,3]oxazin-12(1H)-one 1416767-43-5 C30H27NO2
4,4-dibenzyl-2,3,4,4a-tetrahydronaphtho[2,3-e]pyrido[2,1-b][1,3]oxazin-12(1H)-one
—— 1392323-51-1 C20H17BrN2O2
—— ethyl 5-[3-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]phenyl]pentanoate 383671-45-2 C39H47ClN2O9
ethyl 5-[3-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]phenyl]pentanoate
—— (E)-2-(7-trifluoromethyl-spiro[chroman-2,1'-cyclobutane]-4-ylidene)-N-(3,4-dihydro-2,2-dioxo-1H-2,1,3-benzothiadiazin-5-yl)acetamide 1042971-29-8 C22H20F3N3O4S
(E)-2-(7-trifluoromethyl-spiro[chroman-2,1'-cyclobutane]-4-ylidene)-N-(3,4-dihydro-2,2-dioxo-1H-2,1,3-benzothiadiazin-5-yl)acetamide
—— tert-butyl (((2R,8R,9S)-14-amino-11-((S)-1-((4-methoxybenzyl)oxy)propan-2-yl)-2,9-dimethyl-12-oxo-3,4,5,6,9,10,11,12-octahydro-2H,8H-benzo[b][1,9]dioxa[5]azacyclotetradecin-8-yl)methyl)(methyl)carbamate 1255213-60-5 C35H53N3O7
tert-butyl (((2R,8R,9S)-14-amino-11-((S)-1-((4-methoxybenzyl)oxy)propan-2-yl)-2,9-dimethyl-12-oxo-3,4,5,6,9,10,11,12-octahydro-2H,8H-benzo[b][1,9]dioxa[5]azacyclotetradecin-8-yl)methyl)(methyl)carbamate
—— 2-[2-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]ethyl]furan-3-carboxylic acid 383654-30-6 C33H37ClN2O10
2-[2-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]ethyl]furan-3-carboxylic acid
—— 2-fluoro-N-({4-methyl-6-[7-(2-methyl-1H-benzimidazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-5-(1-methylethyl)pyrimidin-2-yl}methyl)ethanamine 1256952-61-0 C28H33FN6O
2-fluoro-N-({4-methyl-6-[7-(2-methyl-1H-benzimidazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-5-(1-methylethyl)pyrimidin-2-yl}methyl)ethanamine
—— 10-chloro-2-methoxy-6-methyl-1-nitro-12H-benzo[5,6][1,4]oxazino[2,3-c]quinoline 54486-47-4 C17H12ClN3O4
10-chloro-2-methoxy-6-methyl-1-nitro-12H-benzo[5,6][1,4]oxazino[2,3-c]quinoline
—— [2-[(3R,5S)-1-(3-acetyloxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]acetyl] 2,2-dimethylpropanoate 871934-70-2 C31H38ClNO9
[2-[(3R,5S)-1-(3-acetyloxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]acetyl] 2,2-dimethylpropanoate
—— methyl 2-((R)-1,5-dimethyl-3-((S)-2-methyl-5-oxo-2,5-dihydrofuran-2-yl)-2-oxoindolin-3-yl)acrylate 1360462-13-0 C19H19NO5
methyl 2-((R)-1,5-dimethyl-3-((S)-2-methyl-5-oxo-2,5-dihydrofuran-2-yl)-2-oxoindolin-3-yl)acrylate
—— 3-[(3R,5S)-3-(2-amino-2-oxoethyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-2,3-dihydro-4,1-benzoxazepin-1(5H)-yl]-2,2-dimethylpropyl acetate 839724-58-2 C26H31ClN2O7
3-[(3R,5S)-3-(2-amino-2-oxoethyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-2,3-dihydro-4,1-benzoxazepin-1(5H)-yl]-2,2-dimethylpropyl acetate
—— 2-(1-isopropyl-1H-1,2,4-triazol-5-yl)-N-(1-isopropylazetidin-3-yl)-4,5-dihydrobenzo[b]pyrazolo[1,5-d][1,4]oxazepine-9-carboxamide 1282512-18-8 C23H29N7O2
2-(1-isopropyl-1H-1,2,4-triazol-5-yl)-N-(1-isopropylazetidin-3-yl)-4,5-dihydrobenzo[b]pyrazolo[1,5-d][1,4]oxazepine-9-carboxamide
—— 8-(4-Bromo-benzyloxy)-2,2-dimethyl-3,4-dihydro-2H-benzo[f][1,4]oxazepin-5-one 144537-28-0 C18H18BrNO3
8-(4-Bromo-benzyloxy)-2,2-dimethyl-3,4-dihydro-2H-benzo[f][1,4]oxazepin-5-one
—— ethyl 4-[2-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-4-(4-chlorophenyl)-1,3-thiazol-5-yl]butanoate 383673-01-6 C41H45Cl2N3O9S
ethyl 4-[2-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-4-(4-chlorophenyl)-1,3-thiazol-5-yl]butanoate
—— ethyl 3-[3-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]aminophenyl]propionate 383663-35-2 C37H43ClN2O9
ethyl 3-[3-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]aminophenyl]propionate
—— methyl 2-[4-[[2-[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-3-fluorophenyloxy]acetate 383671-60-1 C35H38ClFN2O10
methyl 2-[4-[[2-[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-3-fluorophenyloxy]acetate
—— ethyl 6-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-5-(2,3-dimethoxyphenyl)-7-chloro-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-2-pyridinecarboxylate 383672-30-8 C34H38ClN3O9
ethyl 6-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-5-(2,3-dimethoxyphenyl)-7-chloro-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-2-pyridinecarboxylate
—— ethyl 4-[4-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]phenyl]butanoate 383666-63-5 C38H45ClN2O9
ethyl 4-[4-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]phenyl]butanoate
—— (Z)-4,11-dimethyldibenzo[b,f][1,4]oxazepine 1316273-88-7 C15H13NO
(Z)-4,11-dimethyldibenzo[b,f][1,4]oxazepine
—— (3R,5S)-N-(3-acetoxypropyl)sulfonyl-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetamide 383653-20-1 C31H39ClN2O11S
(3R,5S)-N-(3-acetoxypropyl)sulfonyl-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetamide
—— 1-methylpyrido[4',3':6,7]oxepino[4,3,2-cd]isoindol-2(1H)-one 1453172-71-8 C15H10N2O2
1-methylpyrido[4',3':6,7]oxepino[4,3,2-cd]isoindol-2(1H)-one
—— methyl 3-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino-2-thiophenecarboxylate 383667-69-4 C32H35ClN2O9S
methyl 3-[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino-2-thiophenecarboxylate
—— 2,3,4,5-Tetrahydro-1,4-benzoxazepin-8-ol hydrochloride 1803599-64-5 C9H12ClNO2
2,3,4,5-Tetrahydro-1,4-benzoxazepin-8-ol hydrochloride
—— N-[(3R,5S)-7-chloro-1-(3-hydroxy-2-hydroxymethyl-2-methylpropyl)-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetyl]-4-hydroxypiperidine-4-acetic acid methyl ester 189060-16-0 C32H41ClN2O10
N-[(3R,5S)-7-chloro-1-(3-hydroxy-2-hydroxymethyl-2-methylpropyl)-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetyl]-4-hydroxypiperidine-4-acetic acid methyl ester
—— (12R,18S)-2,5-dioxa-13,17-diazatricyclo[17.4.0.06,11]tricosa-1(23),6,8,10,19,21-hexaene-12,18-dicarboxylic acid 1333237-96-9 C21H24N2O6
(12R,18S)-2,5-dioxa-13,17-diazatricyclo[17.4.0.06,11]tricosa-1(23),6,8,10,19,21-hexaene-12,18-dicarboxylic acid
—— 920739-76-0 C39H48N8O3
—— 2-phenylbenzo[b]pyrrolo[1,2-d][1,4]oxazepin-7(6H)-one 1417565-97-9 C18H13NO2
2-phenylbenzo[b]pyrrolo[1,2-d][1,4]oxazepin-7(6H)-one
—— 1,3-diphenyl-1H-pyrazolo[4,3-b][1,5]benzoxazepine 1263218-13-8 C22H15N3O
1,3-diphenyl-1H-pyrazolo[4,3-b][1,5]benzoxazepine
—— 4-(2-oxopiperazin-1-yl)-7-(trifluoromethyl)-3,4-dihydro-2H-1-benzopyrane 1313034-85-3 C14H15F3N2O2
4-(2-oxopiperazin-1-yl)-7-(trifluoromethyl)-3,4-dihydro-2H-1-benzopyrane
—— 1-methyl-3-(5-(4-methyl-5-oxo-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepin-8-yl)-4-((5-methylpyridin-3-yl)oxy)pyridin-2-yl)urea 1442682-02-1 C23H23N5O4
1-methyl-3-(5-(4-methyl-5-oxo-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepin-8-yl)-4-((5-methylpyridin-3-yl)oxy)pyridin-2-yl)urea
—— 8-fluoro-1,2-dihydro-benz[<i>d</i>][1,3]oxazin-4-one 387-98-4 C8H6FNO2
8-fluoro-1,2-dihydro-benz[<i>d</i>][1,3]oxazin-4-one
—— ethyl 3-[3-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-2-methylphenyl]propionate 383663-76-1 C38H45ClN2O9
ethyl 3-[3-[[[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]amino]-2-methylphenyl]propionate
—— 149161-98-8 C18H16MnN3O2S
—— tert-butyl 2-[5,5-bis(3-chlorophenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-7-yl]-5-cyano-1H-pyrrole-1-carboxylate 865670-00-4 C31H25Cl2N3O4
tert-butyl 2-[5,5-bis(3-chlorophenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-7-yl]-5-cyano-1H-pyrrole-1-carboxylate
—— 7-(2-methyl-1H-benzimidazol-6-yl)-N-(1-methylethyl)-N-(phenylmethyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide 1257298-98-8 C28H30N4O2
7-(2-methyl-1H-benzimidazol-6-yl)-N-(1-methylethyl)-N-(phenylmethyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide
—— 5-(5'-Chloro-2'-nitrophenyl)-2,3-dihydro-1,4-benzoxazepine Hydrochloride 83725-63-7 C15H11ClN2O3*ClH
5-(5'-Chloro-2'-nitrophenyl)-2,3-dihydro-1,4-benzoxazepine Hydrochloride
—— (3S)-3,4-dihydro-3-methyl-1-[N-phthaloyl-3-cyclohexyl-(S)-alanyl]-2H-[1,4]benzoxazine 1416453-34-3 C26H28N2O4
(3S)-3,4-dihydro-3-methyl-1-[N-phthaloyl-3-cyclohexyl-(S)-alanyl]-2H-[1,4]benzoxazine
—— 7-bromo-5,5-di(3-furyl)-1,5-dihydro-4.1-benzoxazepin-2(3H)-one 865671-54-1 C17H12BrNO4
7-bromo-5,5-di(3-furyl)-1,5-dihydro-4.1-benzoxazepin-2(3H)-one
—— methyl 2-((R)-5-chloro-1-methyl-3-((S)-2-methyl-5-oxo-2,5-dihydrofuran-2-yl)-2-oxoindolin-3-yl)acrylate 1360462-17-4 C18H16ClNO5
methyl 2-((R)-5-chloro-1-methyl-3-((S)-2-methyl-5-oxo-2,5-dihydrofuran-2-yl)-2-oxoindolin-3-yl)acrylate
—— 1,1-dimethylethyl 7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate 1257301-21-5 C22H25N3O3
1,1-dimethylethyl 7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate
—— 1,1,1,3,3,3-hexafluoro-2-(2,3,4,5-tetrahydro-benzo[<i>b</i>][1,4]oxazepin-8-yl)-propan-2-ol 71260-06-5 C12H11F6NO2
1,1,1,3,3,3-hexafluoro-2-(2,3,4,5-tetrahydro-benzo[<i>b</i>][1,4]oxazepin-8-yl)-propan-2-ol
—— (3-Chloro-4-fluoro-phenyl)-(5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 875926-20-8 C17H10ClFN4O
(3-Chloro-4-fluoro-phenyl)-(5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine
—— (3S)-1-{[7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}pyrrolidin-3-ol 1257298-78-4 C22H24N4O3
(3S)-1-{[7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}pyrrolidin-3-ol
—— 4-benzylamino-5-oxo-2,3,4,5-tetrahydro-benzo[f][1,4]oxazepine-2-carboxylic acid 2-morpholin-4-yl-ethyl ester 19011-92-8 C23H27N3O5
4-benzylamino-5-oxo-2,3,4,5-tetrahydro-benzo[f][1,4]oxazepine-2-carboxylic acid 2-morpholin-4-yl-ethyl ester
—— (1-β-deuteriotetrahydroisoquinolyl)oxazoline 106681-12-3 C15H20N2O
(1-β-deuteriotetrahydroisoquinolyl)oxazoline