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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-methoxy-4-(2-pyrrolidin-1-ylethoxy)phenyl]-5-(4-methyl-2,3-dihydro-1,4-benzoxazin-7-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1142939-73-8 C28H32N6O3
N-[3-methoxy-4-(2-pyrrolidin-1-ylethoxy)phenyl]-5-(4-methyl-2,3-dihydro-1,4-benzoxazin-7-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— 7-(3,5-dichlorophenyl)-5-ethyl-5-(2-furyl)-1,5-dihydro-4,1-benzoxazepin-2(3H)-one 865669-74-5 C21H17Cl2NO3
7-(3,5-dichlorophenyl)-5-ethyl-5-(2-furyl)-1,5-dihydro-4,1-benzoxazepin-2(3H)-one
—— Dibenzo[b,f][1,4]oxazepin-11-ylmethyl-dimethyl-amine 19970-54-8 C16H16N2O
Dibenzo[b,f][1,4]oxazepin-11-ylmethyl-dimethyl-amine
—— 9-methyl-3-oxo-N-[4-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide 1067226-57-6 C18H15F3N2O3
9-methyl-3-oxo-N-[4-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide
—— 1-(3-Methoxymethyl-4H-5-oxa-1,9b-diaza-cyclopenta[a]naphthalen-2-yl)-ethanone 114627-56-4 C14H14N2O3
1-(3-Methoxymethyl-4H-5-oxa-1,9b-diaza-cyclopenta[a]naphthalen-2-yl)-ethanone
—— methyl 5-({2-[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-1,2,3,5-tetrahydro-2-oxo-4,1-benzoxazepin-3-yl]acetyl}amino)-4-oxopentanoate 839724-54-8 C32H39ClN2O10
methyl 5-({2-[(3R,5S)-1-(3-acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-1,2,3,5-tetrahydro-2-oxo-4,1-benzoxazepin-3-yl]acetyl}amino)-4-oxopentanoate
—— N-propyl-6-[5-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,5-benzoxazepine-2,4'-piperidine]-1'-yl]pyridazine-3-carboxamide 1262756-94-4 C29H32F3N5O2
N-propyl-6-[5-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,5-benzoxazepine-2,4'-piperidine]-1'-yl]pyridazine-3-carboxamide
—— [2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]{7-[6-(propan-2-ylamino)pyridin-3-yl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl}methanone 1251158-14-1 C27H30FN3O4S
[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]{7-[6-(propan-2-ylamino)pyridin-3-yl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl}methanone
—— 5<i>H</i>-benzo[<i>d</i>][1,2,3]oxadiazeto[3,2-<i>b</i>][1,2,3]oxadiazine 29150-10-5 C8H8N2O2
5<i>H</i>-benzo[<i>d</i>][1,2,3]oxadiazeto[3,2-<i>b</i>][1,2,3]oxadiazine
—— 4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-methylaniline 1251158-43-6 C26H27FN2O4S
4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-methylaniline
—— [7-(2-ethoxypyrimidin-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl][2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]methanone 1251161-64-4 C25H26FN3O5S
[7-(2-ethoxypyrimidin-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl][2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]methanone
—— 4,5-dihydro-1<i>H</i>-benzo[<i>e</i>][1,2]oxazepine-3-carboxylic acid dimethylamide 38090-36-7 C12H16N2O2
4,5-dihydro-1<i>H</i>-benzo[<i>e</i>][1,2]oxazepine-3-carboxylic acid dimethylamide
—— {(salicylaldehyde o-mercaptoanil)(o-phenanthroline)oxomolybdenum} 80630-34-8 C25H17MoN3O2S
{(salicylaldehyde o-mercaptoanil)(o-phenanthroline)oxomolybdenum}
—— 3-chloro-8,9,10,11-tetrahydro-7H-12-oxa-6a-azoniacyclonona[de]naphthalene bromide 1026668-17-6 Br*C14H15ClNO
3-chloro-8,9,10,11-tetrahydro-7H-12-oxa-6a-azoniacyclonona[de]naphthalene bromide
—— tert-butyl (((2R,8S,9S)-14-amino-11-((R)-1-((4-methoxybenzyl)oxy)propan-2-yl)-2,9-dimethyl-12-oxo-3,4,5,6,9,10,11,12-octahydro-2H,8H-benzo[b][1,9]dioxa[5]azacyclotetradecin-8-yl)methyl)(methyl)carbamate 1255213-63-8 C35H53N3O7
tert-butyl (((2R,8S,9S)-14-amino-11-((R)-1-((4-methoxybenzyl)oxy)propan-2-yl)-2,9-dimethyl-12-oxo-3,4,5,6,9,10,11,12-octahydro-2H,8H-benzo[b][1,9]dioxa[5]azacyclotetradecin-8-yl)methyl)(methyl)carbamate
—— 2-Methyl-2,3,3a,4-tetrahydrobenzpyranopyrrol 63238-58-4 C12H13NO
2-Methyl-2,3,3a,4-tetrahydrobenzpyranopyrrol
—— N-(2-cyclopropylethyl)-2-[5-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,5-benzoxazepine-2,4'-piperidine]-1'-yl]-1,3-thiazole-5-carboxamide 1262755-93-0 C30H33F3N4O2S
N-(2-cyclopropylethyl)-2-[5-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,5-benzoxazepine-2,4'-piperidine]-1'-yl]-1,3-thiazole-5-carboxamide
—— 3-[(3R,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-3-(2-oxoethyl)-2,3-dihydro-4,1-benzoxazepin-1(5H)-yl]-2,2-dimethylpropyl acetate 839725-03-0 C26H30ClNO7
3-[(3R,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-3-(2-oxoethyl)-2,3-dihydro-4,1-benzoxazepin-1(5H)-yl]-2,2-dimethylpropyl acetate
—— 7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-(1-methylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine 1256945-82-0 C24H25N5O
7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-(1-methylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 4-{[3-fluoro-2-methyl-4-(methylsulfonyl)phenyl]carbonyl}-7-(1H-indazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251155-43-7 C25H22FN3O4S
4-{[3-fluoro-2-methyl-4-(methylsulfonyl)phenyl]carbonyl}-7-(1H-indazol-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— N-[4-(4-{[4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)phenyl]acetamide 1251157-49-9 C25H24N2O5S
N-[4-(4-{[4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)phenyl]acetamide
—— 1-(6-{4-[(4-bromo-2-methylphenyl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1H-benzimidazol-2-yl)-N-methylmethanamine 1251151-45-7 C26H25BrN4O2
1-(6-{4-[(4-bromo-2-methylphenyl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1H-benzimidazol-2-yl)-N-methylmethanamine
—— N-ethyl-N-({4-methyl-6-[7-(2-methyl-1H-benzimidazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-5-(1-methylethyl)pyrimidin-2-yl}methyl)ethanamine 1256952-73-4 C30H38N6O
N-ethyl-N-({4-methyl-6-[7-(2-methyl-1H-benzimidazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-5-(1-methylethyl)pyrimidin-2-yl}methyl)ethanamine
—— 6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-[2-(methyloxy)ethyl]pyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine 1256952-39-2 C26H31N7O2S
6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-[2-(methyloxy)ethyl]pyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine
—— 4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-piperidin-4-ylbenzamide 1251163-12-8 C31H34FN3O5S
4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-piperidin-4-ylbenzamide
—— 7-(1H-benzimidazol-6-yl)-4-{[4-(ethylsulfonyl)-3-fluoro-2-methylphenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251155-17-5 C26H24FN3O4S
7-(1H-benzimidazol-6-yl)-4-{[4-(ethylsulfonyl)-3-fluoro-2-methylphenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— [3-fluoro-2-methyl-4-(methylsulfonyl)phenyl][7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]methanone 1251149-35-5 C26H24FN3O4S
[3-fluoro-2-methyl-4-(methylsulfonyl)phenyl][7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]methanone
—— 6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-prop-2-en-1-ylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine 1256952-43-8 C26H29N7OS
6-(4-(2-[(dimethylamino)methyl]-6-methyl-5-prop-2-en-1-ylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)[1,3]thiazolo[5,4-b]pyridin-2-amine
—— 2-allyl-1-methyl-1,2,4,5-tetrahydro-benzo[<i>d</i>][1,2]oxazepine 37939-24-5 C13H17NO
2-allyl-1-methyl-1,2,4,5-tetrahydro-benzo[<i>d</i>][1,2]oxazepine
—— 3,3-Dimethyl-7-methylsulfonyl-5-(2-pyridyl N-oxide)-2,3-dihydro-1-benzoxepine 157987-21-8 C18H19NO4S
3,3-Dimethyl-7-methylsulfonyl-5-(2-pyridyl N-oxide)-2,3-dihydro-1-benzoxepine
—— (R)-2-bromo-6-ethyl-6-(p-tolyl)benzo[b]pyrrolo[1,2-d][1,4]oxazepin-7(6H)-one 1452816-02-2 C21H18BrNO2
(R)-2-bromo-6-ethyl-6-(p-tolyl)benzo[b]pyrrolo[1,2-d][1,4]oxazepin-7(6H)-one
—— (E)-2-(8-trifluoromethyl-3,4-dihydrobenzo[b]oxepin-5(2H)-yliden)-N-(3-oxo-1,2,3,4-tetrahydroquinolin-5-yl)acetamide 1042969-76-5 C22H19F3N2O3
(E)-2-(8-trifluoromethyl-3,4-dihydrobenzo[b]oxepin-5(2H)-yliden)-N-(3-oxo-1,2,3,4-tetrahydroquinolin-5-yl)acetamide
—— tert-butyl 9-(morpholin-4-ylcarbonyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate 1055881-02-1 C19H26N2O5
tert-butyl 9-(morpholin-4-ylcarbonyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate
—— [7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]{1-methyl-5-[4-(propan-2-ylsulfonyl)phenyl]-1H-pyrrol-2-yl}methanone 1251162-66-9 C32H32N4O4S
[7-(2-methyl-1H-benzimidazol-6-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]{1-methyl-5-[4-(propan-2-ylsulfonyl)phenyl]-1H-pyrrol-2-yl}methanone
—— 7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-methyl-5-(1-phenylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine 1256945-97-7 C30H29N5O
7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-methyl-5-(1-phenylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 4-{[7-(6-aminopyridin-3-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}-3-methyl-N-(1-methylethyl)benzenesulfonamide 1251158-42-5 C25H28N4O4S
4-{[7-(6-aminopyridin-3-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}-3-methyl-N-(1-methylethyl)benzenesulfonamide
—— 5-{4-[(4-chloro-2-methylphenyl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}pyridin-2-amine 1251157-97-7 C22H20ClN3O2
5-{4-[(4-chloro-2-methylphenyl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}pyridin-2-amine
—— 4-{[7-(1H-indazol-3-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}benzenesulfonamide 1251163-41-3 C23H20N4O4S
4-{[7-(1H-indazol-3-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}benzenesulfonamide
—— N-ethyl-4-(4-{[2-ethyl-4-(ethylsulfonyl)-3-fluorophenyl]-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)benzamide 1251154-04-7 C29H31FN2O5S
N-ethyl-4-(4-{[2-ethyl-4-(ethylsulfonyl)-3-fluorophenyl]-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)benzamide
—— N-methyl-1-[6-(4-{[4-(trifluoromethyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1H-benzimidazol-2-yl]methanamine 1251152-83-6 C26H23F3N4O2
N-methyl-1-[6-(4-{[4-(trifluoromethyl)phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1H-benzimidazol-2-yl]methanamine
—— 4-{[3-fluoro-2-methyl-4-(methylsulfonyl)phenyl]carbonyl}-7-(1H-indazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251156-43-0 C25H22FN3O4S
4-{[3-fluoro-2-methyl-4-(methylsulfonyl)phenyl]carbonyl}-7-(1H-indazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— propane-1-sulfonic acid [2-(5-benzyl-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepin-7-yloxy)ethyl]amide 1410790-74-7 C21H28N2O4S
propane-1-sulfonic acid [2-(5-benzyl-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepin-7-yloxy)ethyl]amide
—— 3-(2',6'-Dichlorphenyl)-7-nitro-4H-1,2,4-benzoxadiazin 66288-34-4 C13H7Cl2N3O3
3-(2',6'-Dichlorphenyl)-7-nitro-4H-1,2,4-benzoxadiazin
—— (4H,10H-9-Oxa-3a-aza-benzo[f]azulen-10-ylmethyl)-propyl-amine 63880-40-0 C16H20N2O
(4H,10H-9-Oxa-3a-aza-benzo[f]azulen-10-ylmethyl)-propyl-amine
—— 4-{[7-(1,2-benzisoxazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}benzenesulfonamide 1251162-89-6 C23H19N3O5S
4-{[7-(1,2-benzisoxazol-5-yl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]carbonyl}benzenesulfonamide
—— N-(4-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-thiophenecarboximidamide 216008-21-8 C16H19N3OS
N-(4-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-thiophenecarboximidamide
—— [1-sec-butyl-7-methyl-2,3-dihydro-1H-4-oxa-1,6-diaza-naphthalen-5-yl]-(2,4,6trimethyl-phenyl)-amine 1349474-01-6 C21H29N3O
[1-sec-butyl-7-methyl-2,3-dihydro-1H-4-oxa-1,6-diaza-naphthalen-5-yl]-(2,4,6trimethyl-phenyl)-amine
—— N’-(4-chloro-5-(2-oxo-2H-spiro[benzofuran-3,4’-piperidin]-1‘-yl)pyridazin-3-yl)-3,3,3-trifluoropropanehydrazide 1519049-41-2 C19H17ClF3N5O3
N’-(4-chloro-5-(2-oxo-2H-spiro[benzofuran-3,4’-piperidin]-1‘-yl)pyridazin-3-yl)-3,3,3-trifluoropropanehydrazide
—— N-Desmethyl-(+/-)-oxo-lycoramin-acetat 18797-76-7 C18H21NO5
N-Desmethyl-(+/-)-oxo-lycoramin-acetat
—— 7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-methyl-5-(1-methylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine 1256945-89-7 C25H27N5O
7-(2-methyl-1H-benzimidazol-6-yl)-4-[6-methyl-5-(1-methylethyl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine