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—— 2-[1-[2-(4-methoxy-7-pyrazin-2-yl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxo-acetyl]-4-piperidylidene]-2-phenyl-acetamide 676489-73-9 C27H24N6O4
2-[1-[2-(4-methoxy-7-pyrazin-2-yl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxo-acetyl]-4-piperidylidene]-2-phenyl-acetamide
—— methyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate 676489-65-9 C31H26N4O5
methyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(4-fluorophenyl)phenylmethylene]- 676489-89-7 C29H26FN3O4
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(4-fluorophenyl)phenylmethylene]-
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(3,5-dimethyl-isoxazol-4-ylphenylmethylene)- 676489-84-2 C28H28N4O5
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(3,5-dimethyl-isoxazol-4-ylphenylmethylene)-
—— 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoic acid 676489-67-1 C30H24N4O5
4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoic acid
—— 1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[oxazol-2-yl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione 676489-86-4 C26H24N4O5
1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[oxazol-2-yl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione
—— 1-(4-methoxy-7-pyrazin-2-yl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[oxazol-5-yl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione 676490-30-5 C29H24N6O4
1-(4-methoxy-7-pyrazin-2-yl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[oxazol-5-yl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione
—— 1-[4-(1-phenyl-1-(3-hydroxymethylphenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-22-5 C32H30N6O4
1-[4-(1-phenyl-1-(3-hydroxymethylphenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— 1-[4-(1-phenyl-1-(5-trifluoromethyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676489-77-3 C26H22F3N5O5
1-[4-(1-phenyl-1-(5-trifluoromethyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— Piperidine, 1-[2-(7-chloro-4-methoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(cyano-3-pyridinylmethylene)- 676489-46-6 C22H18ClN5O3
Piperidine, 1-[2-(7-chloro-4-methoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(cyano-3-pyridinylmethylene)-
—— 1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-14-5 C28H26N8O4
1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— 1-[4-(1-phenyl-1-(pyridin-3-yl)-methylene)-piperidin-1-yl]-2-(4-methoxy-7-pyrazinyl-6-azaindol-3-yl)-ethane-1,2-dione 676489-96-6 C31H26N6O3
1-[4-(1-phenyl-1-(pyridin-3-yl)-methylene)-piperidin-1-yl]-2-(4-methoxy-7-pyrazinyl-6-azaindol-3-yl)-ethane-1,2-dione
—— 1-[4-[chloro(phenyl)methylene]-1-piperidyl]-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione 676489-29-5 C23H22ClN3O4
1-[4-[chloro(phenyl)methylene]-1-piperidyl]-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione
—— isopropyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate 676489-64-8 C33H30N4O5
isopropyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate
—— 1-[4-(1-phenyl-1-(5-hydroxy-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-20-3 C27H24N8O5
1-[4-(1-phenyl-1-(5-hydroxy-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— 1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[methylsulfonyl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione 676489-36-4 C24H25N3O6S
1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-[methylsulfonyl(phenyl)methylene]-1-piperidyl]ethane-1,2-dione
—— Piperidine, 4-(cyano-2-pyridinylmethylene)-1-[2-[4-methoxy-7-(5-aminopyrazinyl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]- 676489-53-5 C26H22N8O3
Piperidine, 4-(cyano-2-pyridinylmethylene)-1-[2-[4-methoxy-7-(5-aminopyrazinyl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(4-methyl-thiophen-2-ylphenylmethylene)- 676489-79-5 C28H27N3O4S
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(4-methyl-thiophen-2-ylphenylmethylene)-
—— 1-[4-(1-phenyl-1-(3-hydroxymethylphenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(1,2,3-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-10-1 C31H28N6O4
1-[4-(1-phenyl-1-(3-hydroxymethylphenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(1,2,3-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— 1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4-methoxy-7-pyrazinyl-6-azaindol-3-yl)-ethane-1,2-dione 676489-98-8 C29H25N7O4
1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4-methoxy-7-pyrazinyl-6-azaindol-3-yl)-ethane-1,2-dione
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(2-methoxyphenyl)phenylmethylene]- 676489-90-0 C30H29N3O5
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(2-methoxyphenyl)phenylmethylene]-
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(3-fluorophenyl)phenylmethylene]- 676489-92-2 C29H26FN3O4
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(3-fluorophenyl)phenylmethylene]-
—— 1-[4-(1-phenyl-1-(5-isopropyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-16-7 C30H30N8O4
1-[4-(1-phenyl-1-(5-isopropyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzamide 676489-61-5 C30H25N5O4
4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzamide
—— 1-[4-(1-cyano-1-benzothiazol-2-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676490-61-2 C25H21N5O4S
1-[4-(1-cyano-1-benzothiazol-2-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— 1-[4-(1-cyano-1-thiazol-5-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676490-62-3 C21H19N5O4S
1-[4-(1-cyano-1-thiazol-5-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— 1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-(1-phenylethylidene)-1-piperidyl]ethane-1,2-dione 676489-32-0 C24H25N3O4
1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-[4-(1-phenylethylidene)-1-piperidyl]ethane-1,2-dione
—— 1-[4-[(3-fluorophenyl)-phenyl-methylene]-1-piperidyl]-2-[4-methoxy-7-(3-methylpyrazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]ethane-1,2-dione 676490-36-1 C32H28FN5O3
1-[4-[(3-fluorophenyl)-phenyl-methylene]-1-piperidyl]-2-[4-methoxy-7-(3-methylpyrazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]ethane-1,2-dione
—— 1-[4-(1-phenyl-1-(3,5-difluorophenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione 676490-23-6 C31H26F2N6O3
1-[4-(1-phenyl-1-(3,5-difluorophenyl)-methylene)-piperidin-1-yl]-2-[4-methoxy-7-(3-methyl-1,2,4-triazol-1-yl)-6-azaindol-3-yl]-ethane-1,2-dione
—— Piperidine, 4-(cyanophenylmethylene)-1-[2-[4-methoxy-7-[4-(1-pyrrolidinylcarbonyl)phenyl]-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]- 676489-62-6 C34H31N5O4
Piperidine, 4-(cyanophenylmethylene)-1-[2-[4-methoxy-7-[4-(1-pyrrolidinylcarbonyl)phenyl]-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(pyrazin-2-ylphenylmethylene)- 676489-80-8 C27H25N5O4
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-(pyrazin-2-ylphenylmethylene)-
—— 1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676489-76-2 C26H25N5O5
1-[4-(1-phenyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzonitrile 676489-70-6 C30H23N5O3
4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzonitrile
—— ethyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate 676489-66-0 C32H28N4O5
ethyl 4-[3-[2-[4-[cyano(phenyl)methylene]-1-piperidyl]-2-oxo-acetyl]-4-methoxy-1H-pyrrolo[2,3-c]pyridin-7-yl]benzoate
—— Piperidine, 4-(cyanophenylmethylene)-1-[2-[4-methoxy-7-(5-aminopyrazinyl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]- 676489-52-4 C27H23N7O3
Piperidine, 4-(cyanophenylmethylene)-1-[2-[4-methoxy-7-(5-aminopyrazinyl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-
—— 2-[1-[2-(7-chloro-4-methoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxo-acetyl]-4-piperidylidene]-2-phenyl-acetamide 676489-72-8 C23H21ClN4O4
2-[1-[2-(7-chloro-4-methoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxo-acetyl]-4-piperidylidene]-2-phenyl-acetamide
—— 1-[4-(1-cyano-1-thien-3-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676490-64-5 C22H20N4O4S
1-[4-(1-cyano-1-thien-3-yl-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— (1-{2-[7-(3-amino-pyrazol-1-yl)-4-fluoro-1H-pyrrolo[2,3-c]pyridin-3-yl]-2-oxo-acetyl}-piperidin-4-ylidene)-phenyl-acetonitrile 676490-49-6 C25H20FN7O2
(1-{2-[7-(3-amino-pyrazol-1-yl)-4-fluoro-1H-pyrrolo[2,3-c]pyridin-3-yl]-2-oxo-acetyl}-piperidin-4-ylidene)-phenyl-acetonitrile
—— Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(4-methoxyphenyl)phenylmethylene]- 676489-87-5 C30H29N3O5
Piperidine, 1-[2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-1,2-dioxoethyl]-4-[(4-methoxyphenyl)phenylmethylene]-
—— 1-[4-(1-phenyl-1-(2-phenylethyn-1-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione 676490-56-5 C31H27N3O4
1-[4-(1-phenyl-1-(2-phenylethyn-1-yl)-methylene)-piperidin-1-yl]-2-(4,7-dimethoxy-6-azaindol-3-yl)-ethane-1,2-dione
—— (2Z)-2-[1-[2-(1H-indol-3-yl)-2-oxo-acetyl]-3-methyl-4-piperidylidene]-2-phenyl-acetonitrile 676489-39-7 C24H21N3O2
(2Z)-2-[1-[2-(1H-indol-3-yl)-2-oxo-acetyl]-3-methyl-4-piperidylidene]-2-phenyl-acetonitrile
—— 1-(4-benzhydrylidene-1-piperidyl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione 676489-81-9 C29H27N3O4
1-(4-benzhydrylidene-1-piperidyl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione
—— Piperidine, 4-(cyano-2-pyridinylmethylene)-1-[2-[4-methoxy-7-[4-(methylsulfonyl)phenyl]-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]- 676489-57-9 C29H25N5O5S
Piperidine, 4-(cyano-2-pyridinylmethylene)-1-[2-[4-methoxy-7-[4-(methylsulfonyl)phenyl]-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-
—— N-acetylrifabutin 645406-18-4 C48H64N4O12
N-acetylrifabutin
—— (S)-6-(3-chloro-2-fluorobenzyl)-1-[2,2-dimethyl-1-(hydroxymethyl)propyl]-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 697761-99-2 C24H25ClFNO5
(S)-6-(3-chloro-2-fluorobenzyl)-1-[2,2-dimethyl-1-(hydroxymethyl)propyl]-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
—— 2-(4-aminomethyl-2,6-dimethyl-phenoxy)-N-{(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-acetamide 660410-70-8 C33H43N5O5S2
2-(4-aminomethyl-2,6-dimethyl-phenoxy)-N-{(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-acetamide
—— N-{(1S,2R)-3-[(2-amino-benzothiazole-6-sulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxypropyl}-3-fluoro-2-methyl-benzamide 660410-53-7 C29H33FN4O4S2
N-{(1S,2R)-3-[(2-amino-benzothiazole-6-sulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxypropyl}-3-fluoro-2-methyl-benzamide
—— {(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-carbamic acid thiazol-5-ylmethyl ester 660410-56-0 C27H33N5O5S3
{(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-carbamic acid thiazol-5-ylmethyl ester
—— N-{(1S,2R)-3-[(2-amino-benzothiazole-6-sulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxypropyl}-2-(4-aminomethyl-2,6-dimethyl-phenoxy)-acetamide 660410-54-8 C32H41N5O5S2
N-{(1S,2R)-3-[(2-amino-benzothiazole-6-sulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxypropyl}-2-(4-aminomethyl-2,6-dimethyl-phenoxy)-acetamide
—— 2-(4-amino-2,6-dimethyl-phenoxy)-N-{(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-acetamide 660410-72-0 C32H41N5O5S2
2-(4-amino-2,6-dimethyl-phenoxy)-N-{(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl-(2-methylamino-benzothiazole-6-sulfonyl)-amino]-propyl}-acetamide