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中文名称 英文名称 CAS号 化学式 结构式图片
—— isopropyl (2-((3-(3-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl)amino)ethyl)(methyl)-carbamate 1454555-21-5 C19H24N6O3
isopropyl (2-((3-(3-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl)amino)ethyl)(methyl)-carbamate
—— methyl 3,3,3-trichloro-N-(4-methylbenzoyl)-2-(pyrazin-2-ylamino)alaninate 1289404-92-7 C16H15Cl3N4O3
methyl 3,3,3-trichloro-N-(4-methylbenzoyl)-2-(pyrazin-2-ylamino)alaninate
—— 3-methyl-1-phenyl-7,8-dihydro-6H-pyrazolo[3,4-b]quinoxalin-5-one 1380215-10-0 C16H14N4O
3-methyl-1-phenyl-7,8-dihydro-6H-pyrazolo[3,4-b]quinoxalin-5-one
—— 3-((1R,3R,4S)-3-ethyl-4-(6-tosyl-6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)cyclopentyl)propanenitrile 1428243-64-4 C24H26N6O2S
3-((1R,3R,4S)-3-ethyl-4-(6-tosyl-6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)cyclopentyl)propanenitrile
—— 1-(2-(methoxymethoxy)-6-(methoxymethyl)phenyl)ethanone 161358-57-2 C12H16O4
1-(2-(methoxymethoxy)-6-(methoxymethyl)phenyl)ethanone
—— (R)-1-(4-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine 1326240-46-3 C13H13ClN2
(R)-1-(4-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine
—— N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-2-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1229611-81-7 C28H18F4N6O2S
N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-2-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— methyl 3,3,3-trichloro-2-methoxy-N-(4-methylbenzoyl)alaninate 1289404-76-7 C13H14Cl3NO4
methyl 3,3,3-trichloro-2-methoxy-N-(4-methylbenzoyl)alaninate
—— (S)-tert-butyl (1-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)pyrrolidin-3-yl)carbamate 1454558-31-6 C15H20BrN5O2
(S)-tert-butyl (1-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)pyrrolidin-3-yl)carbamate
—— (5S,6S,7S)-2,6-dihydroxy-2,5,7-trimethylnon-8-en-4-one 1292811-38-1 C12H22O3
(5S,6S,7S)-2,6-dihydroxy-2,5,7-trimethylnon-8-en-4-one
—— (S)-2-amino-1-(4-(3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)piperazin-1-yl)-4-methylpentan-1-one 1454555-41-9 C22H29N7O2
(S)-2-amino-1-(4-(3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)piperazin-1-yl)-4-methylpentan-1-one
—— 5-(3-isopropoxyphenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde 1256163-25-3 C16H16N4O2
5-(3-isopropoxyphenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde
—— MeOC6H3ICH(NHBoc)CONHCH(CH3)COOH 1004524-45-1 C17H23IN2O6
MeOC6H3ICH(NHBoc)CONHCH(CH3)COOH
—— 1-[3-Methyl-2-(phenylmethoxycarbonylamino)pentanoyl]pyrrolidine-2-carboxylic acid 13211-37-5 C19H26N2O5
1-[3-Methyl-2-(phenylmethoxycarbonylamino)pentanoyl]pyrrolidine-2-carboxylic acid
—— (S)-3-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-4-(4-fluorophenyl)oxazolidin-2-one 1269646-16-3 C15H10BrFN4O2
(S)-3-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-4-(4-fluorophenyl)oxazolidin-2-one
—— methyl 3,3,3-trichloro-2-[(4-chlorophenyl)thio]-N-(4-methylbenzoyl)alaninate 1289404-81-4 C18H15Cl4NO3S
methyl 3,3,3-trichloro-2-[(4-chlorophenyl)thio]-N-(4-methylbenzoyl)alaninate
—— 5-(3-(2-methyl-1H-imidazol-1-yl)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde 1256163-04-8 C17H14N6O
5-(3-(2-methyl-1H-imidazol-1-yl)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde
—— 3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-(pyridin-2-yl)oxazolidin-2-one 1269644-74-7 C22H15FN8O2
3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-(pyridin-2-yl)oxazolidin-2-one
—— 5-(methoxymethyl)-4-oxo-4H-1-benzopyran-3-carboxaldehyde 161358-66-3 C12H10O4
5-(methoxymethyl)-4-oxo-4H-1-benzopyran-3-carboxaldehyde
—— 5-(4-isopropoxyphenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde 1256163-44-6 C16H16N4O2
5-(4-isopropoxyphenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde
—— Ac-Phe-Tyr-OMe 15852-46-7 C21H24N2O5
Ac-Phe-Tyr-OMe
—— 5-(3-(2-morpholinoethoxy)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde 1256163-23-1 C19H21N5O3
5-(3-(2-morpholinoethoxy)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde
—— 5-isopropyl-3-(4-(3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)piperazin-1-yl)-1,2,4-oxadiazole 1454555-40-8 C21H24N8O2
5-isopropyl-3-(4-(3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)piperazin-1-yl)-1,2,4-oxadiazole
—— Carbonic acid benzyl ester (2S,3R,4S,5R,6R)-4,5-bis-benzyloxycarbonyloxy-2-methoxy-6-[(4-methoxy-phenyl)-diphenyl-methoxymethyl]-tetrahydro-pyran-3-yl ester 197630-98-1 C51H48O13
Carbonic acid benzyl ester (2S,3R,4S,5R,6R)-4,5-bis-benzyloxycarbonyloxy-2-methoxy-6-[(4-methoxy-phenyl)-diphenyl-methoxymethyl]-tetrahydro-pyran-3-yl ester
—— 5-(3-((1H-imidazol-1-yl)methyl)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde 1256163-12-8 C17H14N6O
5-(3-((1H-imidazol-1-yl)methyl)phenylamino)pyrazolo[1,5-a]pyrimidine-3-carbaldehyde
—— isopropyl 3-hydroxybiphenyl-2-carboxylate 1416168-26-7 C16H16O3
isopropyl 3-hydroxybiphenyl-2-carboxylate
—— 3,4-dimethyl-octa-1,4,6-triene 17208-42-3 C10H16
3,4-dimethyl-octa-1,4,6-triene
—— (S)-2-(2-(3-bromopyrazolo[1,5-a]pyrimidin-5-ylamino)-3-methylbutyl)isoindoline-1,3-dione 1269647-58-6 C19H18BrN5O2
(S)-2-(2-(3-bromopyrazolo[1,5-a]pyrimidin-5-ylamino)-3-methylbutyl)isoindoline-1,3-dione
—— 5-chloro-8-methoxy-1-(4-methylphenylcarbamoyl)-2-methylnaphtho[2,1-b]furan 1134953-17-5 C22H18ClNO3
5-chloro-8-methoxy-1-(4-methylphenylcarbamoyl)-2-methylnaphtho[2,1-b]furan
—— 2-(α-Piperidino-benzyl)-[1]naphthol 102756-54-7 C22H23NO
2-(α-Piperidino-benzyl)-[1]naphthol
—— (S)-4-isopropyl-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one 1269646-25-4 C27H34N6O3Si
(S)-4-isopropyl-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one
—— 1-(methoxymethoxy)-3-(methoxymethyl)benzene 161358-51-6 C10H14O3
1-(methoxymethoxy)-3-(methoxymethyl)benzene
—— methyl 3,3,3-trichloro-N-(4-methylbenzoyl)-2-(morpholin-4-yl)alaninate 1289404-95-0 C16H19Cl3N2O4
methyl 3,3,3-trichloro-N-(4-methylbenzoyl)-2-(morpholin-4-yl)alaninate
—— (S)-1-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-5-isopropylimidazolidin-2-one 1269647-63-3 C12H14BrN5O
(S)-1-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-5-isopropylimidazolidin-2-one
—— 1-benzyl-4-[4-((S)-3-methoxy-2-methyl-propoxymethyl)-phenyl]-3-trityloxymethyl-piperidin-4-ol 1006865-31-1 C44H49NO4
1-benzyl-4-[4-((S)-3-methoxy-2-methyl-propoxymethyl)-phenyl]-3-trityloxymethyl-piperidin-4-ol
—— (S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-phenyloxazolidin-2-one 1269643-42-6 C24H18N6O2
(S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-phenyloxazolidin-2-one
—— (S)-4-(4-fluorophenyl)-3-(3-(4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one 1269645-20-6 C24H18FN7O2
(S)-4-(4-fluorophenyl)-3-(3-(4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one
—— (S)-N2-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-3-methylbutane-1,2-diamine 1269647-61-1 C11H16BrN5
(S)-N2-(3-bromopyrazolo[1,5-a]pyrimidin-5-yl)-3-methylbutane-1,2-diamine
—— N-(4-(2-(4-((2-(dimethylamino)ethyl)(methyl)carbamoyl)phenyl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1229611-84-0 C36H30F4N6O3S
N-(4-(2-(4-((2-(dimethylamino)ethyl)(methyl)carbamoyl)phenyl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— (3S,4R,1'S)-4-methoxycarbonyl-4-methyl-1-(1'-phenyleth-1'-yl)-3-trichloroacetylaminopyrrolidin-2-one 1206626-12-1 C17H19Cl3N2O4
(3S,4R,1'S)-4-methoxycarbonyl-4-methyl-1-(1'-phenyleth-1'-yl)-3-trichloroacetylaminopyrrolidin-2-one
—— (S)-4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)-N'-(1-iminoethyl)benzohydrazide 1269650-07-8 C24H20FN7O3
(S)-4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)-N'-(1-iminoethyl)benzohydrazide
—— LCRF-0004 1229611-73-7 C28H18F4N6O2S
LCRF-0004
—— (S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-isopropyloxazolidin-2-one 1269643-37-9 C21H20N6O2
(S)-3-(3-(4-(1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-isopropyloxazolidin-2-one
—— (S)-4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)benzohydrazide 1269650-05-6 C22H17FN6O3
(S)-4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)benzohydrazide
—— 3-Isopropyl-5-methylhydantoin 19347-82-1 C7H12N2O2
3-Isopropyl-5-methylhydantoin
—— (S)-tert-butyl 4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)benzoate 1269650-01-2 C26H23FN4O4
(S)-tert-butyl 4-(5-(4-(4-fluorophenyl)-2-oxooxazolidin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)benzoate
—— (S)-N-(3-fluoro-4-(2-(4-((N-(1-methoxypropan-2-yl)acetamido)methyl)phenyl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1127327-80-3 C37H31F4N5O4S
(S)-N-(3-fluoro-4-(2-(4-((N-(1-methoxypropan-2-yl)acetamido)methyl)phenyl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— N-(4-(2-(1-acetyl-1,2,3,6-tetrahydropyridin-4-yl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1229611-88-4 C31H23F4N5O3S
N-(4-(2-(1-acetyl-1,2,3,6-tetrahydropyridin-4-yl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— (S)-3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-phenyloxazolidin-2-one 1269644-76-9 C23H16FN7O2
(S)-3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-phenyloxazolidin-2-one
—— (S)-2-(4-isopropyl-2-oxo-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)imidazolidin-1-yl)ethyl 4-methylbenzenesulfonate 1269647-84-8 C35H44N8O5SSi
(S)-2-(4-isopropyl-2-oxo-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)imidazolidin-1-yl)ethyl 4-methylbenzenesulfonate