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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid 1031440-98-8 C12H10N2O2
4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid
—— 6-methoxy-2(3'-fluorophenyl)-quinolin-4-yl-phosphate 1032315-45-9 C16H13FNO5P
6-methoxy-2(3'-fluorophenyl)-quinolin-4-yl-phosphate
—— 4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide 1031440-81-9 C12H11N3O
4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide
—— 2-amino-5-(2,2-dimethyl-3,4-dihydro-2H-chromen-6-yl)-5-(6-fluoro-3'-methoxybiphenyl-3-yl)-3-methyl-3,5-dihydro-4H-imidazol-4-one hydrochloride 1034669-54-9 C28H28FN3O3*ClH
2-amino-5-(2,2-dimethyl-3,4-dihydro-2H-chromen-6-yl)-5-(6-fluoro-3'-methoxybiphenyl-3-yl)-3-methyl-3,5-dihydro-4H-imidazol-4-one hydrochloride
—— cyclopentyl (2S)-cyclohexyl[(4-([((1-[5-(hydroxycarbamoyl)pyrimidin-2-yl]piperidin-4-yl)methyl)amino]methyl)benzyl)amino]acetate 1022928-81-9 C32H46N6O4
cyclopentyl (2S)-cyclohexyl[(4-([((1-[5-(hydroxycarbamoyl)pyrimidin-2-yl]piperidin-4-yl)methyl)amino]methyl)benzyl)amino]acetate
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-1H-imidazo[4,5-c]pyridin-1-yl)-L-phenylalanine 1031342-23-0 C29H26BrN5O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-1H-imidazo[4,5-c]pyridin-1-yl)-L-phenylalanine
—— methyl 4-{1-[(3S)-4-{[3-chloro-5-(trifIuoromethyl)benzoyl](methyl)amino}-3-(4-fluorophenyl)butyl]azetidin-3-yl}-piperazine-1-carboxylate 1034407-42-5 C28H33ClF4N4O3
methyl 4-{1-[(3S)-4-{[3-chloro-5-(trifIuoromethyl)benzoyl](methyl)amino}-3-(4-fluorophenyl)butyl]azetidin-3-yl}-piperazine-1-carboxylate
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-(cyclopropylmethyl)-7-[(cyclopropylmethyl)amino]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine 1031343-07-3 C32H36BrN5O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-(cyclopropylmethyl)-7-[(cyclopropylmethyl)amino]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine
—— N-{1-[2-(dimethylamino)-2-oxo-1-phenylethyl]azepan-4-yl}-N-[4-fluoro-3-(trifluoromethyl)benzyl]-1-methyl-1H-imidazole-4-carboxamide 1031291-58-3 C29H33F4N5O2
N-{1-[2-(dimethylamino)-2-oxo-1-phenylethyl]azepan-4-yl}-N-[4-fluoro-3-(trifluoromethyl)benzyl]-1-methyl-1H-imidazole-4-carboxamide
—— (2S)-cyclohexyl[((3-[5-(hydroxycarbamoyl)pyrimidin-2-yl]-3-azabicyclo[3.1.0]hex-6-yl)methyl)amino]acetic acid 1023296-50-5 C19H27N5O4
(2S)-cyclohexyl[((3-[5-(hydroxycarbamoyl)pyrimidin-2-yl]-3-azabicyclo[3.1.0]hex-6-yl)methyl)amino]acetic acid
—— tert-butyl [(2S)-3-phenyl-2-({[1-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinolin-3-yl]carbonyl}amino)propyl]carbamate 1031440-83-1 C28H31F3N4O3
tert-butyl [(2S)-3-phenyl-2-({[1-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinolin-3-yl]carbonyl}amino)propyl]carbamate
—— 2-(3'-fluorophenyl)-6,7-methylenedioxyquinolin-4-yl-phosphate 1032315-64-2 C16H11FNO6P
2-(3'-fluorophenyl)-6,7-methylenedioxyquinolin-4-yl-phosphate
—— N-(2-chlorophenyl)-N-((3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)methyl)methanesulfonamide 1135417-36-5 C16H13ClFN3O3S
N-(2-chlorophenyl)-N-((3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)methyl)methanesulfonamide
—— 3-[4-(3,3-Dimethyl-butoxy)-phenyl]-3-phenyl-propionic acid 1040738-61-1 C21H26O3
3-[4-(3,3-Dimethyl-butoxy)-phenyl]-3-phenyl-propionic acid
—— 5'-O-[({(1S)-1-benzyl-2-[(2,2-dimethylpropanoyl)oxy]ethyl}amino)(phenoxy)phosphoryl]-2'-C-methylcytidine 1142811-73-1 C30H39N4O9P
5'-O-[({(1S)-1-benzyl-2-[(2,2-dimethylpropanoyl)oxy]ethyl}amino)(phenoxy)phosphoryl]-2'-C-methylcytidine
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-isobutyl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine 1031341-22-6 C28H31BrN4O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-isobutyl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine
—— 4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-2-carboxylic acid 1031441-80-1 C12H10N2O2
4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-2-carboxylic acid
—— N-(2-chloro-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-1H-imidazo[4,5-c]pyridin-1-yl)-L-phenylalanine 1031342-26-3 C29H26ClN5O3
N-(2-chloro-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-1H-imidazo[4,5-c]pyridin-1-yl)-L-phenylalanine
—— {5-Chloro-2-[4-(2-oxo-2,3-dihydro-benzooxazol-7-yl)-piperidine-1-carbonyl]-1H-indol-7-yl}-acetonitrile 1032715-06-2 C23H19ClN4O3
{5-Chloro-2-[4-(2-oxo-2,3-dihydro-benzooxazol-7-yl)-piperidine-1-carbonyl]-1H-indol-7-yl}-acetonitrile
—— ethyl 2-(4-(benzyloxy)-2-oxopyridin-1(2H)-yl)-1,5-dimethyl-1H-imidazole-4-carboxylate 1105690-67-2 C20H21N3O4
ethyl 2-(4-(benzyloxy)-2-oxopyridin-1(2H)-yl)-1,5-dimethyl-1H-imidazole-4-carboxylate
—— (1R)-3-[6-(azetidin-1-ylcarbonyl)-4-(benzyloxy)-1,2-dimethyl-1H-benzimidazol-5-yl]-1-(2-methylphenyl)propan-1-ol 1034771-34-0 C30H33N3O3
(1R)-3-[6-(azetidin-1-ylcarbonyl)-4-(benzyloxy)-1,2-dimethyl-1H-benzimidazol-5-yl]-1-(2-methylphenyl)propan-1-ol
—— 2-phenyl-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide 1031440-61-5 C18H13N3O
2-phenyl-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide
—— (R/S)-2-hydroxy-N-((S)-6-oxo-6,7-dihydro-5H-dibenzo[b,d]azepin-7-yl)-N'-(2,2,3,3,3-pentafluoro-propyl)-2-propyl-malonamide 1043963-76-3 C23H22F5N3O4
(R/S)-2-hydroxy-N-((S)-6-oxo-6,7-dihydro-5H-dibenzo[b,d]azepin-7-yl)-N'-(2,2,3,3,3-pentafluoro-propyl)-2-propyl-malonamide
—— 6-(cyclopentylamino)-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]nicotinamide 1032568-69-6 C29H37N7O4
6-(cyclopentylamino)-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]nicotinamide
—— N-(8-{3-[2-(hydroxymethyl)morpholin-4-yl]propoxy}-7-methoxy-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl)nicotinamide 1032568-57-2 C25H30N6O5
N-(8-{3-[2-(hydroxymethyl)morpholin-4-yl]propoxy}-7-methoxy-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl)nicotinamide
—— (7Z)-1-(cyclohexylamino)-8-methyl-6,13,15,16-tetrahydro-3H,5H-14,16a-ethano-9,12-ethenoimidazo[1,5-a][1,5]diazacyclotetradecin-3-one 1019773-42-2 C25H34N4O
(7Z)-1-(cyclohexylamino)-8-methyl-6,13,15,16-tetrahydro-3H,5H-14,16a-ethano-9,12-ethenoimidazo[1,5-a][1,5]diazacyclotetradecin-3-one
—— 5-(5-(cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide 1020106-18-6 C29H30Cl2N4OS
5-(5-(cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
—— (5-chloro-2,4-dihydroxy-phenyl)-[(R)-2-(pyrrolidine-1-carbonyl)-pyrrolidin-1-yl]-methanone 1023885-50-8 C16H19ClN2O4
(5-chloro-2,4-dihydroxy-phenyl)-[(R)-2-(pyrrolidine-1-carbonyl)-pyrrolidin-1-yl]-methanone
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-[4-(dimethylamino)pyridin-2-yl]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine 1031341-60-2 C31H31BrN6O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-[4-(dimethylamino)pyridin-2-yl]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine
—— 2-[3-(4-chlorophenyl)-2-oxo-1-azaspiro[4.5]dec-3-en-1-yl]-N-(3,5-difluorophenyl)acetamide 1044282-46-3 C23H21ClF2N2O2
2-[3-(4-chlorophenyl)-2-oxo-1-azaspiro[4.5]dec-3-en-1-yl]-N-(3,5-difluorophenyl)acetamide
—— 1-methyl-2-phenyl-1,7-dihydro-1,6,7-triaza-as-indacene-3-carboxylic acid amide 1031440-34-2 C17H14N4O
1-methyl-2-phenyl-1,7-dihydro-1,6,7-triaza-as-indacene-3-carboxylic acid amide
—— N-[(7R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydroazepino[3,4-e]indazol-7-yl]-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[c]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide 1033608-21-7 C28H21ClF3N7O3
N-[(7R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydroazepino[3,4-e]indazol-7-yl]-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[c]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide
—— ethyl 2-(4-(2-cyclopropylethoxy)-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylate 1105690-82-1 C17H20N2O4S
ethyl 2-(4-(2-cyclopropylethoxy)-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylate
—— 2'-oxo-N-{(7R)-8-oxo-9-[4-(trifluoromethyl)benzyl]-3,6,7,8,9,10-hexahydroazepino[3,4-e]indazol-7-yl}-1',2',5,7-tetrahydrospiro[cyclopenta[c]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide 1033608-17-1 C34H26F3N7O3
2'-oxo-N-{(7R)-8-oxo-9-[4-(trifluoromethyl)benzyl]-3,6,7,8,9,10-hexahydroazepino[3,4-e]indazol-7-yl}-1',2',5,7-tetrahydrospiro[cyclopenta[c]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide
—— (4-morpholin-4-yl-phenyl)-[5-(1H-pyrazol-4-yl)-imidazo[1,2-a]pyridin-8-yl]amine 1031284-76-0 C20H20N6O
(4-morpholin-4-yl-phenyl)-[5-(1H-pyrazol-4-yl)-imidazo[1,2-a]pyridin-8-yl]amine
—— 7-(2,6-difluorophenyl)-3-[(5-fluoro-6-methylpyridin-2-yl)amino]-2-{[(3R)-3-hydroxypyrrolidin-1-yl]carbonyl}thieno[2,3-b]pyridin-6(7H)-one 1030833-68-1 C24H19F3N4O3S
7-(2,6-difluorophenyl)-3-[(5-fluoro-6-methylpyridin-2-yl)amino]-2-{[(3R)-3-hydroxypyrrolidin-1-yl]carbonyl}thieno[2,3-b]pyridin-6(7H)-one
—— (2S)-5-(1,3,5-Trimethyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 1044513-01-0 C16H21N3
(2S)-5-(1,3,5-Trimethyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydronaphthalen-2-amine
—— N-{1-[4-(hydroxycarbamoyl)phenyl]piperidin-4-yl}-L-leucine 1022929-21-0 C18H27N3O4
N-{1-[4-(hydroxycarbamoyl)phenyl]piperidin-4-yl}-L-leucine
—— cyclopentyl N-{4-[({1-[5-(hydroxycarbamoyl)pyrimidin-2-yl]piperidin-4-yl}amino)methyl]benzyl}-L-leucinate 1022928-52-4 C29H42N6O4
cyclopentyl N-{4-[({1-[5-(hydroxycarbamoyl)pyrimidin-2-yl]piperidin-4-yl}amino)methyl]benzyl}-L-leucinate
—— trans-5R,7S-6-(3-fluorophenyl)-1'-(3-isopropoxybenzyl)-2-isopropyl-2'-methylspiro[imidazo[1,5-a]imidazole-7,4'-piperidin]-5(6H)-one 1038772-13-2 C29H35FN4O2
trans-5R,7S-6-(3-fluorophenyl)-1'-(3-isopropoxybenzyl)-2-isopropyl-2'-methylspiro[imidazo[1,5-a]imidazole-7,4'-piperidin]-5(6H)-one
—— 1-(4-Ethyl-pyridin-2-yl)-3-[4-(1-methyl-1H-pyrazolo[3,4-c]pyridin-4-yl)-phenyl]-urea 1032943-18-2 C21H20N6O
1-(4-Ethyl-pyridin-2-yl)-3-[4-(1-methyl-1H-pyrazolo[3,4-c]pyridin-4-yl)-phenyl]-urea
—— cyclopentyl N-[(2R)-3-(3-{[5-amino-1-(2,4-difluorophenyl)-1H-pyrazol-4-yl]carbonyl}phenoxy)-2-hydroxypropyl]-L-leucinate 1032826-68-8 C30H36F2N4O5
cyclopentyl N-[(2R)-3-(3-{[5-amino-1-(2,4-difluorophenyl)-1H-pyrazol-4-yl]carbonyl}phenoxy)-2-hydroxypropyl]-L-leucinate
—— 7-(2,6-difluorophenyl)-3-[(5-fluoro-6-methylpyridin-2-yl)amino]-2-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]carbonyl}thieno[2,3-b]pyridin-6(7H)-one 1030833-70-5 C25H21F3N4O3S
7-(2,6-difluorophenyl)-3-[(5-fluoro-6-methylpyridin-2-yl)amino]-2-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]carbonyl}thieno[2,3-b]pyridin-6(7H)-one
—— 1-methyl-3-(4-methyl-piperazin-1-yl)-1H-indazole-6-carboxylic acid 2-methoxy-benzylamide 1027257-31-3 C22H27N5O2
1-methyl-3-(4-methyl-piperazin-1-yl)-1H-indazole-6-carboxylic acid 2-methoxy-benzylamide
—— 2-amino-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]-4-propylpyrimidine-5-carboxamide 1032568-51-6 C26H34N8O4
2-amino-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]-4-propylpyrimidine-5-carboxamide
—— 4-methyl-2-(2-oxo-4-phenylpyridin-1(2H)-yl)thiazole-5-carboxylic acid 1105690-69-4 C16H12N2O3S
4-methyl-2-(2-oxo-4-phenylpyridin-1(2H)-yl)thiazole-5-carboxylic acid
—— (7S,8R,9R)-7-cyclopropyl-7-(2-methoxyethoxy)-2-methyl-9-phenyl-8,9-dihydro-7H-imidazo[1,2-a]pyrano[2,3-c]pyridin-8-ol 1027002-62-5 C23H26N2O4
(7S,8R,9R)-7-cyclopropyl-7-(2-methoxyethoxy)-2-methyl-9-phenyl-8,9-dihydro-7H-imidazo[1,2-a]pyrano[2,3-c]pyridin-8-ol
—— Nelonicline 1026687-03-5 C17H19N3OS
Nelonicline
—— ethyl 2-(4-methoxy-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylate 1105690-81-0 C13H14N2O4S
ethyl 2-(4-methoxy-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylate
—— (2E)-3-{5-chloro-6-[(2-phenoxyethyl)amino]-3-pyridinyl}-N-hydroxyacrylamide hydrochloride 1035217-24-3 C16H16ClN3O3*ClH
(2E)-3-{5-chloro-6-[(2-phenoxyethyl)amino]-3-pyridinyl}-N-hydroxyacrylamide hydrochloride