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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-4-benzyl-3-[1-hydroxy-2-(2-oxo-propyl)-cyclopropyl]-oxazolidin-2-one 1057968-23-6 C16H19NO4
(S)-4-benzyl-3-[1-hydroxy-2-(2-oxo-propyl)-cyclopropyl]-oxazolidin-2-one
—— 8-Methoxycarbonyloctyl 3-O-[2-O-(4-O-methyl-α-D-glucopyranosyl)-α-D-glucopyranosyl]-α-D-glucopyranoside 186419-95-4 C29H52O18
8-Methoxycarbonyloctyl 3-O-[2-O-(4-O-methyl-α-D-glucopyranosyl)-α-D-glucopyranosyl]-α-D-glucopyranoside
—— N2-(3-iodo-1,6-dimethyl-1H-indazol-5-yl)-N2-{2-[(5-fluoro-1,3-dihydro-2H-isoindol-2-yl)(methyl)amino]-2-oxoethyl}-N1-{2-[(tert-butoxycarbonyl)(ethyl)amino]ethyl}glycinamide 1190896-54-8 C31H41FIN7O4
N2-(3-iodo-1,6-dimethyl-1H-indazol-5-yl)-N2-{2-[(5-fluoro-1,3-dihydro-2H-isoindol-2-yl)(methyl)amino]-2-oxoethyl}-N1-{2-[(tert-butoxycarbonyl)(ethyl)amino]ethyl}glycinamide
—— 2-benzyl-6-(4-methoxybenzyl)-4-(4-phenylpiperazin-1-yl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylene 1246670-87-0 C32H33N7O
2-benzyl-6-(4-methoxybenzyl)-4-(4-phenylpiperazin-1-yl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylene
—— tert-butyl 4-[(6,8-dioxo-6,8-dihydropyrazolo[3,4-b]pyrrolo[3,4-d]pyridin-7(3H)-yl)methyl]piperidine-1-carboxylate 1246615-73-5 C19H23N5O4
tert-butyl 4-[(6,8-dioxo-6,8-dihydropyrazolo[3,4-b]pyrrolo[3,4-d]pyridin-7(3H)-yl)methyl]piperidine-1-carboxylate
—— phenyl 2-ethyl-N-(4-methylphenyl)-3-(3-methylphenyloxy)-2-propenimidate 1154685-13-8 C25H25NO2
phenyl 2-ethyl-N-(4-methylphenyl)-3-(3-methylphenyloxy)-2-propenimidate
—— 4-(nitromethyl)-4H-thieno[3,2-c]chromene 1310427-59-8 C12H9NO3S
4-(nitromethyl)-4H-thieno[3,2-c]chromene
—— N-[6-(1,3-benzothiazol-6-yl)-2-methylpyrimidin-4-yl]-1,2,3,4-tetrahydroquinolin-4-amine 1404105-02-7 C21H19N5S
N-[6-(1,3-benzothiazol-6-yl)-2-methylpyrimidin-4-yl]-1,2,3,4-tetrahydroquinolin-4-amine
—— 3-methyl-2-[2-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]ethyl]-1H-quinolin-4-one;hydrochloride 1135028-37-3 C22H28N2O2*ClH
3-methyl-2-[2-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]ethyl]-1H-quinolin-4-one;hydrochloride
—— 2-(5-{2-(4-Fluorophenyl)-5-[(2-methoxypyrimidin-5-yl)thio]-1,3-oxazol-4-yl}pyridin-2-yl)propan-2-ol 1207745-70-7 C22H19FN4O3S
2-(5-{2-(4-Fluorophenyl)-5-[(2-methoxypyrimidin-5-yl)thio]-1,3-oxazol-4-yl}pyridin-2-yl)propan-2-ol
—— 5-(3,4-Diethoxyphenyl)-3-pyridin-4-yl-1,2-oxazole 1201447-19-9 C18H18N2O3
5-(3,4-Diethoxyphenyl)-3-pyridin-4-yl-1,2-oxazole
—— N-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide 1033841-51-8 C23H26FN5O
N-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide
—— N-(3-cyclopropyl-1-((1-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1H-indazol-4-yl)-7-(2-(pyrrolidin-1-yl)ethoxy)imidazo[1,2-a]pyridine-3-carboxamide 1313408-28-4 C31H33N7O3
N-(3-cyclopropyl-1-((1-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1H-indazol-4-yl)-7-(2-(pyrrolidin-1-yl)ethoxy)imidazo[1,2-a]pyridine-3-carboxamide
—— (R)-2-(2-chlorophenyl)-1-((R)-3-(2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)pyrimidin-4-ylamino)piperidin-1-yl)-2-hydroxyethanone 1313280-75-9 C24H22ClFN6O2
(R)-2-(2-chlorophenyl)-1-((R)-3-(2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)pyrimidin-4-ylamino)piperidin-1-yl)-2-hydroxyethanone
—— (S)-2-ethoxy-N-(4-(1-ethyl-3-methyl-1H-pyrazole-5-carboxamido)-1-phenylbutan-2-yl)-N,6-dimethylisonicotinamide 1312559-85-5 C27H35N5O3
(S)-2-ethoxy-N-(4-(1-ethyl-3-methyl-1H-pyrazole-5-carboxamido)-1-phenylbutan-2-yl)-N,6-dimethylisonicotinamide
—— tert-butyl 4-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,4-dioxo-6-phenyl-1,4-dihydrothieno[3,2-d]pyrimidin-3(2H)-yl}piperidine-1-carboxylate 1312599-70-4 C26H29N5O5S
tert-butyl 4-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,4-dioxo-6-phenyl-1,4-dihydrothieno[3,2-d]pyrimidin-3(2H)-yl}piperidine-1-carboxylate
—— (R)-N-(3-ethyl-1-((6-methylpyridin-2-yl)methyl)-1H-indazol-4-yl)-7-(3-hydroxypyrrolidin-1-yl)imidazo[1,2-a]pyridine-3-carboxamide 1313408-40-0 C28H29N7O2
(R)-N-(3-ethyl-1-((6-methylpyridin-2-yl)methyl)-1H-indazol-4-yl)-7-(3-hydroxypyrrolidin-1-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— 4-{4-[4-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)pyridin-2-yl]-piperazin-1-yl}butan-1-ol 1312461-39-4 C27H39N3O
4-{4-[4-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)pyridin-2-yl]-piperazin-1-yl}butan-1-ol
—— methyl 5-[4-({[6-(3-fluorophenyl)pyridin-3-yl]carbonyl}amino)piperidin-1-yl]pyrazine-2-carboxylate 1033839-29-0 C23H22FN5O3
methyl 5-[4-({[6-(3-fluorophenyl)pyridin-3-yl]carbonyl}amino)piperidin-1-yl]pyrazine-2-carboxylate
—— rac-N-(3-{4-[5-(5-diethylaminomethyl-4-methyl-thiophen-2-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-2-hydroxy-propyl)-sulfamic acid dimethyl-amide 1160955-81-6 C23H33N5O4S2
rac-N-(3-{4-[5-(5-diethylaminomethyl-4-methyl-thiophen-2-yl)-[1,2,4]oxadiazol-3-yl]-phenyl}-2-hydroxy-propyl)-sulfamic acid dimethyl-amide
—— N-methyl-4-(1-(naphthalen-1-ylsulfonyl)piperidin-4-yloxy)picolinamide 1073503-02-2 C22H23N3O4S
N-methyl-4-(1-(naphthalen-1-ylsulfonyl)piperidin-4-yloxy)picolinamide
—— 4-[(4-{2-[((1R,2S)-1-amino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylamino}-butyl)-methyl-amino]-butyric acid methyl ester 1051392-64-3 C22H34N4O5S
4-[(4-{2-[((1R,2S)-1-amino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylamino}-butyl)-methyl-amino]-butyric acid methyl ester
—— (2S,4R)-4-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-2-[(1R,2S)-1-(2-{2-[2-(2-methoxycarbonyl-ethoxy)-ethoxy]-acetylamino}-benzenesulfonylaminocarbonyl)-2-vinyl-cyclopropylcarbamoyl]-pyrrolidine-1-carboxylic acid tert-butyl ester 1051392-24-5 C46H57N7O13S2
(2S,4R)-4-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-2-[(1R,2S)-1-(2-{2-[2-(2-methoxycarbonyl-ethoxy)-ethoxy]-acetylamino}-benzenesulfonylaminocarbonyl)-2-vinyl-cyclopropylcarbamoyl]-pyrrolidine-1-carboxylic acid tert-butyl ester
—— 6-amino-2-(butyloxy)-9-{4-[4-(1-methylethyl)-1-piperazinyl]butyl}-7,9-dihydro-8H-purin-8-one 1207679-93-3 C20H35N7O2
6-amino-2-(butyloxy)-9-{4-[4-(1-methylethyl)-1-piperazinyl]butyl}-7,9-dihydro-8H-purin-8-one
—— 7-cyclopentyl-2-{5-[4-(2-hydroxyethyl)piperazin-1-yl]-pyridin-2-ylamino}-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide 1211440-85-5 C25H34N8O2
7-cyclopentyl-2-{5-[4-(2-hydroxyethyl)piperazin-1-yl]-pyridin-2-ylamino}-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide
—— 3-[7-(9,9-Dimethylfluoren-2-yl)-9,9-dimethylfluoren-2-yl]benzo[c]phenanthrene 1310543-27-1 C48H36
3-[7-(9,9-Dimethylfluoren-2-yl)-9,9-dimethylfluoren-2-yl]benzo[c]phenanthrene
—— 7-acetonyloxy-3-ethyl-4,5-dimethylcoumarin 1494571-36-6 C16H18O4
7-acetonyloxy-3-ethyl-4,5-dimethylcoumarin
—— (R)-1-(4-aminobenzyl)-3-(2-(2-((4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl)methyl)pyrrolidin-1-yl)-2-oxoethyl)urea 1313214-46-8 C18H25N7O3
(R)-1-(4-aminobenzyl)-3-(2-(2-((4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl)methyl)pyrrolidin-1-yl)-2-oxoethyl)urea
—— N-[1-(3,6-diethylpyrazin-2-yl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide 1033839-33-6 C25H28FN5O
N-[1-(3,6-diethylpyrazin-2-yl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide
—— N-(3-{3-[2-({4-[2-(dimethylamino)ethyl]phenyl}amino)pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl}phenyl)-2-(thiophen-2-yl)acetamide 1301134-73-5 C33H31N7OS
N-(3-{3-[2-({4-[2-(dimethylamino)ethyl]phenyl}amino)pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl}phenyl)-2-(thiophen-2-yl)acetamide
—— tert-butyl 4-[1-{[1-(methoxymethyl)-1H-tetrazol-5-yl]methyl}-2,4-dioxo-6-phenyl-1,4-dihydrothieno[3,2-d]pyrimidin-3(2H)-yl]piperidine-1-carboxylate 1312599-95-3 C26H31N7O5S
tert-butyl 4-[1-{[1-(methoxymethyl)-1H-tetrazol-5-yl]methyl}-2,4-dioxo-6-phenyl-1,4-dihydrothieno[3,2-d]pyrimidin-3(2H)-yl]piperidine-1-carboxylate
—— 5-(5-(3-(1-tert-butyl-3-(2,2-dimethyl-3-oxopiperazine-1-carbonyl)-1H-pyrazol-4-yl)ureido)-2-methylphenyl)-N-ethylpyridine-2-carboxamide 1207877-28-8 C30H38N8O4
5-(5-(3-(1-tert-butyl-3-(2,2-dimethyl-3-oxopiperazine-1-carbonyl)-1H-pyrazol-4-yl)ureido)-2-methylphenyl)-N-ethylpyridine-2-carboxamide
—— 1-(5-tert-butyl-3-(2,2-dimethyl-3-oxopiperazine-1-carbonyl)thiophen-2-yl)-3-(4-methyl-3-(pyridin-3-yl)phenyl)urea 1207876-34-3 C28H33N5O3S
1-(5-tert-butyl-3-(2,2-dimethyl-3-oxopiperazine-1-carbonyl)thiophen-2-yl)-3-(4-methyl-3-(pyridin-3-yl)phenyl)urea
—— 7-[5-chloro-4-(2-methoxy-4-morpholin-4-yl-phenylamino)-pyrimidin-2-ylamino]-6-methoxy-1-methyl-1,3,4,5-tetrahydro-benzo[b]azepin-2-one 1022960-58-2 C27H31ClN6O4
7-[5-chloro-4-(2-methoxy-4-morpholin-4-yl-phenylamino)-pyrimidin-2-ylamino]-6-methoxy-1-methyl-1,3,4,5-tetrahydro-benzo[b]azepin-2-one
—— (2S,5R)-5-(2-chlorophenyl)-1-(2'-cyano-4'-methoxy-[1,1'-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid 1312802-87-1 C26H21ClN2O4
(2S,5R)-5-(2-chlorophenyl)-1-(2'-cyano-4'-methoxy-[1,1'-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid
—— 1-(4-acetylphenyl)-3-{(4-(methylsulfonyl)phenyl)amino}-1H-pyrazole-4-carbonitrile 1207176-42-8 C19H16N4O3S
1-(4-acetylphenyl)-3-{(4-(methylsulfonyl)phenyl)amino}-1H-pyrazole-4-carbonitrile
—— 5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-2-[2-(S)-(hydroxymethyl)morpholin-4-yl]-1,3-thiazol-4(5H)-one 1312703-96-0 C24H20ClF3N4O3S
5-({1-[4-chloro-2-(trifluoromethyl)benzyl]-1H-indazol-5-yl}methylidene)-2-[2-(S)-(hydroxymethyl)morpholin-4-yl]-1,3-thiazol-4(5H)-one
—— (2S,5R)-1-(2-([1,1'-biphenyl]-4-yl)acetyl)-5-(2-chlorophenyl)pyrrolidine-2-carboxylic acid 1312799-83-9 C25H22ClNO3
(2S,5R)-1-(2-([1,1'-biphenyl]-4-yl)acetyl)-5-(2-chlorophenyl)pyrrolidine-2-carboxylic acid
—— N-(5-((3R,8aS)-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]pyrazine-2-carbonyl)-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)picolinamide 1072100-09-4 C22H29N7O3
N-(5-((3R,8aS)-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]pyrazine-2-carbonyl)-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)picolinamide
—— 3-[1-[3-fluoro-5-(5-fluoro-3-methylindol-1-yl)benzyl]-5-((S)-2-methylaminopropionylamino)-6-oxo-1,6-dihydropyrimidin-2-yl]-N-methylbenzamide 1032999-77-1 C32H30F2N6O3
3-[1-[3-fluoro-5-(5-fluoro-3-methylindol-1-yl)benzyl]-5-((S)-2-methylaminopropionylamino)-6-oxo-1,6-dihydropyrimidin-2-yl]-N-methylbenzamide
—— 8-(2-{[(1R,2S)-1-({(2S,4R)-4-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-pyrrolidine-2-carbonyl}-amino)-2-vinyl-cyclopropanecarbonyl]-sulfamoyl}-phenylcarbamoyl)-octanoic acid 1051395-11-9 C42H51N7O9S2
8-(2-{[(1R,2S)-1-({(2S,4R)-4-[2-(2-isopropylamino-thiazol-4-yl)-7-methoxy-quinolin-4-yloxy]-pyrrolidine-2-carbonyl}-amino)-2-vinyl-cyclopropanecarbonyl]-sulfamoyl}-phenylcarbamoyl)-octanoic acid
—— (1R,2S,2'R,6'S,24a'S)-6'-[(morpholin-4-ylcarbonyl)amino]-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate 1051390-44-3 C40H50FN7O9S
(1R,2S,2'R,6'S,24a'S)-6'-[(morpholin-4-ylcarbonyl)amino]-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate
—— 2-methyl-pyrimidine-5-carboxylic acid (1-{[3-methyl-5-(2-trifluoromethyl-phenylamino)-pyridin-2-ylmethyl]-carbamoyl}-cyclopropyl)-amide 1242455-55-5 C24H23F3N6O2
2-methyl-pyrimidine-5-carboxylic acid (1-{[3-methyl-5-(2-trifluoromethyl-phenylamino)-pyridin-2-ylmethyl]-carbamoyl}-cyclopropyl)-amide
—— 4-ethyl-2,4-dihydro-5-((6-(4-bromophenyl)imidazo[2,1-b]thiazol-3-yl)methyl)-3H-1,2,4-triazole-3-thione 1212415-46-7 C16H14BrN5S2
4-ethyl-2,4-dihydro-5-((6-(4-bromophenyl)imidazo[2,1-b]thiazol-3-yl)methyl)-3H-1,2,4-triazole-3-thione
—— 2-{5-[5-[(5-Chloropyrimidin-2-yl)thio]-2-(3,4-difluorophenyl)-1,3-oxazol-4-yl]pyridin-2-yl}propan-2-ol 1207745-82-1 C21H15ClF2N4O2S
2-{5-[5-[(5-Chloropyrimidin-2-yl)thio]-2-(3,4-difluorophenyl)-1,3-oxazol-4-yl]pyridin-2-yl}propan-2-ol
—— {5-[5-bromo-6-(2-chloro-phenoxy)-pyridine-3-sulfonylamino]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid 1208100-01-9 C23H20BrClN2O6S
{5-[5-bromo-6-(2-chloro-phenoxy)-pyridine-3-sulfonylamino]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid
—— (R)-cyclopentylhydroxyphenylacetic acid 1-(N-benzofuran-5-ylmethylcarbamimidoyl)piperidin-4-yl ester 1128093-05-9 C28H33N3O4
(R)-cyclopentylhydroxyphenylacetic acid 1-(N-benzofuran-5-ylmethylcarbamimidoyl)piperidin-4-yl ester
—— N-[4-[(2S)-morpholin-2-yl]phenyl]-6-(trifluoromethyl)pyridine-3-carboxamide 1312571-05-3 C17H16F3N3O2
N-[4-[(2S)-morpholin-2-yl]phenyl]-6-(trifluoromethyl)pyridine-3-carboxamide
—— 1-(2-pyrrolidin-1-yl-ethyl)-1H-indole-3-carboxylic acid hydrochloride 1313042-66-8 C15H18N2O2*ClH
1-(2-pyrrolidin-1-yl-ethyl)-1H-indole-3-carboxylic acid hydrochloride
—— 7-[2-(1,1-dioxidothiomorpholin-4-yl)ethyl]pyrazolo[3,4-b]pyrrolo[3,4-d]pyridine-6,8(3H,7H)-dione 1246615-65-5 C14H15N5O4S
7-[2-(1,1-dioxidothiomorpholin-4-yl)ethyl]pyrazolo[3,4-b]pyrrolo[3,4-d]pyridine-6,8(3H,7H)-dione