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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-{2-(4-tert-butyl-phenyl)-2-[4-(2',4'-dichlorobiphenyl-4-yl)-1H-imidazol-2-yl]-ethyl}benzoylamino)-ethanesulfonic acid 1208222-93-8 C36H35Cl2N3O4S
2-(4-{2-(4-tert-butyl-phenyl)-2-[4-(2',4'-dichlorobiphenyl-4-yl)-1H-imidazol-2-yl]-ethyl}benzoylamino)-ethanesulfonic acid
—— 7-cyclopentyl-2-(5-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide 1211440-98-0 C27H38N8O3
7-cyclopentyl-2-(5-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide
—— 4-(3-(2-chlorophenyl)-4-(methoxy(4-(1-propylazetidin-3-yloxy)phenyl)methyl)-isoxazol-5-yl)phenol 1383928-64-0 C29H29ClN2O4
4-(3-(2-chlorophenyl)-4-(methoxy(4-(1-propylazetidin-3-yloxy)phenyl)methyl)-isoxazol-5-yl)phenol
—— —— 132308-64-6 C16H13N5O2
—— ethyl 2-<2'-<<2''-(butoxycarbonylaminomethyl)thiazole>-4''-carboxamidomethyl>thiazole-4'-carboxamidomethyl>-thiazole-4-carboxylate 120455-34-7 C22H26N6O6S3
ethyl 2-<2'-<<2''-(butoxycarbonylaminomethyl)thiazole>-4''-carboxamidomethyl>thiazole-4'-carboxamidomethyl>-thiazole-4-carboxylate
—— 3-benzyl-3,4-dihydro-quinazolin-8-ol 100969-12-8 C15H14N2O
3-benzyl-3,4-dihydro-quinazolin-8-ol
—— 1-(N-methylpiperazino)methyl-3-[4'-(4''-nitrobenzyloxy)benzohydrazono]isatin 1314798-76-9 C28H28N6O5
1-(N-methylpiperazino)methyl-3-[4'-(4''-nitrobenzyloxy)benzohydrazono]isatin
—— 4-methoxyphenyl (2-O-acetyl-3-O-benzyl-4,6-O-benzylidene-α-D-galactopyranosyl)-(1->3)-2-azido-4,6-O-benzylidene-2-deoxy-α-D-glucopyranoside 1370599-41-9 C42H43N3O12
4-methoxyphenyl (2-O-acetyl-3-O-benzyl-4,6-O-benzylidene-α-D-galactopyranosyl)-(1->3)-2-azido-4,6-O-benzylidene-2-deoxy-α-D-glucopyranoside
—— 1-(L-leucyl-L-alanyl-L-arginylglycyl-L-tyrosyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazole-5-carboxamide 1071446-47-3 C34H47N11O8
1-(L-leucyl-L-alanyl-L-arginylglycyl-L-tyrosyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazole-5-carboxamide
—— 9-[(1R,2S,5R)-menthoxycarbonyl]cyclobrassinin 1417888-91-5 C22H28N2O2S2
9-[(1R,2S,5R)-menthoxycarbonyl]cyclobrassinin
—— 5-(benzylideneamino)-6-cyano-7H-7-(4-methoxyphenyl)-2-(4-sulphamoylphenylamino)pyrano[2,3-d]thiazole 1382846-48-1 C27H21N5O4S2
5-(benzylideneamino)-6-cyano-7H-7-(4-methoxyphenyl)-2-(4-sulphamoylphenylamino)pyrano[2,3-d]thiazole
—— hydroxy<N-(3-methyl-3-butenyl)N-(methoxycarbonyl)amino>acetic acid dimethyl ester 136294-42-3 C10H17NO5
hydroxy<N-(3-methyl-3-butenyl)N-(methoxycarbonyl)amino>acetic acid dimethyl ester
—— —— 132738-71-7 C20H28O2Si
—— 7-cyclopentyl-2-{5-[(S)-4-(2-hydroxy-ethyl)-3-methyl-piperazin-1-yl]-pyridin-2-ylamino}-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide 1211442-17-9 C26H36N8O2
7-cyclopentyl-2-{5-[(S)-4-(2-hydroxy-ethyl)-3-methyl-piperazin-1-yl]-pyridin-2-ylamino}-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide
—— N-[3-(2,4-dichloro-phenyl)-2,6-dimethyl-pyrazolo[5,1-b]oxazol-7-yl]-N-ethyl-propionamide 1207257-87-1 C18H19Cl2N3O2
N-[3-(2,4-dichloro-phenyl)-2,6-dimethyl-pyrazolo[5,1-b]oxazol-7-yl]-N-ethyl-propionamide
—— 4-[4-(2,4-difluorophenyl)-8-(2,6-difluorophenyl)-7-oxy-1,7-naphthyridin-2-yloxy]-piperidine-1-carboxylic acid tert-butyl ester 1006380-37-5 C30H27F4N3O4
4-[4-(2,4-difluorophenyl)-8-(2,6-difluorophenyl)-7-oxy-1,7-naphthyridin-2-yloxy]-piperidine-1-carboxylic acid tert-butyl ester
—— (S)-2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-4-(1-(4-fluorophenyl)butylamino)pyrimidine-5-carboxamide 1313281-12-7 C22H20F2N6O
(S)-2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-4-(1-(4-fluorophenyl)butylamino)pyrimidine-5-carboxamide
—— ethyl (3-dimethylamino-4-methoxyphenyl)acetate 1012071-59-8 C13H19NO3
ethyl (3-dimethylamino-4-methoxyphenyl)acetate
—— (R)-N-allyl-N-(1-phenylethyl)pivalamide 1529788-01-9 C16H23NO
(R)-N-allyl-N-(1-phenylethyl)pivalamide
—— 1-(5-tert-butoxycarbonyl-3-ethyl-4-methyl-2-pyrrolylmethyl)indole-3-carbaldehyde 1352632-60-0 C22H26N2O3
1-(5-tert-butoxycarbonyl-3-ethyl-4-methyl-2-pyrrolylmethyl)indole-3-carbaldehyde
—— tert-butyl 4-{N-[5-(N-benzylsulfamoyl)-2-methoxyphenyl]-N-methyl amino} piperidine-1-carboxylate 1245239-20-6 C25H35N3O5S
tert-butyl 4-{N-[5-(N-benzylsulfamoyl)-2-methoxyphenyl]-N-methyl amino} piperidine-1-carboxylate
—— (+)-2-[4’-((S)-3-methylpentyloxy)phenyl]-5-(4’-hexyloxyphenyl)styrene 1469925-57-2 C32H40O2
(+)-2-[4’-((S)-3-methylpentyloxy)phenyl]-5-(4’-hexyloxyphenyl)styrene
—— (R)-1-[3-((R)-cyclohexyl-hydroxy-phenyl-methyl)-isoxazol-5-ylmethyl]-3-(2,3-dihydro-benzofuran-5-yloxy)-1-azonia-bicyclo[2.2.2]octane chloride 1208426-54-3 C32H39N2O4*Cl
(R)-1-[3-((R)-cyclohexyl-hydroxy-phenyl-methyl)-isoxazol-5-ylmethyl]-3-(2,3-dihydro-benzofuran-5-yloxy)-1-azonia-bicyclo[2.2.2]octane chloride
—— 2-chloro-N-[(1R)-6-(8-pyridin-4-yl-3,8-diazaspiro[4.5]decane-3-carbonyl)-2,3-dihydro-1H-inden-1-yl]-N-(2,2,2-trifluoro-ethyl)-benzamide 1246498-59-8 C32H32ClF3N4O2
2-chloro-N-[(1R)-6-(8-pyridin-4-yl-3,8-diazaspiro[4.5]decane-3-carbonyl)-2,3-dihydro-1H-inden-1-yl]-N-(2,2,2-trifluoro-ethyl)-benzamide
—— tert-butyl (S)-3-(pyridin-4-yloxy)pyrrolidine-1-carboxylate 1138448-27-7 C14H20N2O3
tert-butyl (S)-3-(pyridin-4-yloxy)pyrrolidine-1-carboxylate
—— 2-[2-(1H-benzotriazol-5-ylcarbamoyl)ethyl]-5-[3-(4-chlorophenyl)ureido]-1H-imidazole-4-carboxamide 1143506-92-6 C20H18ClN9O3
2-[2-(1H-benzotriazol-5-ylcarbamoyl)ethyl]-5-[3-(4-chlorophenyl)ureido]-1H-imidazole-4-carboxamide
—— N'-[1-[3-bromo-4-(3-hydroxypropoxy)phenyl]ethyl]-N-(4-carbamimidoylphenyl)propanediamide 1100769-48-9 C21H25BrN4O4
N'-[1-[3-bromo-4-(3-hydroxypropoxy)phenyl]ethyl]-N-(4-carbamimidoylphenyl)propanediamide
—— [4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-[7-cyclopropyl-1-(2-methoxy-ethyl)-1H-indol-3-yl]-methanone hydrochloride 1313040-21-9 C27H32FN3O2*ClH
[4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-[7-cyclopropyl-1-(2-methoxy-ethyl)-1H-indol-3-yl]-methanone hydrochloride
—— 2-amino-1-[2-(4-fluorophenyl)-3-{[4-(trifluoromethyl)phenyl]amino}-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]-2-methylpropan-1-one 1261110-58-0 C23H23F4N5O
2-amino-1-[2-(4-fluorophenyl)-3-{[4-(trifluoromethyl)phenyl]amino}-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]-2-methylpropan-1-one
—— N-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide 1033840-99-1 C24H28FN5O
N-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide
—— (2S,5R)-1-(3'-carbamoyl-4'-cyano-[1,1'-biphenyl]-4-carbonyl)-5-(2-chlorophenyl)pyrrolidine-2-carboxylic acid 1312802-72-4 C26H20ClN3O4
(2S,5R)-1-(3'-carbamoyl-4'-cyano-[1,1'-biphenyl]-4-carbonyl)-5-(2-chlorophenyl)pyrrolidine-2-carboxylic acid
—— (2S,5R)-5-(2-chlorophenyl)-1-(4-(4,6-dimethoxypyrimidin-5-yl)benzoyl)pyrrolidine-2-carboxylic acid 1312803-43-2 C24H22ClN3O5
(2S,5R)-5-(2-chlorophenyl)-1-(4-(4,6-dimethoxypyrimidin-5-yl)benzoyl)pyrrolidine-2-carboxylic acid
—— (RS)-N-[4-(1-(2-phenyl)ethyl-pyrrolidin-3-yl)-phenyl]-4-chloro-benzamide 1312559-34-4 C25H25ClN2O
(RS)-N-[4-(1-(2-phenyl)ethyl-pyrrolidin-3-yl)-phenyl]-4-chloro-benzamide
—— (2-aminomethyl-thiazolidin-3-yl)-[5-(3-fluoro-phenyl)-thiazol-4-yl]-methanone 1204585-98-7 C14H14FN3OS2
(2-aminomethyl-thiazolidin-3-yl)-[5-(3-fluoro-phenyl)-thiazol-4-yl]-methanone
—— N-[3-(6-(3-aminophenyl)pyrimidin-4-ylamino)benzyl]methanesulfonamide 1313219-39-4 C18H19N5O2S
N-[3-(6-(3-aminophenyl)pyrimidin-4-ylamino)benzyl]methanesulfonamide
—— N-{1-[(6-fluoro-1H-indol-3-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide 1033839-70-1 C26H24F2N4O
N-{1-[(6-fluoro-1H-indol-3-yl)methyl]piperidin-4-yl}-6-(3-fluorophenyl)nicotinamide
—— ethyl 2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-4-(pyridin-3-ylmethylamino)pyrimidin-5-carboxylate 1313279-64-9 C20H17FN6O2
ethyl 2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-4-(pyridin-3-ylmethylamino)pyrimidin-5-carboxylate
—— (2S,3S)-3-hydroxypyrrolidine-2-carboxylic acid [6'-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-3,4,5,6-tetrahydro-2H-1,2'-bipyridinyl-4-yl]amide 1312462-19-3 C29H40N4O2
(2S,3S)-3-hydroxypyrrolidine-2-carboxylic acid [6'-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-3,4,5,6-tetrahydro-2H-1,2'-bipyridinyl-4-yl]amide
—— N-(8-methoxytetralin-2-yl)-N-propyl-2-(2-biphenyl-4-yl)acetamide 1313030-59-9 C28H31NO2
N-(8-methoxytetralin-2-yl)-N-propyl-2-(2-biphenyl-4-yl)acetamide
—— (R)-3-(tert-butoxycarbonylamino)-1-(4-methyl-5-isoquinolinesulfonyl)-piperidine 1052078-68-8 C20H27N3O4S
(R)-3-(tert-butoxycarbonylamino)-1-(4-methyl-5-isoquinolinesulfonyl)-piperidine
—— —— 1443771-43-4 C16H17IN2O
—— [5-[2-(dimethylamino)ethyl-methylamino]pyrazin-2-yl]-[2-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-3-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone 1421502-99-9 C31H34FN9O2
[5-[2-(dimethylamino)ethyl-methylamino]pyrazin-2-yl]-[2-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-3-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone
—— 6-(thiazol-4-yl)-2-(4-trifluoromethylthiazol-2-yl)pyrimidin-4-ol 1251166-60-5 C11H5F3N4OS2
6-(thiazol-4-yl)-2-(4-trifluoromethylthiazol-2-yl)pyrimidin-4-ol
—— 2-(3-chloropyridin-2-yl)-N-[2-(cyanomethylcarbamoyl)-4,6-dimethylphenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229655-39-3 C23H18ClF3N10O2
2-(3-chloropyridin-2-yl)-N-[2-(cyanomethylcarbamoyl)-4,6-dimethylphenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
—— 6-({3-(aminocarbonyl)-5-[2-fluoro-4-(1-hydroxy-1-methylethyl)phenyl]-2-thienyl}amino)-N-(2-hydroxyethyl)pyridine-2-carboxamide 1093874-63-5 C22H23FN4O4S
6-({3-(aminocarbonyl)-5-[2-fluoro-4-(1-hydroxy-1-methylethyl)phenyl]-2-thienyl}amino)-N-(2-hydroxyethyl)pyridine-2-carboxamide
—— 6-[(R)-1-acetylpyrrolidin-2-yl]-5-(6-methoxymethylpyridin-3-yloxy)-2-(pyrazin-2-yl)-1H-indole 1207627-62-0 C25H25N5O3
6-[(R)-1-acetylpyrrolidin-2-yl]-5-(6-methoxymethylpyridin-3-yloxy)-2-(pyrazin-2-yl)-1H-indole
—— 5-(3-Chlorophenyl)-4-(1-methyltetrazol-5-yl)sulfanylthieno[2,3-d]pyrimidine 1370338-76-3 C14H9ClN6S2
5-(3-Chlorophenyl)-4-(1-methyltetrazol-5-yl)sulfanylthieno[2,3-d]pyrimidine
—— 6-(3-fluorophenyl)-N-{1-[2-(2-hydroxyethoxy)benzyl]piperidin-4-yl}nicotinamide 1033840-78-6 C26H28FN3O3
6-(3-fluorophenyl)-N-{1-[2-(2-hydroxyethoxy)benzyl]piperidin-4-yl}nicotinamide
—— 1-(4-(7-phenyl-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-6-yl)phenyl)cyclobutanamine 1313438-69-5 C23H23N3O
1-(4-(7-phenyl-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-6-yl)phenyl)cyclobutanamine
—— 4-(3-oxothiolan-2-ylidenemethyl)phenylacetic acid 1012312-14-9 C13H12O3S
4-(3-oxothiolan-2-ylidenemethyl)phenylacetic acid